Opioid Receptor
Opioid receptors are a group of G protein-coupled receptors that mediate the effects of endogenous and exogenous opioids. These receptors play a central role in pain modulation, mood regulation, and addictive behaviors. Opioid receptor agonists and antagonists are extensively used in pain management and addiction treatment, as well as in research on neurological and psychiatric disorders. At CymitQuimica, we provide a comprehensive selection of high-quality opioid receptor modulators to support your research in neurobiology, pain management, and addiction therapy.
Found 327 products of "Opioid Receptor"
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ADL-5747
CAS:ADL-5747 (ADL-5747 (free base)) (free base) is a delta opioid receptor agonist used in the treatment of neurological disorders, skin and musculoskeletalFormula:C24H28N2O3Purity:98.94% - 99.74%Color and Shape:SolidMolecular weight:392.49ML-335
CAS:ML-335, a μ-δ targeted agonist and MOR/DOR ligand, may lead to isomer-biased drugs with pain-relief properties.Formula:C25H32N2O3Purity:98.58%Color and Shape:SolidMolecular weight:408.53Ref: TM-T23002
5mg44.00€10mg64.00€25mg112.00€50mg175.00€100mg253.00€200mg359.00€1mL*10mM (DMSO)33.00€JNJ-20788560
CAS:JNJ-20788560 is a delta opioid receptor (DOR) agonist with analgesic activity. It is more selective for DOR than for mu opioid receptors (MOR).
Formula:C25H28N2O2Purity:98.02%Color and Shape:SolidMolecular weight:388.5Bevenopran
CAS:Bevenopran (CB-5945) is a peripheral antagonist of μ-opioid receptor and can be used in studies about the treatment of opioid-induced bowel dysfunction.Formula:C20H26N4O4Purity:98.69% - 98.9%Color and Shape:SolidMolecular weight:386.44Ref: TM-T14551
1mg62.00€5mg130.00€10mg187.00€25mg299.00€50mg408.00€100mg532.00€200mg705.00€1mL*10mM (DMSO)142.00€SCH-486757
CAS:SCH-486757 is an agonist of nociceptin-1 (NOP1) and orphanin FQ peptide receptors and is used in the study of cough.Formula:C24H23Cl2N3OPurity:99.53% - >99.99%Color and Shape:SolidMolecular weight:440.37Trimebutine CTB salt
CAS:Trimebutine CTB salt (GIC-1001) is an opioid receptor agonist used in the study of pain.Formula:C29H36N2O8S2Purity:99.85% - >99.99%Color and Shape:SolidMolecular weight:604.74ICI 199,441 hydrochloride
CAS:ICI 199,441 hydrochloride is a potent, selective agonist of κ-opioid receptor.Formula:C21H25Cl3N2OPurity:99.57%Color and Shape:SolidMolecular weight:427.8Ref: TM-T22849
2mg33.00€5mg52.00€10mg75.00€25mg138.00€50mg215.00€100mg314.00€200mg442.00€1mL*10mM (DMSO)58.00€Frakefamide
CAS:Frakefamide: potent analgesic, μ-selective agonist, non-CNS penetrating.Formula:C30H34FN5O5Purity:98%Color and Shape:SolidMolecular weight:563.62Mu opioid receptor antagonist 7
CAS:Compound 24, also known as Mu opioid receptor antagonist 7, is a potent, centrally-acting µ-opioid receptor (µOR) antagonist with an inhibitory concentration (Formula:C22H27ClN2O2Purity:98%Color and Shape:SolidMolecular weight:386.91μ opioid receptor agonist 3
CAS:Compound 20, identified as μ opioid receptor agonist 3, is a potent µOR agonist that exhibits an EC50 value of 0.87 nM.Formula:C22H28N2O2Purity:98%Color and Shape:SolidMolecular weight:352.47ICI 204448
CAS:ICI 204448 is a potent and peripherally selective κ-opioid agonist.Formula:C23H26Cl2N2O4Color and Shape:SolidMolecular weight:465.37Icalcaprant
CAS:Icalcaprant is a kappa-opioid receptor antagonist [1].Formula:C23H26N4O3Purity:98%Color and Shape:SolidMolecular weight:406.48DPI-3290
CAS:DPI-3290 is a specific agonist of opioid receptors (Ki: 0.18 nM, 0.46 nM, and 0.62 nM for δ-, μ-, and κ-opioid receptors, respectively) with potentFormula:C30H34FN3O2Purity:98%Color and Shape:SolidMolecular weight:487.61CYT-1010
CAS:CYT-1010, a mu-opioid receptor agonist; EC50: β-arrestin, 13.1 nM; cAMP, 0.0053 nM. Extracted from patent WO2013173730A2.Formula:C35H40N6O5Purity:98%Color and Shape:SolidMolecular weight:624.73N-Benzylnaltrindole hydrochloride
CAS:δ2 opioid receptor antagonistFormula:C33H33ClN2O3Purity:98%Color and Shape:SolidMolecular weight:541.08Deltakephalin
CAS:Deltakephalin is a synthetic, potent specific opiate delta receptors agonist.Formula:C34H48N6O10Purity:98%Color and Shape:SolidMolecular weight:700.78MR2034
CAS:MR2034 is an agonist of kappa-Opioid receptor. MR2034 stimulates hypothalamic-pituitary-adrenal axis.Formula:C19H27NO2Color and Shape:SolidMolecular weight:301.42Naloxonazine
CAS:Naloxonazine, a potent, selective opiate mu-1 (μ1) antagonist, also influences leishmania through the modulation of host coding function.Formula:C38H42N4O6Color and Shape:SolidMolecular weight:650.76ADL-08-0011
CAS:ADL-08-0011 is an metabolite of alvimopan.Formula:C23H29NO3Color and Shape:SolidMolecular weight:367.49R-84760 hydrochloride
CAS:R-84760, a potent κ-opioid receptor agonist, relieves tonic pain via supraspinal/spinal pathways, activating noradrenergic descent.Formula:C19H25Cl3N2OSColor and Shape:SolidMolecular weight:435.84Trap-101 hydrochloride
CAS:nociceptin/orphanin FQ (NOP) receptor antagonistFormula:C24H36ClN3O2Purity:98%Color and Shape:SolidMolecular weight:434.02μ opioid receptor agonist 1
CAS:μ opioid receptor agonist 1 (Compound H-1a) is an optically pure oxyheterocyclic substituted pyrroloxypyrazole derivative and an MOR receptor agonist that canFormula:C26H38N4OColor and Shape:SolidMolecular weight:422.61Ro 48-6791
CAS:Ro 48-6791, a GABA receptor agonist, is used potentially for anesthesia.Formula:C21H25FN6O2Color and Shape:SolidMolecular weight:412.46ADL 08-0011 HCl
CAS:ADL 08-0011, a μ-opioid antagonist with Ki 0.25 nM, is derived from alvimopan by gut microbes and counteracts loperamide effects in rats.Formula:C23H30ClNO3Color and Shape:SolidMolecular weight:403.947Salvinorin A Carbamate
CAS:Salvinorin A carbamate, a potent κ-opioid receptor (KOR) full agonist, exhibits nearly the same potency as salvinorin A, with EC50 values of 6.2 and 4.5 nM, respectively, for activating the human KOR to augment the binding of [35S]GTPγS. Enhancing biological stability, the addition of a carbamate group to salvinorin A reduces deacetylation.Formula:C22H27NO8Color and Shape:SolidMolecular weight:433.457Prodilidine hydrochloride
CAS:Prodilidine hydrochloride is an opioid analgesic.Formula:C15H22ClNO2Color and Shape:SolidMolecular weight:283.79PD 117302
CAS:PD 117302: nonpeptide, kappa-opioid agonist, anti-arrhythmic, anticonvulsant, impacts locomotion, diuresis.Formula:C21H28N2OSColor and Shape:SolidMolecular weight:356.52Naloxonazine dihydrochloride
CAS:μ1 receptor antagonistFormula:C38H43ClN4O6Purity:98%Color and Shape:SolidMolecular weight:687.22SNC 162
CAS:SNC 162 is a potent and selective delta-opioid receptor (δ-opioid) agonist with analgesic, antidepressant and antiarrhythmic effects.Formula:C27H37N3OPurity:98%Color and Shape:SolidMolecular weight:419.6FK 33-824
CAS:FK 33-824, a stable synthetic analog of methionine enkephalin, reversible with naloxone.Formula:C29H41N5O7SPurity:98%Color and Shape:SolidMolecular weight:603.73Naldemedine tosylate
CAS:Naldemedine (S-297995) tosylate, a PAMORA, targets μ-, δ-, κ-opioid receptors, aiding OIC research, may bind to SARS-CoV2's 3CL pro.Formula:C39H42N4O9SColor and Shape:SolidMolecular weight:742.84DS34942424
DS34942424 is an orally potent analgesic which did not exhibit mu opioid receptor agonist activity.Formula:C15H17FN2OColor and Shape:SolidMolecular weight:260.31BU72
CAS:BU72 is a potent, long-lasting agonist for μ and κ opioid receptors, with partial agonistic activity at the δ opioid receptor (EC50 values of 0.054, 0.033, and 0.58 nM, respectively). It provides strong, enduring analgesic effects primarily mediated through μ opioid receptors. BU72 also exhibits a prolonged duration of activity and can partially reverse morphine-induced analgesia. It is applicable in studies of opioid dependence.Formula:C28H32N2O2Color and Shape:SolidMolecular weight:428.57Mu opioid receptor antagonist 5
Compound NAP: MOR antagonist, crosses blood-brain barrier, EC50: 1.14 nM, Ki: 0.37 nM, useful for OUD research.Formula:C26H29N3O4Color and Shape:SolidMolecular weight:447.53σ1 Receptor/μ Opioid receptor modulator 2
CAS:Compound 4x, also known as σ1 Receptor/μOpioid receptormodulator 2, acts as a μOR agonist and a σ1R antagonist, exhibiting a potent μOR EC50 of 0.6 nM and strong σ1R inhibitory activity (Ki: 363.7 nM). It demonstrates significant analgesic effects in various pain models.Formula:C23H31N3OMolecular weight:365.51Daeatal
CAS:Dynorphin A ethylamide (1-9), the opioid activities were examined in the bioassays.Formula:C56H93N19O10Purity:98%Color and Shape:SolidMolecular weight:1192.46BNTX maleate
CAS:δ1 opioid receptor antagonistFormula:C31H31NO8Purity:98%Color and Shape:SolidMolecular weight:545.58BW 443C
CAS:BW 443C is a selective agonist of mu-opioid receptor.Formula:C33H46N10O10Color and Shape:SolidMolecular weight:742.791Mu opioid receptor antagonist 2
Compound 25: potent, selective MOR antagonist, crosses blood-brain barrier (Ki: 0.37 nM, EC50: 0.44 nM), for OUD research.Formula:C25H28N2O4SColor and Shape:SolidMolecular weight:452.57Salvinorin A Propionate
CAS:Salvinorin A propionate: partial KOR agonist, Ki=32.6 nM, EC50=4.7 nM; ignores μ/δ/ORL-1, non-opioid receptors; less potent analgesic vs. salvinorin A.Formula:C24H30O8Color and Shape:SolidMolecular weight:446.49Phenethyl 4-ANPP
CAS:Phenethyl 4-ANPP is a MOR (μ-opioid receptor) agonist with a structure similar to known opioids.Formula:C27H32N2Color and Shape:SolidMolecular weight:384.56SB-612111
CAS:SB-612111: potent ORL-1 antagonist, Ki=0.33 nM; μ-, κ-, δ-receptor Ki=57.6, 160.5, 2109 nM; blocks nociceptin's pain effect.Formula:C24H29Cl2NOColor and Shape:SolidMolecular weight:418.40CCG258747
CAS:CCG258747 is a novel, selective inhibitor of the GRK2 subfamily.Formula:C28H27FN4O4Color and Shape:SolidMolecular weight:502.54Sunobinop
CAS:Sunobinop (S 117957) is an opioid receptor-like orphan receptor (ORL1) modulator.Formula:C26H33N3O3Color and Shape:SolidMolecular weight:435.56NOP agonist-1
CAS:NOP agonist-1 (compound 4) is a nociceptin opioid receptor (NOP) partial agonist that attenuates Parkinsonian disabilities in 6-OHDA hemilesioned rats [1].Formula:C22H34N2Molecular weight:326.52Mu opioid receptor antagonist 4
Compound 31: Potent, selective MOR antagonist; crosses blood-brain barrier; Ki & EC50: 0.38 nM; useful for OUD research.Formula:C25H28N2O4SColor and Shape:SolidMolecular weight:452.57SB-612111 hydrochloride
SB-612111 is a potent ORL-1 antagonist, with high affinity (Ki: 0.33 nM) and µ-receptor activity (Ki: 57.6 nM), blocking Nociceptin-induced pain.Formula:C24H30Cl3NOColor and Shape:SolidMolecular weight:454.86MTI013
MTI013 is a selective inhibitor of SARS-CoV-2 nsp14 Mtase (IC50: 2.98 µM) and an antiviral agent (IC50: 10.33 µM in HCoV-229E infected Huh7 cells). Additionally, MTI013 demonstrates synergistic antiviral effects when used in conjunction with the RdRp inhibitor SHEN26.Formula:C24H26N6O4SColor and Shape:SolidMolecular weight:494.57RX 809055AX
CAS:RX 809055AX is a long lasting opioid antagonist at mu and delta receptors.Formula:C29H29ClN2O4Color and Shape:SolidMolecular weight:505SC13
CAS:SC13, a novel mitragynine analog, exhibits low-efficacy agonism at Mu opioid receptors and provides antinociception while minimizing adverse effects.Formula:C26H30N2O5Color and Shape:SolidMolecular weight:450.53
