Opioid Receptor
Opioid receptors are a group of G protein-coupled receptors that mediate the effects of endogenous and exogenous opioids. These receptors play a central role in pain modulation, mood regulation, and addictive behaviors. Opioid receptor agonists and antagonists are extensively used in pain management and addiction treatment, as well as in research on neurological and psychiatric disorders. At CymitQuimica, we provide a comprehensive selection of high-quality opioid receptor modulators to support your research in neurobiology, pain management, and addiction therapy.
Found 327 products of "Opioid Receptor"
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BU09059
CAS:BU09059 is a potent, selective, short-acting antagonist of the κ-opioid receptor (KOR).Formula:C28H37N3O5Purity:98%Color and Shape:SolidMolecular weight:495.61Mu opioid receptor antagonist 3
Potent, selective MOR antagonist (compound 26); crosses blood-brain barrier. Ki: 0.24 nM, EC50: 0.54 nM; for studying OUD.Formula:C25H28N2O4SColor and Shape:SolidMolecular weight:452.57Allyphenyline oxalate
CAS:The pKi values of Allyphenyline oxalate (compound 9) for the α2-adrenergic receptor subtypes α2A, α2B, and α2C are 7.24, 6.47, and 7.07, respectively.Formula:C16H20N2O5Color and Shape:SolidMolecular weight:320.34rel-SB-612111 hydrochloride
CAS:NOP receptor antagonistFormula:C24H30Cl3NOPurity:98%Color and Shape:SolidMolecular weight:454.86(S)-MCOPPB
CAS:(S)-MCOPPB is the S-enantiomer of MCOPPB, an orally active selective agonist for the Nociceptin/Orphanin FQ-Receptor. It inhibits signal transduction in mouse brain NOP receptors and is utilized in anxiety disorder research.Formula:C26H40N4Color and Shape:SolidMolecular weight:408.623Opioid receptor antagonist 1
CAS:Opioid receptor antagonist 1 (Compound 10) is an Orvinol-based antagonist of opioid receptors. It exhibits activity as an antagonist against the analgesic properties of morphine.
Formula:C24H29ClF3NO4Color and Shape:SolidMolecular weight:487.94Naltrindole 5′-isothiocyanate
CAS:Naltrindole 5′-isothiocyanate (5'-NTII) is an irreversible delta opioid receptor antagonist that counters the analgesic effects induced by DSLET without altering the effects caused by DPDPE.Formula:C27H25N3O3SColor and Shape:SolidMolecular weight:471.571Norbinaltorphimine dihydrochloride
CAS:Norbinaltorphimine dihydrochloride is a selective and potent κ opioid receptor antagonist that induces itch-associated responses in mice.Formula:C40H45Cl2N3O6Purity:98.17% - 99.88%Color and Shape:SolidMolecular weight:734.71Ref: TM-T12241
1mg35.00€5mg80.00€10mg114.00€25mg224.00€50mg388.00€100mg618.00€200mg859.00€1mL*10mM (DMSO)117.00€JDTic Dihydrochloride
CAS:JDTic Dihydrochloride is a high-affinity and selective κ-opioid receptor (KOR) antagonist that blocks dynorphin-KOR signalling,antidepressant.Formula:C28H41Cl2N3O3Purity:98%Color and Shape:SolidMolecular weight:538.55Bromadoline
CAS:Bromadoline is an opioid compound that exhibits anti-nociceptive properties in rodents.Formula:C15H21BrN2OColor and Shape:SolidMolecular weight:325.244Anilopam
CAS:Anilopam is an opioid analgesic belonging to the benzazepine class and acts as an agonist at opioid receptors.Formula:C20H26N2OColor and Shape:SolidMolecular weight:310.4322-Thiocyanatosalvinorin A
CAS:22-Thiocyanatosalvinorin A (RB-64) is a potent selective agonist for the kappa-opioid receptor, exhibiting an EC50 value of 0.077 nM.Formula:C24H27NO8SColor and Shape:SolidMolecular weight:489.54KNT-127
CAS:KNT-127 is an agonist of δ-Opioid receptor.Formula:C24H24N2O2Purity:98%Color and Shape:SolidMolecular weight:372.46(±)-J 113397
CAS:(±)-J-113397 is a potent and selective non-peptidyl ORL1 receptor antagonist (K(i): cloned human ORL1=1.8 nM).Formula:C24H37N3O2Color and Shape:SolidMolecular weight:399.575′-Guanidinonaltrindole
CAS:5′-Guanidinonaltrindole (GNTI) is a selective antagonist of the kappa opioid receptor.Formula:C27H29N5O3Color and Shape:SolidMolecular weight:471.551GNTI dihydrochloride
CAS:κ opioid receptor antagonistFormula:C27H30ClN5O3Purity:98%Color and Shape:SolidMolecular weight:508.01J-113397
CAS:J-113397 is a potent and selective NOP receptor antagonist (IC50 = 2.3 nM).Formula:C24H37N3O2Purity:98%Color and Shape:SolidMolecular weight:399.57BNTX
CAS:BNTX (7-Benzylidenenaltrexone) is a selective δ1-opioid receptor antagonist. It competitively counteracts the antisecretory effects of DPDPE, Deltorphin 2, and DAMGO. BNTX is applicable in research focused on antinociceptive effects.Formula:C27H27NO4Color and Shape:SolidMolecular weight:429.5086β-Naltrexol
CAS:6β-Naltrexol is a peripherally selective opioid antagonist that reduces constipation from opioids while minimizing central nervous system effects.Formula:C20H25NO4Purity:99.933%Color and Shape:SolidMolecular weight:343.42Mu opioid receptor antagonist 8
CAS:Muopioid Receptor Antagonist 8 (368) serves as an antagonist to the μ-opioid receptor, significantly inhibiting the activation of Gi induced by met-enkephalin at the µOR.Formula:C36H35N3O4SColor and Shape:SolidMolecular weight:605.75Riminkefon
CAS:Riminkefon is a kappa opioid receptor agonist .Formula:C38H57N7O6Color and Shape:SolidMolecular weight:707.9Propiram fumarate HCl
CAS:Propiram fumarate HClis an orally available Opioid receptors agonist with analgesic activity for the study of musculoskeletal pain.
Formula:C16H25N3O·xClHPurity:99.25%Color and Shape:SoildSR17018
CAS:SR17018 is an mu-opioid-receptor (MOR) agonist, binding with GTPγS, with an EC50 of 97 nM.
Formula:C19H18Cl3N3OPurity:99.89%Color and Shape:SolidMolecular weight:410.72Cebranopadol
CAS:Cebranopadol (GRT6005) is an analgesic NOP and opioid receptor agonist with Kis of 0.9 nM, 0.7 nM, 2.6 nM, 18 nM for human NOP, μ-opioid (MOP), κ-opioid (KOP)
Formula:C24H27FN2OPurity:98.32% - 99.78%Color and Shape:SolidMolecular weight:378.48SR14150
CAS:SR14150 is a partial agonist of high-affinity NOP receptor.Formula:C21H30N2OPurity:98%Color and Shape:SolidMolecular weight:326.48Bromadoline maleate
CAS:Bromadoline is an opioid analgesic selective for the μ-opioid receptor.Formula:C19H25BrN2O5Purity:98%Color and Shape:SolidMolecular weight:441.322MOR agonist-1
CAS:MOR Agonist-1 is a μ-opioid receptor (MOR) agonist noted for its potent analgesic properties and is utilized in research concerning pain and associated
Formula:C22H26ClFN2O2Purity:98%Color and Shape:SolidMolecular weight:404.91
