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Opioid Receptor

Opioid Receptor

Opioid receptors are a group of G protein-coupled receptors that mediate the effects of endogenous and exogenous opioids. These receptors play a central role in pain modulation, mood regulation, and addictive behaviors. Opioid receptor agonists and antagonists are extensively used in pain management and addiction treatment, as well as in research on neurological and psychiatric disorders. At CymitQuimica, we provide a comprehensive selection of high-quality opioid receptor modulators to support your research in neurobiology, pain management, and addiction therapy.

Found 296 products of "Opioid Receptor"

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  • Norbinaltorphimine

    CAS:
    <p>nor-Binaltorphimine dihydrochloride is a long-acting potent and highly selective kappa opioid receptor antagonist.</p>
    Formula:C40H43N3O6
    Color and Shape:Solid
    Molecular weight:661.79
  • GSK1521498 free base

    CAS:
    <p>GSK1521498 free base is an effective and selective μ-opioid receptor antagonist with potential applications in obesity, alcoholism, and drug addiction.</p>
    Formula:C24H20F2N4
    Purity:99.85%
    Color and Shape:Solid
    Molecular weight:402.44
  • ADL-5747

    CAS:
    <p>ADL-5747 (ADL-5747 (free base)) (free base) is a delta opioid receptor agonist used in the treatment of neurological disorders, skin and musculoskeletal</p>
    Formula:C24H28N2O3
    Purity:98.94% - 99.74%
    Color and Shape:Solid
    Molecular weight:392.49
  • GR 89696 fumarate

    CAS:
    <p>GR 89696 fumarate is a highly selective κ2 opioid receptor agonist (IC50 = 0.04nM) with anti-pruritchy, anti-injury and neuroprotective effects.</p>
    Formula:C23H29Cl2N3O7
    Purity:99.84%
    Color and Shape:Solid
    Molecular weight:530.4
  • NNC 63-0532

    CAS:
    <p>NNC 63-0532 is a potentnociceptin receptor agonist, Ki=7.3 nM, EC50=305 nM.</p>
    Formula:C27H29N3O3
    Purity:99.53%
    Color and Shape:Solid
    Molecular weight:443.54
  • SCH-486757

    CAS:
    <p>SCH-486757 is an agonist of nociceptin-1 (NOP1) and orphanin FQ peptide receptors and is used in the study of cough.</p>
    Formula:C24H23Cl2N3O
    Purity:99.53% - >99.99%
    Color and Shape:Solid
    Molecular weight:440.37
  • Trimebutine CTB salt

    CAS:
    <p>Trimebutine CTB salt (GIC-1001) is an opioid receptor agonist used in the study of pain.</p>
    Formula:C29H36N2O8S2
    Purity:99.85% - >99.99%
    Color and Shape:Solid
    Molecular weight:604.74
  • IPAG

    CAS:
    <p>IPAG is a potent σ-receptor antagonist (pKi=4.3). IPAG can induce cell apoptosis.</p>
    Formula:C17H22IN3
    Purity:99.65%
    Color and Shape:Solid
    Molecular weight:395.28
  • ICI 199,441 hydrochloride

    CAS:
    <p>ICI 199,441 hydrochloride is a potent, selective agonist of κ-opioid receptor.</p>
    Formula:C21H25Cl3N2O
    Purity:99.57%
    Color and Shape:Solid
    Molecular weight:427.8
  • ICI 204,448

    CAS:
    <p>ICI 204,448 is a potent κ-opioid agonist with potential analgesic activity for the study of neurological diseases.</p>
    Formula:C23H27Cl3N2O4
    Purity:>99.99%
    Color and Shape:Solid
    Molecular weight:501.83
  • Bevenopran

    CAS:
    <p>Bevenopran (CB-5945) is a peripheral antagonist of μ-opioid receptor and can be used in studies about the treatment of opioid-induced bowel dysfunction.</p>
    Formula:C20H26N4O4
    Purity:98.69% - 98.9%
    Color and Shape:Solid
    Molecular weight:386.44
  • JNJ-20788560

    CAS:
    <p>JNJ-20788560 is a delta opioid receptor (DOR) agonist with analgesic activity. It is more selective for DOR than for mu opioid receptors (MOR).</p>
    Formula:C25H28N2O2
    Purity:98.02%
    Color and Shape:Solid
    Molecular weight:388.5
  • ML-335

    CAS:
    <p>ML-335, a μ-δ targeted agonist and MOR/DOR ligand, may lead to isomer-biased drugs with pain-relief properties.</p>
    Formula:C25H32N2O3
    Purity:98.52%
    Color and Shape:Solid
    Molecular weight:408.53
  • AT-121

    CAS:
    <p>AT-121 is a dual μ-opioid and neuropeptide receptor partial agonist (Kis 16.49 and 3.67 nM, respectively).</p>
    Formula:C24H38N4O3S
    Purity:98.49% - 99.73%
    Color and Shape:Solid
    Molecular weight:462.65
  • SNC 162

    CAS:
    <p>SNC 162 is a potent and selective delta-opioid receptor (δ-opioid) agonist with analgesic, antidepressant and antiarrhythmic effects.</p>
    Formula:C27H37N3O
    Purity:98%
    Color and Shape:Solid
    Molecular weight:419.6
  • CYT-1010

    CAS:
    <p>CYT-1010, a mu-opioid receptor agonist; EC50: β-arrestin, 13.1 nM; cAMP, 0.0053 nM. Extracted from patent WO2013173730A2.</p>
    Formula:C35H40N6O5
    Purity:98%
    Color and Shape:Solid
    Molecular weight:624.73
  • Mu opioid receptor antagonist 7

    CAS:
    <p>Compound 24, also known as Mu opioid receptor antagonist 7, is a potent, centrally-acting µ-opioid receptor (µOR) antagonist with an inhibitory concentration (</p>
    Formula:C22H27ClN2O2
    Purity:98%
    Color and Shape:Solid
    Molecular weight:386.91
  • Naloxonazine

    CAS:
    <p>Naloxonazine, a potent, selective opiate mu-1 (μ1) antagonist, also influences leishmania through the modulation of host coding function.</p>
    Formula:C38H42N4O6
    Color and Shape:Solid
    Molecular weight:650.76
  • μ opioid receptor agonist 3

    CAS:
    <p>Compound 20, identified as μ opioid receptor agonist 3, is a potent µOR agonist that exhibits an EC50 value of 0.87 nM.</p>
    Formula:C22H28N2O2
    Purity:98%
    Color and Shape:Solid
    Molecular weight:352.47
  • R-84760 hydrochloride

    CAS:
    <p>R-84760, a potent κ-opioid receptor agonist, relieves tonic pain via supraspinal/spinal pathways, activating noradrenergic descent.</p>
    Formula:C19H25Cl3N2OS
    Color and Shape:Solid
    Molecular weight:435.84