LPA Receptor
AM095 free acid
CAS:1228690-36-5
AM095 (free acid) is a potent LPA1 receptor antagonist (IC50s: 0.98 and 0.73 μM for …
Formula:
C27H24N2O5
Purity:
99.9%
Color and Shape:
Solid
Molecular weight:
456.49
Ref: TM-T10293
1mg | 39.00 € | |
2mg | 51.00 € | |
5mg | 82.00 € | |
10mg | 118.00 € | |
25mg | 208.00 € | |
50mg | 346.00 € | |
100mg | 539.00 € | |
200mg | 777.00 € | |
1ml*10 (DMSO) | 90.00 € |
Estimated delivery in United States, on Friday 24 May 2024
GRI977143
CAS:325850-81-5
GRI977143 is a selective and non-lipid agonist of LPA2 (EC50 = 3.3 μM). GRI977143 inhibits …
Formula:
C22H17NO4S
Purity:
98.07%
Color and Shape:
Solid
Molecular weight:
391.44
Ref: TM-T22812
1mg | 39.00 € | |
5mg | 82.00 € | |
10mg | 129.00 € | |
25mg | 264.00 € | |
50mg | 423.00 € | |
100mg | 625.00 € | |
500mg | 1,333.00 € | |
1ml*10 (DMSO) | 115.00 € |
Estimated delivery in United States, on Tuesday 28 May 2024
TC LPA5 4
CAS:1393814-38-4
TC LPA5 4 is a LPA5 receptor antagonist.
Formula:
C23H23ClN2O3
Purity:
99.05%
Color and Shape:
Solid
Molecular weight:
410.89
Ref: TM-T23438
1mg | 58.00 € | |
5mg | 124.00 € | |
10mg | 183.00 € | |
25mg | 425.00 € | |
50mg | 625.00 € | |
100mg | 891.00 € |
Estimated delivery in United States, on Tuesday 28 May 2024
H2L5186303
CAS:139262-76-3
H2L5186303 is an LPA2 antagonist and can be used in studies about asthma treatment.
Formula:
C26H20N2O8
Purity:
97.23%
Color and Shape:
Solid
Molecular weight:
488.45
Ref: TM-T22835
1mg | 52.00 € | |
5mg | 95.00 € | |
10mg | 172.00 € | |
25mg | 369.00 € | |
50mg | 547.00 € | |
100mg | 786.00 € | |
500mg | 1,606.00 € | |
1ml*10 (DMSO) | 113.00 € |
Estimated delivery in United States, on Tuesday 28 May 2024
Radioprotectin-1
CAS:1622006-09-0
Radioprotectin-1 is a selective agonist of LPA2 with EC50 of 25 nM for murine LPA2 …
Formula:
C23H19ClN2O6S
Purity:
99.43%
Color and Shape:
Solid
Molecular weight:
486.92
Ref: TM-T12684
1mg | 143.00 € | |
2mg | 204.00 € | |
5mg | 346.00 € | |
10mg | 517.00 € | |
25mg | 833.00 € | |
50mg | 1,133.00 € | |
100mg | 1,531.00 € | |
1ml*10 (DMSO) | 371.00 € |
Estimated delivery in United States, on Tuesday 28 May 2024
Ki16198
CAS:355025-13-7
Ki16198 is the methyl ester of Ki16425, which is a LPA antagonist and inhibits LPA1- …
Formula:
C24H25ClN2O5S
Purity:
97.6%
Color and Shape:
Solid
Molecular weight:
488.98
Ref: TM-T6347
1mg | 40.00 € | |
5mg | 86.00 € | |
10mg | 134.00 € | |
25mg | 270.00 € | |
50mg | 423.00 € | |
100mg | 625.00 € | |
500mg | 1,328.00 € | |
1ml*10 (DMSO) | 96.00 € |
Estimated delivery in United States, on Tuesday 28 May 2024
Edg-2 receptor inhibitor 1
CAS:1195941-38-8
Edg-2 receptor inhibitor 1 (SAR-100842) is an Edg-2 receptor inhibitor extracted (IC50: <0.1 μM).
Formula:
C27H27NO5
Purity:
99.69%
Color and Shape:
Solid
Molecular weight:
445.51
Ref: TM-T4521
1mg | 95.00 € | |
2mg | 171.00 € | |
5mg | 268.00 € | |
10mg | 419.00 € | |
25mg | 648.00 € | |
50mg | 925.00 € | |
100mg | 1,240.00 € | |
1ml*10 (DMSO) | 283.00 € |
Estimated delivery in United States, on Tuesday 28 May 2024
DBIBB
CAS:1569309-92-7
DBIBB is a non-lipid agonist of specific lysophosphatidic acid (LPA2) type 2 G-protein-coupled receptor. It …
Formula:
C23H20N2O6S
Purity:
97.26%
Color and Shape:
Solid
Molecular weight:
452.48
Ref: TM-T22070
1mg | 64.00 € | |
5mg | 138.00 € | |
10mg | 212.00 € | |
25mg | 430.00 € | |
50mg | 635.00 € | |
100mg | 907.00 € | |
500mg | 1,810.00 € | |
1ml*10 (DMSO) | 152.00 € |
Estimated delivery in United States, on Tuesday 28 May 2024
LPA1 receptor antagonist 1
CAS:1396006-71-5
LPA1 receptor antagonist 1(LPA1 R antagonist 1) is a selective and potent lysophosphatidic acid (LPA1) …
Formula:
C28H26N4O4
Purity:
99.58%
Color and Shape:
Solid
Molecular weight:
482.53
Ref: TM-T15785
1mg | 142.00 € | |
5mg | 341.00 € | |
10mg | 545.00 € | |
25mg | 853.00 € | |
50mg | 1,141.00 € | |
100mg | 1,549.00 € |
Estimated delivery in United States, on Tuesday 28 May 2024
BMS-986278
CAS:2170126-74-4
BMS-986278 is an orally active and potent hemophosphatidic acid receptor 1 (LPA1) antagonist with Kb …
Formula:
C22H31N5O5
Purity:
99.86%
Color and Shape:
Solid
Molecular weight:
445.51
Ref: TM-T39647
5mg | 540.00 € | |
10mg | 862.00 € | |
25mg | 1,747.00 € | |
50mg | 2,775.00 € | |
100mg | 3,709.00 € | |
1ml*10 (DMSO) | 595.00 € |
Estimated delivery in United States, on Tuesday 28 May 2024
TAK-615
CAS:1664335-55-0
TAK-615 is commonly used to study pulmonary fibrosis and is a negative allosteric modulator of …
Formula:
C25H22FNO4
Purity:
98%
Color and Shape:
Solid
Molecular weight:
419.44
Ref: TM-T9699
1mg | 112.00 € | |
5mg | 267.00 € | |
10mg | 423.00 € | |
25mg | 699.00 € | |
50mg | 989.00 € | |
100mg | 1,328.00 € | |
500mg | 2,654.00 € | |
1ml*10 (DMSO) | 296.00 € |
Estimated delivery in United States, on Tuesday 28 May 2024
H2L 5765834
CAS:420841-84-5
H2L 5765834 is a lysophosphatidic acid receptors antagonist
Formula:
C21H12N2O7
Purity:
99.47%
Color and Shape:
Solid
Molecular weight:
404.33
Ref: TM-T22834
1mg | 60.00 € | |
5mg | 118.00 € | |
10mg | 184.00 € | |
25mg | 423.00 € | |
50mg | 624.00 € | |
100mg | 888.00 € | |
500mg | 1,782.00 € | |
1ml*10 (DMSO) | 129.00 € |
Estimated delivery in United States, on Friday 31 May 2024
AM095
CAS:1345614-59-6
AM095 is a potent LPA1 receptor antagonist with IC50 values of 0.98 and 0.73 μM …
Formula:
C27H23N2NaO5
Purity:
99.62%
Color and Shape:
Solid
Molecular weight:
478.47
Ref: TM-T2000
1mg | 48.00 € | |
2mg | 64.00 € | |
5mg | 94.00 € | |
10mg | 132.00 € | |
25mg | 240.00 € | |
50mg | 417.00 € | |
100mg | 601.00 € |
Estimated delivery in United States, on Friday 31 May 2024
LX-1031
CAS:945976-76-1
LX-1031 is an effective inhibitor of tryptophan 5-hydroxylase. LX-1031 decreases serotonin (5-HT) synthesis peripherally.
Formula:
C28H25F3N4O4
Purity:
97.97%
Color and Shape:
Solid
Molecular weight:
538.52
Ref: TM-T15796
1mg | 73.00 € | |
2mg | 94.00 € | |
5mg | 175.00 € | |
10mg | 304.00 € | |
25mg | 518.00 € | |
50mg | 741.00 € | |
100mg | 1,019.00 € | |
1ml*10 (DMSO) | 207.00 € |
Estimated delivery in United States, on Friday 31 May 2024
AM966
CAS:1228690-19-4
AM966, a excellent affinity, specific, oral LPA1(IC50=17 nM) antagonist, suppresses LPA-stimulated intracellular calcium release.
Formula:
C27H23ClN2O5
Purity:
99.49%
Color and Shape:
Solid
Molecular weight:
490.93
Ref: TM-T4278
2mg | 40.00 € | |
5mg | 59.00 € | |
10mg | 96.00 € | |
25mg | 158.00 € | |
50mg | 259.00 € | |
100mg | 416.00 € | |
500mg | 927.00 € | |
1ml*10 (DMSO) | 65.00 € |
Estimated delivery in United States, on Friday 31 May 2024
BMS-986020
CAS:1257213-50-5
BMS-986020 (AM152) is a selective antagonist of LPA1.
Formula:
C29H26N2O5
Purity:
100%
Color and Shape:
Solid
Molecular weight:
482.53
Ref: TM-T4016
1mg | 51.00 € | |
5mg | 82.00 € | |
10mg | 118.00 € | |
25mg | 207.00 € | |
50mg | 346.00 € | |
100mg | 520.00 € | |
1ml*10 (DMSO) | 88.00 € |
Estimated delivery in United States, on Friday 31 May 2024
1-Oleoyl lysophosphatidic acid sodium
CAS:325465-93-8
1-Oleoyl lysophosphatidic acid sodium (1-Oleoyl lysophosphatidic acid sodium salt) salt is an Endogenous agonist of …
Formula:
C21H42O7P·Na
Purity:
99.24%
Color and Shape:
Solid
Molecular weight:
459.51
Ref: TM-T21654
1mg | 70.00 € | |
5mg | 149.00 € | |
10mg | 169.00 € | |
25mg | 342.00 € | |
50mg | 510.00 € |
Estimated delivery in United States, on Friday 31 May 2024
Ki16425
CAS:355025-24-0
Ki16425 (Debio 0719) is a competitive, potent and reversible antagonist to LPA1, LPA2 and LPA3 …
Formula:
C23H23ClN2O5S
Purity:
98.54%
Color and Shape:
Solid
Molecular weight:
474.96
Ref: TM-T6108
2mg | 41.00 € | |
5mg | 56.00 € | |
10mg | 87.00 € | |
25mg | 184.00 € | |
50mg | 360.00 € | |
100mg | 503.00 € | |
1ml*10 (DMSO) | 59.00 € |
Estimated delivery in United States, on Friday 31 May 2024
ONO-7300243
CAS:638132-34-0
ONO-7300243 is an antagonist of lysophosphatidic acid receptor 1 (LPA1; IC50 : 0.16 μM).
Formula:
C28H31NO5
Purity:
98%
Color and Shape:
Solid
Molecular weight:
461.55
Ref: TM-T7393
1mg | 45.00 € | |
2mg | 59.00 € | |
5mg | 95.00 € | |
10mg | 142.00 € | |
25mg | 305.00 € | |
50mg | 531.00 € | |
100mg | 765.00 € | |
1ml*10 (DMSO) | 87.00 € |
Estimated delivery in United States, on Friday 31 May 2024
Tetradecyl Phosphonate
CAS:4671-75-4
Tetradecyl phosphonate is a pan-antagonist of lysophosphatidic acid 1 (LPA1), LPA2, and LPA3 receptors.
Formula:
C14H31O3P
Purity:
98%
Color and Shape:
White To Off-White Powder
Molecular weight:
278.37
Ref: TM-T7689
5mg | 54.00 € | |
10mg | 81.00 € | |
25mg | 124.00 € | |
50mg | 180.00 € | |
100mg | 267.00 € | |
200mg | 402.00 € | |
500mg | 662.00 € |
Estimated delivery in United States, on Friday 31 May 2024