Other Inhibitors
This category encompasses a wide variety of inhibitors that do not fit into the standard classifications but are still critical for various biochemical and pharmacological research. These inhibitors may target unique or less-studied pathways, enzymes, and molecular interactions, providing valuable tools for specialized research areas. At CymitQuimica, we offer a diverse selection of high-quality inhibitors across multiple biological targets and research disciplines, enabling you to explore novel therapeutic avenues and deepen your understanding of complex biological processes.
Found 37931 products of "Other Inhibitors"
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MMG-11 quarterhydrate
<p>MMG-11 quarterhydrate, a potent hTLR2 antagonist, inhibits TLR2/1 and TLR2/6 with IC50s of 1.7μM and 5.7μM; low toxicity.</p>Formula:C15H16O8Color and Shape:SolidMolecular weight:310.78H 218-54
CAS:<p>H 218-54 is a renin inhibitor.</p>Formula:C37H56N2O5SColor and Shape:SolidMolecular weight:640.92(-)-Adenophorine
CAS:<p>(-)-Adenophorine is a moderate alpha-l-fucosidase inhibitor.</p>Formula:C8H17NO4Color and Shape:SolidMolecular weight:191.22Tezampanel hydrate
CAS:<p>Tezampanel is used for the treatment of migraine, neuropathic pain.</p>Formula:C13H23N5O3Color and Shape:SolidMolecular weight:297.35YEATS4 binder-1
<p>YEATS4 binder-1(4e) is an effective and selective compound that targets the KAc recognition site within the YEATS structural domain, exhibiting a binding</p>Formula:C23H34N4O3Color and Shape:SolidMolecular weight:414.54SML-10-70-1
CAS:<p>SML-10-70-1 is a Novel Active Site Inhibitor of Oncogenic K-Ras G12C.</p>Formula:C25H42ClN7O13P2Color and Shape:SolidMolecular weight:746.04PARP1-IN-5
<p>PARP1-IN-5 is a potent, selective, orally active, low-toxicity PARP-1 inhibitor with an IC50 value of 14.7 nM. PARP1-IN-5 can be used in cancer research.</p>Formula:C25H24N2O5SColor and Shape:SolidMolecular weight:464.53Odiparcil
CAS:<p>Odiparcil is an orally active beta-d-thioxyloside analog.</p>Formula:C15H16O6SPurity:98%Color and Shape:SolidMolecular weight:324.35Nanaomycin D
CAS:<p>Nanaomycin D is an antibiotic with antibacterial properties.</p>Formula:C16H12O6Color and Shape:SolidMolecular weight:300.2632,4-Diaminoanisole
CAS:<p>2,4-Diaminoanisole is a carcinogenic aromatic primary amine compound.</p>Formula:C7H10N2OColor and Shape:SolidMolecular weight:138.172-Hydroxygentamicin B1
CAS:<p>2-Hydroxygentamicin B1 is an aminoglycoside antibiotic that exhibits activity against both Gram-positive and Gram-negative bacteria.</p>Formula:C20H40N4O11Color and Shape:SolidMolecular weight:512.552SID 125240931
CAS:<p>SID 125240931 is a regulator of fluorine-activated proteins (FAPs). This compound disrupts the binding between fluoride and FAPs.</p>Formula:C19H24N4O3SColor and Shape:SolidMolecular weight:388.48Antibiotic LL Z1640-2
CAS:<p>Antibiotic LL Z1640-2 is an inhibitor against the TAK1 activity.</p>Formula:C19H22O7Color and Shape:SolidMolecular weight:362.38Ep vinyl quinidine
CAS:<p>3-Epiquinine is a Quinidine stereoisomer, used in malaria, antiarrhythmic, inhibits P450db, and blocks K+ channels, IC50: 19.9 μM.</p>Formula:C20H24N2O2Color and Shape:SolidMolecular weight:324.42Belatacept
CAS:<p>Belatacept (BMS 224818), a T-cell costimulation inhibitor, targets CD80/86 for transplant immunosuppression.</p>Color and Shape:LiquidCI 922
CAS:<p>CI 922 is an anaphylaxis mediator release inhibitor. It inhibits the activation of human neutrophils.</p>Formula:C26H30N10O6Color and Shape:SolidMolecular weight:578.58LI-3948
CAS:<p>IP6K-IN-2 (compound 29c) is an IP6K inhibitor that demonstrates oral bioavailability and the ability to permeate the blood-brain barrier (IC 50 : 15.8 nM), making it suitable for research on central nervous system diseases.</p>Formula:C19H16Cl2FN3O3Color and Shape:SolidMolecular weight:424.25DDCPPB-Glu
CAS:<p>DDCPPB-Glu is a 6-5 fused ring heterocycle antifolate that shows antitumor activity.</p>Formula:C22H27N5O5Purity:98%Color and Shape:SolidMolecular weight:441.48Ceclazepide
CAS:<p>Ceclazepide is an antagonist of cholecystokinin receptor.</p>Formula:C30H32N6O5Purity:98%Color and Shape:SolidMolecular weight:556.61TP-030-2
CAS:<p>TP-030-2 is a RIPK1 inhibitor (human K i =0.43 nM ; mouse IC 50 =100 nM) .</p>Formula:C23H21BrN4O3Color and Shape:SolidMolecular weight:481.34DMP 728
CAS:<p>DMP 728 is an antagonist of Glycoprotein IIb-IIIa.</p>Formula:C26H40N8O10SPurity:98%Color and Shape:SolidMolecular weight:656.71ZIKV-IN-5
<p>ZIKV-IN-5 is an acid-stable, low cytotoxic anti-ZIKV agent with an EC50 value of 0.71 μM. ZIKV-IN-5 showed effective inhibition of ZIKV NS5 MTase activity.</p>Formula:C36H45NO4SiColor and Shape:SolidMolecular weight:583.83Heme Oxygenase-1-IN-3
CAS:<p>Heme Oxygenase-1-IN-3 (compound 4) serves as a potent and selective inhibitor of heme oxygenase-1 (HO-1) with a dissociation constant (Kd) of 141 nM, making it suitable for use in cancer and neurodegenerative disease research.</p>Formula:C22H18BrFN4O2SColor and Shape:SolidMolecular weight:501.37Carbacyclin
CAS:<p>Carbacyclin, a PGI2 analog, is a prostacyclin (PGI2) receptor agonist and vasodilator with potent inhibitory platelet aggregation.</p>Formula:C21H34O4Purity:98%Color and Shape:SolidMolecular weight:350.49(R)-FL118
CAS:<p>FL118 inhibits human survivinion expression and activates tumor suppressor p53 as a MOA in p53 wild-type cancer cells.</p>Formula:C21H16N2O6Color and Shape:SolidMolecular weight:392.36PD 113271
CAS:<p>PD 113,271 is an analog of the fermentation products fostriecin with antitumor activity in vitro and in vivo.</p>Formula:C19H27O10PPurity:98%Color and Shape:SolidMolecular weight:446.39Adecypenol
CAS:<p>Adecypenol is a unique adenosine deaminase inhibitor. It shows effective inhibitory activity against calf intestinal adenosine deaminase.</p>Formula:C12H16N4O4Purity:98%Color and Shape:SolidMolecular weight:280.28MDK-3298
CAS:<p>MDK-3298 is a reversible covalent inhibitor of Mcl-1, a target of protein-protein interaction (PPI).</p>Formula:C35H32BN3O7Purity:98%Color and Shape:SolidMolecular weight:617.46Detajmium
CAS:<p>Detajmium is an anti-arrhythmia compound. It is an Na(+)-channel-blocking drug with an extremely long recovery from use-dependent sodium channel block.</p>Formula:C27H42N3O3Purity:98%Color and Shape:SolidMolecular weight:456.64Coleon-U-quinone
CAS:<p>Coleon-U-quinone, a P-gp inhibitor, reduces cancer cell viability and enhances Doxorubicin sensitivity in resistant cells.</p>Formula:C20H24O5Color and Shape:SolidMolecular weight:344.4(25S)-δ7-Dafachronic acid
CAS:<p>(25S)-delta7-Dafachronic acid, an orphan nuclear receptor DAF-12 ligand, inhibits the dauer-promoting activity of DAF-12.</p>Formula:C27H42O3Purity:98%Color and Shape:SolidMolecular weight:414.62nNOS-IN-25
CAS:<p>nNOS-IN-25 is an effective, selective, and cell-permeable inhibitor of neuronal nitric oxide synthase.</p>Formula:C21H22N4Purity:98%Color and Shape:SolidMolecular weight:330.43AT-IAP
CAS:<p>AT-IAP is an effective dual antagonist of XIAP and cIAP1.</p>Formula:C29H40FN5O2Purity:98%Color and Shape:SolidMolecular weight:509.66Ici D1542
CAS:<p>Ici D1542: potent TXS inhibitor & TXA2 receptor antagonist, effective thromboxane blocker in vitro.</p>Formula:C25H30N2O7Purity:98%Color and Shape:SolidMolecular weight:470.51MEIS-IN-3
<p>MEIS-IN-3 is a potent inhibitor of MEIS.</p>Formula:C25H26N2O4Color and Shape:SolidMolecular weight:418.48SB 204070 hydrochloride
CAS:<p>SB 204070 hydrochloride is an inhibitor of beta-lactamase, it is isolated from Spondias mombin.</p>Formula:C19H27ClN2O4Purity:98%Color and Shape:SolidMolecular weight:382.88eIF4A3-IN-4
<p>eIF4A3-IN-4 is a novel inhibitor of eIF4A (IC50: 8.6 μM).</p>Formula:C24H20N2O5Color and Shape:SolidMolecular weight:416.43Bcl-2-IN-8
<p>Bcl-2-IN-8: potent, hinders cell growth/migration, induces apoptosis, promising in triple-negative breast cancer research.</p>Formula:C36H44O6Color and Shape:SolidMolecular weight:572.73Chrymutasin C
CAS:<p>Chrymutasin C is a glycoside antitumor antibiotic with cytotoxic properties.</p>Formula:C39H43NO17Color and Shape:SolidMolecular weight:797.755AY-22,252
CAS:<p>AY-22,252 is an inhibitor of beef heart & rat brain nucleoside-3',5'- monophosphate phosphodiesterase.</p>Formula:C27H37NaO7Color and Shape:SolidMolecular weight:496.57BRD-9526
CAS:<p>BRD-9526 is a potent and selective inhibitor of Sonic Hedgehog (Shh).</p>Formula:C26H31Cl2N3O6SPurity:98%Color and Shape:SolidMolecular weight:584.512-Hydroxygentamicin C2
CAS:<p>2-Hydroxygentamicin C2 is an aminoglycoside antibiotic that exhibits activity against both Gram-positive and Gram-negative bacteria.</p>Formula:C20H41N5O8Color and Shape:SolidMolecular weight:479.568L 767679
CAS:<p>L 767679 is an antagonist of the fibrinogen receptors.</p>Formula:C20H24N4O4Purity:98%Color and Shape:SolidMolecular weight:384.43Polyoxin H
CAS:<p>Polyoxin H is a nucleoside antifungal antibiotic that exhibits significant efficacy against rice sheath blight.</p>Formula:C23H32N6O13Color and Shape:SolidMolecular weight:600.53SSR-182289A (Free)
CAS:<p>SSR-182289A (Free) is a thrombin inhibitor.</p>Formula:C30H33F2N5O4SPurity:98%Color and Shape:SolidMolecular weight:597.68Dinordrin
CAS:<p>Dinordrin is an implantation inhibitor and hormone.</p>Formula:C27H36O4Purity:98%Color and Shape:SolidMolecular weight:424.57Asperenone
CAS:<p>Asperenone is a 15-lipoxygenase (15-LOX) inhibitor with an IC50 of 0.3 mM. Additionally, it acts as a platelet aggregation inhibitor with an IC50 of 0.23 mM. Asperenone also exhibits antifungal properties, inhibiting the growth of pathogenic fungi Ophiostoma crassivaginatum and O. piliferum, and may be utilized in research related to cardiovascular diseases and anti-infective treatments.</p>Formula:C20H22OColor and Shape:SolidMolecular weight:278.388Granaticin B
CAS:<p>Granaticin B inhibits the initial phase of RNA biosynthesis and exhibits activity against Gram-positive bacteria, mycobacteria (weak), and Trichomonas vaginalis, along with the ability to suppress tumor cells.</p>Formula:C28H30O12Color and Shape:SolidMolecular weight:558.531Dihydroabikoviromycin
CAS:<p>Dihydroabikoviromycin is a secondary metabolite of Streptomyces anulatus and acts as a polyketide synthase inhibitor.</p>Formula:C10H13NOColor and Shape:SolidMolecular weight:163.216Epelmycin D
CAS:<p>Epelmycin D exhibits activity against both Gram-positive and Gram-negative bacteria, as well as Candida albicans, and demonstrates efficacy against leukemia (L1210).</p>Formula:C30H35NO11Color and Shape:SolidMolecular weight:585.599Pluracidomycin C2
CAS:<p>Pluracidomycin C2 is a carbapenem antibiotic with activity against both Gram-positive and Gram-negative bacteria.</p>Formula:C11H15NO9S2Color and Shape:SolidMolecular weight:369.37PD-149163
CAS:<p>PD-149163: brain-penetrating, selective NTR1 agonist; shows pro-cognitive, anti-psychotic, anxiolytic effects.</p>Formula:C42H71N9O6Color and Shape:SolidMolecular weight:798.07Danavorexton
CAS:<p>Danavorexton is an orexin receptor agonist.</p>Formula:C21H32N2O5SColor and Shape:SolidMolecular weight:424.55Halomicin D
CAS:<p>Halomicin D is an ansamycin-class antibiotic that exhibits activity against both Gram-positive and Gram-negative bacteria.</p>Formula:C43H56N2O12Color and Shape:SolidMolecular weight:792.911Lactoquinomycin B
CAS:<p>Lactoquinomycin B is a quinone antibiotic with activity against Gram-positive bacteria and some Gram-negative bacteria, though its efficacy against Gram-negative species is weaker and it does not affect fungi. It inhibits various cell lines, including lymphoma L5178Y parental cells, doxorubicin-resistant cells, bleomycin-resistant cells, human leukemia K562 cells, and murine leukemia L-1210 and P388 cells, with ID50 (μg/mL) values of 0.43, 0.21, 0.19, 0.16, 0.2, and 0.12, respectively.</p>Formula:C24H27NO9Color and Shape:SolidMolecular weight:473.473A 70450
CAS:<p>A 70450, an inhibitor of aspartyl proteinase, can be used as an antifungal agent and may have a role in HIV protease inhibition therapy.</p>Formula:C42H71ClN6O5Purity:98%Color and Shape:SolidMolecular weight:775.50Feigrisolide C
CAS:<p>Feigrisolide C is a lactone produced by the bacterium Streptomyces griseus.</p>Formula:C21H36O7Color and Shape:SolidMolecular weight:400.506Deoxyfrenolicin
CAS:<p>Deoxyfrenolicin is a quinone antibiotic that can be isolated from the fermentation broth of the Streptomyces roseofulvus strain AM-3867 and belongs to the frenolicin class of antibiotics. This compound exhibits in vitro antibacterial activity and is effective in inhibiting the activity of Mycoplasma gallisepticum.</p>Formula:C18H18O6Color and Shape:SolidMolecular weight:330.332Chitinovorin C
CAS:<p>Chitinovorin C is a β-lactam class antibiotic (antibiotic) that exhibits weak inhibitory activity against Gram-negative bacteria.</p>Formula:C15H20N4O8SColor and Shape:SolidMolecular weight:416.406Pulvomycin
CAS:<p>Pulvomycin is a protein biosynthesis inhibitor preventing ternary complex formation between elongation factor Tu, GTP, and aminoacyl-tRNA.</p>Formula:C47H66O13Purity:98%Color and Shape:SolidMolecular weight:839.032ZD6021
CAS:<p>ZD6021 is an antagonist of neurokinin 1 receptor.</p>Formula:C35H35Cl2N3O2SPurity:98%Color and Shape:SolidMolecular weight:632.64Org-31710
CAS:<p>Org-31710 is a progesterone receptor antagonist potentially for contraception.</p>Formula:C30H39NO2Purity:98%Color and Shape:SolidMolecular weight:445.64Cortistatin A
CAS:<p>Cortistatin A is a potent and selective mediator-associated kinase CDK8 and its paralogue CDK19 inhibitor.</p>Formula:C30H36N2O3Purity:98%Color and Shape:SolidMolecular weight:472.62ONO-8809
CAS:<p>ONO-8809: Thromboxane A2 antagonist, reduces airway hyperresponse, macrophage accumulation, and MMP-9 in SHRSP brains.</p>Formula:C30H46BrNO4SPurity:98%Color and Shape:SolidMolecular weight:596.66Methyl Streptonigrin
CAS:<p>Methyl Streptonigrin is an ABCG2 transporter function inhibitor.</p>Formula:C26H24N4O8Purity:98%Color and Shape:SolidMolecular weight:520.49GSK579289A
CAS:<p>GSK579289A is an inhibitor of benzimidazole thiophene.</p>Formula:C26H27ClN4O3SPurity:98%Color and Shape:SolidMolecular weight:511.04Retelliptine
CAS:<p>Retelliptine, a DNA topoisomerase II inhibitor, is used potentially for the treatment of cancer.</p>Formula:C25H32N4OPurity:98%Color and Shape:SolidMolecular weight:404.55L 739749
CAS:<p>L 739749 is a CAAX peptidomimetic. It is also an inhibitor of farnesyl-protein transferase.</p>Formula:C24H41N3O6S2Purity:98%Color and Shape:SolidMolecular weight:531.73SX 3202
CAS:<p>SX 3202 is an aldose reductase inhibitor being developed for the treatment of diabetic neuropathy.</p>Formula:C17H11BrFN3O4Color and Shape:SolidMolecular weight:420.19Naltalimide
CAS:<p>Naltalimide: µ-opioid receptor partial agonist, improves bladder storage by affecting spinal cord reflex.</p>Formula:C28H28N2O5Purity:98%Color and Shape:SolidMolecular weight:472.53Pamiparib maleate
CAS:<p>Pamiparib (BGB-290) is a selective PARP inhibitor that blocks DNA repair and promotes apoptosis.</p>Formula:C44H42F2N8O14Purity:98%Color and Shape:SolidMolecular weight:944.859Ambelline
CAS:<p>Ambelline has antitumor activity.</p>Formula:C18H21NO5Purity:98%Color and Shape:SolidMolecular weight:331.36GSK699
CAS:<p>GSK699 is a potent, cell penetrant PCAF/GCN5 PROTAC.</p>Formula:C45H51BrN8O7Color and Shape:SolidMolecular weight:895.84G-9791
CAS:<p>G-9791 is an effective and selective inhibitor of group-I PAK.</p>Formula:C26H26ClFN6O2Purity:98%Color and Shape:SolidMolecular weight:508.98MPO-IN-8
CAS:<p>MPO-IN-8, an orally active myeloperoxidase (MPO) inhibitor, effectively inhibits the production of hypochlorous acid in neutrophils and the release of extracellular traps (NETosis). In mice exhibiting gouty arthritis, it reduces swelling, decreases peroxidase activity, and lowers IL-1β levels.</p>Formula:C12H9N3O2Color and Shape:SolidMolecular weight:227.22Dimesna free acid
CAS:<p>Dimesna (BNP-778), when used in conjunction with active cancer chemotherapy agents, can reduce the toxicity associated with uremia.</p>Formula:C4H10O6S4Color and Shape:SolidMolecular weight:282.38LY 190388
CAS:<p>LY 190388 is a penicillamine-containing enkephalin analog used as an mu receptor agonist with analgesia activity.</p>Formula:C30H41N5O7SPurity:98%Color and Shape:SolidMolecular weight:615.74Emd 52297
CAS:<p>Emd 52297 is an inhibitor of renin.</p>Formula:C39H59N11O7Purity:98%Color and Shape:SolidMolecular weight:793.96AFP-07 free acid
CAS:<p>AFP 07 free acid is a 7,7-difluoroprostacyclin derivative. It also acts as a selective and highly potent agonist for the IP receptor.</p>Formula:C22H30F2O5Purity:98%Color and Shape:SolidMolecular weight:412.47Antitrypanosomal agent 6
<p>Compound 18a: potent vs. T. brucei (IC50: 0.47 μM), >2x efficacy compared to Nifurtimox, good ADME, binds AT-rich DNA.</p>Formula:C22H29Cl2N5OColor and Shape:SolidMolecular weight:450.4Netobimin
CAS:<p>Netobimin is an anthelmintic effective against naturally acquired gastrointestinal nematodes in cows.</p>Formula:C14H20N4O7S2Color and Shape:SolidMolecular weight:420.46RN941
CAS:<p>RN941 is a highly potent Bruton's tyrosine kinase (BTK) inhibitor.</p>Formula:C34H34FN7O5Purity:98%Color and Shape:SolidMolecular weight:639.687β,16α-Dihydroxybufalin
CAS:<p>7β,16α-Dihydroxybufalin, a dihydroxylated derivative of bufalin, demonstrates cytotoxic properties against various cancer cell lines.</p>Formula:C24H34O6Color and Shape:SolidMolecular weight:418.52Dup-714
CAS:<p>Dup-714 is a thrombin inhibitor.</p>Formula:C21H33BN6O5Purity:98%Color and Shape:SolidMolecular weight:460.33Foroxymithine
CAS:<p>Foroxymithine is an inhibitor of angiotensin-converting enzyme.</p>Formula:C22H37N7O11Purity:98%Color and Shape:SolidMolecular weight:575.57Flurdihydroergotamine
CAS:<p>Flurdihydroergotamine, a serotonin 5HT1 receptor agonist, is used as an antimigraine drug.</p>Formula:C34H36F3N5O5Purity:98%Color and Shape:SolidMolecular weight:651.68SMP-797 HCl
CAS:<p>SMP-797 HCl, an ACAT (acyl-CoA-cholesterol acyltransferase) inhibitor, is used potentially for the treatment of Hyperlipidemia.</p>Formula:C34H44ClN5O4Purity:98%Color and Shape:SolidMolecular weight:622.20S24-14
CAS:<p>S24-14 serves as an effective anti-osteoporosis agent by inhibiting osteoclastogenesis, promoting osteoblast differentiation, and reducing bone resorption.</p>Formula:C19H12N2O3SColor and Shape:SolidMolecular weight:348.38JBJ-08-178-01
CAS:<p>JBJ-08-178-01, a mutant-selective tyrosine kinase inhibitor, targets (HER2) human epidermal growth factor receptor 2 and exhibits antitumoral activity. This compound not only diminishes HER2's kinase activity and protein levels through the induction of proteasomal degradation of the receptor but also shows promise in non-small-cell lung cancer research.</p>Formula:C31H30N8O3Color and Shape:SolidMolecular weight:562.62BRD4-IN-9
CAS:<p>BRD4-IN-9, an orally active BRD4 inhibitor, demonstrates a potent IC50 of 9.4 nM. In a murine melanoma xenograft model, it effectively inhibits tumor growth.</p>Formula:C24H23N3O3Color and Shape:SolidMolecular weight:401.46Tyk2-IN-10
CAS:<p>Tyk2-IN-10 acts as an inhibitor of the Tyrosine Kinase 2 (Tyk2)-mediated signaling pathway, which plays a role in inflammation regulation.</p>Formula:C25H27N5O3Color and Shape:SolidMolecular weight:445.51Arterolane maleate
CAS:<p>Arterolane, an adenosine triphosphatase inhibitor, is used potentially for the treatment of malaria.</p>Formula:C26H40N2O8Purity:98%Color and Shape:SolidMolecular weight:508.612Enprostil
CAS:<p>Enprostil: synthetic PGE2 analog, reduces gastric acid, protects mucosa, lowers post-meal gastrin, treats ulcers effectively and safely.</p>Formula:C23H28O6Purity:98%Color and Shape:SolidMolecular weight:400.46CHNQD-01255
CAS:<p>CHNQD-01255 is an orally active inhibitor of Arf-GEFs that is effective against hepatocellular carcinoma (HCC).</p>Formula:C23H29NO6Color and Shape:SolidMolecular weight:415.48OP-2507
CAS:<p>OP-2507, a prostacyclin agonist, is used potentially for the treatment of hepatic insufficiency and hypertension.</p>Formula:C25H41NO4Purity:98%Color and Shape:SolidMolecular weight:419.6CH-38083
CAS:<p>CH-38083 is a selective and effective alpha-2 adrenoceptors antagonist.</p>Formula:C18H24ClNO3Purity:98%Color and Shape:SolidMolecular weight:337.84Pradimicin T2
CAS:<p>Pradimicin T2 is an antibiotic with activity against filamentous fungi and yeast-like fungi.</p>Formula:C37H37NO19Color and Shape:SolidMolecular weight:799.685Pyrisulfoxin A
CAS:<p>Pyrisulfoxin A is an antibiotic that can be found in Streptomyces callfornicus [BS-75].</p>Formula:C13H13N3O3SColor and Shape:SolidMolecular weight:291.326PI3K-IN-27
CAS:<p>PI3K-IN-27 is a potent PI3K inhibitor, relevant for cancer and immune disease research. See patent WO2021233227A1.</p>Formula:C30H26F2N6O2SColor and Shape:SolidMolecular weight:572.63Seldomycin factor 1
CAS:<p>Seldomycin factor 1 (XK 88-1) is an aminoglycoside antibiotic known for its broad-spectrum antibacterial activity.</p>Formula:C17H34N4O10Color and Shape:SolidMolecular weight:454.473PZ-3022
CAS:<p>PZ-3022 is an orally active, conformational PanK activator that counteracts C3-CoA inhibition. In a mouse model of propionic acidemia, it elevates hepatic CoASH and C2-CoA levels while reducing C3-CoA, making it useful for studying mitochondrial defects in propionic acidemia.</p>Formula:C20H21N5OColor and Shape:SolidMolecular weight:347.414-Chloropyridine
CAS:<p>4-Chloropyridine acts as an inhibitor of Nicotinamide N-methyltransferase (NNMT). Serving as a substrate for NNMT, this compound enhances the electrophilicity at the C4 position through methylation of the pyridine nitrogen. This modification facilitates an aromatic nucleophilic substitution reaction with the non-catalytic cysteine (C159) in NNMT, ultimately leading to suicidal activity inhibition of the enzyme. 4-Chloropyridine is a promising candidate for the development of activity-based probes targeting NNMT functions.</p>Formula:C5H4ClNColor and Shape:SolidMolecular weight:113.55Pacidamycin D
CAS:<p>Pacidamycin D is an antibiotic of the Pacidamycin class, demonstrating activity against Pseudomonas aeruginosa with a minimum inhibitory concentration (MIC) of 4-16 μg/mL. It shows no efficacy against other Gram-negative or Gram-positive bacteria, nor does it affect drug-resistant strains of Pseudomonas aeruginosa.</p>Formula:C32H41N9O10Color and Shape:SolidMolecular weight:711.722Epoxyquinomicin A
CAS:<p>Epoxyquinomicin A is an antibiotic isolated from Amycolatopsissp. It exhibits inhibitory activity against Micrococcus luteus, Bacillus subtilis, Pasteurella piscicida, and Staphylococcus aureus with MIC values of 3-12.5 µg/mL. Additionally, it shows cytotoxicity in cancer cells L1210, B16, and S180, with an IC50 of 2-8 µg/mL. Furthermore, Epoxyquinomicin A demonstrates anti-inflammatory effects in collagen-induced arthritis.</p>Formula:C14H10ClNO6Color and Shape:SolidMolecular weight:323.685PIKfyve-IN-1
<p>PIKfyve-IN-1: potent, cell-active inhibitor for PIKfyve research, IC50=6.9 nM.</p>Formula:C20H21N5Color and Shape:SolidMolecular weight:331.41SORT1-IN-3
CAS:<p>SORT1-IN-3 (compound 5) is a SORT1 inhibitor characterized by its ability to permeate the blood-brain barrier.</p>Formula:C16H26ClNO3Color and Shape:SolidMolecular weight:315.84(±)-ANAP hydrochloride (1185251-08-4 free base)
<p>(±)-ANAP hydrochloride is the amino acid analog of prodan. It can be used as a fluorescent probes and enhance environmental sensitivity.</p>Formula:C15H17ClN2O3Purity:98%Color and Shape:SolidMolecular weight:308.76(R)-NVS-ZP7-4
CAS:<p>(R)-NVS-ZP7-4, an R-isomer, inhibits ZIP7 to study ER zinc impact & Notch pathway.</p>Formula:C28H28FN5OSPurity:98%Color and Shape:SolidMolecular weight:501.62Polyoxin E
CAS:<p>Polyoxin E is a nucleoside antifungal antibiotic that demonstrates significant effectiveness against rice sheath blight.</p>Formula:C17H23N5O13Color and Shape:SolidMolecular weight:505.39Acetoxycycloheximide
CAS:<p>Acetoxycycloheximide triggers TNF receptor 1, prompts apoptosis, and cytochrome c release by activating c-Jun N-terminal kinase.</p>Formula:C17H25NO6Color and Shape:SolidMolecular weight:339.38Micacocidin A
CAS:<p>Micacocidin A is an antibiotic showing excellent activity against Mycoplasma species.</p>Formula:C27H37N3O4S3ZnColor and Shape:SolidMolecular weight:629.20C20 Sphingomyelin (d18:1/20:1)
CAS:<p>C20 Sphingomyelin (d18:1/20:1) (Compound SM:20:1) is a type of sphingolipid. This compound shows potential for research related to motor neuron diseases, such as amyotrophic lateral sclerosis (ALS) and primary lateral sclerosis (PLS).</p>Formula:C43H85N2O6PColor and Shape:SolidMolecular weight:757.119Antiviral agent 7
<p>Antiviral agent 7 is a peptide-based coating that kills viruses.</p>Formula:C29H31F2N3O6Color and Shape:SolidMolecular weight:555.57Phosmidosine
CAS:<p>Phosmidosine inhibits cell cycle progression and morphological recovery in srcts-NRK cells. Additionally, Phosmidosine exhibits antifungal properties.</p>Formula:C16H24N7O8PColor and Shape:SolidMolecular weight:473.38Pinselin
CAS:<p>Pinselin is a nitrogen-containing heterocyclic antibiotic with yeast-inhibiting properties.</p>Formula:C16H12O6Color and Shape:SolidMolecular weight:300.263BW-10
CAS:<p>BW-10 potently inhibits bombesin evoked release of gastrointestinal hormones in vitro and in vivo.</p>Formula:C57H72N14O8Color and Shape:SolidMolecular weight:1081.27Cetoniacytone B
CAS:<p>Cetoniacytone B inhibits the growth of HEPG2 and MCF7 human tumor cell lines, with a GI50 of 4.4 μM.</p>Formula:C7H9NO4Color and Shape:SolidMolecular weight:171.151DMP-728 free base
CAS:<p>DMP-728 free base is a highly potent and selective GPIIbDIIa antagonist</p>Formula:C25H36N8O7Color and Shape:SolidMolecular weight:560.60Ro-24-4736
CAS:<p>Ro 24-4736 is an effective and selective platelet-activating factor antagonist.</p>Formula:C31H20ClN5OSPurity:98%Color and Shape:SolidMolecular weight:546.04SCP1-IN-1
CAS:<p>SCP1-IN-1 (SH T-62) is a potent inhibitor of SCP1, promoting REST degradation and potentially aiding glioblastoma research.</p>Formula:C20H19F3N2O7S2Purity:99.53%Color and Shape:SoildMolecular weight:520.5KF 20274
CAS:<p>KF 20274 is an adenosine A1 antagonist; purinergic receptor antagonist.</p>Formula:C21H29N5OColor and Shape:SolidMolecular weight:367.49PARP10/15-IN-1
<p>PARP10/15-IN-1 (compound 8l) is a dual PARP10 and PARP15 inhibitor with IC50s of 160 nM and 370 nM, respectively. It can be used in cancer research[1].</p>Formula:C13H10N2O3SColor and Shape:SolidMolecular weight:274.3NSC 357754
CAS:<p>NSC 357754 is an inhibitor of Claudin. It can enhance transepithelial electrical resistance and reduce specific cation permeability. NSC 357754 is useful for research involving Claudin-2 and/or Claudin-15 mediated intestinal disorders.</p>Formula:C26H20N4O2Color and Shape:SolidMolecular weight:420.463Azonafide-PEABA
CAS:<p>Azonafide-PEABA is a drug moiety with cytotoxic [1].</p>Formula:C32H33N5O4Purity:98%Color and Shape:SolidMolecular weight:551.641-Deamino-1-hydroxysagamicin
CAS:<p>1-Deamino-1-hydroxysagamicin (AntibioticSUM-3) is an aminoglycoside antibiotic that is effective against both Gram-positive and Gram-negative bacteria.</p>Formula:C20H40N4O8Color and Shape:SolidMolecular weight:464.554Phenazostatin B
CAS:<p>Phenazostatin B is a phenazine derivative known for its neuroprotective properties. It acts by scavenging free radicals, protecting N18-RE 105 neuronal cells from glutamate-induced toxicity, and inhibiting lipid peroxidation. It inhibits glutamate toxicity in N18-RE-105 cells, with an EC50 of 0.33 μg/mL.</p>Formula:C32H26N4O4Color and Shape:SolidMolecular weight:530.57Methylenomycin A
CAS:<p>Methylenomycin A is a cyclopentanone-derived antibiotic effective against both Gram-negative and Gram-positive bacteria.</p>Formula:C9H10O4Color and Shape:SolidMolecular weight:182.173Ekatetrone
CAS:<p>Ekatetrone displays activity against both Gram-positive and Gram-negative bacteria, with particularly strong inhibitory effects on Mycobacterium tuberculosis.</p>Formula:C19H13NO7Color and Shape:SolidMolecular weight:367.309GDC-6036-NH
CAS:<p>GDC-6036-NH is a precursor of compound 17a /b, which is a RAS inhibitor that can be used in cancer research.</p>Formula:C26H30ClF4N7OPurity:99.84%Color and Shape:SolidMolecular weight:568.01ZIKV-IN-4
<p>ZIKV-IN-4 is a low cytotoxic, acid-stable anti-ZIKV agent with an EC50 value of 3.49 μM. ZIKV-IN-4 exhibited potent inhibition of ZIKV NS5 MTase.</p>Formula:C33H37NO4Color and Shape:SolidMolecular weight:511.65SARS-CoV-2 nsp3-IN-1
<p>Compound 15c selectively inhibits SARS-CoV-2 nsp3 Mac1 with IC50 of 6.1 μM.</p>Formula:C17H15N5O2Color and Shape:SolidMolecular weight:321.33AVE 0991
CAS:<p>AVE 0991 is a nonpeptide analog of angiotensin-(1-7), a Mas agonist with inhibitory effects on [125I]-Ang-(1-7) and on neuroinflammation in Alzheimer's disease.</p>Formula:C29H32N4O5S2Purity:98.69%Color and Shape:SolidMolecular weight:580.72L2H2-6OTD
CAS:<p>L2H2-6OTD is a telomerase inhibitor with G-quadruplex loops; IC50: 15 nM.</p>Formula:C30H30N10O8Color and Shape:SolidMolecular weight:658.62Heme Oxygenase-2-IN-1
<p>Heme Oxygenase-2-IN-1 is a selective HO-2 inhibitor with IC50s: 14.9 μM (HO-1), 0.9 μM (HO-2).</p>Formula:C19H17N3O2Color and Shape:SolidMolecular weight:319.366-Deoxyilludin M
CAS:<p>6-Deoxyilludin M is an antitumor antibiotic with anti-leukemic properties. It can be isolated from the culture broth of a basidiomycetous fungus belonging to the genus Pleurotus (Pleurotus japonicas).</p>Formula:C15H20O2Color and Shape:SolidMolecular weight:232.318Flavipucine
CAS:<p>Flavipucine (Flavipucin) is a glutarimide antibiotic found in the Aspergillus flavipes F-2090/7 strain. It exhibits antibacterial activity against Bacillus subtilis, possesses antiprotozoal properties, and demonstrates cytotoxic effects on various cancer cells.</p>Formula:C12H15NO4Color and Shape:SolidMolecular weight:237.252Amidomycin
CAS:<p>Amidomycin is an antibiotic that primarily targets yeast.</p>Formula:C40H68N4O12Color and Shape:SolidMolecular weight:796.99mPGES1-IN-4
CAS:<p>mPGES1-IN-4 (compound 32) is a multi-substituted pyrimidine compound acting as a submicromolar inhibitor of PGE2 production. It primarily exerts its anti-inflammatory effects by inhibiting mPGES-1 and significantly suppresses acute inflammation models in vivo.</p>Formula:C27H25F2N3OColor and Shape:SolidMolecular weight:445.50Unoprostone
CAS:<p>Unoprostone is a prostaglandin F2α analogs (PGAs), and reduces intraocular pressure and is used topically for glaucoma or ocular hypertension.</p>Formula:C22H38O5Purity:98%Color and Shape:SolidMolecular weight:382.53Miyakamide B2
CAS:<p>Miyakamide B2 is an antibiotic with insecticidal properties. It suppresses the growth of brine shrimp and shows weak activity against Xanthomonas species. The IC50 for inhibition of P388 cells by Miyakamide B2 is 7.6 μg/mL.</p>Formula:C31H32N4O4Color and Shape:SolidMolecular weight:524.61Taprostene
CAS:<p>Taprostene (CG-4203), a stable Prostacyclin analogue, protects endothelium and myocardium post-ischemia in cats, with minimal hemodynamic impact.</p>Formula:C24H30O5Color and Shape:SolidMolecular weight:398.49Atiratecan
CAS:<p>Atiratecan (TP300), a CH0793076-based camptothecin prodrug, combats BCRP+/- tumors; doesn't affect AChE.</p>Formula:C31H34N6O6Purity:98%Color and Shape:SolidMolecular weight:586.645-Hydroxy-3,4,7-triphenyl-2,6-benzofurandione
CAS:<p>5-Hydroxy-3,4,7-triphenyl-2,6-benzofurandione is an inhibitor of xanthine oxidase (XO) found in the fungus Peniophora sanguinea.</p>Formula:C26H16O4Color and Shape:SolidMolecular weight:392.40MMP408
CAS:<p>MMP408 acts as an inhibitor of MMP-12.</p>Formula:C19H20N2O7SColor and Shape:SolidMolecular weight:420.44Anti-inflammatory agent 18
<p>Anti-inflammatory agent 18: NO activity blocker (IC50: 15.94 μM), hampers HMGB1-induced inflammation, potential for COVID-19, sepsis study.</p>Formula:C30H50O6Color and Shape:SolidMolecular weight:506.71Antileishmanial agent-5
<p>Antileishmanial agent-4, a ribonucleoside analogue, targets L.infantum and T.cruzi with EC50s of 0.68 μM and 0.83 μM.</p>Formula:C17H17ClN4O4Color and Shape:SolidMolecular weight:376.79Nothramicin
CAS:<p>Nothramicin is an anthracycline antibiotic that exhibits antimycobacterial activity.</p>Formula:C30H37NO11Color and Shape:SolidMolecular weight:587.615Sovesudil hydrochloride
<p>Sovesudil (PHP-201) HCl: potent local ROCK inhibitor; targets ROCK I/II (IC50: 3.7/2.3 nM); lowers IOP, non-congesting.</p>Formula:C23H23ClFN3O3Color and Shape:SolidMolecular weight:443.9Hydroxyakalone
CAS:<p>Hydroxyakalone is an inhibitor of the enzyme xanthine oxidase (XOD, EC 1.2.3.2) and has an IC50 of 4.6 μM for XOD.</p>Formula:C5H5N5O2Color and Shape:SolidMolecular weight:167.126AH22921
CAS:<p>AH22921 is an EP4 prostaglandin receptor antagonist with the ability to antagonize the activation of adenylyl cyclase by prostaglandins in CHO cells. It induces a rightward shift in the PGE? concentration-response curve in these cells, functioning as a non-competitive antagonist. AH22921 is selective for the EP4 receptor, inhibiting its activity in CHO cells without affecting the PGE? concentration-response curve in NPE cells that contain the EP2 receptor.</p>Formula:C29H35NO5Color and Shape:SolidMolecular weight:477.59SARS-CoV-2-IN-99
CAS:<p>SARS-CoV-2-IN-99 (compound 58) is an inhibitor of the main protease of SARS-CoV-2.</p>Formula:C20H16Br2NO4PColor and Shape:SolidMolecular weight:525.13PDE4B-IN-3
<p>PDE4B-IN-3 is a potent inhibitor of PDE4B (IC50: 0.94 μM) and exhibits anti-inflammatory effects.</p>Formula:C30H35N3O4S2Color and Shape:SolidMolecular weight:565.75MRS4865
CAS:<p>MRS4865 (compound 7a) serves as a chimeric antagonist for the P2Y14 receptor and an agonist for UDP-glucose, offering protection against neuropathic pain.</p>Formula:C39H39F3N4O7Color and Shape:SolidMolecular weight:732.74α-Prumycin hydrochloride
CAS:<p>α-Prumycin hydrochloride is a carbohydrate antibiotic with antifungal properties and weak antibacterial activity.</p>Formula:C8H19Cl2N3O4Color and Shape:SolidMolecular weight:292.16Thielavin B
CAS:<p>Thielavin B, from Thielavia terricola, inhibits prostaglandin E2 synthesis and reduces rat oedema.</p>Formula:C31H34O10Color and Shape:SolidMolecular weight:566.6Hexedine
CAS:<p>Hexedine is a biochemical.</p>Formula:C22H45N3Color and Shape:SolidMolecular weight:351.61TSWV-IN-1
<p>TSWV-IN-1 is an anti-TSWV drug with potential TSWV N.</p>Formula:C26H31FO4S2Color and Shape:SolidMolecular weight:490.65Vicanicin
CAS:<p>Vicanicin is an aryl phenol ether compound found in lichens. It inhibits the expression of Hsp70, modulates intracellular redox-sensitive mechanisms, increases reactive oxygen species (ROS) in cancer cells, alters the Bax/Bcl-2 ratio, activates caspase-3, and induces apoptosis. Vicanicin suppresses cell growth and promotes apoptosis in androgen-sensitive (LNCaP) and androgen-insensitive (DU-145) human prostate cancer cells. It holds potential for prostate cancer research.</p>Formula:C18H16Cl2O5Color and Shape:SolidMolecular weight:383.223PDE4-IN-14
CAS:<p>PDE4-IN-14 (Compound 1) serves as an inhibitor of phosphodiesterase 4 (PDE4), applicable in research concerning diseases associated with PDE4, including</p>Formula:C19H20F2N4O3SColor and Shape:SolidMolecular weight:422.45Carmegliptin dihydrochloride
CAS:<p>Carmegliptin dihydrochloride (RG-1579, RO4876904) is a salt of Camegliptin, a DPP-4 inhibitor for type 2 diabetes.</p>Formula:C20H30Cl2FN3O3Color and Shape:SolidMolecular weight:450.38Kalafungin
CAS:<p>Kalafungin inhibits various fungi, yeasts, protozoa, and gram-positive bacteria, less so for gram-negative bacteria.</p>Formula:C16H12O6Color and Shape:SolidMolecular weight:300.26Cilazapril HCl
CAS:<p>Cilazapril, also known as Ro 31 2848, is a potent ACE inhibitor used for hypertension.</p>Formula:C22H32ClN3O5Color and Shape:SolidMolecular weight:453.96Anti-TSWV agent 1
<p>Anti-TSWV agent 1 is a highly effective inactivator (EC50:144 μg/mL) of tomato spotted wilt virus (TSWV).</p>Formula:C22H27ClN4OS3Color and Shape:SolidMolecular weight:495.12Iroxanadine hydrobromide
CAS:<p>Iroxanadine hydrobromide is a MAPK p38 inhibitor potentially for the treatment of atherosclerosis.</p>Formula:C14H21BrN4OColor and Shape:SolidMolecular weight:341.25ND-654
CAS:<p>ND-654 is an acetyl CoA carboxylase inhibitor.</p>Formula:C29H33N3O8SColor and Shape:SolidMolecular weight:583.65Flusoxolol
CAS:<p>Flusoxolol is a beta-adrenoceptor partial agonist.</p>Formula:C22H30FNO4Color and Shape:SolidMolecular weight:391.48RXR antagonist 2
<p>RXR antagonist 2 is a potent antagonist of RXR (Ki: 0.391 μM, Kd: 0.281 μM). RXR antagonist 2 has shown research potential for RXR-related diseases.</p>Formula:C29H35F3N2O3Color and Shape:SolidMolecular weight:516.6Freselestat quarterhydrate
<p>ONO-6818 quarterhydrate: oral neutrophil elastase inhibitor, Ki 12.2 nM; >100x less effective on other proteases; strong anti-inflammatory.</p>Formula:C23H30N6O5Color and Shape:SolidMolecular weight:457.03FTI-2153 TFA
<p>FTI-2153 TFA inhibits farnesyltransferase with high selectivity (IC50: 1.4 nM), over 3000x more than Rap1A processing.</p>Formula:C27H31F3N4O5SColor and Shape:SolidMolecular weight:580.62Anticancer agent 35
<p>Compound 10, a sulfonylurea, inhibits A549, A431, PACA2 cells with IC50s: 18.1, 4.0, 18.9 μg/mL.</p>Formula:C15H13N3O3S3Color and Shape:SolidMolecular weight:379.48Kaitocephalin
CAS:<p>Kaitocephalin: naturally occurring, non-selective antagonist blocking glutamate receptors, made by Eupenicillium shearii fungus.</p>Formula:C18H21Cl2N3O9Color and Shape:SolidMolecular weight:494.28GZN39838
CAS:<p>GZN39838, a natural Kv1.2 blocker, induces C-type inactivation without blocking the outer pore.</p>Formula:C22H30O6Color and Shape:SolidMolecular weight:390.47Glutaminyl cyclases-IN-1
<p>Glutaminyl cyclase inhibitor IsoQC-IN-1: IC50=12 nM for QC, 73 nM for isoQC; blocks CD47/SIRPα; boosts THP-1, U937 macrophage phagocytosis.</p>Formula:C25H30N6O2SColor and Shape:SolidMolecular weight:478.61Antibiotic MA 144M1
CAS:<p>Antibiotic MA 144M1, an anthracycline, targets gram-positive bacteria and animal tumors; derived from Streptomyces fermentation or aclacinomycin A conversion.</p>Formula:C42H55NO15Color and Shape:SolidMolecular weight:813.88P-gp modulator 1
CAS:<p>P-gp modulator 1 is a high affinity and orally available P-glycoprotein (Pgp) modulator</p>Formula:C41H72N2O6Purity:98%Color and Shape:SolidMolecular weight:689.02Antileishmanial agent-6
<p>Antileishmanial agent-6: potent against Leishmania donovani, IC50 0.54μM; cytotoxic IC50 10.2μM.</p>Formula:C24H26O8Color and Shape:SolidMolecular weight:442.46YW3-56
CAS:<p>YW3-56 is a potent peptidylarginine deiminase (PAD) inhibitor, with an IC50 of 1-5 μM for PAD4.</p>Formula:C27H32ClN5O2Color and Shape:SolidMolecular weight:494.03Fandosentan
CAS:<p>Fandosentan is an endothelin receptor antagonist.</p>Formula:C25H18F3NO6SColor and Shape:SolidMolecular weight:517.47Encephalitic alphavirus-IN-1
<p>Alphavirus-IN-1 blocks VEEV (EC50: 0.24 μM) & EEEV (EC50: 0.16 μM), non-toxic, stable in mice plasma.</p>Formula:C27H25FN6O2Color and Shape:SolidMolecular weight:484.52FCE-27262
CAS:<p>FCE-27262 is a prostaglandin H2/thromboxane A2 receptor antagonist.</p>Formula:C23H31N3O3Color and Shape:SolidMolecular weight:397.51DWN-12088 HCl
CAS:<p>DWN-12088 HCl is the salt form of DWN-12088 Free Base, an orally administered small molecule prolyl-tRNA synthetase (PRS) inhibitor</p>Formula:C15H21Cl4N3OColor and Shape:SolidMolecular weight:401.15ASB14780
<p>ASB14780 is a 4-phenoxy derivative and an inhibitor of cytoplasmic phospholipase cPLA2α (IC50: 20 nM).</p>Color and Shape:SolidGSK3527497
CAS:<p>GSK3527497 is a novel potent and selective inhibitor of transient receptor potential vanilloid-4 (TRPV4).</p>Formula:C17H16ClFN4O4SColor and Shape:SolidMolecular weight:426.85MDL-43291
CAS:<p>MDL-43291 is a leukotriene receptor antagonist.</p>Formula:C25H42O4SColor and Shape:SolidMolecular weight:438.66Anticancer agent 12
<p>Anticancer agent 12 shows cytotoxic activity in malignant cells with no hepatotoxicity.</p>Formula:C16H17BrN4O2SColor and Shape:SolidMolecular weight:409.3METTL3-IN-2
CAS:<p>METTL3-IN-2, a potent METTL3 inhibitor, exhibits an IC50 value of 6.1 nM, effectively impairing the proliferation of Caov3 cancer cells.</p>Formula:C25H26N8OColor and Shape:SolidMolecular weight:454.53NCI-006
CAS:<p>NCI-006, an LDH inhibitor, slows tumor growth and enhances pyruvate's role in mitochondrial metabolism.</p>Formula:C31H24F2N4O4S3Color and Shape:SolidMolecular weight:650.74TP-6076
CAS:<p>TP-6076 is a fluorocycline antibiotic, inhibiting bacterial protein synthesis, exhibiting great antimicrobial activity against carbapenem-resistant A.</p>Formula:C28H32F3N3O7Color and Shape:SolidMolecular weight:579.56NB-216
CAS:<p>NB-216 is a macrocyclic peptidic BACE-1 inhibitor.</p>Formula:C35H45N3O4Color and Shape:SolidMolecular weight:571.75MEN-10354
CAS:<p>MEN-10354 is a less potent and less selective NK-2 tachykinin receptor antagonist compared to the linear analog, R 396.</p>Formula:C37H46N8O9Color and Shape:SolidMolecular weight:746.81AZD-3199 dihydrobromide
CAS:<p>AZD-3199 dihydrobromide is a β2 adrenergic receptor agonist potentially for the treatment of asthma and chronic obstructive.</p>Formula:C32H44Br2N4O4SColor and Shape:SolidMolecular weight:740.59AFM-30a hydrochloride
<p>AFM-30a hydrochloride: selective PAD2 inhibitor, EC50 9.5 μM; blocks H3 guanylation, EC50 0.4 μM; used for cancer and autoimmune research.</p>Formula:C24H28ClFN6O3Color and Shape:SolidMolecular weight:502.974α-PDD
CAS:<p>4alpha-PDD activates transient receptor potential vanilloid 4 (TRPV4) channels and is inactive for signaling through PKC.</p>Formula:C40H64O8Color and Shape:SolidMolecular weight:672.93Freselestat
CAS:<p>Freselestat (ONO-6818) inhibits neutrophil elastase, reduces interleukin 8, C5B-9, and inflammation in cardiopulmonary bypass.</p>Formula:C23H28N6O4Color and Shape:SolidMolecular weight:452.513-IN-PP1
CAS:<p>3-IN-PP1: PKD inhibitor (IC50: 94-108 nM for PKD1/2/3), broad anticancer agent for research.</p>Formula:C17H18N6Color and Shape:SolidMolecular weight:306.36ONO-AE1-329
CAS:<p>ONO-AE1-329 is a novel agonist of the prostaglandin PGE2 receptor EP4.</p>Formula:C22H30O6S2Color and Shape:SolidMolecular weight:454.6MtDTBS-IN-1
<p>MtDTBS-IN-1 is a notably potent binder (K_D = 57 nM) and inhibitor (K_i = 5 μM) of MtDTBS.</p>Formula:C16H16N4O5Color and Shape:SolidMolecular weight:344.32BMS-554417
CAS:<p>BMS-554417 inhibits IGF-IR/insulin receptors, curbing cell proliferation and tumor growth, with IC50 values of 120 nm–>8.5 μmol/L.</p>Formula:C28H30ClN7O2Color and Shape:SolidMolecular weight:532.04PEN-866
CAS:<p>PEN-866, a conjugate of HSP90i and SN-38, may control early NSCLC tumor growth.</p>Formula:C49H49N7O9Color and Shape:SolidMolecular weight:879.95O-Propargyl-Puromycin
CAS:<p>O-Propargyl-Puromycin (OP-puro) is a potent protein synthesis inhibitor, a puromycin acetylene analog.</p>Formula:C24H29N7O5Purity:97.83% - 99.70%Color and Shape:SolidMolecular weight:495.53
