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Other Inhibitors

Other Inhibitors

This category encompasses a wide variety of inhibitors that do not fit into the standard classifications but are still critical for various biochemical and pharmacological research. These inhibitors may target unique or less-studied pathways, enzymes, and molecular interactions, providing valuable tools for specialized research areas. At CymitQuimica, we offer a diverse selection of high-quality inhibitors across multiple biological targets and research disciplines, enabling you to explore novel therapeutic avenues and deepen your understanding of complex biological processes.

Found 37827 products of "Other Inhibitors"

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  • Heme Oxygenase-2-IN-1


    <p>Heme Oxygenase-2-IN-1 is a selective HO-2 inhibitor with IC50s: 14.9 μM (HO-1), 0.9 μM (HO-2).</p>
    Formula:C19H17N3O2
    Color and Shape:Solid
    Molecular weight:319.36
  • RTIOX-372

    CAS:
    <p>RTIOX-372 is a potent and selective orexin-1 receptor antagonist.</p>
    Formula:C30H39N5O3
    Color and Shape:Solid
    Molecular weight:517.66
  • Monamycin H1

    CAS:
    <p>Monamycin H1 is an ester peptide antibiotic that exhibits activity against Gram-positive bacteria.</p>
    Formula:C34H56ClN7O8
    Color and Shape:Solid
    Molecular weight:726.30
  • Gepotidacin hydrochloride

    CAS:
    <p>Gepotidacin (GSK-2140944) is a potent DNA topoisomerase inhibitor, a novel antibacterial efficacious against various anaerobes.</p>
    Formula:C24H29ClN6O3
    Color and Shape:Solid
    Molecular weight:484.98
  • Artemisiane E

    CAS:
    <p>Artemisiane E is a potent PI3K/AKT pathway inhibitor with an IC 50 of 8.9 μM .</p>
    Formula:C20H22O5
    Color and Shape:Solid
    Molecular weight:342.39
  • 3-O-Demethylmonensin A

    CAS:
    <p>3-O-Demethylmonensin A is a polyether antibiotic produced by Streptomyces cinnamonensis (strain LO-63).</p>
    Formula:C35H60O11
    Color and Shape:Solid
    Molecular weight:656.84
  • Epoxyquinomicin C

    CAS:
    <p>Epoxyquinomicin C is an antibiotic that can be isolated from Amycolatopsis sp. It exhibits anti-inflammatory properties against collagen-induced arthritis and is also utilized in the synthesis of the NF-κB inhibitor DHMEQ.</p>
    Formula:C14H13NO6
    Color and Shape:Solid
    Molecular weight:291.256
  • Kahweol linoleate

    CAS:
    <p>Kahweol linoleate, a semi-synthetic from coffee, blocks osteoclast creation, fights cancerous cells, prevents DNA damage, and reduces oxidative stress.</p>
    Formula:C38H56O4
    Color and Shape:Solid
    Molecular weight:576.85
  • GRPR antagonist-2


    <p>GRPR antagonist-2 blocks GRPR, kills some cancer cells, effective on HGC-27 (IC50: 0.77 μM) &amp; Pan02 (IC50: 2.5 μM).</p>
    Formula:C28H32F3N5O4
    Color and Shape:Solid
    Molecular weight:559.58
  • Amdinocillin methylacetate

    CAS:
    <p>Amdinocillin methylacetate is a Synthetic penicillin.</p>
    Formula:C18H27N3O4S
    Color and Shape:Solid
    Molecular weight:381.49
  • Plumbemycin A

    CAS:
    <p>Plumbemycin A is isolated from Streptomyces plumbeus; an L-threonine antagonist.</p>
    Formula:C12H20N3O9P
    Color and Shape:Solid
    Molecular weight:381.28
  • Feigrisolide D

    CAS:
    <p>Feigrisolide D is a lactone produced by Streptomyces griseus. It exhibits moderate inhibitory activity against 3α-hydroxysteroid dehydrogenase.</p>
    Formula:C22H38O7
    Color and Shape:Solid
    Molecular weight:414.533
  • Topoisomerase I/II inhibitor 2


    <p>Compound 1a inhibits Topoisomerase I/II, shrinks mouse liver tumors, IC50: 6.83/9.82 μM for LM9/Huh7 cells.</p>
    Formula:C19H16N2O4
    Color and Shape:Solid
    Molecular weight:336.34
  • MRS2179 tetrasodium hydrate


    <p>MRS2179 blocks turkey P2Y1 receptor (Kb 102 nM, pA2 6.99), affects platelet aggregation, and has varying IC50s on P2 receptors.</p>
    Formula:C11H15N5Na4O10P2
    Color and Shape:Solid
    Molecular weight:576.21
  • DAD dichloride


    <p>DAD dichloride is a 3rd-gen photoelectric switch, blocks K+ channels, and helps in visual function research.</p>
    Formula:C26H42Cl2N6O
    Color and Shape:Solid
    Molecular weight:525.56
  • PI3K-IN-23


    <p>PI3K-IN-23 is a (E)-9-oxooctadec-10-en-12-ynoic acid analogue that promotes glucose uptake (EC50: 7.00 μM).</p>
    Formula:C24H33NO4S
    Color and Shape:Solid
    Molecular weight:431.59
  • DMP-728 free base

    CAS:
    <p>DMP-728 free base is a highly potent and selective GPIIbDIIa antagonist</p>
    Formula:C25H36N8O7
    Color and Shape:Solid
    Molecular weight:560.60
  • GSK866

    CAS:
    <p>GSK866 is a selective glucocorticoid receptor agonist (SEGRA).</p>
    Formula:C23H21Cl2F4N5O3
    Color and Shape:Solid
    Molecular weight:562.34
  • HS-731

    CAS:
    <p>HS-731 is a μ-Opioid Receptor Agonist.</p>
    Formula:C20H26N2O5
    Color and Shape:Solid
    Molecular weight:374.43
  • 1-Deamino-1-hydroxygentamicin C1a

    CAS:
    <p>1-Deamino-1-hydroxygentamicin C1a (AntibioticSU-2) is an aminoglycoside antibiotic effective against both gram-positive and gram-negative bacteria.</p>
    Formula:C19H38N4O8
    Color and Shape:Solid
    Molecular weight:450.527
  • Retezorogant

    CAS:
    <p>Retezorogant is a retinoic acid receptor-related orphan receptor gamma (RORγ) antagonist.</p>
    Formula:C23H33ClN2O3
    Color and Shape:Solid
    Molecular weight:420.97
  • ER Thermo Yellow

    CAS:
    <p>ER Thermo Yellow is a high-sensitivity (3.9%/°C) fluorescent probe designed for temperature visualization specifically targeting the endoplasmic reticulum.</p>
    Formula:C27H20BClF5N3O3
    Molecular weight:575.72
  • PPARγ agonist 1


    <p>PPARγ agonist 1 is a potent agonist of PPARγ that efficiently activates hPPARγ without causing full agonism, thereby avoiding adverse effects.</p>
    Formula:C34H39NO3
    Color and Shape:Solid
    Molecular weight:509.68
  • Peridinin

    CAS:
    <p>Peridinin is an exceptionally potent and membrane-embedded inhibitor of bilayer lipid peroxidation.</p>
    Formula:C39H50O7
    Color and Shape:Solid
    Molecular weight:630.81
  • BDZ-h

    CAS:
    <p>BDZ-h inhibits both closed/open states of all 4 homomeric &amp; 2 GluA2R-complex AMPA receptors.</p>
    Formula:C21H21N5O3S
    Color and Shape:Solid
    Molecular weight:423.49
  • RK-582

    CAS:
    <p>RK-582: oral spiroindolinone tankyrase inhibitor, halts colon cancer growth in COLO-320DM mouse model.</p>
    Formula:C27H35FN6O3
    Color and Shape:Solid
    Molecular weight:510.6
  • AKR1C3-IN-7


    <p>AKR1C3-IN-7 (Compound 13) is an effective and selective AKR1C3 inhibitor (IC50=0.19 μM). AKR1C3-IN-7 has antitumor activity.</p>
    Formula:C24H20N2O4
    Color and Shape:Solid
    Molecular weight:400.43
  • TRPC4/5-IN-1


    <p>TRPC4/5-IN-1, a TRPC5/4 inhibitor with IC50s 0.54 μM/2.06 μM, targets skin inflammation and proteinuric kidney diseases.</p>
    Formula:C21H21N3O
    Color and Shape:Solid
    Molecular weight:331.41
  • Piperazinomycin

    CAS:
    <p>Piperazinomycin is an antifungal antibiotic, showing inhibitory activity against fungi and yeasts, especially against Trichophyton.</p>
    Formula:C18H20N2O2
    Color and Shape:Solid
    Molecular weight:296.36
  • Anticancer agent 80


    <p>Anticancer agent 80 (Compound 3c) is an anticancer agent that exhibits a significant dark toxic effect on T47-D (IC50: 10.14 μM).</p>
    Formula:C19H12BrNO5
    Color and Shape:Solid
    Molecular weight:414.21
  • AKR1C3-IN-8


    <p>AKR1C3-IN-8 (Compound 5) is an effective and selective AKR1C3 inhibitor (IC50=0.069 μM). AKR1C3-IN-8 has antitumor activity.</p>
    Formula:C23H20N4O3
    Color and Shape:Solid
    Molecular weight:400.43
  • AVE-1330A sodium

    CAS:
    <p>AVE-1330A sodium is a beta-Lactamase inhibitor.</p>
    Formula:C7H10N3NaO6S
    Color and Shape:Solid
    Molecular weight:287.23
  • PF-06815345 hydrochloride

    CAS:
    <p>PF-06815345 HCl is an oral, potent PCSK9 inhibitor, IC50 13.4 μM, lowers PCSK9 in mice.</p>
    Formula:C27H30Cl2FN9O4
    Color and Shape:Solid
    Molecular weight:634.49
  • PIKfyve-IN-1


    <p>PIKfyve-IN-1: potent, cell-active inhibitor for PIKfyve research, IC50=6.9 nM.</p>
    Formula:C20H21N5
    Color and Shape:Solid
    Molecular weight:331.41
  • Nolpitantium Free Base

    CAS:
    <p>Nolpitantium is a potent, selective NK1 receptor antagonist that inhibits substance P without affecting NK2/NK3 receptors.</p>
    Formula:C37H45Cl2N2O2
    Color and Shape:Solid
    Molecular weight:620.67
  • Pefcalcitol

    CAS:
    <p>Pefcalcitol is a novel antipsoriatic prodrug candidate containing a 16-en-22-oxa-vitamin D3 structure.</p>
    Formula:C26H34F5NO4
    Color and Shape:Solid
    Molecular weight:519.54
  • LAS195319

    CAS:
    <p>LAS195319 is a potent and selective inhaled PI3Kδ Inhibitor (IC50 = 0.5 nM) for the Treatment of Respiratory Diseases.</p>
    Formula:C29H26N10O3S
    Color and Shape:Solid
    Molecular weight:594.65
  • TrxR-IN-2


    <p>TrxR-IN-2 is a potential thioredoxin reductase (TrxR) inhibitor. TrxR-IN-2 has research value in the chemotherapy of drug-resistant hepatocellular carcinoma.</p>
    Formula:C22H22N4O4
    Color and Shape:Solid
    Molecular weight:406.43
  • Mepixetil


    <p>Mepixetil is a potent angiotensin II receptor antagonist[1].</p>
    Formula:C12H18N2O3
    Color and Shape:Solid
    Molecular weight:238.28
  • 22-HDHA

    CAS:
    <p>22-HDHA is an oxidation product of docosahexaenoic acid .</p>
    Formula:C22H32O3
    Color and Shape:Solid
    Molecular weight:344.49
  • Topoisomerase I inhibitor 8

    CAS:
    <p>Topoisomerase I inhibitor 8, a hexacyclic analogue of camptothecin, is also a potent inhibitor of topoisomerase I and is toxic to tumour cells.</p>
    Formula:C24H21FN2O4
    Color and Shape:Solid
    Molecular weight:420.43
  • MurB-IN-1


    <p>MurB-IN-1 (compound 44) inhibits key bacterial enzyme MurB with 3.57 μM affinity, offering treatment potential against P. aeruginosa.</p>
    Formula:C12H7Cl2F3N2O2
    Color and Shape:Solid
    Molecular weight:339.1
  • Antibacterial agent 70


    <p>Antibacterial agent 70 is a new dihydropyrimidinone-imidazole hybrid antimicrobial agent (MIC: 0.5 μg/ml).</p>
    Formula:C25H32ClN7O6S
    Color and Shape:Solid
    Molecular weight:594.08
  • 5(S),6(R)-DiHETE

    CAS:
    <p>5(S),6(R)-DiHETE is a dihydroxy fatty acid from LTA4 hydrolysis and weak LTD4 agonist with ED50 of 1.3 μM for guinea pig ileum contraction.</p>
    Formula:C20H32O4
    Color and Shape:Solid
    Molecular weight:336.47
  • SSTR5 antagonist 2 hydrochloride


    <p>SSTR5 antagonist 2 hydrochloride: potent, oral SSTR5 blocker with potential in type 2 diabetes research.</p>
    Formula:C32H36ClFN2O5
    Color and Shape:Solid
    Molecular weight:583.09
  • Indinavir monohydrate

    CAS:
    <p>Indinavir monohydrate is a potent and specific HIV protease inhibitor that appears to have good oral bioavailability.</p>
    Formula:C36H49N5O5
    Color and Shape:Solid
    Molecular weight:631.82
  • Tacrolimus anhydrous 8-epimer

    CAS:
    <p>Tacrolimus anhydrous 8-epimer, an immunosuppressive l-pipecolic acid macrolide, blocks T cell growth by hindering IL-2.</p>
    Formula:C44H69NO12
    Color and Shape:Solid
    Molecular weight:804.02
  • 9(R)-HETE

    CAS:
    <p>9(R)-HETE, 50% of racemic mix, activates RXRγ 1.5x at 300 nM; identified by HPLC comparison.</p>
    Formula:C20H32O3
    Color and Shape:Solid
    Molecular weight:320.47
  • GW-597901 cinnamate

    CAS:
    <p>GW-597901 cinnamate is a long-acting beta(2)-agonist.</p>
    Formula:C34H46N2O8S
    Color and Shape:Solid
    Molecular weight:642.80
  • Queenslandon

    CAS:
    <p>Queenslandon exhibits moderate antifungal activity against fungi such as Streptomyces, Penicillium, Aspergillus fumigatus, and Aspergillus flavus, and has no effect on bacteria.</p>
    Formula:C20H26O8
    Color and Shape:Solid
    Molecular weight:394.42