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Other Inhibitors

Other Inhibitors

This category encompasses a wide variety of inhibitors that do not fit into the standard classifications but are still critical for various biochemical and pharmacological research. These inhibitors may target unique or less-studied pathways, enzymes, and molecular interactions, providing valuable tools for specialized research areas. At CymitQuimica, we offer a diverse selection of high-quality inhibitors across multiple biological targets and research disciplines, enabling you to explore novel therapeutic avenues and deepen your understanding of complex biological processes.

Found 37926 products of "Other Inhibitors"

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  • 16(R)-Iloprost

    CAS:
    <p>Iloprost, a potent prostacyclin analog, binds IP &amp; EP1 receptors (Ki 11 nM), contains 16(S/R) isomers, and inhibits platelets (IC50 65 nM).</p>
    Formula:C22H32O4
    Color and Shape:Solid
    Molecular weight:360.49
  • Purine phosphoribosyltransferase-IN-2


    <p>Purine PRTase-IN-2 inhibits Pf, Pv, Tbr PRT; Ki: 30, 20, 2 nM.</p>
    Formula:C11H15N5Na4O10P2
    Color and Shape:Solid
    Molecular weight:531.17
  • AFM-30a hydrochloride


    <p>AFM-30a hydrochloride: selective PAD2 inhibitor, EC50 9.5 μM; blocks H3 guanylation, EC50 0.4 μM; used for cancer and autoimmune research.</p>
    Formula:C24H28ClFN6O3
    Color and Shape:Solid
    Molecular weight:502.97
  • Luffolide

    CAS:
    <p>Luffolide, a Luffariella sponge metabolite, shares manoalide's anti-inflammatory traits and fully inhibits PLA2's cleavage of phosphatidylcholine.</p>
    Formula:C27H40O6
    Color and Shape:Solid
    Molecular weight:460.60
  • Carbacyclin

    CAS:
    <p>Carbacyclin, a PGI2 analog, is a prostacyclin (PGI2) receptor agonist and vasodilator with potent inhibitory platelet aggregation.</p>
    Formula:C21H34O4
    Purity:98%
    Color and Shape:Solid
    Molecular weight:350.49
  • TCMDC-125431


    <p>TCMDC-125431 is a novel inhibitor of Plasmodium calcium kinetics with minimal inhibition of haemoglobin crystals.</p>
    Formula:C25H27N3O2S
    Color and Shape:Solid
    Molecular weight:433.57
  • Saprisartan potassium

    CAS:
    <p>Saprisartan potassium is an Angiotensin II Type 1 receptor antagonist and antihypertensive agent.</p>
    Formula:C25H21BrF3KN4O4S
    Color and Shape:Solid
    Molecular weight:649.52
  • PX-316

    CAS:
    <p>PX-316: AKT inhibitor, reduces Akt activity by 78% in HT-29 xenografts, effective against MCF-7 and HT-29 cancers, well-tolerated intravenously.</p>
    Formula:C28H57O10P
    Color and Shape:Solid
    Molecular weight:584.72
  • BMS-554417

    CAS:
    <p>BMS-554417 inhibits IGF-IR/insulin receptors, curbing cell proliferation and tumor growth, with IC50 values of 120 nm–&gt;8.5 μmol/L.</p>
    Formula:C28H30ClN7O2
    Color and Shape:Solid
    Molecular weight:532.04
  • GSK2945 hydrochloride


    <p>GSK2945 HCl is a specific Rev-erbα antagonist, EC50: 21.5 μM (mouse), 20.8 μM (human), increases cholesterol 7α-hydroxylase.</p>
    Formula:C20H19Cl3N2O2S
    Color and Shape:Solid
    Molecular weight:457.8
  • TRK-IN-19


    <p>TRK-IN-19 (I-10) inhibits TRKA (1.1 nM IC50) &amp; TRKAG595R (5.3 nM), promising for cancer research.</p>
    Formula:C22H26FN5O2
    Color and Shape:Solid
    Molecular weight:411.47
  • ORP-101

    CAS:
    <p>ORP-101: large, stable molecule with partial μ agonist, full κ antagonist properties.</p>
    Formula:C60H84N2O8
    Color and Shape:Solid
    Molecular weight:961.32
  • (±)-ANAP hydrochloride (1185251-08-4 free base)


    <p>(±)-ANAP hydrochloride is the amino acid analog of prodan. It can be used as a fluorescent probes and enhance environmental sensitivity.</p>
    Formula:C15H17ClN2O3
    Purity:98%
    Color and Shape:Solid
    Molecular weight:308.76
  • AGN-204396

    CAS:
    <p>AGN-204396 is an antagonist that selectively blocks the activity of prostamides (prostaglandin-ethanolamides).</p>
    Formula:C32H44FN3O4
    Color and Shape:Solid
    Molecular weight:553.71
  • ATX inhibitor 12


    <p>Oral ATX inhibitor 12 (IC50: 1.72 nM) at 60 mg/kg prevents lung damage in C57Bl/6J mice.</p>
    Formula:C30H34FN5O2
    Color and Shape:Solid
    Molecular weight:515.62
  • Antimalarial agent 9


    <p>Antimalarial 9, a quinoline-imidazole derivative, effectively targets CQ-susceptible (IC50-0.14 μM) and MDR strains (IC50-0.41 μM) with low toxicity.</p>
    Formula:C28H32BrN3O2
    Color and Shape:Solid
    Molecular weight:522.48
  • AS1940477

    CAS:
    <p>AS1940477 selectively inhibits p38 MAPK α/β, blocks proinflammatory cytokines in cells, and has anti-inflammatory effects in rats.</p>
    Formula:C24H22FN5O2
    Color and Shape:Solid
    Molecular weight:431.46
  • SHR0687

    CAS:
    <p>SHR0687: potent KOR agonist, selective, favorable PK, effective in rat pain model, minimal BBB penetration, less CNS side effects.</p>
    Formula:C39H60N8O5
    Color and Shape:Solid
    Molecular weight:720.94
  • Epiderstatin

    CAS:
    <p>Epiderstatin is isolated from Streptomyces pulveraceus subsp. epiderstagenes; inhibits mitogenic activity of epidermal growth factor.</p>
    Formula:C15H20N2O4
    Color and Shape:Solid
    Molecular weight:292.33
  • E-3030 free acid

    CAS:
    <p>E-3030 free acid, a PPAR agonist, lowers blood glucose, triglycerides, and insulin; boosts adiponectin; reduces apo C-III; and raises lipoprotein lipase.</p>
    Formula:C22H23ClFNO5
    Purity:98%
    Color and Shape:Solid
    Molecular weight:435.87
  • TLN-232

    CAS:
    <p>TLN-232, a synthetic heptapeptide, may inhibit cancer by targeting M2PK to disrupt tumor cell energy production.</p>
    Formula:C36H49N9O7S2
    Color and Shape:Solid
    Molecular weight:783.96
  • MV061194

    CAS:
    <p>MV061194 is a potent and selective cathepsin K (Cat K) inhibitor.</p>
    Formula:C28H37N5O4S
    Color and Shape:Solid
    Molecular weight:539.69
  • NCI-006

    CAS:
    <p>NCI-006, an LDH inhibitor, slows tumor growth and enhances pyruvate's role in mitochondrial metabolism.</p>
    Formula:C31H24F2N4O4S3
    Color and Shape:Solid
    Molecular weight:650.74
  • Ascofuranone

    CAS:
    <p>Ascofuranone is an inhibitor of the ubiquinol oxidase activity of Trypanosoma brucei mitochondrial alternative oxidase (TAO), as well as an inhibitor of HsDHODH</p>
    Formula:C23H29ClO5
    Color and Shape:Solid
    Molecular weight:420.93
  • Epelmycin C

    CAS:
    <p>Epelmycin C exhibits antibacterial activity against both Gram-positive and Gram-negative bacteria, as well as antifungal activity against Candida albicans. It also shows activity against leukemia L1210.</p>
    Formula:C36H45NO14
    Color and Shape:Solid
    Molecular weight:715.741
  • MDL-43291

    CAS:
    <p>MDL-43291 is a leukotriene receptor antagonist.</p>
    Formula:C25H42O4S
    Color and Shape:Solid
    Molecular weight:438.66
  • VEGFR-2-IN-26

    CAS:
    <p>VEGFR-2-IN-26 inhibits VEGFR-2 (IC50: 15.5 nM), combating various cancers' cell growth.</p>
    Formula:C24H19F3N6O2
    Color and Shape:Solid
    Molecular weight:480.44
  • Anticancer agent 79


    <p>Anticancer agent 79 (3d) has potent activity against breast cancer, with cytotoxic effects on T47-D, IC50=13.64±0.26μM.</p>
    Formula:C20H12F3NO5
    Color and Shape:Solid
    Molecular weight:403.31
  • Anti-TSWV agent 1


    <p>Anti-TSWV agent 1 is a highly effective inactivator (EC50:144 μg/mL) of tomato spotted wilt virus (TSWV).</p>
    Formula:C22H27ClN4OS3
    Color and Shape:Solid
    Molecular weight:495.12
  • MCTR2

    CAS:
    <p>MCTR2, synthesized from DHA in macrophages, aids in tissue repair and reduces inflammation by promoting eicosanoid PGD2 and PGF2α decrease.</p>
    Formula:C27H40N2O6S
    Color and Shape:Solid
    Molecular weight:520.68
  • Enpp-1-IN-11


    <p>Enpp-1-IN-11 inhibits ENPP1 with a 45 nM Ki, is plasma stable, and has low clearance in human/mouse livers, potentially aiding cancer research.</p>
    Formula:C15H15N5O3S
    Color and Shape:Solid
    Molecular weight:345.38
  • Ezomycin D2

    CAS:
    <p>Ezomycin D2 is an antifungal antibiotic effective primarily against plant pathogens such as Sclerotinia sclerotiorum and Botrytis cinerea. It helps control diseases like sclerotinia blight and gray mold in crops, as well as candidiasis.</p>
    Formula:C19H27N5O14
    Color and Shape:Solid
    Molecular weight:549.443
  • Griseusin B

    CAS:
    <p>Griseusin B is a quinone antibiotic primarily effective against Gram-positive bacteria.</p>
    Formula:C22H22O10
    Color and Shape:Solid
    Molecular weight:446.404
  • PD-149163

    CAS:
    <p>PD-149163: brain-penetrating, selective NTR1 agonist; shows pro-cognitive, anti-psychotic, anxiolytic effects.</p>
    Formula:C42H71N9O6
    Color and Shape:Solid
    Molecular weight:798.07
  • SX 3202

    CAS:
    <p>SX 3202 is an aldose reductase inhibitor being developed for the treatment of diabetic neuropathy.</p>
    Formula:C17H11BrFN3O4
    Color and Shape:Solid
    Molecular weight:420.19
  • NPEC-caged-(S)-3,4-DCPG

    CAS:
    <p>mGlu8a agonist</p>
    Formula:C19H16N2O10
    Purity:98%
    Color and Shape:Solid
    Molecular weight:432.34
  • Chrymutasin B

    CAS:
    <p>Chrymutasin B is a glycoside antitumor antibiotic known for its cytotoxic properties.</p>
    Formula:C32H31NO13
    Color and Shape:Solid
    Molecular weight:637.587
  • 6"'-Deamino-6"'-hydroxyparomomycin I

    CAS:
    <p>6"'-Deamino-6"'-hydroxyparomomycin I is an aminoglycoside antibiotic produced by Streptomyces rimosus forma paromomycinus A67 15, exhibiting activity against both Gram-positive and Gram-negative bacteria. It serves as an intermediate in the biosynthesis of paromomycin.</p>
    Formula:C23H44N4O15
    Color and Shape:Solid
    Molecular weight:616.613
  • AKR1C3-IN-7


    <p>AKR1C3-IN-7 (Compound 13) is an effective and selective AKR1C3 inhibitor (IC50=0.19 μM). AKR1C3-IN-7 has antitumor activity.</p>
    Formula:C24H20N2O4
    Color and Shape:Solid
    Molecular weight:400.43
  • Tacrolimus anhydrous 8-epimer

    CAS:
    <p>Tacrolimus anhydrous 8-epimer, an immunosuppressive l-pipecolic acid macrolide, blocks T cell growth by hindering IL-2.</p>
    Formula:C44H69NO12
    Color and Shape:Solid
    Molecular weight:804.02
  • Antibacterial agent 70


    <p>Antibacterial agent 70 is a new dihydropyrimidinone-imidazole hybrid antimicrobial agent (MIC: 0.5 μg/ml).</p>
    Formula:C25H32ClN7O6S
    Color and Shape:Solid
    Molecular weight:594.08
  • Diolmycin A1

    CAS:
    <p>Diolmycin A1 is an antibiotic known for its anticoccidial activity.</p>
    Formula:C18H19NO3
    Color and Shape:Solid
    Molecular weight:297.348
  • Hydrolyzed Fumonisin B2

    CAS:
    <p>Hydrolyzed Fumonisin B2 (HFB2) is a hydrolysis product of fumonisins (HF), which retains biological activity. It exhibits phytotoxicity.</p>
    Formula:C22H47NO4
    Purity:98%
    Color and Shape:Solid
    Molecular weight:389.61
  • Cacospongionolide B

    CAS:
    <p>Cacospongionolide B from Fasciospongia cavernosa inhibits secretory phospholipase A2, curbing inflammation.</p>
    Formula:C25H36O4
    Color and Shape:Solid
    Molecular weight:400.55
  • PF-06815345 hydrochloride

    CAS:
    <p>PF-06815345 HCl is an oral, potent PCSK9 inhibitor, IC50 13.4 μM, lowers PCSK9 in mice.</p>
    Formula:C27H30Cl2FN9O4
    Color and Shape:Solid
    Molecular weight:634.49
  • Gilvusmycin

    CAS:
    <p>Gilvusmycin is an antibiotic with potent antitumor properties. It effectively inhibits the proliferation of P388, K562, A431, and MKN28 cells, with IC50 values (ng/mL) of 0.08, 0.86, 0.72, and 0.75, respectively.</p>
    Formula:C38H34N6O8
    Color and Shape:Solid
    Molecular weight:702.712
  • Heparastatin

    CAS:
    <p>Heparastatin is an inhibitor of heparanase.</p>
    Formula:C8H11F3N2O5
    Purity:98%
    Color and Shape:Solid
    Molecular weight:272.18
  • Steroid sulfatase-IN-4


    <p>Steroid sulfatase-IN-4 irreversibly inhibits human STS with a 25 nM IC50, useful for endometriosis research.</p>
    Formula:C19H17ClN2O5S
    Color and Shape:Solid
    Molecular weight:420.87
  • BDZ-h

    CAS:
    <p>BDZ-h inhibits both closed/open states of all 4 homomeric &amp; 2 GluA2R-complex AMPA receptors.</p>
    Formula:C21H21N5O3S
    Color and Shape:Solid
    Molecular weight:423.49
  • PPARγ agonist 1


    <p>PPARγ agonist 1 is a potent agonist of PPARγ that efficiently activates hPPARγ without causing full agonism, thereby avoiding adverse effects.</p>
    Formula:C34H39NO3
    Color and Shape:Solid
    Molecular weight:509.68