Building Blocks

Versatile small molecule scaffold

Versatile small molecule scaffold

Versatile small molecule scaffold

Versatile small molecule scaffold

<p>Versatile small molecule scaffold</p>

<p>Versatile small molecule scaffold</p>

Versatile small molecule scaffold

5,7-Dichlorobenzo[d]thiazol-2-amine is a carbonyl compound that binds to receptors and inhibits the binding of natural ligands. It has been shown to have affinity for dopamine receptors, serotonin receptors, histamine receptors, and adrenergic receptors. This drug also blocks the binding of a wide range of drugs such as amphetamine, phencyclidine, cocaine, and morphine. 5,7-Dichlorobenzo[d]thiazol-2-amine has been shown to inhibit the binding of these drugs due to its ability to act as an antagonist by blocking the receptor site.

<p>Versatile small molecule scaffold</p>

<p>Versatile small molecule scaffold</p>

3-Quinolinecarboxylic acid, 1,2-dihydro-1-(1-methylethyl)-2-oxo-, hydrochloride (3QCA) is a compound that belongs to the class of amides. It has been shown to have a 5HT4 receptor agonist activity in vitro and in vivo experiments. 3QCA is used for the treatment of chronic constipation, as it stimulates bowel motility by increasing the peristaltic reflex. It also has an analgesic effect on the bowel, which may be due to its ability to inhibit pain transmission in the spinal cord. 3QCA has been shown to be effective in treating patients with bowel syndrome by increasing the volume of stool and reducing abdominal pain.

<p>Versatile small molecule scaffold</p>

<p>Versatile small molecule scaffold</p>

Versatile small molecule scaffold

<p>Methyl 4-methanesulfonyl-2-nitrobenzoate is a crystalline compound that belongs to the class of organic compounds. It is a white solid that is soluble in methanol and chloroform. The crystal structure of methyl 4-methanesulfonyl-2-nitrobenzoate has been determined by X-ray diffraction. This compound has a dihedral angle of about 23 degrees, and the nitro group is stabilized by a chloride ion.</p>

Versatile small molecule scaffold

Versatile small molecule scaffold

Versatile small molecule scaffold

<p>Versatile small molecule scaffold</p>

Versatile small molecule scaffold

Versatile small molecule scaffold

<p>Versatile small molecule scaffold</p>

<p>Versatile small molecule scaffold</p>

Versatile small molecule scaffold

<p>Versatile small molecule scaffold</p>

Versatile small molecule scaffold

Versatile small molecule scaffold

<p>Versatile small molecule scaffold</p>

Rupatadine is a drug that has been shown to have antihistamine and anticholinergic properties. It is used for the treatment of allergic rhinitis, chronic idiopathic urticaria, and pruritus. Rupatadine has also been investigated for its potential use in the treatment of solid tumours. Rupatadine belongs to a class of drugs called histamine H1 receptor antagonists. In experimental models, it has been shown to inhibit the growth of certain types of cancer cells by blocking the activity of histamine receptors on cell membranes and inhibiting protein synthesis. The drug also inhibits cardiac potassium channels, which may lead to cardiac effects such as arrhythmias or heart block. Rupatadine fumarate is metabolized into rupatadine (RUP) by esterases and oxidized by cytochrome P450 enzymes or conjugated with glucuronic acid. This active form binds to proteins

Versatile small molecule scaffold

Versatile small molecule scaffold

Versatile small molecule scaffold

Versatile small molecule scaffold

Versatile small molecule scaffold

Versatile small molecule scaffold

Versatile small molecule scaffold

Versatile small molecule scaffold

Versatile small molecule scaffold

Versatile small molecule scaffold

Versatile small molecule scaffold

Versatile small molecule scaffold

Versatile small molecule scaffold

Versatile small molecule scaffold

<p>Versatile small molecule scaffold</p>

Versatile small molecule scaffold

Versatile small molecule scaffold

<p>Versatile small molecule scaffold</p>

Versatile small molecule scaffold

Versatile small molecule scaffold

Ethynylcycloheptane is a cyclic ether that contains a ring of seven carbon atoms. It has two isomers: the homologous isomer and the positional isomer. The homologous isomer has the same number of hydrogen atoms on each carbon atom, while the positional isomer has different numbers of hydrogen atoms on some of its carbons. The odorant property of this chemical makes it useful as an additive in perfumes.