Protacs and Impurities
RSS0680
CAS:2769753-48-0
RSS0680 is a protein kinase degrader that degrades a variety of kinases and can be …
Formula:
C52H64N10O6S3
Purity:
98.02%
Color and Shape:
Solid
Molecular weight:
1021.32
Ref: TM-T74643
| 1mg | 370.00 € |
Estimated delivery in United States, on Tuesday 3 Dec 2024
PROTAC EED degrader-1
PROTAC EED degrader-1 is a PROTAC targeting EED (pKD = 9.02), is a inhibitor of …
Formula:
C55H60FN11O8S
Purity:
98%
Color and Shape:
Solid
Molecular weight:
1054.2
Ref: TM-T12553
| 100mg | To inquire | ||
| 500mg | To inquire |
Estimated delivery in United States, on Tuesday 3 Dec 2024
SIAIS178
CAS:2376047-73-1
SIAIS178 is a potent and selective degrader of BCR-ABL based on PROTAC technology (IC50 of …
Formula:
C50H62ClN11O6S2
Purity:
98%
Color and Shape:
Solid
Molecular weight:
1012.68
Ref: TM-T12907
| 1mg | 163.00 € | ||
| 5mg | 375.00 € | ||
| 10mg | 509.00 € | ||
| 50mg | 1,520.00 € | ||
| 100mg | 2,152.00 € | ||
| 200mg | To inquire | ||
| 500mg | To inquire | ||
| 1mL*10mM (DMSO) | 414.00 € |
Estimated delivery in United States, on Tuesday 3 Dec 2024
TL13-12
CAS:2229037-04-9
TL13-12 is a selective degrader of ALK-PROTAC and inhibits ALK activity (IC50: 0.69 nM).
Formula:
C45H53ClN10O10S
Purity:
98%
Color and Shape:
Solid
Molecular weight:
961.49
Ref: TM-T13930
| 5mg | 1,015.00 € |
Estimated delivery in United States, on Tuesday 3 Dec 2024
PROTAC EED degrader-2
PROTAC EED degrader-2 is a PROTAC targeting EED (pKD of 9.27),is a inhibitor of polycomb …
Formula:
C50H58FN11O6S
Purity:
98%
Color and Shape:
Solid
Molecular weight:
960.13
Ref: TM-T12554
| 100mg | To inquire | ||
| 500mg | To inquire |
Estimated delivery in United States, on Tuesday 3 Dec 2024
PROTAC BET degrader-2
CAS:2093388-33-9
PROTAC BET degrader-2 is a highly potent degrader of Bromodomain and Extra-Terminal (BET) proteins (IC50 …
Formula:
C41H42N10O6
Purity:
98%
Color and Shape:
Solid
Molecular weight:
770.84
Ref: TM-T12559
| 5mg | 376.00 € | ||
| 10mg | 596.00 € | ||
| 25mg | 1,104.00 € | ||
| 50mg | To inquire | ||
| 100mg | To inquire | ||
| 1mL*10mM (DMSO) | 602.00 € |
Estimated delivery in United States, on Tuesday 3 Dec 2024
ARCC-4
CAS:1973403-00-7
ARCC-4: A VHL-recruiting, low-nanomolar (DC50=5nM) AR degrader; outshines enzalutamide; degrades AR mutants resistant to therapy.
Formula:
C53H56F3N7O7S2
Purity:
98%
Color and Shape:
Solid
Molecular weight:
1024.18
Ref: TM-T14318
| 5mg | 1,025.00 € |
Estimated delivery in United States, on Tuesday 3 Dec 2024
dFKBP-1
CAS:1799711-22-0
dFKBP-1 is a potent and PROTAC-based FKBP12 degrader. dFKBP-1 incorporates the ligand SLF of FKBP12, …
Formula:
C53H64N6O14
Purity:
98%
Color and Shape:
Solid
Molecular weight:
1009.11
Ref: TM-T18597
| 100mg | To inquire | ||
| 500mg | To inquire |
Estimated delivery in United States, on Tuesday 3 Dec 2024
PROTAC ER Degrader-4
CAS:2361114-15-8
PROTAC ER Degrader-4 is a PROATC degrader of estrogen receptor (ER)(IC50 of 0.8 nM).
Formula:
C53H67F3N6O8S
Purity:
98%
Color and Shape:
Solid
Molecular weight:
1005.2
Ref: TM-T13839
| 100mg | To inquire | ||
| 500mg | To inquire |
Estimated delivery in United States, on Tuesday 3 Dec 2024
BETd-246
CAS:2140289-17-2
BETd-246 is an inhibitor of second-generation and PROTAC-based BET bromodomain (BRD), show antitumor activity.
Formula:
C48H55N11O10
Purity:
98%
Color and Shape:
Solid
Molecular weight:
946.02
Ref: TM-T14549
| 5mg | 509.00 € | ||
| 10mg | 745.00 € | ||
| 25mg | 1,520.00 € | ||
| 50mg | 2,303.00 € | ||
| 100mg | To inquire | ||
| 200mg | To inquire |
Estimated delivery in United States, on Tuesday 3 Dec 2024
PROTAC CRBN Degrader-1
CAS:2358775-70-7
PROTAC CRBN Degrader-1: a compound with CRBN and VHL binding groups linked, serving as a …
Formula:
C53H72N8O13S
Purity:
98%
Color and Shape:
Solid
Molecular weight:
1061.25
Ref: TM-T18604
| 5mg | 936.00 € |
Estimated delivery in United States, on Tuesday 3 Dec 2024
PROTAC FLT-3 degrader 1
CAS:2230826-81-8
PROTAC FLT-3 degrader 1 is a PROTAC FLT-3 degrader of internal tandem duplication (ITD)(IC50 0.6 …
Formula:
C52H61N9O9S2
Purity:
98%
Color and Shape:
Solid
Molecular weight:
1020.23
Ref: TM-T12555
| 100mg | To inquire | ||
| 500mg | To inquire |
Estimated delivery in United States, on Tuesday 3 Dec 2024
PROTAC MDM2 Degrader-2
CAS:2249944-99-6
PROTAC MDM2 Degrader-2: A potent MDM2-targeting compound with PROTAC tech for E3 ligase-mediated degradation.
Formula:
C70H76Cl4N10O12
Purity:
98%
Color and Shape:
Solid
Molecular weight:
1391.22
Ref: TM-T18632
| 100mg | To inquire | ||
| 500mg | To inquire |
Estimated delivery in United States, on Tuesday 3 Dec 2024
PROTAC IRAK4 degrader-1
CAS:2360533-90-8
PROTAC IRAK4 degrader-1 is a degrader of PROTAC interleukin-1 receptor-associated kinase 4 (IRAK4).
Formula:
C44H39F3N12O7
Purity:
98%
Color and Shape:
Solid
Molecular weight:
904.85
Ref: TM-T13842
| 100mg | To inquire | ||
| 500mg | To inquire |
Estimated delivery in United States, on Tuesday 3 Dec 2024
ARD-266
ARD-266: Potent VHL-based AR degrader; degrades AR in prostate cancer cells with DC50s of 0.2-1 …
Formula:
C52H59ClN6O7
Purity:
98%
Color and Shape:
Solid
Molecular weight:
915.51
Ref: TM-T13552
| 100mg | To inquire | ||
| 500mg | To inquire |
Estimated delivery in United States, on Tuesday 3 Dec 2024
PROTAC ERα Degrader-1
PROTAC ERα Degrader-1 is a chemical compound.
Formula:
C66H69N7O10
Purity:
98%
Color and Shape:
Solid
Molecular weight:
1120.29
Ref: TM-T18636
| 100mg | To inquire | ||
| 500mg | To inquire |
Estimated delivery in United States, on Tuesday 3 Dec 2024
PROTAC RIPK degrader-2
CAS:1801547-16-9
PROTAC RIPK degrader-2 is a nonpeptidic PROTAC ,and potently targets serine-threonine kinase RIPK2 and has …
Formula:
C52H65N7O11S3
Purity:
98%
Color and Shape:
Solid
Molecular weight:
1060.31
Ref: TM-T13846
| 100mg | To inquire | ||
| 500mg | To inquire |
Estimated delivery in United States, on Tuesday 3 Dec 2024
iRucaparib-AP6
CAS:2410557-00-3
iRucaparib-AP6: a specific, non-trapping PARP1 degrader; inhibits the enzyme's activity and scaffolding.
Formula:
C46H55FN6O11
Purity:
98%
Color and Shape:
Solid
Molecular weight:
886.96
Ref: TM-T13737
| 1mg | 431.00 € | ||
| 5mg | 1,284.00 € | ||
| 10mg | 2,227.00 € | ||
| 50mg | To inquire | ||
| 100mg | To inquire |
Estimated delivery in United States, on Tuesday 3 Dec 2024
PROTAC FAK degrader 1
CAS:2301916-69-6
PROTAC FAK degrader 1 is a selective and potent degrader of focal adhesion kinase (Fak) …
Formula:
C47H56F3N9O8S2
Purity:
98%
Color and Shape:
Solid
Molecular weight:
996.13
Ref: TM-T13840
| 1mg | 431.00 € | ||
| 5mg | 768.00 € | ||
| 10mg | 1,171.00 € | ||
| 50mg | To inquire | ||
| 100mg | To inquire |
Estimated delivery in United States, on Tuesday 3 Dec 2024
TL13-112
CAS:2229037-19-6
TL13-112 is a selective degrader of ALK-PROTAC and inhibits ALK activity (IC50: 0.14 nM).
Formula:
C49H60ClN9O10S
Purity:
98%
Color and Shape:
Solid
Molecular weight:
1002.57
Ref: TM-T13929
| 5mg | 1,025.00 € |
Estimated delivery in United States, on Tuesday 3 Dec 2024
