Protacs and Impurities
Tri-GalNAc-DBCO
Tri-GalNAc-DBCO, a compound with high affinity for the hepatocyte-specific asialoglycoprotein receptor (ASGPR), can bind to …
Formula:
C82H127N11O29
Purity:
99.92% - 99.92%
Color and Shape:
Liquid
Molecular weight:
1730.94
Ref: TM-T77948
1mg | 465.00 € |
Estimated delivery in United States, on Tuesday 3 Dec 2024
Folate-MS432
CAS:2769735-56-8
Folate-MS432 is a PROTAC that degrades MEKs selectively in cancer cells via folate receptor-dependent pathways.
Formula:
C77H94F3IN18O12S
Purity:
98%
Color and Shape:
Liquid
Molecular weight:
1679.65
Ref: TM-T82378
5mg | To inquire | ||
50mg | To inquire |
Estimated delivery in United States, on Tuesday 3 Dec 2024
PROTAC TTK degrader-1
CAS:2953426-43-0
PROTAC TTK degrader-1, a potent threonine tyrosine kinase (TTK) PROTAC degrader, demonstrates DC50 values of …
Formula:
C47H53N9O7
Purity:
98%
Color and Shape:
Liquid
Molecular weight:
855.98
Ref: TM-T81375
5mg | To inquire | ||
50mg | To inquire |
Estimated delivery in United States, on Tuesday 3 Dec 2024
PZ703b TFA
PZ703b TFA, a Bcl-xl PROTAC degradation agent, promotes apoptosis and halts bladder cancer cell proliferation, …
Formula:
C82H103ClF6N10O13S4
Purity:
98%
Color and Shape:
Liquid
Molecular weight:
1714.46
Ref: TM-T77913
5mg | To inquire | ||
50mg | To inquire |
Estimated delivery in United States, on Tuesday 3 Dec 2024
PROTAC Her3 Degrader-8
CAS:2103331-95-7
PROTAC Her3 Degrader-8 (Compound PP2) is a proteolysis targeting chimera (PROTAC) capable of degrading the …
Formula:
C49H55N11O6S
Purity:
98%
Color and Shape:
Liquid
Molecular weight:
926.1
Ref: TM-T77976
5mg | To inquire | ||
50mg | To inquire |
Estimated delivery in United States, on Tuesday 3 Dec 2024
Pomalidomid-C6-PEG3-butyl-N3
CAS:2300178-66-7
Pomalidomid-C6-PEG3-butyl-N3 is a click chemistry reagent featuring an azide group and serves as a crosslinker-E3 …
Formula:
C29H40N6O8
Purity:
98%
Color and Shape:
Liquid
Molecular weight:
600.66
Ref: TM-T81422
5mg | To inquire | ||
50mg | To inquire |
Estimated delivery in United States, on Tuesday 3 Dec 2024
Dovitinib-RIBOTAC
CAS:2759351-68-1
Dovitinib RIBOTAC is a potent, selective targeted RNA degrader that cleaves pre-miR-21.
Formula:
C51H56FN9O10S
Purity:
98%
Color and Shape:
Liquid
Molecular weight:
1006.11
Ref: TM-T77929
5mg | To inquire | ||
50mg | To inquire |
Estimated delivery in United States, on Tuesday 3 Dec 2024
SIAIS164018 hydrochloride
SIAIS164018 hydrochloride is a PROTAC-based degrader targeting ALK and EGFR, exhibiting IC50 values of 2.5 …
Formula:
C43H49Cl2N10O7P
Purity:
98%
Color and Shape:
Liquid
Molecular weight:
919.79
Ref: TM-T77942
5mg | To inquire | ||
50mg | To inquire |
Estimated delivery in United States, on Tuesday 3 Dec 2024
PROTAC SOS1 degrader-4
PROTAC SOS1 Degrader-4 (compound 10) is a potent degrader of SOS1 and exhibits antiproliferative activity …
Formula:
C53H65ClN8O7S
Purity:
98%
Color and Shape:
Liquid
Molecular weight:
993.65
Ref: TM-T79098
5mg | To inquire | ||
50mg | To inquire |
Estimated delivery in United States, on Tuesday 3 Dec 2024
SA-VA
SA-VA, an intracellular self-assembled PROTAC featuring azide and alkyne groups, selectively degrades VEGFR-2 and EphB4 …
Formula:
C50H53ClF3N11O7S
Purity:
98%
Color and Shape:
Liquid
Molecular weight:
1044.54
Ref: TM-T79531
5mg | To inquire | ||
50mg | To inquire |
Estimated delivery in United States, on Tuesday 3 Dec 2024
PROTAC BRD9 Degrader-3
CAS:2633632-05-8
PROTAC BRD9 Degrader-3 is a bifunctional degrader targeting BRD9, utilized in cancer research.
Formula:
C41H47ClN6O6
Purity:
98%
Color and Shape:
Liquid
Molecular weight:
755.3
Ref: TM-T81384
5mg | To inquire | ||
50mg | To inquire |
Estimated delivery in United States, on Tuesday 3 Dec 2024
PROTAC TTK degrader-2
CAS:2953426-48-5
PROTAC TTK Degrader-2 is a potent threonine tyrosine kinase (TTK) PROTAC degrader, achieving DC50 values …
Formula:
C49H57N9O7
Purity:
98%
Color and Shape:
Liquid
Molecular weight:
884.03
Ref: TM-T81374
5mg | To inquire | ||
50mg | To inquire |
Estimated delivery in United States, on Tuesday 3 Dec 2024
PROTAC KRAS G12C degrader-1
PROTAC KRAS G12C degrader-1, a cereblon-based degrader, promotes CRBN/KRAS G12C dimerization and facilitates the degradation …
Formula:
C50H54ClFN8O6
Purity:
98%
Color and Shape:
Liquid
Molecular weight:
917.47
Ref: TM-T77926
5mg | To inquire | ||
50mg | To inquire |
Estimated delivery in United States, on Tuesday 3 Dec 2024
PROTAC NSD3 degrader-1
PROTAC NSD3 degrader-1 (compound 56) is a targeted degradation agent for the Nuclear receptor binding …
Purity:
98%
Ref: TM-T81377
5mg | To inquire | ||
50mg | To inquire |
Estimated delivery in United States, on Tuesday 3 Dec 2024
PROTAC α-synuclein degrader 5
CAS:2781922-42-5
PROTAC α-synuclein degrader 5 is a highly selective (PROTAC) compound that targets and degrades α-synuclein …
Formula:
C39H41N7O10
Purity:
98%
Color and Shape:
Liquid
Molecular weight:
767.78
Ref: TM-T79250
5mg | 936.00 € |
Estimated delivery in United States, on Tuesday 3 Dec 2024
HDAC6 degrader-1
CAS:2439058-23-6
HDAC6 degrader-1, a proteolysis-targeting chimeric molecule (PROTAC), incorporates the selective HDAC6 inhibitor Nexturastat A (Nex …
Formula:
C40H45N9O9
Purity:
98%
Color and Shape:
Liquid
Molecular weight:
795.84
Ref: TM-T77922
5mg | To inquire | ||
50mg | To inquire |
Estimated delivery in United States, on Tuesday 3 Dec 2024
SA-PA
SA-PA, a self-assembled intracellular PROTAC leveraging azide-alkyne click chemistry, selectively degrades VEGFR-2, PDGFR-β, and EphB4 …
Formula:
C40H32ClF3N10O8
Purity:
98%
Color and Shape:
Liquid
Molecular weight:
873.19
Ref: TM-T79530
5mg | To inquire | ||
50mg | To inquire |
Estimated delivery in United States, on Tuesday 3 Dec 2024
GBD-9
CAS:2864408-92-2
GBD-9, a dual-mechanism degrader, effectively promotes the degradation of BTK and GSPT1 through recruitment of …
Formula:
C44H47N9O6
Purity:
98%
Color and Shape:
Liquid
Molecular weight:
797.9
Ref: TM-T79139
5mg | To inquire | ||
50mg | To inquire |
Estimated delivery in United States, on Tuesday 3 Dec 2024
PPM-3
PPM-3, a selective PROTAC ERK5 degrader, exhibits a potent inhibitory concentration (IC 50) of 62.4 …
Formula:
C54H69N11O6S
Purity:
98%
Color and Shape:
Liquid
Molecular weight:
1000.26
Ref: TM-T78901
5mg | To inquire | ||
50mg | To inquire |
Estimated delivery in United States, on Tuesday 3 Dec 2024
CFT-2718
CFT-2718 is an advanced BRD4-targeting PROTAC (proteolysis-targeting chimera) known for its improved catalytic efficiency and …
Purity:
98%
Ref: TM-T82742
5mg | To inquire | ||
50mg | To inquire |
Estimated delivery in United States, on Tuesday 3 Dec 2024