G-protein Coupled Receptors and 7-TM Receptors

G-protein coupled receptors (GPCRs) and 7-transmembrane (7-TM) receptors are a large family of membrane proteins that play key roles in cellular communication and signal transduction. These receptors are involved in a wide range of physiological processes, including sensory perception, immune response, and hormone regulation. GPCRs are major targets in drug discovery, making them essential for research in pharmacology and medicine. At CymitQuimica, we offer a comprehensive selection of high-quality reagents and compounds related to GPCRs and 7-TM receptors to support your research and drug development efforts.

Found 5800 products of "G-protein Coupled Receptors and 7-TM Receptors"

Purity (%)

100

products per page.

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RF9 acetate
RF9 acetate is an effective and selective antagonist of Neuropeptide FF receptor with Ki values of 58 and 75 nM for hNPFF1R and hNPFF2R, respectively.
Formula:C₂₈H₄₂N₆O₅
Purity:99.77%
Color and Shape:Solid
Molecular weight:542.67
Ref: TM-T16738L
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Kisspeptin-10, human
CAS:
- 374675-21-5
Kisspeptin-10, human is an effective vasoconstrictor and inhibitor of angiogenesis.
Formula:C₆₃H₈₃N₁₇O₁₄
Purity:98%
Color and Shape:Solid
Molecular weight:1302.462
Ref: TM-TP1396
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GB-110 hydrochloride
GB-110 HCl: potent, nonpeptidic oral PAR2 agonist; triggers Ca2+ release in HT29 cells; EC50 0.28 μM.
Formula:C₃₃H₄₉ClN₆O₅
Color and Shape:Solid
Molecular weight:645.23
Ref: TM-T73854
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Setmelanotide Acetate(920014-72-8 free base)
CAS:
- 2759937-80-7
Setmelanotide Acetate(920014-72-8 free base) (RM-493 Acetate) is a selective agonist of melanocortin 4 receptor (MC4R)(human and rat MC4R with EC50s of 0.27 nM
Formula:C₅₁H₇₂N₁₈O₁₁S₂
Purity:99.71%
Color and Shape:Solid
Molecular weight:1177.35
Ref: TM-T12882L
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4-Chloromethamphetamine hydrochloride
CAS:
- 30572-91-9
4-Chloromethamphetamine hydrochloride is a novel psychoactive substance belonging to the amphetamine class.
Formula:C₁₀H₁₅Cl₂N
Color and Shape:Solid
Molecular weight:220.14
Ref: TM-T203542
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TRPV1/CB2 agonist 1
TRPV1/CB2 agonist 1 (compound 41) is a dual agonist targeting hTRPV1 and CB2 receptors, with an EC50 value of 26.8 μM for hTRPV1. It is applicable in research related to the nervous system.
Color and Shape:Odour Solid
Ref: TM-T200749
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Apelin-17(human, bovine)
CAS:
- 217082-57-0
Endogenous apelin receptor agonist. Potently inhibits forskolin-stimulated cAMP accumulation (pIC50 = 9.94).
Formula:C₉₆H₁₅₆N₃₄O₂₀S
Purity:98%
Color and Shape:Solid
Molecular weight:2138.56
Ref: TM-TP2092
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4-Butyl-α-agarofuran
CAS:
- 272126-07-5
4-Butyl-alpha-agarofuran, a Gharu-wood derivative, is an anxiolytic, antidepressant, and aids neurological research.
Formula:C₁₈H₃₀O
Color and Shape:Solid
Molecular weight:262.43
Ref: TM-T75257
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[Pro34]Neuropeptide Y, porcine
CAS:
- 128768-54-7
[Pro34]Neuropeptide Y, porcine functions as a selective agonist for the NPY (Y1) receptor and induces vasoconstriction in the guinea pig's caval vein [1].
Formula:C₁₉₀H₂₈₆N₅₄O₅₆
Color and Shape:Solid
Molecular weight:4222.63
Ref: TM-TP2523
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PEN (human)
CAS:
- 597578-70-6
PEN (human) is an Endogenous peptide GPR83 agonist. ProSAAS-derived neuropeptide.
Formula:C₉₇H₁₅₉N₂₇O₃₂
Purity:98%
Color and Shape:Solid
Molecular weight:2215.49
Ref: TM-TP1949
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Etelcalcetide
CAS:
- 1262780-97-1
Etelcalcetide (AMG 416), a synthetic peptide CaSR activator, treats secondary hyperparathyroidism in hemodialysis patients.
Formula:C₃₈H₇₃N₂₁O₁₀S₂
Purity:98%
Color and Shape:Solid
Molecular weight:1048.26
Ref: TM-TP1235
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Succinate/succinate receptor antagonist 1
CAS:
- 2361972-29-2
Potent succinate receptor antagonist with IC50 of 20 μM; blocks gingival succinate signaling, may treat periodontal disease.
Formula:C₁₇H₁₅N₃O
Purity:99.53%
Color and Shape:Soild
Molecular weight:277.32
Ref: TM-T67915
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Cagrilintide
CAS:
- 1415456-99-3
Cagrilintide: a long-acting amylin analogue, potential obesity treatment, reduces appetite and weight.
Formula:C₁₉₄H₃₁₂N₅₄O₅₉S₂
Color and Shape:Solid
Molecular weight:4409.01
Ref: TM-T76262
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Prostaglandin F2α 1,11-lactone
CAS:
- 62410-84-8
Prostaglandin F2α 1,11-lactone (PGF2α 1,11-lactone) is a lipid-soluble prodrug of Prostaglandin F2α and can be used in studies about treating glaucoma.
Formula:C₂₀H₃₂O₄
Purity:98%
Color and Shape:Solid
Molecular weight:336.47
Ref: TM-T37326
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BMS-604992 dihydrochloride
CAS:
- 1469750-46-6
BMS-604992 dihydrochloride is a selective GHSR agonist with high affinity (Ki=2.3 nM) and potent activity (EC50=0.4 nM), stimulating rodent appetite.
Formula:C₂₄H₃₃Cl₂N₇O₅
Color and Shape:Solid
Molecular weight:570.47
Ref: TM-T38959
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(D-Ser4,D-Ser(tBu)6,Azagly10)-LHRH
CAS:
- 1926163-39-4
Analog of LHRH, stimulates LH and FSH release, controls reproduction.
Formula:C₅₉H₈₄N₁₈O₁₄
Color and Shape:Solid
Molecular weight:1269.41
Ref: TM-T76616
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Bombinakinin M
CAS:
- 509151-65-9
Potent, selective bradykinin receptor agonist 50x stronger than bradykinin, contracts guinea pig ileum muscle at EC50 4.0 nM.
Formula:C₁₀₀H₁₅₉N₃₁O₂₄
Purity:98%
Color and Shape:Solid
Molecular weight:2179.55
Ref: TM-TP2075
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NI-203
NI-203 is a monoclonal antibody inhibitor that targets amylin and shows potential for research in type 2 diabetes.
Color and Shape:Odour Liquid
Ref: TM-T9901A-993
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BMS-753426
CAS:
- 1004536-52-0
BMS-753426 is a potent and orally bioavailable antagonist of CCR2 .
Formula:C₂₅H₃₃F₃N₆O₂
Color and Shape:Solid
Molecular weight:506.574
Ref: TM-T38397
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CYN 154806
CAS:
- 183658-72-2
CYN 154806: potent sst2 antagonist; pIC50: 8.58 (sst2), 5.41 (sst1), 6.07 (sst3), 5.76 (sst4), 6.48 (sst5).
Formula:C₅₆H₆₈N₁₂O₁₄S₂
Purity:98%
Color and Shape:Solid
Molecular weight:1197.34
Ref: TM-TP1877