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G-protein Coupled Receptors and 7-TM Receptors

G-protein Coupled Receptors and 7-TM Receptors

G-protein coupled receptors (GPCRs) and 7-transmembrane (7-TM) receptors are a large family of membrane proteins that play key roles in cellular communication and signal transduction. These receptors are involved in a wide range of physiological processes, including sensory perception, immune response, and hormone regulation. GPCRs are major targets in drug discovery, making them essential for research in pharmacology and medicine. At CymitQuimica, we offer a comprehensive selection of high-quality reagents and compounds related to GPCRs and 7-TM receptors to support your research and drug development efforts.

Found 5800 products of "G-protein Coupled Receptors and 7-TM Receptors"

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    Secretin (28-54), human TFA

    <p>Secretin (28-54), human TFA is a 27-amino acid peptide that works on the human Secretin receptor.</p>
    Formula:C132H221N44F3O42
    Purity:98%
    Color and Shape:Solid
    Molecular weight:3153.48

    Ref: TM-TP1135

  • 20-Carboxy-Leukotriene B4
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    20-Carboxy-Leukotriene B4

    CAS:
    <p>20-COOH LTB4, a metabolite of LTB4, binds BLT1 receptor and inhibits LTB4-induced neutrophil responses.</p>
    Formula:C20H30O6
    Color and Shape:Solid
    Molecular weight:366.45

    Ref: TM-T73793

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    U-46619 serinol amide

    U-46619 serinol amide is a derivative of U-46619, acting as a stable analog of Thromboxane A2 (TXA2). It effectively functions as a TXA2 agonist, capable of inducing platelet shape change and aggregation.
    Formula:C24H41NO5
    Color and Shape:Solid
    Molecular weight:423.29847

    Ref: TM-T207554

  • 11-deoxy Prostaglandin E1
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    11-deoxy Prostaglandin E1

    CAS:
    <p>11-deoxy Prostaglandin E1 is a prostaglandin E1 analogue that has bronchodilator activity and can inhibit histamine-induced bronchoconstriction and cause</p>
    Formula:C20H34O4
    Color and Shape:Solid
    Molecular weight:338.48

    Ref: TM-T36770

  • Mabuterol free base
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    Mabuterol free base

    CAS:
    Mabuterol: selective β2 agonist, inhibits isoprenaline, affects rat uterus and rabbit jejunum, alters intestinal propulsion.
    Formula:C13H18ClF3N2O
    Purity:98%
    Color and Shape:Solid
    Molecular weight:310.74

    Ref: TM-T27970

  • Luseogliflozin
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    Luseogliflozin

    CAS:
    Luseogliflozin inhibits SGLT2 for glucose uptake with 1.10 nM potency.
    Formula:C23H30O6S
    Color and Shape:Solid
    Molecular weight:434.55

    Ref: TM-T21399

  • Lys-[Des-Arg9]Bradykinin TFA
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    Lys-[Des-Arg9]Bradykinin TFA

    CAS:
    <p>Lys-[Des-Arg9]Bradykinin TFA: natural kinin, selective B1 agonist; Ki: 0.12 nM (human), 1.7 nM (mouse), 0.23 nM (rabbit); weak on B2 receptors.</p>
    Formula:C54H75F6N13O15
    Color and Shape:Solid
    Molecular weight:1260.24

    Ref: TM-T73646

  • VU0453379
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    VU0453379

    CAS:
    VU0453379 is a highly selective and central nervous system penetrant positive allosteric modulator of glucagon-like peptide-1R (EC50: 1.3 μM).
    Formula:C26H34N4O2
    Purity:98%
    Color and Shape:Solid
    Molecular weight:434.57

    Ref: TM-T17242

  • HS014
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    HS014

    CAS:
    Potent MC4 antagonist; Ki: 3.16 nM (MC4), 108 (MC1), 54.4 (MC3), 694 (MC5). Boosts rat appetite, mouse pain, blocks IL-1β Fos in hypothalamus.
    Formula:C71H94N20O17S2
    Purity:98%
    Color and Shape:Solid
    Molecular weight:1563.77

    Ref: TM-TP2015

  • HL2-m5
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    HL2-m5

    CAS:
    HL2-m5 is an inhibitor of the sonic hedgehog/patched (Shh/PTCH1) interaction, with a Kd for Shh of 170 nM. It effectively inhibits the activation of the Hedgehog signaling pathway and the transcription of Gli-controlled genes, with an IC50 of 230 nM.
    Formula:C70H101N15O24S3
    Color and Shape:Solid
    Molecular weight:1632.83

    Ref: TM-TP3102

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    D5R agonist 1

    D5R Agonist 1 (Compound 5j) is a selective, orally active partial agonist of the D5 receptor that can penetrate the blood-brain barrier (EC50: 269.7 nM). It has been demonstrated to enhance cognitive abilities in a scopolamine-induced amnesia model.
    Color and Shape:Odour Solid

    Ref: TM-T200501

  • HHS-0701
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    HHS-0701

    CAS:
    HHS-0701: SuTEx ligand, strong PTGR2 inhibitor, blocks 15-Keto-PGE2 metabolism.
    Formula:C20H20N4O3S
    Purity:97.24%
    Color and Shape:Soild
    Molecular weight:396.46

    Ref: TM-T67766

  • Somatostatin 1-28 acetate
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    Somatostatin 1-28 acetate

    Somatostatin 1-28 acetate circulates in human plasma.
    Purity:99.22%
    Color and Shape:Soild

    Ref: TM-TP2124L

  • Succinate/succinate receptor antagonist 1
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    Succinate/succinate receptor antagonist 1

    CAS:
    <p>Potent succinate receptor antagonist with IC50 of 20 μM; blocks gingival succinate signaling, may treat periodontal disease.</p>
    Formula:C17H15N3O
    Purity:99.53%
    Color and Shape:Soild
    Molecular weight:277.32

    Ref: TM-T67915

  • Imipramine N-oxide
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    Imipramine N-oxide

    CAS:
    Imipramine N-oxide is a tricyclic antidepressant (TCA) and imipramine analogue used to treat depression.
    Formula:C19H24N2O
    Purity:99.80%
    Color and Shape:Solid
    Molecular weight:296.41

    Ref: TM-T74205

  • Apraglutide
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    Apraglutide

    CAS:
    Apraglutide (FE 203799 is a synthetic 33-amino acid peptide and long-acting glp-2 analogue.
    Formula:C172H263N43O52
    Purity:98%
    Color and Shape:Solid
    Molecular weight:3765.25

    Ref: TM-TP1172

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    JKC363 TFA

    JKC363 TFA is an MC4 receptor antagonist with 90x more affinity than MC3 (IC50: 0.5 nM vs 44.9 nM), blocks α-MSH's effect on TRH, and is anti-hyperalgesic.
    Formula:C71H93F3N19O18S2
    Color and Shape:Solid
    Molecular weight:1620.73

    Ref: TM-T75850

  • N-0500 HCl
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    N-0500 HCl

    CAS:
    <p>N-0500 HCl, a potent DA receptor agonist, displaces [3H]DP_x005f_x0002_5,6-ADTN with an IC50 of 3nM.</p>
    Formula:C15H22ClNO2
    Purity:98.85% - 99.54%
    Color and Shape:Solid
    Molecular weight:283.79

    Ref: TM-T60107

  • Thrombin Receptor Activator for Peptide 5 (TRAP-5)
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    Thrombin Receptor Activator for Peptide 5 (TRAP-5)

    CAS:
    Thrombin Receptor Activator for Peptide 5 (TRAP-5) is also called Coagulation Factor II Receptor (1-5), used in the research of coronary heart disease (CHD).
    Formula:C30H50N8O7
    Purity:98%
    Color and Shape:Solid
    Molecular weight:634.77

    Ref: TM-T7496

  • Propranolol hydrochloride
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    Propranolol hydrochloride

    CAS:
    Propranolol hydrochloride is a widely used non-cardioselective beta-adrenergic antagonist. Propranolol has been used for MYOCARDIAL INFARCTION; ARRHYTHMIA; ANGINA PECTORIS; HYPERTENSION; HYPERTHYROIDISM; MIGRAINE; PHEOCHROMOCYTOMA; and ANXIETY but adverse
    Formula:C16H22ClNO2
    Purity:99.94% - >99.99%
    Color and Shape:White Or Almost White Powder White Powder
    Molecular weight:295.80

    Ref: TM-T0812