G-protein Coupled Receptors and 7-TM Receptors
G-protein coupled receptors (GPCRs) and 7-transmembrane (7-TM) receptors are a large family of membrane proteins that play key roles in cellular communication and signal transduction. These receptors are involved in a wide range of physiological processes, including sensory perception, immune response, and hormone regulation. GPCRs are major targets in drug discovery, making them essential for research in pharmacology and medicine. At CymitQuimica, we offer a comprehensive selection of high-quality reagents and compounds related to GPCRs and 7-TM receptors to support your research and drug development efforts.
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16,16-Dimethyl prostaglandin E2
CAS:39746-25-3
16,16-Dimethyl prostaglandin E2 regulates hematopoietic stem cells via EP2/EP4 and Wnt, taken orally.
Formula:
C22H36O5
Purity:
98%
Color and Shape:
Solid
Molecular weight:
380.52
Ref: TM-T10046
| 1mg | 205.00 € | ||
| 5mg | 949.00 € | ||
| 10mg | 1,786.00 € |
Estimated delivery in United States, on Monday 2 Jun 2025
AZD5462
CAS:2787501-83-9
AZD5462 is a potent orally available relaxin receptor RXFP1 agonist for the study of heart …
Formula:
C30H41FN2O6
Purity:
99.63%
Color and Shape:
Liquid
Molecular weight:
544.65
Ref: TM-T63838
| 1mg | 354.00 € | ||
| 5mg | 850.00 € | ||
| 10mg | 1,206.00 € | ||
| 25mg | 1,882.00 € | ||
| 50mg | 2,642.00 € | ||
| 100mg | 3,345.00 € |
Estimated delivery in United States, on Monday 2 Jun 2025
BMS-986141
CAS:1478711-48-6
BMS-986141(UDM-003183) is a selective and potent protease-activated receptor-4 (PAR-4) antagonist with oral activity and an …
Formula:
C27H23N5O5S2
Purity:
98.36% - 99.11%
Color and Shape:
Liquid
Molecular weight:
561.63
Ref: TM-T63966
| 1mg | 747.00 € | ||
| 5mg | 1,501.00 € | ||
| 10mg | 1,872.00 € | ||
| 25mg | 2,680.00 € | ||
| 50mg | 3,591.00 € | ||
| 100mg | 4,874.00 € |
Estimated delivery in United States, on Monday 2 Jun 2025
Orvepitant maleate
CAS:579475-24-4
Orvepitant maleate, a selective NK-1 receptor antagonist (pKi 10.2), may treat depression and CRC; crosses …
Formula:
C35H39F7N4O6
Purity:
98%
Color and Shape:
Solid
Molecular weight:
744.7
Ref: TM-T16406
| 25mg | 653.00 € | ||
| 50mg | 868.00 € | ||
| 100mg | 1,293.00 € |
Estimated delivery in United States, on Monday 2 Jun 2025
Taranabant
CAS:701977-09-5
Taranabant: potent CB1 receptor inverse agonist; inhibits agonists with 0.13 nM Ki in vitro.
Formula:
C27H25ClF3N3O2
Purity:
99.06% - 99.06%
Color and Shape:
Solid
Molecular weight:
515.96
Ref: TM-T13080L
| 1mg | 98.00 € |
Estimated delivery in United States, on Monday 2 Jun 2025
Vofopitant dihydrochloride
CAS:168266-51-1
Vofopitant dihydrochloride (GR 205171A) is a tachykinin NK1 receptor antagonist and a potential compound for …
Formula:
C21H25Cl2F3N6O
Purity:
98.99%
Color and Shape:
Solid
Molecular weight:
505.36
Ref: TM-T13329L
| 1mg | 99.00 € | ||
| 5mg | 235.00 € | ||
| 10mg | 376.00 € | ||
| 25mg | 712.00 € | ||
| 50mg | 1,064.00 € | ||
| 100mg | 1,454.00 € | ||
| 500mg | 2,822.00 € | ||
| 1mL*10mM (DMSO) | 261.00 € |
Estimated delivery in United States, on Monday 2 Jun 2025
(±)-Penbutolol
CAS:36507-48-9
(±)-Penbutolol ((Rac)-Penbutolol) is the racemic form of Penbutolol. It acts as an orally active β-adrenergic …
Formula:
C18H29NO2
Color and Shape:
Liquid
Molecular weight:
291.43
Ref: TM-T201472
| 10mg | To inquire | ||
| 50mg | To inquire |
Estimated delivery in United States, on Monday 2 Jun 2025
ASP-2205
CAS:1334440-09-3
ASP-2205, a 5-HT2C receptor agonist (human 5-HT2C receptor, EC50=0.85 nM; rat 5-HT2C receptor, EC50=2.5 nM), …
Formula:
C19H28N2O
Color and Shape:
Liquid
Molecular weight:
300.44
Ref: TM-T201450
| 10mg | To inquire | ||
| 50mg | To inquire |
Estimated delivery in United States, on Monday 2 Jun 2025
AB-FUBINACA 3-fluorobenzyl isomer
CAS:1185282-19-2
AB-FUBINACA 3-fluorobenzyl isomer is a synthetic cannabinoid and an indazole derivative, exhibiting high affinity for …
Formula:
C20H21FN4O2
Color and Shape:
Liquid
Molecular weight:
368.41
Ref: TM-T201486
| 10mg | To inquire | ||
| 50mg | To inquire |
Estimated delivery in United States, on Monday 2 Jun 2025
H3R-IN-1 Hydrochloride
CAS:2319790-07-1
H3R-IN-1 Hydrochloride is an inverse agonist of histamine receptor 3( H3R ) .
Formula:
C19H24ClN3O3
Purity:
98%
Color and Shape:
Solid
Molecular weight:
377.86
Ref: TM-T11531
| 25mg | 1,054.00 € | ||
| 50mg | 1,378.00 € | ||
| 100mg | 2,167.00 € |
Estimated delivery in United States, on Monday 2 Jun 2025
Isotodesnitazene
CAS:2732926-27-9
Isotodesnitazene is an opioid compound that primarily targets the μ-opioid receptor (MOR). It exhibits EC50 …
Formula:
C23H31N3O
Color and Shape:
Liquid
Molecular weight:
365.51
Ref: TM-T201840
| 10mg | To inquire | ||
| 50mg | To inquire |
Estimated delivery in United States, on Monday 2 Jun 2025
UNC10099984A
CAS:1354030-25-3
UNC10099984A (Compound 6) is a functionally selective ligand for the dopamine D2 receptor, exhibiting a …
Formula:
C24H29Cl2N3O2
Color and Shape:
Liquid
Molecular weight:
462.41
Ref: TM-T201623
| 10mg | To inquire | ||
| 50mg | To inquire |
Estimated delivery in United States, on Monday 2 Jun 2025
Elzasonan hydrochloride
CAS:220322-05-4
Elzasonan hydrochloride is a serotonin 1B and serotonin 1D receptor antagonist. It is utilized in …
Formula:
C22H24Cl3N3OS
Color and Shape:
Liquid
Molecular weight:
484.87
Ref: TM-T201763
| 10mg | To inquire | ||
| 50mg | To inquire |
Estimated delivery in United States, on Monday 2 Jun 2025
Aclidinium
CAS:727649-81-2
Aclidinium, a dual-action compound, serves as a long-acting muscarinic antagonist and a β2-adrenoceptor (β2-AR) agonist, …
Formula:
C26H30NO4S2
Color and Shape:
Liquid
Molecular weight:
484.65
Ref: TM-T200043
| 10mg | To inquire | ||
| 50mg | To inquire |
Estimated delivery in United States, on Monday 2 Jun 2025
YGZ-331
CAS:1350113-04-0
YGZ-331, a sedative hypnotic, acts by elevating GABA levels as a derivative of the adenosine …
Formula:
C19H23N5O4
Color and Shape:
Liquid
Molecular weight:
385.42
Ref: TM-T200016
| 10mg | To inquire | ||
| 50mg | To inquire |
Estimated delivery in United States, on Monday 2 Jun 2025
D1R antagonist 1
CAS:2983777-67-7
Compound 12a (D1R antagonist 1) is a D1R antagonist that participates in both G-protein-coupled and …
Formula:
C22H26BrNO4
Purity:
98%
Color and Shape:
Liquid
Molecular weight:
448.35
Ref: TM-T78735
| 1mg | 185.00 € | ||
| 5mg | 459.00 € | ||
| 10mg | 657.00 € | ||
| 25mg | 1,026.00 € | ||
| 50mg | 1,415.00 € | ||
| 100mg | 1,872.00 € |
Estimated delivery in United States, on Monday 2 Jun 2025
5-HT2A/5-HT2C inverse agonist 1
CAS:2718990-76-0
5-HT2A/5-HT2C inverse agonist 1 serves as a dual and potent inverse agonist for the 5-HT2A …
Formula:
C24H35N5O2
Color and Shape:
Liquid
Molecular weight:
425.57
Ref: TM-T200089
| 10mg | To inquire | ||
| 50mg | To inquire |
Estimated delivery in United States, on Monday 2 Jun 2025
(S)-Bucindolol
CAS:91548-61-7
(S)-Bucindolol is an enantiomer of bucindolol, specifically a β1-adrenergic receptor antagonist. It is primarily utilized …
Formula:
C22H25N3O2
Color and Shape:
Liquid
Molecular weight:
363.45
Ref: TM-T200285
| 10mg | To inquire | ||
| 50mg | To inquire |
Estimated delivery in United States, on Monday 2 Jun 2025
GLPG0974
CAS:1391076-61-1
GLPG0974 is an antagonist of FFA2/GPR43 with IC50 of 9 nM.
Formula:
C25H25ClN2O4S
Purity:
99.58%
Color and Shape:
Solid
Molecular weight:
484.99
Ref: TM-T15388
| 1mg | 56.00 € | ||
| 5mg | 119.00 € | ||
| 10mg | 187.00 € | ||
| 25mg | 376.00 € | ||
| 50mg | 560.00 € | ||
| 1mL*10mM (DMSO) | 126.00 € |
Estimated delivery in United States, on Monday 2 Jun 2025
TAAR1 agonist 2
CAS:1804128-38-8
TAAR1 agonist 2 (compound 30), a full agonist at trace amine-associated receptor 1 (TAAR1) (pEC50=7.5), …
Formula:
C9H11NO
Color and Shape:
Liquid
Molecular weight:
149.19
Ref: TM-T200140
| 10mg | To inquire | ||
| 50mg | To inquire |
Estimated delivery in United States, on Monday 2 Jun 2025
