G-protein Coupled Receptors and 7-TM Receptors
G-protein coupled receptors (GPCRs) and 7-transmembrane (7-TM) receptors are a large family of membrane proteins that play key roles in cellular communication and signal transduction. These receptors are involved in a wide range of physiological processes, including sensory perception, immune response, and hormone regulation. GPCRs are major targets in drug discovery, making them essential for research in pharmacology and medicine. At CymitQuimica, we offer a comprehensive selection of high-quality reagents and compounds related to GPCRs and 7-TM receptors to support your research and drug development efforts.
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U91356
CAS:152886-85-6
U91356 is an agonist of the dopamine receptors.
Formula:
C13H17N3O
Purity:
98%
Color and Shape:
Solid
Molecular weight:
231.29
Ref: TM-T13240
| 25mg | 2,157.00 € | ||
| 50mg | 2,832.00 € | ||
| 100mg | 3,800.00 € |
Estimated delivery in United States, on Friday 27 Jun 2025
SORT1-IN-5
CAS:3031580-91-0
SORT1-IN-5 (compound 3) is a SORT1 inhibitor capable of crossing the blood-brain barrier. The MSOH …
Formula:
C19H31NO6S
Color and Shape:
Liquid
Molecular weight:
401.52
Ref: TM-T201789
| 10mg | To inquire | ||
| 50mg | To inquire |
Estimated delivery in United States, on Friday 27 Jun 2025
Dinoxyline
CAS:757176-96-8
Dinoxyline is a potent dopamine receptor agonist, with dissociation constants (Ki values) for D1, D2, …
Formula:
C15H13NO3
Color and Shape:
Liquid
Molecular weight:
255.27
Ref: TM-T201856
| 10mg | To inquire | ||
| 50mg | To inquire |
Estimated delivery in United States, on Friday 27 Jun 2025
Butopamine hydrochloride
CAS:74432-68-1
Butopamine hydrochloride is an orally active inotropic compound that is more effective at increasing heart …
Formula:
C18H24ClNO3
Color and Shape:
Liquid
Molecular weight:
337.84
Ref: TM-T201508
| 10mg | To inquire | ||
| 50mg | To inquire |
Estimated delivery in United States, on Friday 27 Jun 2025
22-Thiocyanatosalvinorin A
CAS:1174223-49-4
22-Thiocyanatosalvinorin A (RB-64) is a potent selective agonist for the kappa-opioid receptor, exhibiting an EC50 …
Formula:
C24H27NO8S
Color and Shape:
Liquid
Molecular weight:
489.54
Ref: TM-T201845
| 10mg | To inquire | ||
| 50mg | To inquire |
Estimated delivery in United States, on Friday 27 Jun 2025
CCG258208
CAS:2055990-90-2
GRKs-IN-1 has remarkable potency against and selectivity for G protein-coupled receptor kinase 2 GRK2 (IC50: …
Formula:
C24H25FN4O4
Purity:
98%
Color and Shape:
Solid
Molecular weight:
452.48
Ref: TM-T13714
| 25mg | 2,300.00 € | ||
| 50mg | 3,022.00 € | ||
| 100mg | 4,085.00 € |
Estimated delivery in United States, on Friday 27 Jun 2025
Flucopride
CAS:1639925-34-0
Flucopride (Compound 4a) acts as an acetylcholinesterase inhibitor (AChE) with an IC50 value of 24 …
Formula:
C22H33FN2O2
Color and Shape:
Liquid
Molecular weight:
376.51
Ref: TM-T201815
| 10mg | To inquire | ||
| 50mg | To inquire |
Estimated delivery in United States, on Friday 27 Jun 2025
Anilopam
CAS:53716-46-4
Anilopam is an opioid analgesic belonging to the benzazepine class and acts as an agonist …
Formula:
C20H26N2O
Color and Shape:
Liquid
Molecular weight:
310.43
Ref: TM-T201609
| 10mg | To inquire | ||
| 50mg | To inquire |
Estimated delivery in United States, on Friday 27 Jun 2025
R-137696
CAS:695185-73-0
R-137696 is an orally active 5-HT1A receptor agonist that facilitates the relaxation of the proximal …
Formula:
C17H23N3O2
Color and Shape:
Liquid
Molecular weight:
301.38
Ref: TM-T201501
| 10mg | To inquire | ||
| 50mg | To inquire |
Estimated delivery in United States, on Friday 27 Jun 2025
Pexacerfont
CAS:459856-18-9
Pexacerfont (BMS-562086) is a selective antagonist of the corticotropin-releasing factor receptor (IC50: 6.1±0.6 nM for …
Formula:
C18H24N6O
Purity:
99.74%
Color and Shape:
Solid
Molecular weight:
340.42
Ref: TM-T16475
| 1mg | 48.00 € | ||
| 5mg | 87.00 € | ||
| 1mL*10mM (DMSO) | 97.00 € |
Estimated delivery in United States, on Friday 27 Jun 2025
SB-224289 hydrochloride
CAS:180084-26-8
SB-224289 hydrochloride (SB-224289A) is a selective antagonist of 5-HT1B receptor, with anxiolytic effect.
Formula:
C32H33ClN4O3
Purity:
97.82% - 98.09%
Color and Shape:
Solid
Molecular weight:
557.08
Ref: TM-T12841
| 5mg | 97.00 € | ||
| 10mg | 146.00 € | ||
| 25mg | To inquire | ||
| 50mg | To inquire | ||
| 1mL*10mM (DMSO) | 116.00 € |
Estimated delivery in United States, on Friday 27 Jun 2025
Rodatristat ethyl
CAS:1673571-51-1
Rodatristat ethyl is an oral TPH1 inhibitor reducing 5-HT levels & lowering PAH at low …
Formula:
C29H31ClF3N5O3
Purity:
98%
Color and Shape:
Solid
Molecular weight:
590.04
Ref: TM-T16779
| 25mg | 2,270.00 € | ||
| 50mg | 3,676.00 € | ||
| 100mg | 5,919.00 € |
Estimated delivery in United States, on Friday 27 Jun 2025
SCH 563705
CAS:473728-58-4
SCH 563705 is a CXCR2 and CXCR1 antagonist used in the study of acute respiratory …
Formula:
C23H27N3O5
Purity:
98.03%
Color and Shape:
Solid
Molecular weight:
425.48
Ref: TM-T16864
| 1mg | 313.00 € | ||
| 5mg | 747.00 € | ||
| 10mg | 1,169.00 € | ||
| 25mg | 1,738.00 € | ||
| 50mg | 2,357.00 € | ||
| 1mL*10mM (DMSO) | 838.00 € |
Estimated delivery in United States, on Friday 27 Jun 2025
FR-145715
CAS:149917-31-7
FR-145715 is a histamine H2 receptor antagonist characterized by its specific anti-Helicobacter pylori activity. This …
Formula:
C16H21N5O2S
Color and Shape:
Liquid
Molecular weight:
347.44
Ref: TM-T201582
| 10mg | To inquire | ||
| 50mg | To inquire |
Estimated delivery in United States, on Friday 27 Jun 2025
O-1269
CAS:336615-64-6
O-1269 acts as a partial agonist for the cannabinoid receptor 1 (CB1R), with a binding …
Formula:
C22H22Cl3N3O
Color and Shape:
Liquid
Molecular weight:
450.79
Ref: TM-T201557
| 10mg | To inquire | ||
| 50mg | To inquire |
Estimated delivery in United States, on Friday 27 Jun 2025
SGL5213
CAS:1240305-17-2
SGL5213 is a potent oral SGLT1 inhibitor (IC50: 29 nM) with potential for treating type …
Formula:
C37H55N3O8
Purity:
98%
Color and Shape:
Solid
Molecular weight:
669.85
Ref: TM-T12892
| 25mg | 3,535.00 € | ||
| 50mg | 4,446.00 € | ||
| 100mg | 5,890.00 € |
Estimated delivery in United States, on Friday 27 Jun 2025
Tiprenolol hydrochloride
CAS:13379-87-8
Tiprenolol hydrochloride is a β-adrenoceptor (β-adrenoceptor) antagonist. This compound is effective in eliminating ventricular arrhythmias …
Formula:
C13H22ClNO2S
Color and Shape:
Liquid
Molecular weight:
291.84
Ref: TM-T201760
| 10mg | To inquire | ||
| 50mg | To inquire |
Estimated delivery in United States, on Friday 27 Jun 2025
Tipindole
CAS:7489-66-9
Tipindole is a serotonin antagonist utilized in research related to depression.
Formula:
C16H20N2O2S
Color and Shape:
Liquid
Molecular weight:
304.41
Ref: TM-T201819
| 10mg | To inquire | ||
| 50mg | To inquire |
Estimated delivery in United States, on Friday 27 Jun 2025
BAY 38-7271
CAS:212188-60-8
BAY 38-7271: potent neuroprotective, selective CB1/CB2 agonist, Ki of 1.85 nM (CB1) & 5.96 nM …
Formula:
C20H21F3O5S
Purity:
98%
Color and Shape:
Solid
Molecular weight:
430.44
Ref: TM-T14504
| 25mg | 2,442.00 € | ||
| 50mg | 3,212.00 € | ||
| 100mg | 4,370.00 € |
Estimated delivery in United States, on Friday 27 Jun 2025
Dersimelagon
CAS:1835256-48-8
Dersimelagon (MT-7117) is an orally active, selective melanocortin 1 receptor (MC1R) agonist.Cost-effective and quality-assured.
Formula:
C36H45F4N3O5
Purity:
97.35% - 98.23%
Color and Shape:
Solid
Molecular weight:
675.75
Ref: TM-T25310
| 1mg | 79.00 € | ||
| 5mg | 180.00 € | ||
| 10mg | 264.00 € | ||
| 25mg | 452.00 € | ||
| 50mg | 647.00 € |
Estimated delivery in United States, on Friday 27 Jun 2025
