G-protein Coupled Receptors and 7-TM Receptors
G-protein coupled receptors (GPCRs) and 7-transmembrane (7-TM) receptors are a large family of membrane proteins that play key roles in cellular communication and signal transduction. These receptors are involved in a wide range of physiological processes, including sensory perception, immune response, and hormone regulation. GPCRs are major targets in drug discovery, making them essential for research in pharmacology and medicine. At CymitQuimica, we offer a comprehensive selection of high-quality reagents and compounds related to GPCRs and 7-TM receptors to support your research and drug development efforts.
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LTB4 antagonist 1
CAS:2929239-84-7
LTB4 Antagonist 1, a carboxamide-acid derivative, potently inhibits Leukotriene B4 (LTB4) activity with an IC50 …
Formula:
C26H23NO6
Purity:
98%
Color and Shape:
Liquid
Molecular weight:
445.46
Ref: TM-T72625
| 25mg | 1,872.00 € | ||
| 50mg | 2,452.00 € | ||
| 100mg | 3,230.00 € |
Estimated delivery in United States, on Friday 30 May 2025
Tedalinab
CAS:916591-01-0
Tedalinab is an effective and selective cannabinoid receptor 2 agonist.
Formula:
C19H21F2N3O
Purity:
98%
Color and Shape:
Solid
Molecular weight:
345.39
Ref: TM-T17027
| 25mg | 1,084.00 € | ||
| 50mg | 1,415.00 € | ||
| 100mg | 2,242.00 € |
Estimated delivery in United States, on Friday 30 May 2025
LTB4 antagonist 3
CAS:2929239-87-0
Compound 24e, a leukotriene B4 (LTB4) antagonist, exhibits an inhibitory concentration 50 (IC50) of 477 …
Formula:
C29H27NO6
Purity:
98%
Color and Shape:
Liquid
Molecular weight:
485.53
Ref: TM-T78678
| 25mg | 1,872.00 € | ||
| 50mg | 2,452.00 € | ||
| 100mg | 3,230.00 € |
Estimated delivery in United States, on Friday 30 May 2025
CaSR antagonist-1
CAS:1219811-83-2
CaSR Antagonist-1 is a potent inhibitor of the calcium-sensing receptor (CaSR) with an inhibitory concentration …
Formula:
C29H24FN3O2S
Purity:
98%
Color and Shape:
Liquid
Molecular weight:
497.58
Ref: TM-T79023
| 5mg | To inquire | ||
| 50mg | To inquire |
Estimated delivery in United States, on Friday 30 May 2025
(S)-FTY720-phosphonate
CAS:1142015-10-8
FTY720 (S)-Phosphate, an S1P receptor 1 (S1PR1) agonist, is utilized in studying acute inflammatory diseases, …
Formula:
C20H36NO4P
Purity:
98%
Color and Shape:
Liquid
Molecular weight:
385.48
Ref: TM-T78091
| 5mg | To inquire | ||
| 50mg | To inquire |
Estimated delivery in United States, on Friday 30 May 2025
NUCC-390 dihydrochloride (1060524-97-1 free base)
NUCC-390 dihydrochloride is selective agonist of small-molecule CXCR4 receptor.
Formula:
C23H35Cl2N5O
Purity:
98%
Color and Shape:
Solid
Molecular weight:
468.46
Ref: TM-T12269L
| 25mg | 1,444.00 € | ||
| 50mg | 1,882.00 € | ||
| 100mg | 2,375.00 € | ||
| 500mg | To inquire |
Estimated delivery in United States, on Friday 30 May 2025
ATP-γ-S tetrasodium
CAS:88453-52-5
Collagen, Type I, from bovine achilles tendon is a type I collagen extracted from bovine …
Formula:
C10H12N5Na4O12P3S
Color and Shape:
Liquid
Molecular weight:
611.17
Ref: TM-T83827
| 2600µg | 379.00 € |
Estimated delivery in United States, on Friday 30 May 2025
Deriglidole
CAS:122830-14-2
Deriglidole (SL 86-0715), an alpha2 receptor inhibitor, blocks colistin/Idazoxan but not prazosin/α2-adrenergic receptors.
Formula:
C16H21N3
Purity:
98.24% - 99.45%
Color and Shape:
Solid
Molecular weight:
255.36
Ref: TM-T10998
| 1mg | 437.00 € | ||
| 5mg | 1,008.00 € | ||
| 10mg | 1,349.00 € | ||
| 25mg | 1,995.00 € | ||
| 50mg | 2,452.00 € | ||
| 100mg | 3,230.00 € | ||
| 1mL*10mM (DMSO) | 752.00 € |
Estimated delivery in United States, on Friday 30 May 2025
AMG 837
CAS:865231-46-5
Prinaberel (ERB 041) is an ERβ agonist with anticancer activity and anti-inflammatory activity that inhibits …
Formula:
C26H21F3O3
Purity:
98%
Color and Shape:
Solid
Molecular weight:
438.44
Ref: TM-T14216
| 1mg | 92.00 € | ||
| 5mg | 275.00 € | ||
| 10mg | 507.00 € | ||
| 25mg | 1,149.00 € |
Estimated delivery in United States, on Friday 30 May 2025
Firuglipel
CAS:1371591-51-3
Firuglipel is an orally available and selective agonist of GPR119.
Formula:
C25H26FN3O5
Purity:
98%
Color and Shape:
Solid
Molecular weight:
467.49
Ref: TM-T15283
| 25mg | 1,730.00 € | ||
| 50mg | 2,262.00 € | ||
| 100mg | 2,945.00 € |
Estimated delivery in United States, on Friday 30 May 2025
LGD-6972
CAS:1207989-09-0
LGD-6972 is an antagonist of glucagon receptor.
Formula:
C43H46N2O5S
Purity:
98.8% - 99.33%
Color and Shape:
Solid
Molecular weight:
702.9
Ref: TM-T11845
| 1mg | 88.00 € | ||
| 5mg | 187.00 € | ||
| 10mg | 274.00 € | ||
| 25mg | 472.00 € | ||
| 50mg | 692.00 € | ||
| 100mg | 938.00 € | ||
| 1mL*10mM (DMSO) | 283.00 € |
Estimated delivery in United States, on Tuesday 10 Jun 2025
Vasopressin
CAS:11000-17-2
Vasopressin receptor agonist; antidiuretic
Formula:
C46H65N15O12S2
Purity:
Min. 95%
Color and Shape:
White Powder
Molecular weight:
1,084.23 g/mol
Ref: 3D-FV40959
| 1g | 1,237.00 € | ||
| 50mg | 330.00 € | ||
| 100mg | 465.00 € | ||
| 250mg | 690.00 € | ||
| 500mg | 920.00 € |
Estimated delivery in United States, on Tuesday 10 Jun 2025
AMG 837 calcium hydrate
CAS:1259389-38-2
AMG 837 calcium hydrate is a potent GPR40 agonist with an EC50 of 13 nM.
Formula:
C52H44CaF6O8
Purity:
98.07%
Color and Shape:
Solid
Molecular weight:
950.97
Ref: TM-TQ0020
| 2mg | 37.00 € | ||
| 5mg | 52.00 € | ||
| 10mg | 80.00 € | ||
| 25mg | 150.00 € | ||
| 50mg | 284.00 € | ||
| 100mg | 415.00 € | ||
| 200mg | 567.00 € | ||
| 1mL*10mM (DMSO) | 58.00 € |
Estimated delivery in United States, on Friday 13 Jun 2025
SB-616234-A
CAS:908601-49-0
SB-616234-A is a selective and orally bioavailable antagonist of 5-HT1B receptor, with anxiolytic and antidepressant …
Formula:
C32H36ClN5O3
Purity:
99.68%
Color and Shape:
Solid
Molecular weight:
574.11
Ref: TM-T12847
| 1mg | 105.00 € | ||
| 5mg | 255.00 € | ||
| 10mg | 368.00 € | ||
| 25mg | 557.00 € | ||
| 50mg | 752.00 € | ||
| 100mg | 1,035.00 € | ||
| 200mg | 1,396.00 € | ||
| 1mL*10mM (DMSO) | 321.00 € |
Estimated delivery in United States, on Friday 13 Jun 2025
SR 142948
CAS:184162-64-9
SR 142948 is a neurotensin (NT) receptor antagonist.
Formula:
C39H51N5O6
Purity:
98%
Color and Shape:
Solid
Molecular weight:
685.85
Ref: TM-T23386
| 10mg | 878.00 € |
Estimated delivery in United States, on Friday 13 Jun 2025
Lumateperone
CAS:313368-91-1
Lumateperone (ITI 722) is a 5HT2A receptor antagonist and a dopamine receptor phosphoprotein modulator (DPPM).
Formula:
C24H28FN3O
Purity:
99.77%
Color and Shape:
Solid
Molecular weight:
393.5
Ref: TM-T21069
| 10mg | 39.00 € | ||
| 25mg | 58.00 € | ||
| 50mg | 85.00 € | ||
| 100mg | 116.00 € |
Estimated delivery in United States, on Friday 13 Jun 2025
PSB 1115
CAS:152529-79-8
PSB 1115 is an A2B receptor antagonist and can counteract the inhibitory effect of NECA.
Formula:
C14H14N4O5S
Purity:
100% - 99.24%
Color and Shape:
Solid
Molecular weight:
350.35
Ref: TM-T23201
| 1mg | 66.00 € | ||
| 5mg | To inquire |
Estimated delivery in United States, on Friday 13 Jun 2025
SGLT inhibitor-1
CAS:2247314-23-2
SGLT inhibitor-1 is a potentsodium glucose co-transporter proteins (SGLTs) dual inhibitor(hSGLT1 and hSGLT2 with IC50s …
Formula:
C24H27FO8
Purity:
98%
Color and Shape:
Solid
Molecular weight:
462.46
Ref: TM-T12893
| 25mg | 2,442.00 € | ||
| 50mg | 3,212.00 € | ||
| 100mg | 4,370.00 € |
Estimated delivery in United States, on Friday 27 Jun 2025
Isotodesnitazene
CAS:2732926-27-9
Isotodesnitazene is an opioid compound that primarily targets the μ-opioid receptor (MOR). It exhibits EC50 …
Formula:
C23H31N3O
Color and Shape:
Liquid
Molecular weight:
365.51
Ref: TM-T201840
| 10mg | To inquire | ||
| 50mg | To inquire |
Estimated delivery in United States, on Friday 27 Jun 2025
Elzasonan hydrochloride
CAS:220322-05-4
Elzasonan hydrochloride is a serotonin 1B and serotonin 1D receptor antagonist. It is utilized in …
Formula:
C22H24Cl3N3OS
Color and Shape:
Liquid
Molecular weight:
484.87
Ref: TM-T201763
| 10mg | To inquire | ||
| 50mg | To inquire |
Estimated delivery in United States, on Friday 27 Jun 2025
