Benzimidazole and Imidazole Derivatives
Benzimidazole is a compound consisting of a benzene ring fused to an imidazole ring, a five-membered structure containing two nitrogen atoms. Benzimidazole derivatives, such as albendazole, are known for their antiparasitic and antifungal activity, used in the treatment of parasitic infections and certain parasitic diseases in animals and humans. Imidazole, on the other hand, is a five-membered structure with two nitrogen atoms found in various biologically active compounds. Imidazole derivatives, such as metronidazole, have antimicrobial and antiparasitic properties. These compounds are also used in the pharmaceutical industry for treating bacterial infections, parasitic diseases, and some fungal infections, as well as in organic chemistry as catalysts.
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Found 10345 products of "Benzimidazole and Imidazole Derivatives"
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Benznidazole-d7
CAS:Controlled Product<p>Applications Benznidazole-D7 is a labelled analogue of Benznidazole (B197925).<br></p>Formula:C12H5D7N4O3Color and Shape:NeatMolecular weight:267.29(2-Chlorophenyl)diphenylmethanol
CAS:<p>Impurity Clotrimazole EP Impurity A<br>Applications (2-Chlorophenyl)diphenylmethane (Clotrimazole EP Impurity A) is a triarylmethane with antiproliferative activity. (2-Chlorophenyl)diphenylmethane is a degradation product of the antifungal agent Clotrimazole (C587400). Clotrimazole Related Compound A<br>References Suzuki, M. Iyak. Kenk., 23, 44 (1992); Hajkova, R. et al.: Talanta, 73, 483 (2007); Sabourin, L. et al.: Environ. Toxicol. Chem., 30, 582 (2011);<br></p>Formula:C19H15ClOColor and Shape:NeatMolecular weight:294.77N-(3-(1H-imidazol-1-yl)propyl)-1-(4-fluorophenyl)-2,2-dimethylcyclopropane-1-carboxamide
CAS:Purity:98%Molecular weight:315.3919982910156N-Nitroso Varenicline
CAS:Controlled Product<p>Applications N-Nitroso Varenicline is a derivative of Varenicline (V215635(M)), which is a useful medication for smoking cessation.<br>References Hart, E., et al.: Behavioural Brain Research, 397, 112887 (2021)<br></p>Formula:C13H12N4OColor and Shape:NeatMolecular weight:240.261Itraconazole-d9
CAS:Controlled Product<p>Applications Itraconazole-d9, is the labeled analogue of Itraconazole (I937500, an orally active antimycotic structurally related to Ketoconazole. Antifungal. It is a COVID19-related research product.<br>References Espinel-Ingroff, A., et al.: Antimicrob. Agents Chemother., 26, 5 (1984), Heykants, J., et al.: Mycoses, 32, Suppl 1, 67 (1989), Sugar, A.M., et al.: Curr. Clin. Top. Infect. Dis., 13, 74 (1993),<br></p>Formula:C35H29D9Cl2N8O4Color and Shape:Off-White To BeigeMolecular weight:714.69rac Rivastigmine-d6
CAS:Controlled Product<p>Applications Labelled rac Rivastigmine. A brain selective acetylcholinesterase inhibitor. Nootropic.<br> Not a dangerous good if item is equal to or less than 1g/ml and there is less than 100g/ml in the package<br>References Rosler, M., et al.: Brit. Med. J., 318, 633 (1999), Enz, A., et al.: Prog. Brain Res., 98, 431 (1993),<br></p>Formula:C14H16D6N2O2Color and Shape:NeatMolecular weight:256.37(S)-N-Desethyl Oxybutynin Hydrochloride
CAS:Controlled Product<p>Applications (S)-Metabolite of the drug Oxybutynin. Used in the treatmentment of incontinence.<br>References Ehlert, F., et al.: Life Sci., 74, 355 (2003), Matsui-Sakata, A., et al.: Drug Metab. Pharmacokinet., 20, 187 (2005), Hegde, S., et al.: Br. J. Pharmacol., 147, S80 (2006), Tashiro, M., et al.: Br. J. Clin. Pharmacol., 61, 16 (2006),<br></p>Formula:C20H27NO3·ClHColor and Shape:NeatMolecular weight:365.89Lamotrigine N2-Oxide
CAS:Controlled Product<p>Applications Lamotrigine analog for production of anti-lamotrigine antibodies and use as immunoassay reagent.<br> Not a dangerous good if item is equal to or less than 1g/ml and there is less than 100g/ml in the package<br>References Doig, M.V., et al.: J. Chromatogr., 554, 181 (1991),<br></p>Formula:C9H7Cl2N5OPurity:90%Color and Shape:NeatMolecular weight:272.0911-Keto Oxcarbazepine
CAS:Controlled Product<p>Stability Unstable in Solution<br>Applications A keto impurity of the anticonvulsant Oxcarbazepine (O869250).<br></p>Formula:C15H10N2O3Color and Shape:NeatMolecular weight:266.251-Methyl Mebendazole
CAS:Controlled Product<p>Impurity Mebendazole USP Related Compound D<br>Applications Mebendazole (M200500) related compound as anthelmintic agent. Mebendazole USP Related Compound D.<br>References Dhaneshwar, S.R., et al.: Indian Drugs, 28, 21 (1990),<br></p>Formula:C17H15N3O3Color and Shape:NeatMolecular weight:309.32Miconazole N-(2-Methyl)propanoate
CAS:Controlled Product<p>Applications Miconazole N-(2-Methyl)propanoate is an impurity of Miconazole (M342500). Miconazole EP Impurity E.<br></p>Formula:C22H20Cl4N2O3Color and Shape:NeatMolecular weight:502.22Tioconazole
CAS:Controlled Product<p>Applications Tioconazole is an antifungal that is more active than Fluconazole (F421000) or Voriconazole (V760000) against Candida glabrata mutant strains. Antifungal (topical).<br>References Jevons, S., et al.: Antimicrob. Agents Chemother., 15, 597 (1979), Clayton, Y.M., et al.: Clin. Exp. Dermatol., 7, 543 (1982), Marriott, M.S., et al.: Dermatologica, 166, 1 (1983),<br></p>Formula:C16H13Cl3N2OSColor and Shape:WhiteMolecular weight:387.71Fenbendazole Sulfone-d3
CAS:Controlled Product<p>Applications Labelled version of Fenbendazole Sulfone (F246770), which is a metabolite of Fenbendazole (F246750).<br>References McKellar, Q., et al.: J. Vet. Pharmacol. Ther., 13, 223 (1990), De Ruyck, H., et al.: Food Control., 11, 165 (2000),<br></p>Formula:C15D3H10N3O4SColor and Shape:NeatMolecular weight:334.368-Chloro-6-(2-fluorophenyl)-1-methyl-6H-Imidazo[1,5-a][1,4]benzodiazepine
CAS:Controlled Product<p>Impurity MIdazolam EP Impurity B<br>Applications 8-Chloro-6-(2-fluorophenyl)-1-methyl-6H-Imidazo[1,5-a][1,4]benzodiazepine is an isomer of Midazolam (M343000), an anesthetic, anticonvulsant, sedative and hypotic agent.<br>References Walser, A., et al.: J. Org. Chem., 43, 936 (1978); Dundee, J. W., et al.: Drugs, 28, 519 (1984); Lahat, E., et al.: Br. Med. J., 321, 83 (2000)<br></p>Formula:C18H13ClFN3Color and Shape:NeatMolecular weight:325.775-Chloro-6-(2,3-dichlorophenoxy)-1,3-dihydro-2H-benzimidazol-2-one
CAS:<p>Applications 5-Chloro-6-(2,3-dichlorophenoxy)-1,3-dihydro-2H-benzimidazol-2-one is a metabolite of Triclabendazole (T774175), the only anthelmintic drug, which is active against immature, mature and adult stages of fluke.<br>References Whelan, M., et al.: J. Chromato., 1275, 41 (2013); Barrera, S., et al.; Antimicrob. Agent. Chemother., 56, 3535 (2012);<br></p>Formula:C13H7Cl3N2O2Color and Shape:Off-White To BrownMolecular weight:329.57Hydroxy Voriconazole
Controlled Product<p>Applications A hydroxylated derivative of Voriconazole (V760000), a systemic antifungal and ergosterol biosynthesis inhibitor.<br> Not a dangerous good if item is equal to or less than 1g/ml and there is less than 100g/ml in the package<br>References Sanati, H., et al.: Antimicrob. Ag. Chemother., 41, 2492 (1997).<br></p>Formula:C16H14F3N5O2Color and Shape:NeatMolecular weight:365.313,5-Didesamino-3,5-dioxo Lamotrigine
CAS:Controlled Product<p>Impurity Lamotrigine EP Impurity D<br>Applications 3,5-Didesamino-3,5-dioxo Lamotrigine (Lamotrigine EP Impurity D) is an impurity of the anticonvulsant Lamotrigine (L173250).<br>References Hlavac, J. et al.: ARKIVOC, 1, 22 (2003);<br></p>Formula:C9H5Cl2N3O2Color and Shape:NeatMolecular weight:258.06(3aR,7aS)-rel-Hexahydro-1,3-isobenzofurandione
CAS:Controlled Product<p>Applications (3aR,7aS)-rel-Hexahydro-1,3-isobenzofurandione is a reagent used in the synthesis of Pregabalin (P704800), a GABA analogue used as an anticonvulsant. Also used to prepare P2X7 receptor antagonists.<br>References Taylor, C.P., at al.: Epilepsy Res., 14, 11 (1993), Field, M.J., et al.: Pain, 80, 391 (1999); Eur. J. Org. Chem., 2013, 4495 (2013); Yang, H. et al.: Chinese. Chem. Lett., 24, 553 (2013);<br></p>Formula:C8H10O3Color and Shape:NeatMolecular weight:154.16Lamotrigine 5,5-Dimer
Controlled Product<p>Applications Lamotrigine 5,5-Dimer is a dimer impurity of the anticonvulsant Lamotrigine (L173250).<br>References Miller, A.A., et al.: Epilepsia, 27, 483 (1986), Grunze, et al.: Neuropsychobiology, 38, 131 (1998), Calabrese, J.R., et al.: J. Clin. Psychiatry, 60, 79 (1999),<br></p>Formula:C19H14Cl4N10Color and Shape:Off White SolidMolecular weight:524.19Omeprazole sulfide N-Oxide
CAS:<p>Applications 5-Methoxy-2-[[(4-methoxy-3,5-dimethyl-2-pyridinyl)methyl]thio]-1H-benzimidazole N-Oxide is a metabolite of Omeprazole (O635000), an proton inhibitor used as an antiulcerative agent.<br>References Muller, P., et al.: Arzneimittel-Forsch., 33, 1685 (1983), Wallmark, B., et al.: Biochim. Biophys. Acta., 778, 549 (1984), Morii, M., et al.: J. Biol. chem., 268, 21553 (1993), Ritter, M., et al.: Br. J. Pharmacol., 124, 627 (1998)<br></p>Formula:C17H19N3O3SColor and Shape:Off-WhiteMolecular weight:345.42
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