Benzodiazepine Derivatives
Benzodiazepines are organic compounds with a fused bicyclic benzodiazepine core, widely used in the development of drugs with anxiolytic, sedative, anticonvulsant, and muscle relaxant properties. Their derivatives include modified structures that enhance selectivity and pharmacokinetic profiles, enabling the creation of new molecules with advanced therapeutic applications. These compounds are used in the formulation of APIs for the treatment of sleep disorders, anxiety, epilepsy, and muscle spasms. Additionally, benzodiazepine derivatives are essential in the research of new psychotropic agents and in optimising neurological treatments.
At CymitQuimica, we offer high-purity benzodiazepine derivatives for applications in chemical synthesis, pharmaceutical development, and neuroscience.
Found 332 products of "Benzodiazepine Derivatives"
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3-Amino-6-chloro-3,4-dihydro-2-methyl-4-phenyl-4-quinazolinol
CAS:Controlled ProductFormula:C15H14ClN3OColor and Shape:NeatMolecular weight:287.742-Amino-5-nitrobenzophenone
CAS:Controlled ProductFormula:C13H10N2O3Color and Shape:NeatMolecular weight:242.23Flumazenil Carboxylic Acid-D3
Controlled Product<p>Applications Flumazenil Carboxylic Acid-D3 is an isotope labelled form of Flumazenil Carboxylic Acid (F500455); a derivative of Flumazenil (F500455), a benzodiazepine antagonist that can prevent or abolish (at the receptor level) the effects of a benzodiazepine.<br>References Brogden, R. & Goa, K.: Drugs, 35, 448 (1988); Klotz, U. & Kanto, J.: Clin. Pharmacokinet., 14, 1 (1988)<br></p>Formula:C13H7D3FN3O3Color and Shape:NeatMolecular weight:278.257-Aminonorflunitrazepam
CAS:Controlled ProductFormula:C15H12FN3OColor and Shape:Light YellowMolecular weight:269.272-(2-Acetylhydrazino)-7-chloro-5-phenyl-3H-1,4-benzodiazepine
CAS:Controlled Product<p>Applications 2-(2-Acetylhydrazino)-7-chloro-5-phenyl-3H-1,4-benzodiazepine is an impurity of Alprazolam (A575650.<br>References Hester, J.B., et al.: J. Org. Chem., 44, 2688, (1979); Anjaneyulu, Y., et al.: Asian. J. Chem., 19, 3375 (2007);<br></p>Formula:C17H15ClN4OColor and Shape:White To Off-WhiteMolecular weight:326.783-Methyl Clobazam
CAS:Controlled Product<p>Applications 3-Methyl Clobazam is a metabolite of Clobazam (C582500), a benzodiazepine psychotherapeutic agent that has proven efficacy against multiple seizure types. An anxiolytic; anticonvulsant.<br>References Gastaut, H., et al.: Epilepsia, 20, 437 (1979); Guberman, A., et al.: Can J. Neurol. Sci., 17, 311 (1990); Munn, R., et al.: Pediatr. Neurol. 9, 465 (1993)<br></p>Formula:C17H15ClN2O2Color and Shape:NeatMolecular weight:314.77Clobazam CIV
CAS:Controlled Product<p>Clobazam (inn) and methyprylon (inn)</p>Formula:C16H13ClN2O2Color and Shape:White Crystalline PowderMolecular weight:300.066562-(2-Amino-5-bromobenzoyl)pyridine
CAS:<p>2-(2-Amino-5-bromobenzoyl)pyridine (2ABBP) is a chemical compound with the molecular formula C10H7BrN3. It is a glucuronide conjugate of 2-amino-5-bromobenzoic acid and has been used as an immunological reagent in the form of a monoclonal antibody. 2ABBP binds to dryopteris, which is a plant species that contains polyphenols called pteridines. 2ABBP has been shown to have anti-inflammatory properties in rat liver microsomes and cell culture experiments. The mechanism of action may involve inhibition of cyclooxygenase enzymes, which are involved in prostaglandin synthesis. 2ABBP also binds to human serum albumin and chaperones, proteins that bind other proteins or small molecules. The biological activity of 2ABBP may be due to its ability to form coval</p>Formula:C12H9BrN2OPurity:Min. 95%Molecular weight:277.12 g/molRef: 4Z-E-153009
Discontinued productRef: 4Z-A-231026
Discontinued product7-Amino Clonazepam-d4
CAS:Controlled Product<p>Applications A labelled major metabolite of Clonazepam (C587080).<br>References Clark, D., et al.: Drugs, 29, 342 (1985), Colmenero, J., et al.: Antimicrob. Agents Chemother., 38, 2798 (1994), Grant, D., et al.: Pharmacology, 61, 204 (2000), Negrusz, A., et al.: Anal. Bioanal. Chem., 376, 1198 (2003),<br></p>Formula:C152H4H8ClN3OColor and Shape:NeatMolecular weight:289.75
