Endokrinologie/Hormone

NE 52-QQ57 is a selective, and orally available antagonist of GPR4(IC50 : 70 nM),with anti-inflammatory …

ZT 52656A is a selective agonist of kappa opioid, and used for the prevention or …

L-Thyroxine (NSC 36397) is the major hormone derived from the thyroid gland. L-Thyroxine (NSC 36397) …

Estradiol cypionate (Depofemin), the 17 β-cyclopentylpropinate ester of estradiol, inhibits ET-1 synthesis via estrogen receptor.

Alvimopan (LY 246736) is a synthetic trans-3, 4-dimethyl-4-(3-hydroxyphenyl) piperidine with peripherally selective opioid mu receptor …

Beclometasone dipropionate (Vancenase) is the dipropionate ester of a synthetic glucocorticoid with anti-inflammatory and immunomodulating …

Medroxyprogesterone Acetate (Farlutin) is a synthetic progestin that is derived from 17-hydroxyprogesterone. It is a …

Estradiol benzoate (Benzhormovarine) is the synthetic benzoate ester of estradiol, a steroid sex hormone vital …

N-Desmethyltamoxifen hydrochloride is the major tamoxifen metabolite in humans.

Mestranol (Devocin), a semisynthetic estrogen, is used as an estrogen receptor agonist and must be …

Megestrol acetate (BDH1298) is a progestogen with actions and uses similar to those of the …

UT-155 is a selective and potent antagonist of the androgen receptor (AR) (Ki: 267 nM …

Vincamine (Perval) is a major alkaloid of Vinca minor L., Apocynaceae. It has been used …

Ethynodiol diacetate (Ethynodiol acetate) is a synthetic progestational hormone used alone or in combination with …

Diethylstilbestrol (DES) is used in the treatment of menopausal and postmenopausal disorders.

GSK256073 is an orally active GPR109A agonist. GSK256073 also is a long-lasting and non-flushing HCA2 …

Nimodipine (BAY-e 9736), a 1, 4-dihydropyridine calcium channel blocker, acts primarily on vascular smooth muscle …

AR antagonist 1 is a potent antagonist of the androgen receptor. It binds to E3 …

Flumethasone (RS-2177) is a glucocorticoid receptor agonist, with anti-inflammatory, antipruritic and vasoconstrictive properties.

Elacestrant (RAD1901) with IC50s of 48 and 870 nM for ERα and ERβ, respectively.Elacestrant is …

Norethindrone is a potent synthetic hormone used for amenorrhea, uterine bleeding, endometriosis, and contraception.

Glucagon (1-29), bovine, human, porcine hydrochloride is a peptide hormone, produced by pancreatic α-cells. Glucagon …

Resorcinolnaphthalein is a specific enhancer of angiotensin-converting enzyme 2 (ACE2) (EC50 value of 19.5 μM).

Perindopril erbumine (S9490-3) is the tert-butylamine salt of perindopril, the ethyl ester of a non-sulfhydryl …

2-Thiouracil (Deracil) is a thiolated uracil derivative that is a known anti-hyperthyroid agent.

Eplerenone (CGP 30083) is an aldosterone receptor antagonist and potassium-sparing diuretic used in the therapy …

Betamethasone Dipropionate is the 17, 21-dipropionate ester of betamethasone, a synthetic glucocorticoid with metabolic, immunosuppressive …

Clobetasol propionate (CGP9555) exerts its effect by binding to cytoplasmic glucocorticoid receptors and subsequently activates …

Triamcinolone (Aristocort) is a synthetic glucocorticoid with anti-inflammatory and immunomodulating properties.

Chlormadinone acetate (Gestafortin) is an orally active synthetic progestational hormone used often in combinations as …

Triamcinolone acetonide (Azmacort) is a Corticosteroid. The mechanism of action of triamcinolone acetonide is as …

Ramatroban (BAY u3405) (BAY u3405) is a thromboxane A(2) (TxA(2)) antagonist marketed for allergic rhinitis. …

Altrenogest (Allyltrenbolone)(A35957; RU2267), a progestogen, has structural relation with veterinary steroid trenbolone.

Epalrestat (ONO2235), an aldose reductase inhibitor, is well tolerated in Long-term therapy. It can effectually …

Mirtazapine (6-Azamianserin) is a tetracyclic antidepressant with a somewhat unique mechanism of action. Mirtazapine therapy …

6α-Methylprednisolone 21-hemisuccinate sodium salt (Asmacortone), a water-soluble ester, is used for allergic, cardiac, and hypoxic …

Medrysone is a synthetic glucocorticoid for topical use with anti-inflammatory and anti-allergic effects, altering gene …

Mifepristone (C-1073) is a Progestin Antagonist. The mechanism of action of mifepristone is as a …

Estropipate (Piperazine estrone sulfate) is a natural estrogenic substance composed of estrone sulfate and piperazine.

Cortisone (17-Hydroxy-11-dehydrocorticosterone) is a corticosteroid with potent glucocorticoid activity.

Canrenone (SC14266) is an aldosterone antagonist with potassium-sparing diuretic activity.

PCO371 (2,4-Imidazolidinedione, 1-(3,5-dimethyl-4-(2-((4-oxo-2-(4-(trifluoromethoxy)phenyl)-1,3,8-triazaspiro(4.5)dec-1-en-8-yl)sulfonyl)ethyl)phenyl)-5,5-dimethyl-) is an orally active full agonist of parathyroid hormone receptor 1. It …

Clomiphene citrate (NSC 35770) is a selective estrogen receptor modulator.

Dehydroisoandrosterone 3-acetate (Prasterone acetate) is a primary C19 steroid generated by the adrenal cortex.

N-Desmethyl-Apalutamide is a less potent antagonist of the androgen receptor, is an active Apalutamide metabolite.

G-1 is a nonsteroidal, high-affinity and selective GPR30 agonist (Ki: 11 nM).

AZD5423: Inhaled, potent GR modulator, non-steroidal, curbs allergy asthma symptoms.

Avobenzone is a dibenzoylmethane endocrine disruptor that binds directly to estrogen receptor β, acting as …

ACP-105 is a novel and potent nonsteroidal selective androgen receptor modulator (SARM) with partial agonist …

Quinapril HCl (PD-109452-2) treats hypertension and heart failure; low risk of liver enzyme elevations.

Clobetasone butyrate, a synthetic glucocorticoid with topical anti-inflammatory activity, is effective in treating corticosteroid-responsive dermatoses, …

17α-Hydroxyprogesterone (17-OHP) is a physiological progestin that is produced during glucocorticoid and steroid hormone synthesis …

The test principle applied in this kit is Sandwich enzyme immunoassay. The microtiter plate provided …

The test principle applied in this kit is Sandwich enzyme immunoassay. The microtiter plate provided …

The test principle applied in this kit is Sandwich enzyme immunoassay. The microtiter plate provided …

The test principle applied in this kit is Sandwich enzyme immunoassay. The microtiter plate provided …