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Apoptosis

Apoptosis

Los inhibidores de la apoptosis son compuestos que previenen o retrasan el proceso de muerte celular programada, conocido como apoptosis. Estos inhibidores son vitales para estudiar los mecanismos de supervivencia celular y se utilizan para investigar enfermedades donde la apoptosis está desregulada, como el cáncer, los trastornos neurodegenerativos y las enfermedades autoinmunes. Al modular la apoptosis, estos inhibidores pueden ayudar en el desarrollo de terapias dirigidas a controlar la muerte celular. En CymitQuimica, ofrecemos una amplia selección de inhibidores de la apoptosis de alta calidad para apoyar su investigación en biología celular, oncología y campos relacionados.

Subcategorías de "Apoptosis"

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Se han encontrado 5600 productos de "Apoptosis"

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  • Alisertib Sodium

    CAS:
    <p>Alisertib Sodium (MLN 8237 Sodium)is a selective Aurora A inhibitor that causes G2/M phase arrest and chromosomal misalignment, leading to tumour cell apoptosis.</p>
    Fórmula:C27H19ClFN4NaO4
    Pureza:99.77%
    Forma y color:Solid
    Peso molecular:540.91
  • Tiplaxtinin

    CAS:
    <p>Tiplaxtinin (Tiplasinin)(PAI-039) is a selective and orally efficacious inhibitor of plasminogen activator inhibitor-1 (PAI-1) with IC50 of 2.7 uM.</p>
    Fórmula:C24H16F3NO4
    Pureza:99.16% - 99.93%
    Forma y color:Solid
    Peso molecular:439.38
  • AT9283

    CAS:
    <p>AT9283 (J-504568) is an effective multi-targeted inhibitor of JAK2(IC50=1.2 nM) and JAK3(IC50=1.1 nM), Aurora A, Aurora B and Abl(T315I).</p>
    Fórmula:C19H23N7O2
    Pureza:99.83% - 99.98%
    Forma y color:Solid
    Peso molecular:381.43
  • Se-Methylselenocysteine

    CAS:
    <p>Se-Methylselenocysteine (Se-MSC) is a potent chemopreventive agent in many test systems and has been shown to inhibit tumor promotion and induce apoptosis.</p>
    Fórmula:C4H9NO2Se
    Pureza:99.49% - 99.87%
    Forma y color:White To Slightly Yellow Powder
    Peso molecular:182.08
  • Tamibarotene

    CAS:
    <p>Tamibarotene (Amnolake) is an orally active, synthetic retinoid, developed to overcome all-trans retinoic acid (ATRA) resistance, with potential antineoplastic</p>
    Fórmula:C22H25NO3
    Pureza:98.55% - 99.73%
    Forma y color:Crystalline Solid
    Peso molecular:351.44
  • AGK2

    CAS:
    <p>AGK2(IC50=3.5 μM) is an effective, and specific SIRT2 inhibitor.</p>
    Fórmula:C23H13Cl2N3O2
    Pureza:98.68% - 99.17%
    Forma y color:Solid
    Peso molecular:434.27
  • Leachianone A

    CAS:
    <p>Leachianone A (Isokurarinone) is a potential antitoxic agent, it shows inhibitory effects on cadmium- Induced cytotoxicity.</p>
    Fórmula:C26H30O6
    Pureza:98.53% - 99.79%
    Forma y color:Solid
    Peso molecular:438.51
  • S55746 hydrochloride

    CAS:
    <p>S55746 hydrochloride is a potent, orally active and selective inhibitor of BCL-2(Ki of 1.3 nM and a Kd of 3.9 nM),with antitumor activity with low toxicity.</p>
    Fórmula:C43H43ClN4O6
    Pureza:98%
    Forma y color:Solid
    Peso molecular:747.28
  • PS210

    CAS:
    <p>PS210 selectively activates PDK1 (Kd: 3 μM), doesn't affect PDK1 downstream kinases. Prodrug PS423 inhibits PDK1-mediated S6K phosphorylation.</p>
    Fórmula:C19H15F3O5
    Pureza:99.78%
    Forma y color:Solid
    Peso molecular:380.31
  • Alofanib

    CAS:
    <p>Alofanib (RPT835) selectively inhibits FGFR2 in KATO III cells with IC50 &lt;10 nM; doesn’t affect FGFR1/3 or FGF2-FGFR2 binding.</p>
    Fórmula:C19H15N3O6S
    Pureza:99.53% - 99.81%
    Forma y color:Solid
    Peso molecular:413.4
  • Dinoprost tromethamine salt

    CAS:
    <p>Dinoprost tromethamine salt (PGF2α THAM) is a naturally occurring prostaglandin used in medicine to induce labor and as an abortifacient.</p>
    Fórmula:C24H45NO8
    Pureza:99.73%
    Forma y color:Natural Form Crystals Solid
    Peso molecular:475.62
  • Clovamide

    CAS:
    <p>Trans-Clovamide (trans-Clovamide) is a naturally occurring caffeoyl conjugate identified in the antioxidant polyphenolic fraction of cocoa (T.</p>
    Fórmula:C18H17NO7
    Pureza:97.12% - 97.68%
    Forma y color:Solid
    Peso molecular:359.33
  • RX-3117

    CAS:
    <p>RX-3117 (fluorocyclopentenylcytosine) is a novel a cytidine analog.</p>
    Fórmula:C10H12FN3O4
    Pureza:97.46%
    Forma y color:Solid
    Peso molecular:257.22
  • Cycleanine

    CAS:
    <p>Cycleanine has potent antibacterial, antifungal, antiplasmodial, and cytotoxic activities.</p>
    Fórmula:C38H42N2O6
    Pureza:98.04% - 99.57%
    Forma y color:Solid
    Peso molecular:622.75
  • API-1

    CAS:
    <p>API-1 (NSC-177223) is a potent inhibitor of Akt. It induces GSK3-dependent, β-TrCP- and FBXW7-mediated Mcl-1 degradation, resulting in induction of apoptosis .</p>
    Fórmula:C13H15N5O6
    Pureza:97.15%
    Forma y color:Solid
    Peso molecular:337.29
  • Dapivirine

    CAS:
    <p>Dapivirine (R147681) is a diarylpyrimidine non-nucleoside reverse transcriptase inhibitor.</p>
    Fórmula:C20H19N5
    Pureza:98% - 99.77%
    Forma y color:Solid
    Peso molecular:329.4
  • Melatonin

    CAS:
    <p>Melatonin (Melatonine) is a natural hormone that activates melatonin receptors. Melatonin regulates the biological clock. Cost-effective and quality-assured.</p>
    Fórmula:C13H16N2O2
    Pureza:98% - 99.89%
    Forma y color:Pale Yellow Leaflets From Benzene Solid
    Peso molecular:232.28
  • Chrysosplenol D

    CAS:
    <p>Chrysosplenol D, an efflux pump inhibitor that can potentiate the activity of commercially important antibiotics and antimalarials.</p>
    Fórmula:C18H16O8
    Pureza:97.87% - 99.98%
    Forma y color:Solid
    Peso molecular:360.31
  • R547

    CAS:
    <p>R547 (Ro 4584820) is a potent ATP-competitive inhibitor of CDK1/2/4 with Ki of 2 nM/3 nM/1 nM.</p>
    Fórmula:C18H21F2N5O4S
    Pureza:90% - 99.64%
    Forma y color:Solid
    Peso molecular:441.45
  • Arctigenin

    CAS:
    <p>(-)-Arctigenin ((-)-Arctigenin) is found in burdock.</p>
    Fórmula:C21H24O6
    Pureza:98% - 99.51%
    Forma y color:Solid
    Peso molecular:372.41