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Caspasa

Caspasa

Los inhibidores de caspasas son compuestos que bloquean la actividad de las caspasas, una familia de proteasas que son ejecutores centrales de la apoptosis. Las caspasas escinden sustratos específicos dentro de la célula para desencadenar el proceso apoptótico, lo que conduce a la muerte celular programada. Los inhibidores de caspasas se utilizan para estudiar los mecanismos de la apoptosis, así como para prevenir la muerte celular no deseada en varios modelos de investigación. Estos inhibidores también se exploran en contextos terapéuticos para proteger las células de la apoptosis en enfermedades como la neurodegeneración. En CymitQuimica, ofrecemos una amplia gama de inhibidores de caspasas de alta calidad para apoyar su investigación en apoptosis, muerte celular y campos relacionados.

Se han encontrado 125 productos de "Caspasa"

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  • Almorexant hydrochloride

    CAS:
    <p>Almorexant hydrochloride (ACT 078573 hydrochloride) is a dual orexin receptor antagonist that induces apoptosis and can be used to study sleep disorders.</p>
    Fórmula:C29H32ClF3N2O3
    Pureza:99.85%
    Forma y color:Solid
    Peso molecular:549.02
  • MX1013

    CAS:
    <p>MX1013, a dipeptide pan-caspase inhibitor, inhibits caspase-1, -3, -6, -7, -8, and -9.</p>
    Fórmula:C18H23FN2O6
    Forma y color:Solid
    Peso molecular:382.39
  • J22352

    CAS:
    <p>J22352, a PROTAC (proteolysis-targeting chimeras)-like and highly selective HDAC6 inhibitor with an IC50 value of 4.7 nM, enhances anticancer effects in</p>
    Fórmula:C24H21N3O4
    Forma y color:Solid
    Peso molecular:415.44
  • Paris saponin VII

    CAS:
    <p>Paris saponin VII (Dioscini) shows inhibitory effects on cell proliferation.</p>
    Fórmula:C51H82O21
    Pureza:99.51% - 99.63%
    Forma y color:Solid
    Peso molecular:1031.18
  • Asperosaponin VI

    CAS:
    <p>Asperosaponin VI, from Dipsacus asper rhizome, treats back pain, hematoma, and fractures.</p>
    Fórmula:C47H76O18
    Pureza:97.15% - 99.79%
    Forma y color:Solid
    Peso molecular:929.1
  • KEA1-97

    CAS:
    <p>Kea1-97 is a selective disruptor of interaction between thioredoxin and caspase-3 (IC50 = 10 μ M).</p>
    Fórmula:C15H9Cl2FN4
    Pureza:97.07%
    Forma y color:Solid
    Peso molecular:335.16
  • Taurodeoxycholic acid sodium hydrate

    CAS:
    <p>Taurodeoxycholic acid sodium hydrate (Sodium taurodeoxycholate monohydrate), a hydrophilic bile salt, on bile salt and biliary lipid secretion in the rat.</p>
    Fórmula:C26H46NNaO7S
    Pureza:99.95%
    Forma y color:Solid
    Peso molecular:539.70
  • Z-DEVD-FMK

    CAS:
    <p>Z-DEVD-FMK (Caspase-3 Inhibitor) is a selective, irreversible Caspase-3 inhibitor, and also exhibits effective inhibition activity on caspase-6, caspase-7,</p>
    Fórmula:C30H41FN4O12
    Pureza:96.19% - 99.69%
    Forma y color:Solid
    Peso molecular:668.66
  • Chelidonic acid

    CAS:
    <p>Chelidonic acid, in Chelidonium majus, acts as an analgesic, antimicrobial, CNS sedative, and has anti-inflammatory properties.</p>
    Fórmula:C7H4O6
    Pureza:99.03%
    Forma y color:Solid
    Peso molecular:184.1
  • AVN-944

    CAS:
    <p>AVN-944 (VX-944)(VX-944) is a selective, noncompetitive inhibitor of human IMPDH with Ki of 6-10 nM for IMPDH1/IMPDH2.</p>
    Fórmula:C25H27N5O5
    Pureza:99.07% - ≥95%
    Forma y color:Solid
    Peso molecular:477.51
  • Ac-DEVD-AMC

    CAS:
    <p>Ac-DEVD-AMC (AC-ASP-MET-GLN-ASP-7-AMINO-4-METHYLCOUMARIN) is the substrate of Caspase-3 .</p>
    Fórmula:C30H37N5O13
    Pureza:98.20%
    Forma y color:White Powder
    Peso molecular:675.64
  • 5,7-Dihydroxychromone

    CAS:
    <p>1.</p>
    Fórmula:C9H6O4
    Pureza:99.76% - ≥95%
    Forma y color:Solid
    Peso molecular:178.14
  • Tauroursodeoxycholate

    CAS:
    <p>Tauroursodeoxycholate (UR 906), a hydrophilic bile acid, low in humans, may treat PBC, insulin resistance, and ALS.</p>
    Fórmula:C26H45NO6S
    Pureza:98.77% - 99.93%
    Forma y color:White Solid
    Peso molecular:499.7
  • Diclofenac Potassium

    CAS:
    <p>Diclofenac Potassium (CGP-45840B) is a nonsteroidal anti-inflammatory drug taken to reduce inflammation and as an analgesic reducing pain in certain conditions.</p>
    Fórmula:C14H10Cl2KNO2
    Pureza:99.51%
    Forma y color:White To Yellowish Crystalline Powder
    Peso molecular:334.24
  • CASP3 Activator 1541

    CAS:
    <p>CASP3 Activator 1541 is an activator of the proenzyme forms of caspase-3, and induces cell death.</p>
    Fórmula:C24H17N3O4
    Pureza:98.84%
    Forma y color:Solid
    Peso molecular:411.41
  • 5,​7,​4'-​Trimethoxyflavone

    CAS:
    <p>5,7,4'-Trimethoxyflavone (4',5,7-Trimethoxyflavone) is isolated from Kaempferia parviflora (KP) which is a medicinal plant from Thailand.</p>
    Fórmula:C18H16O5
    Pureza:97.53%
    Forma y color:Solid
    Peso molecular:312.32
  • L67

    CAS:
    <p>L67 (DNA Ligase Inhibitor) is a competitive human DNA ligase inhibitor, inhibits DNA ligases I and III (IC50: 10 μM).</p>
    Fórmula:C16H14Br2N4O4
    Pureza:98.34% - 99.56%
    Forma y color:Solid
    Peso molecular:486.11
  • Belnacasan

    CAS:
    <p>Belnacasan (VX-765) is an orally active IL-converting enzyme/caspase-1 inhibitor.</p>
    Fórmula:C24H33ClN4O6
    Pureza:96.53% - 99.5%
    Forma y color:Solid
    Peso molecular:508.99
  • 2-HBA

    CAS:
    <p>2-HBA, a synthetic analog of curcumin, is an indirect inducer of enzymes that catalyze detoxification reactions through the Keap1-Nrf2-ARE pathway.</p>
    Fórmula:C17H14O3
    Pureza:99.76%
    Forma y color:Solid
    Peso molecular:266.29
  • Arnicolide D

    CAS:
    <p>Arnicolide D is a sesquiterpene lactone.</p>
    Fórmula:C19H24O5
    Pureza:96.66%
    Forma y color:Solid
    Peso molecular:332.39