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Canal de sodio

Canal de sodio

Los canales de sodio son proteínas de membrana esenciales que permiten el paso de iones de sodio (Na+) a través de la membrana celular, generando y propagando señales eléctricas en neuronas, células musculares y otros tejidos excitables. Estos canales son vitales para la iniciación y conducción de potenciales de acción, lo que los hace cruciales en procesos como la transmisión de impulsos nerviosos, la contracción muscular y la función cardíaca. La desregulación de los canales de sodio puede llevar a trastornos neurológicos, arritmias y condiciones de dolor crónico. En CymitQuimica, ofrecemos una variedad de moduladores de canales de sodio para apoyar su investigación en neurobiología, cardiología y manejo del dolor.

Se han encontrado 202 productos de "Canal de sodio"

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  • Brompheniramine maleate

    CAS:
    <p>Brompheniramine maleate (Dimotane) is an antagonist against histamine H1 receptors.</p>
    Fórmula:C16H19BrN2·C4H4O4
    Pureza:99.80%
    Forma y color:Crystal Powder
    Peso molecular:435.31
  • Phenytoin

    CAS:
    <p>Phenytoin: a non-sedative hydantoin, antiepileptic with anticonvulsant effects, stabilizes neurons, prevents seizure spread, and relaxes muscles.</p>
    Fórmula:C15H12N2O2
    Pureza:99.95%
    Forma y color:Needles (Alcohol) Tasteless (Ntp 1992)
    Peso molecular:252.27
  • NaV1.7 inhibitor-1

    CAS:
    <p>NaV1.7 inhibitor-1, an efficacious inhibitor of voltage-gated sodium channel (NaV) 1.7 (IC50 of 0.6 nM for hNaV1.7).</p>
    Fórmula:C23H30FNO4S
    Pureza:99.89%
    Forma y color:Solid
    Peso molecular:435.55
  • Tocainide

    CAS:
    <p>Tocainide is a blocker of the sodium channel and used for the treatment of tinnitus.</p>
    Fórmula:C11H16N2O
    Pureza:99.84%
    Forma y color:Solid
    Peso molecular:192.26
  • Primidone

    CAS:
    <p>Primidone (NCI-C56360) is a potent anticonvulsant agent.</p>
    Fórmula:C12H14N2O2
    Pureza:99.91%
    Forma y color:Crystals (Ntp 1992)
    Peso molecular:218.25
  • Diphenidol hydrochloride

    CAS:
    <p>Diphenidol hydrochloride (Difenidol hydrochloride), a muscarinic antagonist, is employed as an anti-vertigo and as an antiemetic drug.</p>
    Fórmula:C21H28ClNO
    Pureza:99.15% - 99.33%
    Forma y color:Crystals Soluble In Methanol Water
    Peso molecular:345.91
  • Methocarbamol

    CAS:
    <p>Methocarbamol (AHR 85) is a centrally acting muscle relaxant whose mode of action has not been established.</p>
    Fórmula:C11H15NO5
    Pureza:99.96%
    Forma y color:Crystals From Benzene Solid
    Peso molecular:241.24
  • Bupivacaine hydrochloride

    CAS:
    <p>Bupivacaine hydrochloride (Vivacaine) is a long-lasting, amide local anesthetic that blocks sodium channels, inhibiting nerve impulses and sensation.</p>
    Fórmula:C18H28N2O·HCl
    Pureza:99.9% - >99.99%
    Forma y color:Solid
    Peso molecular:324.89
  • Butamben

    CAS:
    <p>Butamben (Butyl 4-aminobenzoate) is a long-duration local anesthetic used for the treatment of chronic pain.</p>
    Fórmula:C11H15NO2
    Pureza:99.43%
    Forma y color:Crystals From Alc Physical Description Yellow Powder Insoluble In Water (Ntp 1992)
    Peso molecular:193.24
  • Lidocaine

    CAS:
    <p>Lidocaine, an amide local anesthetic, reduces pain and inflammation by dampening ICAM-1, cytokines, and neutrophil influx.</p>
    Fórmula:C14H22N2O
    Pureza:99.95% - >99.99%
    Forma y color:Needles From Benzene Or Alcohol Solid
    Peso molecular:234.34
  • Lamotrigine

    CAS:
    <p>Lamotrigine (BW430C) is an Anti-epileptic Agent and Mood Stabilizer.</p>
    Fórmula:C9H7Cl2N5
    Pureza:99.76% - 99.95%
    Forma y color:White To Pale Cream-Colored Powder Crystals From Isopropanol Solid
    Peso molecular:256.09
  • Ropivacaine

    CAS:
    <p>Ropivacaine (LEA-103 HCl) is a local anaesthetic drug belonging to the amino amide group.</p>
    Fórmula:C17H26N2O
    Pureza:97.75% - >99.99%
    Forma y color:Solid
    Peso molecular:274.40
  • Tocainide hydrochloride

    CAS:
    <p>Tocainide hydrochloride (2-amino-n-(2,6-dimethylphenyl)propanamide hydrochloride) is a sodium channel blocker.</p>
    Fórmula:C11H17ClN2O
    Pureza:97%
    Forma y color:Solid
    Peso molecular:228.72
  • DSP-2230

    CAS:
    <p>DSP-2230 is a selective blocker of Nav1.7/Nav1.8.</p>
    Fórmula:C20H20F3N5O2
    Pureza:97.14%
    Forma y color:Solid
    Peso molecular:419.4
  • Eleclazine hydrochloride

    CAS:
    <p>Eleclazine hydrochloride (GS 6615 hydrochloride) is a novel inhibitor of late Na+ current (IC50: 0.7 uM).</p>
    Fórmula:C21H17ClF3N3O3
    Pureza:99.86%
    Forma y color:Solid
    Peso molecular:451.83
  • Disopyramide

    CAS:
    <p>Disopyramide, or Triombrin, a class I anti-arrhythmic with membrane-stabilizing effects, has heart depressant, anticholinergic, and anesthetic properties.</p>
    Fórmula:C21H29N3O
    Pureza:99.62%
    Forma y color:Solid
    Peso molecular:339.47
  • PF-04885614

    CAS:
    <p>PF-04885614 is a potent inhibitor of NaV1.8, has potential for neurological and neurodevelopmental diseases treatment.</p>
    Fórmula:C13H14F3N3O
    Pureza:98.02%
    Forma y color:Solid
    Peso molecular:285.27
  • QX-314 chloride

    CAS:
    <p>QX-314 chloride is a membrane-impermeable permanently charged blocker of sodium channel.</p>
    Fórmula:C16H27ClN2O
    Pureza:99.73%
    Forma y color:Solid
    Peso molecular:298.85
  • Articaine hydrochloride

    CAS:
    <p>Articaine hydrochloride (Hoe-045) is a thiophene-containing local anesthetic pharmacologically similar to MEPIVACAINE.</p>
    Fórmula:C13H21ClN2O3S
    Pureza:99.76%
    Forma y color:White Crystalline Powder
    Peso molecular:320.84
  • Vinpocetine

    CAS:
    <p>Vinpocetine (RGH-4405) is a selective inhibitor of cyclic GMP phosphodiesterase (PDE).</p>
    Fórmula:C22H26N2O2
    Pureza:99.85% - 99.98%
    Forma y color:White Crystalline Solid
    Peso molecular:350.45