AhR
El Receptor de Hidrocarburos Aromáticos (AhR) es un factor de transcripción activado por ligandos que desempeña un papel crítico en la regulación de las respuestas biológicas a contaminantes ambientales, como las dioxinas. AhR también está involucrado en el metabolismo de xenobióticos y en la regulación de las respuestas inmunitarias, la proliferación y la diferenciación celular. La desregulación de la señalización de AhR está vinculada a diversas enfermedades, incluido el cáncer y los trastornos autoinmunes. En CymitQuimica, ofrecemos una gama de inhibidores de AhR para apoyar su investigación en toxicología, biología del cáncer e inmunología.
Se han encontrado 41 productos de "AhR"
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GNF351
CAS:<p>GNF351: Full AHR antagonist, inhibits DRE-dependent/independent activity, low toxicity, binds AHR (IC50: 62 nM).</p>Fórmula:C24H25N7Pureza:98.43%Forma y color:SolidPeso molecular:411.5Diosmin
CAS:<p>Diosmin (Venosmine) is a bioflavonoid that strengthens vascular walls.</p>Fórmula:C28H32O15Pureza:97.90%Forma y color:Greyish-Yellow Or Light Yellow Hygroscopic PowderPeso molecular:608.54Mexiletine hydrochloride
CAS:<p>Mexiletine hydrochloride is a lidocaine-like antiarrhythmic (Class IB) and anesthetic, stabilizing heartbeats by inhibiting sodium in cardiac cells.</p>Fórmula:C11H18ClNOPureza:99.88%Forma y color:White To Off-White SolidPeso molecular:215.72BAY 2416964
CAS:<p>BAY 2416964 is a small molecule inhibitor that selectively targets aromatic receptor (AhR) and is commonly used in tumor research. Cost-effective and quality-assured.</p>Fórmula:C18H18ClN5O3Pureza:99.15% - 99.85%Forma y color:SolidPeso molecular:387.82Leflunomide
CAS:<p>Leflunomide (HWA486) is an immunomodulatory agent used in the therapy of rheumatoid arthritis and psoriatic arthritis.</p>Fórmula:C12H9F3N2O2Pureza:99.52% - 99.96%Forma y color:Off White Crystalline SolidPeso molecular:270.21StemRegenin 1 Hydrochloride
CAS:<p>StemRegenin 1 Hydrochloride is an AhR antagonist (IC₅₀ = 127 nM) that inhibits RANKL-induced osteoclast generation and differentiation.</p>Fórmula:C24H24ClN5OSPureza:99.94%Forma y color:SolidPeso molecular:466KYN-101
CAS:<p>KYN-101 is an and aryl hydrocarbon receptor (AHR) inhibitor with anticancer activity. KYN-101 is used for the study of breast cancer and acute myeloid leukemia.</p>Fórmula:C22H19FN6Pureza:98.35%Forma y color:SolidPeso molecular:386.43MeBIO
CAS:<p>MeBIO is an agonist of aryl hydrocarbon receptor, with IC50 of 44 and 55 μM for GSK-3 and CDK1/CyclinB, respectively. MeBIO does not affect GSK-3β.</p>Fórmula:C17H12BrN3O2Pureza:99.64%Forma y color:SolidPeso molecular:370.2WAY-605471
CAS:<p>WAY-605471 is a AHR antagonist with IC50 of 0.5 - 1 μM.</p>Fórmula:C14H15NO3S2Pureza:99.62%Forma y color:SolidPeso molecular:309.4AHR Inhibitor I-103
CAS:<p>AHR Inhibitor I-103 is an aryl hydrocarbon receptor (AHR) inhibitor with anticancer activity used in the study of breast cancer and acute myeloid leukemia.</p>Fórmula:C21H17FN6Pureza:98.70%Forma y color:SoildPeso molecular:372.43',4'-Dimethoxyflavone
CAS:<p>3',4'-Dimethoxyflavone is a standard compound of flavonoids with numerous medicinal activities.</p>Fórmula:C17H14O4Pureza:98.05%Forma y color:SolidPeso molecular:282.29L-Kynurenine
CAS:<p>L-Kynurenine ((S)-Kynurenine)) is an endogenous agonist of aryl hydrocarbon receptor (AHR) ,inhibits allogeneic T cell proliferation. High-Quality, Low-Cost!</p>Fórmula:C10H12N2O3Pureza:98.44% - 99.91%Forma y color:Light Yellow CrystallinePeso molecular:208.21YL-109
CAS:<p>YL-109, a novel anticancer agent, can inhibit breast Y cell growth and invasiveness in vitro and in vivo.</p>Fórmula:C14H11NO2SPureza:99.77% - ≥95%Forma y color:SolidPeso molecular:257.31ITE
CAS:<p>ITE is a potent endogenous agonist of aryl hydrocarbon receptor (AhR) (Ki : 3 nM), has immunosuppressive activity.</p>Fórmula:C14H10N2O3SPureza:97.91% - 99.14%Forma y color:SolidPeso molecular:286.31PDM11
CAS:<p>PDM11 (1-[2-(4-Chloro-phenyl)-vinyl]-3,5-diMeth) is an antagonist of aryl hydrocarbon receptor (AhR)</p>Fórmula:C16H15ClO2Pureza:99.88%Forma y color:SolidPeso molecular:274.74Benzyl butyl phthalate
CAS:<p>Benzyl butyl phthalate (1,2-benzenedicarboxylic acid) is used as a plasticizer for PVC.</p>Fórmula:C19H20O4Pureza:99.02%Forma y color:Colourless Liquid Oily LiquidPeso molecular:312.36Indole-3-pyruvic acid
CAS:<p>Indole-3-pyruvic acid is a precursor for the plant growth hormone indole-3-acetic acid.</p>Fórmula:C11H9NO3Pureza:98.89% - 99.21%Forma y color:Off White CrystalsPeso molecular:203.19Tapinarof
CAS:<p>Tapinarof (Benvitimod) is targeted as a topical cream treatment for psoriasis, a chronic autoimmune skin disease.</p>Fórmula:C17H18O2Pureza:99.64% - >99.99%Forma y color:SolidPeso molecular:254.32PD98059
CAS:<p>PD98059 is an MEK inhibitor that inhibits MEK1 and MEK2 (IC50=2/50 μM) and is non-ATP-competitive.</p>Fórmula:C16H13NO3Pureza:98.63% - >99.99%Forma y color:Yellow SolidPeso molecular:267.28Carbidopa
CAS:<p>Carbidopa (Lodosyn) is an aromatic-L-amino-acid decarboxylase inhibitor (IC50: 29±2 μM).</p>Fórmula:C10H14N2O4Pureza:98.01% - ≥98%Forma y color:SolidPeso molecular:226.23
