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Proteasas / Proteasoma

Proteasas / Proteasoma

Los inhibidores de proteasas y proteasomas son compuestos que bloquean la actividad de las proteasas y del proteasoma, que están involucrados en la degradación y renovación de proteínas. Estos inhibidores son vitales para estudiar la regulación de la homeostasis proteica, el control del ciclo celular y la apoptosis. Los inhibidores de proteasas y proteasomas también se utilizan en el tratamiento de enfermedades como el cáncer, donde la degradación anormal de proteínas desempeña un papel en la progresión de la enfermedad. Al inhibir las proteasas o el proteasoma, estos compuestos pueden inducir la muerte celular en células cancerosas y son herramientas esenciales tanto en la investigación básica como en el desarrollo terapéutico. En CymitQuimica, ofrecemos una amplia gama de inhibidores de proteasas y proteasomas de alta calidad para apoyar su investigación en bioquímica, biología celular y desarrollo de fármacos.

Subcategorías de "Proteasas / Proteasoma"

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Se han encontrado 1039 productos de "Proteasas / Proteasoma"

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  • Azo-Resveratrol

    CAS:
    <p>Azo-Resveratrol is an analog of Resveratrol used as a potent tyrosinase inhibitor.</p>
    Fórmula:C12H10N2O3
    Forma y color:Solid
    Peso molecular:230.22
  • Sortin1

    CAS:
    Sortin1, a chemical genetic-hit compound, specifically induces mislocalization of both soluble and membrane-associated vacuolar markers in plants and yeast.
    Fórmula:C26H19NO6
    Pureza:98%
    Forma y color:Solid
    Peso molecular:441.43
  • MDK7677

    CAS:
    <p>MDK7677 is a selective inhibitor of cathepsin B endopeptidase and exopeptidase activities.</p>
    Fórmula:C12H10N4O3
    Forma y color:Solid
    Peso molecular:258.23
  • Furaprofen

    CAS:
    <p>Furaprofen is an HCV inhibitor with anti-inflammatory activity that inhibits carrageenan-induced paw edema in rats.</p>
    Fórmula:C17H14O3
    Pureza:98.49% - 99.52%
    Forma y color:Solid
    Peso molecular:266.29
  • (3S,4S)-A2-32-01


    <p>(3S,4S)-A2-32-01, a less active (S,S)-enantiomer of A2-32-01. A2-32-01 is a potent caseinolytic protein proteases (ClpP) inhibitor .</p>
    Fórmula:C19H27NO2
    Forma y color:Solid
    Peso molecular:301.42
  • GEMSA

    CAS:
    <p>GEMSA is a potent inhibitor of enkephalin convertase ( K i =8.8 nM) with analgesic effect[1].</p>
    Fórmula:C7H13N3O4S
    Forma y color:Solid
    Peso molecular:235.26
  • MMP-1-IN-1


    <p>MMP-1-IN-1 is a highly potent MMP-1 inhibitor with an IC 50 of 0.034 μM .</p>
    Fórmula:C14H17ClN2O3
    Forma y color:Solid
    Peso molecular:296.75
  • Gemigliptin Tartrate(911637-19-9 free base)

    CAS:
    <p>Gemigliptin Tartrate (LC15-0444 tartrate) is a highly selective, reversible and competitive inhibitor of dipeptidyl peptidase-4 (DPP-4).</p>
    Fórmula:C22H25F8N5O8
    Pureza:>99.99%
    Forma y color:Solid
    Peso molecular:639.45
  • AK 275

    CAS:
    <p>AK 275 is a calpain inhibitor that prevents degradation of cytoskeletal and myelin proteins in spinal cord in vitro.</p>
    Fórmula:C20H31N3O4
    Forma y color:Solid
    Peso molecular:377.48
  • AZD-9684

    CAS:
    <p>AZD-9684, a carboxypeptidase U inhibitor, is used potentially for the prevention of thrombosis.</p>
    Fórmula:C10H14N2O2S
    Forma y color:Solid
    Peso molecular:226.3
  • SAP2-IN-1

    CAS:
    <p>SAP2-IN-1 inhibits secreted aspartate protease 2 (IC50: 0.92 μM), doesn't work in vitro, and helps research infections.</p>
    Fórmula:C34H29NO7
    Forma y color:Solid
    Peso molecular:563.6
  • ITX-4520

    CAS:
    <p>ITX-4520 novel highly potent, orally bioavailable inhibitor of hepatitis C virus (HCV) entry.</p>
    Fórmula:C24H23F2N3OS
    Forma y color:Solid
    Peso molecular:439.52
  • NAAA-IN-2

    CAS:
    <p>NAAA-IN-2, a selective inhibitor with 50 nM IC50, targets NAAA, an enzyme hydrolyzing PEA/OEA, and may aid inflammation and pain studies.</p>
    Fórmula:C11H13N3O2S
    Forma y color:Solid
    Peso molecular:251.3
  • L 722151

    CAS:
    <p>L 722151 is an FXIIIa inhibitor.</p>
    Fórmula:C8H9ClN2O5S3
    Pureza:98%
    Forma y color:Solid
    Peso molecular:344.82
  • TAPI-0

    CAS:
    <p>TAPI-0 is a matrix metalloprotease (MMP) and TACE inhibitor.</p>
    Fórmula:C24H32N4O5
    Forma y color:Solid
    Peso molecular:456.53
  • Chymase-IN-1

    CAS:
    <p>Chymase-IN-1 is a selective, orally active inhibitor of human mast cell chymase (IC50: 29 nM).</p>
    Fórmula:C20H15ClNO4PS
    Pureza:99.17%
    Forma y color:Solid
    Peso molecular:431.83
  • Tyrosinase-IN-10

    CAS:
    <p>Tyrosinase-IN-10 serves as a partially competitive inhibitor of tyrosinase, demonstrating an inhibition concentration (IC50) value of 1.6 μM against the enzyme'</p>
    Fórmula:C16H12O4
    Forma y color:Solid
    Peso molecular:268.26
  • ADAMTS-5-IN-2

    CAS:
    <p>ADAMTS-5-IN-2 is a potent inhibitor of ADAMTS-5, exhibiting an IC50 of 0.71 µM, and holds potential for osteoarthritis research.</p>
    Fórmula:C17H15N3OS
    Forma y color:Solid
    Peso molecular:309.39
  • Calpain-2-IN-1

    CAS:
    <p>Calpain-2-IN-1 is a selective calpain-2 inhibitor that prolongs ERK activation and thus enhances learning and memory.</p>
    Fórmula:C28H37N3O7
    Forma y color:Solid
    Peso molecular:527.61
  • Safironil

    CAS:
    <p>Safironil, a novel antifibrotic, competitively inhibits collagen synthesis and modulates fibrosis, impacting type I/III collagen levels.</p>
    Fórmula:C15H23N3O4
    Pureza:99.83%
    Forma y color:Solid
    Peso molecular:309.36
  • BR351

    CAS:
    <p>BR351 is a brain penetrant MMP inhibitor (IC50s: 4, 2, 11, 50 nM for MMP2, MMP8, MMP9 and MMP13).</p>
    Fórmula:C20H25FN2O5S
    Pureza:98%
    Forma y color:Solid
    Peso molecular:424.49
  • HCV-IN-35

    CAS:
    <p>HCV-IN-35 is a potent inhibitor of HCV and shows potential for infectious disease research.</p>
    Fórmula:C30H36ClN5
    Forma y color:Solid
    Peso molecular:502.09
  • Calpain Inhibitor XI

    CAS:
    <p>Calpain Inhibitor XI, a reversible covalent inhibitor of calpain-1, is utilized in the research of neurodegenerative disorders.</p>
    Fórmula:C26H40N4O6
    Forma y color:Solid
    Peso molecular:504.62
  • AM 4299 B

    CAS:
    <p>AM 4299 B is a novel inhibitor of a thiol protease.</p>
    Fórmula:C16H27N3O7
    Pureza:98%
    Forma y color:Solid
    Peso molecular:373.4
  • MDL 27399

    CAS:
    <p>MDL 27399 suppresses human neutrophil cathepsin G.</p>
    Fórmula:C26H36N4O8
    Forma y color:Solid
    Peso molecular:532.59
  • CAA0225

    CAS:
    <p>CAA0225 is a selective inhibitor of cathepsin L. CAA0225 is a probe for autophagic proteolysis.</p>
    Fórmula:C28H29N3O5
    Forma y color:Solid
    Peso molecular:487.55
  • Immunoproteasome inhibitor 1

    CAS:
    <p>Potent, reversible immunoproteasome inhibitor; Ki: β5c 1.18 μM, β1i 0.27 μM, β5i 1.91 μM; potential in treating cancer.</p>
    Fórmula:C20H26N2O4
    Forma y color:Solid
    Peso molecular:358.43
  • α-Glucosidase-IN-5

    CAS:
    <p>α-Glucosidase-IN-5 (compound 8) is isolated from a twig extract of Polyalthia cinnamomea which is a potent α-glucosidase inhibitor with an IC50 of 57.9 µM.</p>
    Fórmula:C15H13NO3
    Forma y color:Solid
    Peso molecular:255.27
  • JO146

    CAS:
    <p>JO146为针对沙眼衣原体高温需要蛋白A(CtHtrA)的蛋白酶抑制剂,其对CtHtrA和人中性粒细胞弹性蛋白酶(HNE)的IC50值分别为21.86 μM和1.15 μM,可应用于细菌感染的抑制。</p>
    Fórmula:C31H44N3O7P
    Forma y color:Solid
    Peso molecular:601.67
  • L-873724

    CAS:
    <p>L-873724: Selective, reversible cathepsin K inhibitor; IC50s—cat K: 0.2 nM, cat S: 178 nM, cat L: 264 nM, cat B: 5239 nM; inhibits bone resorption.</p>
    Fórmula:C23H26F3N3O3S
    Pureza:98%
    Forma y color:Solid
    Peso molecular:481.53
  • (R)-ND-336

    CAS:
    <p>(R)-ND-336: potent, selective MMP-9 inhibitor (K i = 19 nM); inhibits MMP-2 (127 nM), MMP-14 (119 nM); studied for diabetic foot ulcers.</p>
    Fórmula:C16H18ClNO3S2
    Forma y color:Solid
    Peso molecular:371.89
  • Adafosbuvir PM

    CAS:
    <p>Adafosbuvir PM (AL-335 PM) is a small molecule NS5B inhibitor that can be used to study chronic hepatitis C.</p>
    Fórmula:C10H13FN2O6
    Pureza:97.08%
    Forma y color:Solid
    Peso molecular:276.22
  • OM-189

    CAS:
    <p>OM-189 is a selective inhibitor of synthetic thrombin.</p>
    Fórmula:C24H36N6O3S
    Pureza:98%
    Forma y color:Solid
    Peso molecular:488.65
  • MMP-2/9-IN-1

    CAS:
    <p>MMP-2/9-IN-1 (Compound 4a) is a potent dual inhibitor of MMP-2 (IC50: 56 nM) and MMP-9 (IC50: 38 nM). leading to DNA fragmentation.</p>
    Fórmula:C14H16IN7S
    Forma y color:Solid
    Peso molecular:441.29
  • GLS1 Inhibitor-3

    CAS:
    <p>GLS1 Inhibitor-3 (compound C147) is a potent inhibitor of GLS1 (IC50: 27.98 nM) and exhibits anti-proliferative effects.</p>
    Fórmula:C30H32N10O2S
    Forma y color:Solid
    Peso molecular:596.71
  • CA 074

    CAS:
    <p>CA 074 is a potent inhibitor of cathepsin B with a Ki value of 2 to 5 nM.CA 074 inhibits ischemic hippocampal neuronal death in primates and attenuates</p>
    Fórmula:C18H29N3O6
    Pureza:97.80%
    Forma y color:Solid
    Peso molecular:383.44
  • XMU-MP-2

    CAS:
    <p>XMU-MP-2 is a potent and selective protease inhibitor with anticancer activity that inhibits the growth of oncogenic BRK-driven tumors in a mouse xenograft</p>
    Fórmula:C32H33F3N8O2
    Pureza:99.29%
    Forma y color:Solid
    Peso molecular:618.65
  • Tyrosinase-IN-1

    CAS:
    <p>Tyrosinase-IN-1: potent inhibitor for skin-whitening &amp; food preservation with uses in cosmetics &amp; medicine.</p>
    Fórmula:C10H9N3O2S2
    Forma y color:Solid
    Peso molecular:267.33
  • HCV-IN-36

    CAS:
    <p>HCV-IN-36: oral HCV inhibitor, EC50 0.016 μM, CC50 8.78 μM, potent antiviral.</p>
    Fórmula:C30H36ClN5
    Forma y color:Solid
    Peso molecular:502.09
  • BMS-363131

    CAS:
    <p>BMS-363131 (BMS363131) is a potent and selective trypsin inhibitor with an IC50 value of &lt;1.7 nM.</p>
    Fórmula:C28H40N6O5
    Pureza:97.99%
    Forma y color:Solid
    Peso molecular:540.65
  • 2',5-Difluoro-2'-deoxycytidine

    CAS:
    <p>2',5-Difluoro-2'-deoxycytidine has potent anti-HCV activity and toxicity to rRNA.</p>
    Fórmula:C9H11F2N3O4
    Pureza:98%
    Forma y color:Solid
    Peso molecular:263.2
  • BRD-8899

    CAS:
    <p>BRD-8899 is a STK33 inhibitor, with an IC 50 of 11 nM [1].</p>
    Fórmula:C17H22N4O3S
    Forma y color:Solid
    Peso molecular:362.45
  • Tyrosinase-IN-5

    CAS:
    <p>Tyrosinase-IN-5 (16c) inhibits tyrosinase with 0.02 μM IC50, reduces melanogenesis, and is low-toxicity.</p>
    Fórmula:C18H13N3O6
    Forma y color:Solid
    Peso molecular:367.31
  • Elasnin

    CAS:
    <p>Elasnin is a reversible inhibitor of elastase for human granulocyte and pancreatic enzymes with IC50 values of 1.3 and 30 µg/ml, respectively.</p>
    Fórmula:C24H40O4
    Forma y color:Solid
    Peso molecular:392.57
  • ASPER-29

    CAS:
    <p>ASPER-29, an Asperphenamate analog, inhibits cathepsins L/S with IC50s of 6.03/5.02 μM, useful in cancer migration/invasion research.</p>
    Fórmula:C31H29BrN2O5S
    Forma y color:Solid
    Peso molecular:621.54
  • Gü1303

    CAS:
    <p>Gü1303 is a highly potent and reversible inhibitor of Cathepsin K (CatK), with a Ki value of 0.91 nM for mature CatK (mCatK).</p>
    Fórmula:C20H22N4O3
    Forma y color:Solid
    Peso molecular:366.41
  • CAY10704

    CAS:
    <p>CAY10704: Potent HCV inhibitor, EC50=17 nM, low cytotoxicity, good in mice, liver-targeted, not hepatotoxic, weak against dengue.</p>
    Fórmula:C18H20Cl2N2
    Forma y color:Solid
    Peso molecular:335.27
  • DPP-4-IN-1

    CAS:
    <p>DPP-4-IN-1 inhibits DPP-4 with 49 nM IC50, ideal for diabetes study, akin to Alogliptin.</p>
    Fórmula:C19H19ClN6
    Forma y color:Solid
    Peso molecular:366.85
  • AA10 TG2 inhibitor

    CAS:
    <p>AA10 is an irreversible inhibitor of transglutaminase 2 (TG2).</p>
    Fórmula:C32H36N4O5
    Forma y color:Solid
    Peso molecular:556.65
  • ABT-770

    CAS:
    <p>ABT-770: an orally potent and selective MMP inhibitor, shown to reduce tumor growth in animal models.</p>
    Fórmula:C22H22F3N3O6
    Forma y color:Solid
    Peso molecular:481.42
  • BAY8040

    CAS:
    <p>BAY8040 is a potent selective human neutrophilic elastase inhibitor with excellent potency and selectivity with promising pharmacokinetic characteristics.</p>
    Fórmula:C21H16F3N5O2
    Forma y color:Solid
    Peso molecular:427.38
  • PK44 phosphate

    CAS:
    <p>PK44 phosphate is a potent inhibitor of dipeptidyl peptidase IV (DPP-IV) (IC50: 15.8 nM).</p>
    Fórmula:C17H19F5N7O5P
    Forma y color:Solid
    Peso molecular:527.349
  • VEL-0230

    CAS:
    <p>VEL-0230 (NC-2300) is a cathespin K inhibitor boosting bone growth and reducing loss, targeting bone diseases and developed by Velcura Therapeutics.</p>
    Fórmula:C14H24NNaO5
    Forma y color:Solid
    Peso molecular:309.33
  • BrBzGCp2

    CAS:
    <p>BrBzGCp2 (p BrBzGSH(Cp)2) is a GLO1 inhibitor with antitumor activities, relieving anxiety, and is useful in researching neurological disorders.</p>
    Fórmula:C27H38BrN3O6S
    Pureza:98.68% - 98.68%
    Forma y color:Solid
    Peso molecular:612.58
  • ACH-806

    CAS:
    <p>ACH-806 is an NS4A antagonist. It can inhibit Hepatitis C Virus (HCV) replication with an EC50 of 14 nM.</p>
    Fórmula:C19H20F3N3O2S
    Pureza:98%
    Forma y color:Solid
    Peso molecular:411.44
  • Antiviral agent 30

    CAS:
    <p>Antiviral Agent 30 (Example 118) is an active compound against HCV and RSV with an inhibitory concentration (IC 50) of greater than 25μM [1].</p>
    Fórmula:C21H32N2O3S
    Forma y color:Solid
    Peso molecular:392.56
  • Alicapistat

    CAS:
    <p>Alicapistat (ABT-957) is a human calpains 1 and 2 inhibitor. It can potentially be used to treat Alzheimer's disease (AD).</p>
    Fórmula:C25H27N3O4
    Pureza:98%
    Forma y color:Solid
    Peso molecular:433.5
  • A-933548

    CAS:
    <p>A-933548: potent calpain inhibitor, selective vs. cathepsins, stable, effective in cell assays.</p>
    Fórmula:C25H21N5O3
    Pureza:98%
    Forma y color:Solid
    Peso molecular:439.47
  • Tyrosinase-IN-6

    CAS:
    <p>Tyrosinase-IN-6 (4B) is a potent tyrosinase inhibitor (IC50=3.80 μM) with good antioxidant activity.</p>
    Fórmula:C24H31N3O2
    Forma y color:Solid
    Peso molecular:393.52
  • SP-Chymostatin B

    CAS:
    <p>SP-Chymostatin B inhibits proteases like chymotrypsin and papain; less effective on human elastase; works at 100-200 μg/ml.</p>
    Fórmula:C30H41N7O6
    Pureza:98%
    Forma y color:Solid
    Peso molecular:595.69
  • Anticancer agent 82

    CAS:
    <p>Anticancer agent 82, a FiVe1 derivative, selectively targets VIM in cancer cells to disrupt mitosis, with improved oral bioavailability.</p>
    Fórmula:C19H18Cl2N4O
    Forma y color:Solid
    Peso molecular:389.28
  • DPP-IV-IN-1

    CAS:
    <p>DPP-IV-IN-1 is an effective inhibitor of dipeptidyl peptidase IV (DPP-IV), a serine protease (IC50: 4.6 nM).</p>
    Fórmula:C11H18FN3O2
    Pureza:98%
    Forma y color:Solid
    Peso molecular:243.28
  • Tyrosinase-IN-3

    CAS:
    <p>Tyrosinase-IN-3 inhibits melanin production; potential for skin whitening and food preservation.</p>
    Fórmula:C21H23NO5
    Forma y color:Solid
    Peso molecular:369.41
  • MK-2048

    CAS:
    <p>MK-2048 is a potent inhibitor of integrase (IN) and INR263K with IC50 of 2.6 nM and 1.5 nM, respectively.</p>
    Fórmula:C21H21ClFN5O4
    Pureza:98%
    Forma y color:Solid
    Peso molecular:461.87
  • Gü2602

    CAS:
    <p>Gü2602 inhibits the cathepsin K zymogen autocatalytic activation that is a potent, reversible inhibitor of cathepsin K (CatK) with a Ki of 0.013 nM for mature</p>
    Fórmula:C16H22N4O3
    Forma y color:Solid
    Peso molecular:318.37
  • AZD5248

    CAS:
    <p>AZD-5248 is a potent, selective, first generation, oral inhibitor of dipeptidyl peptidase 1 (DPP1).</p>
    Fórmula:C22H22N4O2
    Forma y color:Solid
    Peso molecular:374.44
  • HCV-IN-33

    CAS:
    <p>HCV-IN-33 (Compound (S)-3i) is an inhibitor of HCV entry.</p>
    Fórmula:C31H36ClN5
    Forma y color:Solid
    Peso molecular:514.1
  • JNJ-10329670

    CAS:
    <p>JNJ 10329670 is a highly potent (Ki of approximately 30 nM), nonpeptidic, noncovalent inhibitor of human cathepsin S with immunosuppressive activity.</p>
    Fórmula:C30H34ClF3N6O3S
    Forma y color:Solid
    Peso molecular:651.14
  • Gosogliptin

    CAS:
    <p>Gosogliptin is a potent, orally active, highly selective, reversible and competitive inhibitor of DPP-4, increasing the level of intestinal GLP-1 and GIP.</p>
    Fórmula:C17H24F2N6O
    Pureza:99.74%
    Forma y color:Solid
    Peso molecular:366.41
  • (Rac)-Tanomastat

    CAS:
    <p>Tanomastat (BAY 12-9566) is an oral biphenyl MMP inhibitor; blocks MMP-2, -3, -9, -13, with anti-invasive and anti-metastatic properties.</p>
    Fórmula:C23H19ClO3S
    Forma y color:Solid
    Peso molecular:410.91
  • GSK2793660 HCl

    CAS:
    <p>GSK2793660 is a irreversible covalent α,β-unsaturated amide based DPP1 inhibitor.</p>
    Fórmula:C22H32ClN3O3
    Forma y color:Solid
    Peso molecular:421.96
  • Cysteine Protease inhibitor

    CAS:
    <p>Cysteine protease inhibitors are inhibitors of cysteine proteases. Target: Cysteine Protease</p>
    Fórmula:C18H14N4O
    Pureza:98%
    Forma y color:Solid
    Peso molecular:302.33
  • Cysteine Protease inhibitor hydrochloride

    CAS:
    <p>Cysteine Protease inhibitor hydrochloride is a cysteine protease inhibitor.</p>
    Fórmula:C18H15ClN4O
    Pureza:98%
    Forma y color:Solid
    Peso molecular:338.79
  • VA4 TG2 inhibitor

    CAS:
    <p>VA4 is a novel irreversible TG2 transamidase site-specific inhibitor.</p>
    Fórmula:C33H41N5O6S
    Forma y color:Solid
    Peso molecular:635.77
  • Kallikrein 5-IN-2

    CAS:
    <p>Kallikrein 5-IN-2 inhibits KLK5 (pIC50=7.1); may normalize skin shedding, lessen inflammation &amp; itching.</p>
    Fórmula:C23H22N6O
    Forma y color:Solid
    Peso molecular:398.46
  • Tec-IN-21

    CAS:
    <p>Tec-IN-21 is an inhibitor of Tec kinase, it also blocks unconventional secretion of fibroblast growth factor 2 (FGF2).</p>
    Fórmula:C16H15ClN4O2S
    Pureza:98%
    Forma y color:Solid
    Peso molecular:362.83
  • Sheng Gelieting

    CAS:
    <p>CGT-8012 inhibits DP-IV enzyme, aiding type II diabetes research, with an IC50 of 87 nM.</p>
    Fórmula:C17H16F6N4O
    Forma y color:Solid
    Peso molecular:406.33
  • CP-471474

    CAS:
    <p>MMP inhibitor with IC50: MMP-2 (0.7 nM), MMP-13 (0.9 nM), MMP-9 (13 nM), MMP-3 (16 nM), MMP-1 (1170 nM); reduces heart dilation post-infarct.</p>
    Fórmula:C16H17FN2O5S
    Pureza:98%
    Forma y color:Solid
    Peso molecular:368.38
  • SJA6017

    CAS:
    <p>SJA6017: inhibits calpain-1/2, cathepsins B/L; prevents apoptosis, protects spinal cord, boosts function. IC50s: 7.5-78 nM.</p>
    Fórmula:C17H25FN2O4S
    Pureza:98%
    Forma y color:Solid
    Peso molecular:372.45
  • Elastase-IN-1

    CAS:
    <p>Elastase-IN-1 (Compound Q11) is a non-toxic elastase inhibitor with an IC 50 of 0.897 μM [1].</p>
    Fórmula:C17H12N4O3
    Forma y color:Solid
    Peso molecular:320.3
  • SQ 32602

    CAS:
    <p>SQ 32602 is a cathepsin E inhibitor.</p>
    Fórmula:C32H52N3O7P
    Forma y color:Solid
    Peso molecular:621.74
  • Tyrosinase-IN-8


    <p>Tyrosinase-IN-8, a potent inhibitor of tyrosinase, demonstrates an inhibitory concentration (IC 50) value of 1.6 µM and exhibits low cytotoxicity while</p>
    Fórmula:C16H12O4
    Forma y color:Solid
    Peso molecular:268.26
  • DPP-4-IN-2

    CAS:
    <p>DPP-4-IN-2, analog of Alogliptin with 79 nM IC50, is a research tool for diabetes.</p>
    Fórmula:C18H18N6O
    Forma y color:Solid
    Peso molecular:334.38
  • Cysteine protease inhibitor-2

    CAS:
    <p>Cysteine protease inhibitor from US20070032499A1; halts DCT116 at 6.5μM, PC3 at 4.4μM.</p>
    Fórmula:C13H5N5O
    Pureza:98%
    Forma y color:Solid
    Peso molecular:247.21
  • HIV-1 integrase inhibitor 8

    CAS:
    <p>HIV-1 integrase inhibitor 8 is an inhibitor of HIV-1 integrase. Integration is a required step in HIV replication [1].</p>
    Fórmula:C21H24O2
    Pureza:98.91%
    Forma y color:Solid
    Peso molecular:308.41
  • Atevirdine

    CAS:
    <p>Atevirdine is an HIV-1 reverse transcriptase inhibitor with antiviral activity for the study of the AIDS dementia complex (ADC).</p>
    Fórmula:C21H25N5O2
    Pureza:98.20%
    Forma y color:Solid
    Peso molecular:379.46
  • L 756423

    CAS:
    <p>L756423 is a potent, selective HIV protease inhibitor (Ki=0.049 nM), effective against HIV spread in MT25 lymphocytes at 0.1-0.5 nM, useful for AIDS research.</p>
    Fórmula:C39H48N4O5
    Pureza:99.34% - 99.88%
    Forma y color:Solid
    Peso molecular:652.82
  • VRK-IN-1

    CAS:
    VRK-IN-1 is a potent and selective inhibitor of cowpox-associated kinase 1 (VRK1), which can be used in the study of neurological disorders.
    Fórmula:C18H11F4NO2
    Pureza:99.18% - 99.25%
    Forma y color:Solid
    Peso molecular:349.28
  • CPA inhibitor

    CAS:
    <p>CPA inhibitor (Carboxypeptidase inhibitor) is a potent carboxypeptidase A (CPA) inhibitor with a Ki of 0.32 μM.</p>
    Fórmula:C18H19NO4
    Pureza:99.94%
    Forma y color:Solid
    Peso molecular:313.35
  • Uprifosbuvir

    CAS:
    Uprifosbuvir is an inhibitor of uridine nucleotide analog HCV NS5B polymerase.
    Fórmula:C22H29ClN3O9P
    Pureza:99.73% - >99.99%
    Forma y color:Solid
    Peso molecular:545.91
  • Tyrosinase-IN-2

    CAS:
    <p>Tyrosinase-IN-2, a potent tyrosinase inhibitor, may help in skin lightening and food preservation research.</p>
    Fórmula:C8H8N4O2S
    Pureza:99.78%
    Forma y color:Solid
    Peso molecular:224.24
  • AGPS-IN-2i

    CAS:
    AGPS-IN-2i inhibits alkylglycerol phosphate synthase, affecting ether lipid metabolism and reducing cancer cell migration and proliferation.
    Fórmula:C18H17F2N3O2
    Pureza:98.92%
    Forma y color:Solid
    Peso molecular:345.34
  • Gemigliptin

    CAS:
    <p>Gemigliptin (LC15-0444) is a potent dipeptidyl peptidase-4 (DPP-4) inhibitor(KD : 7.25 nM.)</p>
    Fórmula:C18H19F8N5O2
    Pureza:99.72%
    Forma y color:Solid
    Peso molecular:489.36
  • TG2-IN-3h

    CAS:
    <p>TG2-IN-3h is a highly selective, potent, cell-permeable fluorescent irreversible tissue transglutaminase (tg2) inhibitor</p>
    Fórmula:C21H26N4O4S
    Pureza:99.34% - 99.76%
    Forma y color:Solid
    Peso molecular:430.52
  • 2'-C-Methyladenosine

    CAS:
    <p>2'-C-Methyladenosine from C. renalis inhibits HCV, NS5B RNA synthesis (IC50: 0.3, 1.9µM), and LRV1 in L. guyanensis, L. braziliensis.</p>
    Fórmula:C11H15N5O4
    Pureza:99.85%
    Forma y color:Solid
    Peso molecular:281.27
  • Isatoribine

    CAS:
    <p>Isatoribine(ANA245) free base is a potent TLR7 receptor agonist with anti-hepatitis C virus infection activity for the study of HCV infection.</p>
    Fórmula:C10H12N4O6S
    Pureza:98.99% - 99.75%
    Forma y color:Solid
    Peso molecular:316.29
  • P32/98 hemifumarate

    CAS:
    <p>P32/98 hemifumarate is a DPP4 inhibitor with hypoglycemic properties and is used in the study of type 2 diabetes.</p>
    Fórmula:C22H40N4O6S2
    Pureza:99.46%
    Forma y color:Solid
    Peso molecular:520.71
  • BILB-1941

    CAS:
    <p>BILB-1941 (BILB-1941ZW) is an inhibitor of HCV NS5B polymerase and can be used in studies about HCV infection.</p>
    Fórmula:C34H34N4O4
    Pureza:99.51% - 99.65%
    Forma y color:Solid
    Peso molecular:562.66
  • TS-021

    CAS:
    <p>TS-021 is a selective dipeptidyl peptidase 4 (DPP-4) inhibitor with antidiabetic activity for the study of type 2 diabetes.</p>
    Fórmula:C17H24FN3O5S
    Pureza:>99.99% - >99.99%
    Forma y color:Solid
    Peso molecular:401.45
  • GSK-364735

    CAS:
    <p>GSK-364735 is an HIV-1 IN inhibitor.</p>
    Fórmula:C19H18FN3O4
    Pureza:97.73%
    Forma y color:Solid
    Peso molecular:371.36