Proteasas / Proteasoma
Los inhibidores de proteasas y proteasomas son compuestos que bloquean la actividad de las proteasas y del proteasoma, que están involucrados en la degradación y renovación de proteínas. Estos inhibidores son vitales para estudiar la regulación de la homeostasis proteica, el control del ciclo celular y la apoptosis. Los inhibidores de proteasas y proteasomas también se utilizan en el tratamiento de enfermedades como el cáncer, donde la degradación anormal de proteínas desempeña un papel en la progresión de la enfermedad. Al inhibir las proteasas o el proteasoma, estos compuestos pueden inducir la muerte celular en células cancerosas y son herramientas esenciales tanto en la investigación básica como en el desarrollo terapéutico. En CymitQuimica, ofrecemos una amplia gama de inhibidores de proteasas y proteasomas de alta calidad para apoyar su investigación en bioquímica, biología celular y desarrollo de fármacos.
Subcategorías de "Proteasas / Proteasoma"
- Acetil-CoA Carboxilasa(34 productos)
- Cisteína proteasa(96 productos)
- DPP-4(20 productos)
- Glutaminasa(40 productos)
- Proteasa del VIH(449 productos)
- PAI-1(25 productos)
- Inhibidores de la proteasa(50 productos)
- Receptor activado por proteasa(53 productos)
- Proteasoma(94 productos)
- Serina proteasa(50 productos)
- p97(14 productos)
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Se han encontrado 1044 productos de "Proteasas / Proteasoma"
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MK-8325
CAS:<p>MK-8325 is a potent and orally available HCV NS5A inhibitor with replicative activity against a wide range of genotypes.MK-8325 has demonstrated bioavailability</p>Fórmula:C43H54Cl2F2N8O6SiPureza:>99.99%Forma y color:SolidPeso molecular:915.93TG-2-IN-1
CAS:<p>TG-2-IN-1 (Compound D003) is a transglutaminase-2 ( TGM-2 ) inhibitor. TG-2-IN-1 can be used in myopia research[1].</p>Fórmula:C8H13ClN2OSPureza:98.43%Forma y color:SolidPeso molecular:220.72Tyrosinase-IN-2
CAS:<p>Tyrosinase-IN-2, a potent tyrosinase inhibitor, may help in skin lightening and food preservation research.</p>Fórmula:C8H8N4O2SPureza:99.78%Forma y color:SolidPeso molecular:224.24L 756423
CAS:<p>L756423 is a potent, selective HIV protease inhibitor (Ki=0.049 nM), effective against HIV spread in MT25 lymphocytes at 0.1-0.5 nM, useful for AIDS research.</p>Fórmula:C39H48N4O5Pureza:99.34% - 99.88%Forma y color:SolidPeso molecular:652.82UPGL00004
CAS:<p>UPGL00004: potent GAC inhibitor, IC50=29 nM, Kd=27 nM, suppresses triple-negative breast cancer cell growth.</p>Fórmula:C25H26N8O2S2Pureza:97.93%Forma y color:SolidPeso molecular:534.662'-C-Methyladenosine
CAS:<p>2'-C-Methyladenosine from C. renalis inhibits HCV, NS5B RNA synthesis (IC50: 0.3, 1.9µM), and LRV1 in L. guyanensis, L. braziliensis.</p>Fórmula:C11H15N5O4Pureza:99.85%Forma y color:SolidPeso molecular:281.27Lenacapavir
CAS:<p>Lenacapavir (GS-6207) is the first HIV-1 capsid inhibitor approved by the U.S. Food and Drug Administration, the European Medicines Agency, and Health Canada for the treatment of MDR HIV-1 infection.Cost-effective and quality-assured.</p>Fórmula:C39H32ClF10N7O5S2Pureza:99.61% - 99.87%Forma y color:SolidPeso molecular:968.28TY-51469
CAS:<p>TY-51469 is an inhibitor of chymase (IC50s for simian and human chymases: 0.4 and 7.0 nM, respectively).</p>Fórmula:C20H15FN2O6S4Pureza:99.65%Forma y color:SolidPeso molecular:526.6Etarotene
CAS:<p>Etarotene (Arotinoid ethyl sulphone) is an ethylsulfonyl derivative of aloe acid with differentiation-inducing and potentially antitumor activity.Etarotene is a</p>Fórmula:C25H32O2SPureza:99.58% - 99.93%Forma y color:SolidPeso molecular:396.59BDCRB
<p>BDCRB disrupts HCMV DNA maturation by altering terminase cleavage, extending packaging 30 kb until second site.</p>Fórmula:C12H11BrCl2N2O4Pureza:99.41% - 99.43%Forma y color:SoildPeso molecular:398.04MMP2-IN-3
CAS:<p>MMP2-IN-3 is a potent inhibitor of matrix metalloproteinases (MMP-2) (IC50: 31 μM).</p>Fórmula:C23H21N3OPureza:99.38%Forma y color:SolidPeso molecular:355.43BILB-1941
CAS:<p>BILB-1941 (BILB-1941ZW) is an inhibitor of HCV NS5B polymerase and can be used in studies about HCV infection.</p>Fórmula:C34H34N4O4Pureza:99.51% - 99.65%Forma y color:SolidPeso molecular:562.66(2RS)-FPMPA
CAS:<p>(2RS)-FPMPA（FPMPA） has antiviral activity with an IC50 value of 1.85 μM measured in human MT12 cells infected with SHIV (DH4R).</p>Fórmula:C9H13FN5O4PPureza:99.9% - >99.99%Forma y color:SolidPeso molecular:305.2HIV-1 integrase inhibitor 8
CAS:<p>HIV-1 integrase inhibitor 8 is an inhibitor of HIV-1 integrase. Integration is a required step in HIV replication [1].</p>Fórmula:C21H24O2Pureza:98.91%Forma y color:SolidPeso molecular:308.41Gemigliptin
CAS:<p>Gemigliptin (LC15-0444) is a potent dipeptidyl peptidase-4 (DPP-4) inhibitor(KD : 7.25 nM.)</p>Fórmula:C18H19F8N5O2Pureza:99.72%Forma y color:SolidPeso molecular:489.36NP-313
CAS:<p>NP-313 (NSC-4264) is a potent antithrombotic that blocks platelet aggregation via thromboxane A2 synthesis inhibition and targets SOCC-mediated Ca2+ efflux.</p>Fórmula:C12H8ClNO3Pureza:98.97%Forma y color:SolidPeso molecular:249.65BMS-929075
CAS:<p>BMS-929075 is an orally active HCV NS5B replicase (HCV NS5B replicase) palm site variant inhibitor with potency, high oral bioavailability and pharmacokinetic</p>Fórmula:C31H24F2N4O3Pureza:98.44% - 99.94%Forma y color:SolidPeso molecular:538.54GSK-364735
CAS:<p>GSK-364735 is an HIV-1 IN inhibitor.</p>Fórmula:C19H18FN3O4Pureza:97.73%Forma y color:SolidPeso molecular:371.36Emivirine
CAS:<p>Emivirine (MKC-442) is a potent and selective nonnucleoside reverse transcriptase inhibitor of human immunodeficiency virus type 1.</p>Fórmula:C17H22N2O3Pureza:99.8%Forma y color:SolidPeso molecular:302.37PG-116800
CAS:<p>PG-116800 (PG-530742) is a matrix metalloproteinase (MMP) inhibitor. PG-116800 can be used in studies about the treatment of osteoarthritis.</p>Fórmula:C24H27N3O7SPureza:98.03% - 99.66%Forma y color:SolidPeso molecular:501.55BMS-488043
CAS:<p>BMS-488043 is a novel and unique oral small molecule HIV fusion inhibitor that inhibits the attachment of Human Immunodeficiency Virus type 1 (HIV-1) to CD4(+)</p>Fórmula:C22H22N4O5Pureza:99.95%Forma y color:SolidPeso molecular:422.43CP-544439
CAS:<p>CP-544439 is an inhibitor of matrix metalloproteinase-13, which has an effect on adipose tissue development.</p>Fórmula:C18H19FN2O6SPureza:95.02% - 98.66%Forma y color:SolidPeso molecular:410.42JNJ-10311795
CAS:<p>JNJ-10311795 (RWJ-355871) is an inhibitor of neutrophil elastase G and mast cell chymase, demonstrating significant anti-inflammatory effects.</p>Fórmula:C40H35N2O6PPureza:97.43%Forma y color:SolidPeso molecular:670.69P32/98 hemifumarate
CAS:<p>P32/98 hemifumarate is a DPP4 inhibitor with hypoglycemic properties and is used in the study of type 2 diabetes.</p>Fórmula:C22H40N4O6S2Pureza:99.46%Forma y color:SolidPeso molecular:520.71Cathepsin X-IN-1
CAS:<p>Cathepsin X-IN-1 (compound 25) reduces the migration of PC-3 cell with low cytotoxic that is a potent inhibitor of Cathepsin X (IC 50 = 7.13 μM) [1].</p>Fórmula:C15H13N3O3SPureza:99.34%Forma y color:SolidPeso molecular:315.35Sovaprevir
CAS:<p>Sovaprevir is a non-structural 3 (NS3) protease inhibitor with antiviral activity for the treatment of HCV infection.</p>Fórmula:C43H53N5O8SPureza:99.11%Forma y color:SolidPeso molecular:799.97Sirpiglenastat
CAS:<p>Sirpiglenastat (DRP-104) is a glutamine antagonist, a prodrug of DON, with antitumor activity that acts by suppressing the adaptive immune system.</p>Fórmula:C22H27N5O5Pureza:98.01% - 98.37%Forma y color:SolidPeso molecular:441.48DB04760
CAS:<p>DB04760: selective MMP-13 inhibitor, non-zinc-chelating, IC50=8nM, reduces paclitaxel neurotoxicity, anticancer.</p>Fórmula:C22H20F2N4O2Pureza:99.93% - 99.99%Forma y color:SolidPeso molecular:410.42MMP-2/MMP-9 Inhibitor I
CAS:<p>MMP-2/MMP-9-IN-1: oral IV collagenase inhibitor; IC50: 0.24 μM (MMP-9), 0.31 μM (MMP-2); targets cancer.</p>Fórmula:C21H19NO4SPureza:99.74%Forma y color:SolidPeso molecular:381.44Isatoribine
CAS:<p>Isatoribine(ANA245) free base is a potent TLR7 receptor agonist with anti-hepatitis C virus infection activity for the study of HCV infection.</p>Fórmula:C10H12N4O6SPureza:98.99% - 99.75%Forma y color:SolidPeso molecular:316.29Melagatran
CAS:<p>Melagatran is an orally available, direct synthetic thrombin inhibitor that does not require endogenous cofactors other than thrombin.Cost-effective and quality-assured.</p>Fórmula:C22H31N5O4Pureza:98.29% - >99.99%Forma y color:SolidPeso molecular:429.51TG2-IN-3h
CAS:<p>TG2-IN-3h is a highly selective, potent, cell-permeable fluorescent irreversible tissue transglutaminase (tg2) inhibitor</p>Fórmula:C21H26N4O4SPureza:99.34% - 99.76%Forma y color:SolidPeso molecular:430.52Opaviraline
CAS:<p>Opaviraline (GW-420867X) is a potent reverse transcriptase inhibitor that inhibits Human immunodeficiency virus 1 and has the potential to treat HIV infection.</p>Fórmula:C14H17FN2O3Pureza:99.94%Forma y color:SolidPeso molecular:280.29DS-1040 Tosylate
CAS:<p>DS-1040 Tosylate is a thrombin-activated fibrinolysis inhibitor (TAFI) inhibitor and a fibrinolysis enhancer, used for researching thromboembolic diseases.</p>Fórmula:C23H35N3O5SForma y color:SolidPeso molecular:465.61SID 26681509
CAS:<p>SID 26681509 is a selective, reversible and competitive human cathepsin L inhibitor (IC50 of 56 nM).</p>Fórmula:C27H33N5O5SPureza:98.16%Forma y color:SolidPeso molecular:539.65MMP3 inhibitor 1
CAS:<p>MMP3 inhibitor 1 is a potent and highly selective inhibitor of MMP-3 (IC50 of 1 nM).</p>Fórmula:C23H31N3O6SPureza:98%Forma y color:SolidPeso molecular:477.57Human enteropeptidase-IN-1
CAS:<p>Enteropeptidase-IN-1: orally active, potent inhibitor, low systemic exposure, for anti-obesity research.</p>Fórmula:C20H18N4O7Forma y color:SolidPeso molecular:426.38GSK-2485852
CAS:<p>GSK-2485852, a NS5B inhibitor, is used potentially for treatment of HCV infection.</p>Fórmula:C27H25BF2N2O6SForma y color:SolidPeso molecular:554.37PNU-103017
CAS:<p>PNU-103017 is an inhibitor of HIV protease.</p>Fórmula:C28H28N2O5SPureza:98%Forma y color:SolidPeso molecular:504.6MDL 27324
CAS:<p>MDL 27324 is an inhibitor of human neutrophil elastase.</p>Fórmula:C29H38F3N5O6SPureza:98%Forma y color:SolidPeso molecular:641.7LY52
CAS:<p>LY52 is a matrix metalloproteinase-2 inhibitor. It acts by suppressing tumor invasion and metastasis.</p>Fórmula:C22H24N4O6Pureza:98%Forma y color:SolidPeso molecular:440.45HCV-IN-43
CAS:<p>HCV-IN-43 (compound 2), an HCV NS5B protein inhibitor, efficiently inhibits HCV virus replication and is utilized in the study of HCV infection [1].</p>Fórmula:C26H26FN3O5SForma y color:SolidPeso molecular:511.57M867
CAS:<p>M867 is a selective, reversible caspase-3 inhibitor, possessing an IC50 of 1.4 nM and a Ki value of 0.7 nM, demonstrating anti-apoptotic activity [1].</p>Fórmula:C27H43N7O6Pureza:98%Forma y color:SolidPeso molecular:561.67Inogatran
CAS:<p>Inogatran is a synthetic thrombin inhibitor, developed for the possible treatment and prophylaxis of venous and arterial thrombotic diseases.</p>Fórmula:C21H38N6O4Pureza:98%Forma y color:SolidPeso molecular:438.56KCC009
CAS:<p>KCC009 is a potent and selective Transglutaminase 2 Inhibitor.</p>Fórmula:C21H22BrN3O5Forma y color:SolidPeso molecular:476.32XL-784 free base
CAS:<p>XL-784 free base selectively inhibits MMPs with IC50: MMP-1 (1.9µM), MMP-2 (0.81nM), MMP-3 (120nM), MMP-8 (10.8nM), MMP-9 (18nM), MMP-13 (0.56nM).</p>Fórmula:C21H22ClF2N3O8SPureza:98%Forma y color:SolidPeso molecular:549.93BMS-189664
CAS:<p>BMS-189664 is an inhibitor of thrombin.</p>Fórmula:C22H34N6O4SPureza:98%Forma y color:SolidPeso molecular:478.61JW 480
CAS:<p>JW480 is a potent and selective inhibitor of KIAA1363, a serine hydrolase enzyme.</p>Fórmula:C22H23NO2Pureza:99.72%Forma y color:SolidPeso molecular:333.42MMP-3 Inhibitor VIII
CAS:<p>Matrix metalloproteinase-3 (MMP-3), also known as stromelysin-1, is a critical enzyme involved in tissue remodeling and repair through its role in degrading extracellular matrix proteins, facilitating cell migration. This enzyme has been implicated in various physiological processes including vascular remodeling associated with aneurysm formation, wound healing, the progression of atherosclerosis, and tumor initiation. MMP-3 inhibitor VIII, a cell-permeable sulfonamide-based hydroxamic acid, effectively inhibits MMP-3 by binding to its active site (Ki = 23 nM), thus blocking its enzymatic activity. Additionally, this inhibitor has been demonstrated to suppress the activity of mouse macrophage metalloelastase MME/MMP-12, with an IC50 value of 13 nM, highlighting its potential utility in research on tissue remodeling and disease processes involving MMPs.</p>Fórmula:C20H26N2O5SForma y color:SolidPeso molecular:406.5Reverse transcriptase-IN-1
CAS:<p>Reverse transcriptase-IN-1 is a diarylbenzopyrimidine (DABP) analogue and a potent inhibitor of HIV-1 nonnucleoside reverse transcriptase with an IC50of 13.7</p>Fórmula:C25H17N7O2Pureza:99.61%Forma y color:SolidPeso molecular:447.45NS5A-IN-2
CAS:<p>NS5A-IN-2, a potent inhibitor, is highly effective against HCV 1b and shows increased activity for GT 3a with good metabolic stability.</p>Fórmula:C46H45N7O7Pureza:98%Forma y color:SolidPeso molecular:807.89DCLK1-IN-2
CAS:<p>DCLK1-IN-2 (Compound I-5) is a potent inhibitor of DCLK1, exhibiting an IC50 of 171.3 nM, and demonstrates significant antiproliferative effects on SW1990 cell</p>Fórmula:C26H32N8O3SForma y color:SolidPeso molecular:536.65MDL-101146, (R)-
CAS:<p>MDL-101146, (R)- is an effective orally active inhibitor of human neutrophil elastase.</p>Fórmula:C29H37F5N4O6Pureza:98%Forma y color:SolidPeso molecular:632.62HIV-1 protease-IN-9
CAS:<p>HIV-1 protease-IN-9 (compound 5b), a potent HIV-1 protease inhibitor, exhibits strong antiviral efficacy with a dissociation constant (K_i) of 0.028 nM and a</p>Fórmula:C37H41N7O4SPureza:98%Forma y color:SolidPeso molecular:679.83Kallikrein-IN-2
CAS:<p>Kallikrein-IN-2 (compound 1) is an inhibitor of the kinin-releasing enzyme Kallikrein.</p>Fórmula:C28H25F3N4O4Forma y color:SolidPeso molecular:538.52Z-DEVD-CMK
CAS:<p>Z-DEVD-CMK irreversibly inhibits various cathepsins in vitro [1].</p>Fórmula:C27H35ClN4O12Forma y color:SolidPeso molecular:643.04Cyclotheonellazole A
CAS:<p>Cyclotheonellazole A inhibits elastase (IC50=0.034nM) & chymotrypsin (IC50=0.62nM), a natural macrocyclic peptide.</p>Fórmula:C44H54N9NaO14S2Forma y color:SolidPeso molecular:1020.07MK-3281
CAS:<p>MK-3281: Oral, potent HCV NS5B inhibitor with promising properties and efficacy in replication trials, suitable for clinical use.</p>Fórmula:C29H37N3O3Forma y color:SolidPeso molecular:475.62L-689502
CAS:<p>L-689502 is a potent HIV-l protease inhibitor (IC50: 1 nM).</p>Fórmula:C39H51N3O7Pureza:98%Forma y color:SolidPeso molecular:673.84TP0556351
CAS:<p>TP0556351: potent MMP2 inhibitor with 0.2 nM IC50, reduces collagen in pulmonary fibrosis mice.</p>Fórmula:C50H70N10O16Pureza:98%Forma y color:SolidPeso molecular:1067.15GSK-625433
CAS:<p>GSK-625433: Homochiral inhibitor blocks HCV genotypes 1a/1b polymerase.</p>Fórmula:C26H32N4O5SForma y color:SolidPeso molecular:512.62AA74-1
CAS:<p>AA74-1 is a potent, selective APEH inhibitor that significantly enhances T-cell proliferation by inhibiting APEH activity [1].</p>Fórmula:C16H28N4O2Pureza:98%Forma y color:SolidPeso molecular:308.42Petesicatib
CAS:<p>Petesicatib is an inhibitor of cathepsin S. Petesicatib used in the research of immune diseases.</p>Fórmula:C25H23F6N5O4SPureza:99.76%Forma y color:SolidPeso molecular:603.54Cipemastat
CAS:<p>Cipemastat is a competitive inhibitor of human collagenases 1, 2, and 3 (Kis: 3.0, 4.4, and 3.4 nM).</p>Fórmula:C22H36N4O5Pureza:98%Forma y color:SolidPeso molecular:436.55Cathepsin K inhibitor 3
CAS:<p>Cathepsin K inhibitor 3: Selective, IC50 of 0.5 nM, good pharmacokinetics, potential for OA research.</p>Fórmula:C30H31FN4O4SForma y color:SolidPeso molecular:562.65MeOSuc-AAPV-CMK
CAS:<p>MeOSuc-AAPV-CMK (Elastase Inhibitor III) serves as an inhibitor of elastase, as well as cathepsin G and proteinase 3, and impedes leukocyte elastase-mediated</p>Fórmula:C22H35ClN4O7Forma y color:SolidPeso molecular:502.99FK706
CAS:<p>FK706, a human neutrophil elastase inhibitor (IC50: 83 nM, Ki: 4.2 nM), also blocks mouse and porcine elastases. Anti-inflammatory.</p>Fórmula:C26H33F3N4NaO7Forma y color:SolidPeso molecular:593.556XL-784
CAS:<p>XL-784 is a selective MMP inhibitor with low IC50s for MMP-1,2,3,8,9,13, modulating extracellular matrix remodeling, tumor invasion, and metastasis in cancer.</p>Fórmula:C42H42Cl2F4MgN6O16S2Pureza:98%Forma y color:SolidPeso molecular:1122.15Phe-Pro-Ala-pNA
CAS:<p>Phe-Pro-Ala-pNA is a chromogenic substrate utilized for assessing tripeptidyl peptidase activity.</p>Fórmula:C23H27N5O5Forma y color:SolidPeso molecular:453.49Atecegatran metoxil
CAS:<p>Atecegatran Metoxil (AZD0837), an oral thrombin inhibitor in development for stroke prevention in atrial fibrillation, is well-tolerated with favorable PK.</p>Fórmula:C22H23ClF2N4O5Forma y color:SolidPeso molecular:496.89MMP-7-IN-3
CAS:<p>MMP-7-IN-3 (compound 15) is a potent and selective MMP-7 inhibitor, inhibiting renal fibrosis in a unilateral ureteral obstruction mouse model.</p>Fórmula:C34H43ClF3N7O9SPureza:99.915%Forma y color:SolidPeso molecular:818.26Thrombin inhibitor 1
CAS:<p>Thrombin inhibitor 1 is a potent inhibitor of thrombin (Ki: 0.66 nM, 2xaPTT=0.43 μM).</p>Fórmula:C22H20Cl2F2N4O3Pureza:98%Forma y color:SolidPeso molecular:497.32Collagen proline hydroxylase inhibitor
CAS:<p>Collagen proline hydroxylase inhibitor is an inhibitor collagen proline hydroxylase and useful for antifibrotic proliferative agents.</p>Fórmula:C18H18N4O4Pureza:98%Forma y color:SolidPeso molecular:354.36Ro 31-9790
CAS:<p>Ro 31-9790 is a synthetic inhibitor of metalloproteinase (MMP).</p>Fórmula:C15H29N3O4Pureza:98%Forma y color:SolidPeso molecular:315.41Beclabuvir HCl
CAS:<p>Beclabuvir (BMS-791325) is an HCV inhibitor targeting NS5B polymerase with sub-28 nM potency for genotypes 1, 3, 4, 5.</p>Fórmula:C36H46ClN5O5SForma y color:SolidPeso molecular:696.3Azt-pmap
CAS:<p>AZT-PMPA, an aryl phosphate derivative of AZT and a nucleoside analogue, demonstrates anti-HIV activity[1].</p>Fórmula:C20H25N6O8PPureza:98%Forma y color:SolidPeso molecular:508.42HCV-IN-44
CAS:<p>HCV-IN-44 (compound 28) is an inhibitor of the HCV NS5B protein, efficacious in suppressing HCV virus replication and useful for researching HCV infection [1].</p>Fórmula:C24H26FN3O5SForma y color:SolidPeso molecular:487.54Paltimatrectinib
CAS:<p>Paltimatrectinib (PBI-200) is a tyrosine kinase inhibitor with anticancer activity, and is used in the study of bladder, breast, and colorectal cancers.</p>Fórmula:C20H15F5N6Pureza:99.96%Forma y color:SolidPeso molecular:434.37Proteasome β2c/i-IN-1
CAS:<p>Proteasome β2c/i-IN-1 (compound 37) serves as a selective inhibitor targeting the β2c and β2i subunits of the human proteasome [1].</p>Fórmula:C32H48N4O7Pureza:98%Forma y color:SolidPeso molecular:600.75Proteasome-IN-4
<p>Proteasome-IN-4, a potent non-covalent inhibitor (IC50=8.39nM), halts cancer cell growth, useful for oncology studies.</p>Fórmula:C44H58N6O5Forma y color:SolidPeso molecular:750.97KB-R7785
CAS:<p>KB-R7785 is a novel ADAM12/MMP inhibitor improving heart function and insulin sensitivity by blocking HB-EGF and TNF-alpha.</p>Fórmula:C18H27N3O4Forma y color:SolidPeso molecular:349.42NCI-B16
CAS:<p>NCI-B16 is a small-molecule RNA binder that inhibits HCV (hepatitis C virus) replication [1].</p>Fórmula:C27H26N8O4Forma y color:SolidPeso molecular:526.55Z-PDLDA-NHOH
CAS:<p>Z-PDLDA-NHOH is a potent, specific vertebrate collagenase inhibitor [1].</p>Fórmula:C22H32N4O6Forma y color:SolidPeso molecular:448.51Cathepsin Inhibitor 2
CAS:<p>Cathepsin Inhibitor 2 is a potent Cathepsin S inhibitor (Ki: <20 nM).</p>Fórmula:C19H21F6N3OPureza:98%Forma y color:SolidPeso molecular:421.38Mergetpa
CAS:<p>Mergetpa, a carboxypeptidase inhibitor, impedes the conversion of kinins and B2 receptor antagonists into metabolites devoid of the C-terminal arginine [1].</p>Fórmula:C7H15N3O2S2Pureza:98%Forma y color:SolidPeso molecular:237.34Ecallantide
CAS:<p>Ecallantide (DX-88) is a recombinant inhibitor specifically targeting plasma kallikrein, which serves to impede the synthesis of bradykinin.</p>Fórmula:C305H448N88O91S8Forma y color:SolidPeso molecular:7059.88ONO 4817
CAS:ONO-4817 suppresses MMPs, limiting plaque progression and aortic hyperplasia in hyperlipidemic rabbits.Fórmula:C22H28N2O6Forma y color:SolidPeso molecular:416.47Dim16
CAS:<p>Dim16, a dual inhibitor of PCSK9/HMG-CoAR, demonstrates potent activity with an IC50 of 19 nM against PCSK9 and significantly impedes PCSK9-LDLR interaction</p>Fórmula:C29H38IN5Forma y color:SolidPeso molecular:583.55GS-6620
CAS:<p>GS-6620 is a HCV nonstructural protein 5B (NS5B) inhibitor.</p>Fórmula:C29H37N6O9PForma y color:SolidPeso molecular:644.61LU-002i
CAS:<p>LU-002i is a selective inhibitor targeting the human proteasome subunits β2c and β2i, demonstrating an inhibitory concentration (IC50) of 220 nM for β2i [1].</p>Fórmula:C35H52N4O7Pureza:98%Forma y color:SolidPeso molecular:640.81AZD-7295
CAS:<p>AZD-7295 (A-689) is an NS5A inhibitor that may be used to treat HCV infection.</p>Fórmula:C32H35F3N4O5SForma y color:SolidPeso molecular:644.7SSR 69071
CAS:<p>SSR69071: selective neutrophil elastase inhibitor, stronger for humans (Ki=0.0168 nM), may treat COPD, asthma, and reduce heart injury.</p>Fórmula:C27H32N4O7SForma y color:SolidPeso molecular:556.63Proteasome-IN-5
CAS:<p>Proteasome-IN-5, also known as compound 5, acts as a proteasome inhibitor [1].</p>Fórmula:C20H30BN5O7Pureza:98%Forma y color:SolidPeso molecular:463.29PTC725
CAS:<p>PTC725 is a selective HCV 1b replicons inhibitor. It has been shown to target the nonstructural protein 4B.</p>Fórmula:C23H18F4N6O2SPureza:98%Forma y color:SolidPeso molecular:518.49EP1013
CAS:<p>EP1013 is a broad-spectrum selective inhibitor of Caspase used in the study of type 1 diabetes.</p>Fórmula:C18H23FN2O6Pureza:98%Forma y color:SolidPeso molecular:382.38HIV-1 protease-IN-7
CAS:<p>HIV-1 protease-IN-7 (compound 16) is an orally active inhibitor of HIV-1 protease, exhibiting an IC50 of 3.52 nM and an EC50 of 37 nM [1].</p>Fórmula:C68H104N10O12SPureza:98%Forma y color:SolidPeso molecular:1285.68I-XW-053
CAS:<p>I-XW-053 is an inhibitor of capsid targeted HIV-1 replication using the hybrid structure based method to block the interface between CA N-terminal domains (NTD-</p>Fórmula:C22H16N2O2Pureza:99.05%Forma y color:SolidPeso molecular:340.37Neurodegenerative Disorder-Targeting Compound 1
CAS:<p>Neurodegenerative Disorder-Targeting Compound 1 is an inhibitor of calpain [1].</p>Fórmula:C28H28N4O4Pureza:98%Forma y color:SolidPeso molecular:484.55HIV-1 protease-IN-12
CAS:<p>HIV-1 protease-IN-12 (compound 35b) serves as a potent inhibitor of HIV-1 protease, exhibiting an IC50 value of 0.51 nM, and demonstrates efficacy against drug-</p>Fórmula:C25H35N3O5SPureza:98%Forma y color:SolidPeso molecular:489.63MMP-145
CAS:<p>MMP-145 is used as a protease inhibitor.</p>Fórmula:C20H20N2O7SPureza:98%Forma y color:SolidPeso molecular:432.45
