CymitQuimica logo
Proteasas / Proteasoma

Proteasas / Proteasoma

Los inhibidores de proteasas y proteasomas son compuestos que bloquean la actividad de las proteasas y del proteasoma, que están involucrados en la degradación y renovación de proteínas. Estos inhibidores son vitales para estudiar la regulación de la homeostasis proteica, el control del ciclo celular y la apoptosis. Los inhibidores de proteasas y proteasomas también se utilizan en el tratamiento de enfermedades como el cáncer, donde la degradación anormal de proteínas desempeña un papel en la progresión de la enfermedad. Al inhibir las proteasas o el proteasoma, estos compuestos pueden inducir la muerte celular en células cancerosas y son herramientas esenciales tanto en la investigación básica como en el desarrollo terapéutico. En CymitQuimica, ofrecemos una amplia gama de inhibidores de proteasas y proteasomas de alta calidad para apoyar su investigación en bioquímica, biología celular y desarrollo de fármacos.

Subcategorías de "Proteasas / Proteasoma"

Mostrar 3 subcategorías más

Se han encontrado 1044 productos de "Proteasas / Proteasoma"

Ordenar por

Pureza (%)
0
100
|
0
|
50
|
90
|
95
|
100
productos por página.
  • Sucunamostat

    CAS:
    <p>Sucunamostat is an L-aspartic acid enteropeptidase inhibitor.</p>
    Fórmula:C22H22N4O8
    Forma y color:Solid
    Peso molecular:470.438
  • STK33-IN-1

    CAS:
    <p>STK33-IN-1 (compound 1) is a STK33 inhibitor, with an IC 50 of 7 nM.</p>
    Fórmula:C24H27N7O2
    Forma y color:Solid
    Peso molecular:445.527
  • ZG36


    <p>ZG36, a human Caseinolytic protease P (ClpP) agonist, non-selectively degrades respiratory chain complexes and reduces mitochondrial DNA, causing mitochondrial</p>
    Forma y color:Odour Solid
  • Dutogliptin tartrate

    CAS:
    Dutogliptin tartrate is an effective and selective oral dipeptide-peptide-4 (DPP4) inhibitor for the treatment of type 2 diabetes mellitus.
    Fórmula:C14H26BN3O9
    Pureza:98%
    Forma y color:Solid
    Peso molecular:391.18
  • MMP-3 Inhibitor

    CAS:
    <p>MMP-3 Inhibitor is a peptide matrix metalloproteinase-3 (MMP-3) inhibitor with a Ki value of 95 nM.MMP-3 inhibitor has anticancer and antitumor activity.</p>
    Fórmula:C27H46N10O9S
    Pureza:98.87%
    Forma y color:Solid
    Peso molecular:686.78
  • HCV-IN-4

    CAS:
    <p>HCV-IN-4: Potent, oral HCV NS5A inhibitor; effective vs GT1a/b, GT2b, GT3a, Y93H, L31V; EC90s: 3 pM-0.02 nM.</p>
    Fórmula:C52H58FN9O8
    Pureza:98%
    Forma y color:Solid
    Peso molecular:956.07
  • Cathepsin D and E FRET Substrate acetate(839730-93-7 Free base)


    Fluorogenic substrate for cathepsins D & E; cleaves at Phe-Phe bond; not for B, H, L. Useful for assays and studies.
    Forma y color:Odour Solid
  • Cys-TAT(47-57) acetate(583836-55-9 Free base)


    <p>Cys-TAT(47-57) acetate is derived from the HIV-1 transactivating protein. Cys-TAT(47-57) acetate is an arginine rich peptide that can penetrate cells.</p>
    Fórmula:C69H128N34O16S
    Pureza:95.1100%
    Forma y color:Solid
    Peso molecular:1722.04
  • Nitidanin


    <p>Nitidanin is a useful organic compound for research related to life sciences and the catalog number is T125599.</p>
    Fórmula:C21H24O8
    Forma y color:Solid
    Peso molecular:404.415
  • MK-6169

    CAS:
    <p>MK-6169 is an effective Pan-Genotype Hepatitis C Virus NS5A inhibitor. It also has Optimized Activity against Common Resistance-Associated Substitutions.</p>
    Fórmula:C54H62FN9O8S
    Pureza:98%
    Forma y color:Solid
    Peso molecular:1016.2
  • DPP-4-IN-14


    <p>DPP-4-IN-14 (compound 30) is an inhibitor of DPP-4, with an IC50 value of 12.82 nM.</p>
    Fórmula:C33H27N7O3
    Forma y color:Solid
    Peso molecular:569.613
  • Talabostat

    CAS:
    <p>Talabostat (PT100, Val-boroPro) is a potent, nonselective and orally available dipeptidyl peptidase IV (DPP-IV) inhibitor with a Ki of 0.18 nM.</p>
    Fórmula:C9H19BN2O3
    Forma y color:Solid
    Peso molecular:214.07
  • Elastatinal

    CAS:
    <p>Elastatinal is an elastase inhibitor. It is found in culture filtrates of various species of actinomyces.</p>
    Fórmula:C21H36N8O7
    Forma y color:Yellowish Solid
    Peso molecular:512.56
  • JC-10

    CAS:
    <p>JC-10 is a potent inhibitor of metalloproteinases and is often used as a probe.</p>
    Fórmula:C25H29Cl2IN4
    Pureza:95%
    Forma y color:Solid
    Peso molecular:583.34
  • CRA-2059 TFA


    <p>CRA-2059 is a highly specific and selective tryptase inhibitor, with a Ki of 620 pM for recombinant human tryptase-β (rHTβ)[1][2].</p>
    Forma y color:Solid
  • BMS-767778

    CAS:
    <p>BMS-767778, a DPP-4 inhibitor, is used potentially for the treatment of type 2 diabetes.</p>
    Fórmula:C19H20Cl2N4O2
    Forma y color:Solid
    Peso molecular:407.29
  • Sofosbuvir impurity H


    <p>Sofosbuvir impurity H, an diastereoisomer of Sofosbuvir, is the impurity of Sofosbuvir.</p>
    Fórmula:C29H33FN3O10P
    Pureza:98%
    Forma y color:Solid
    Peso molecular:633.56
  • Fotagliptin

    CAS:
    <p>Fotagliptin is a dipeptidyl peptidase IV inhibitor.</p>
    Fórmula:C17H19FN6O
    Forma y color:Solid
    Peso molecular:342.37
  • Dnp-P-Cha-G-Cys(Me)-HA-K(Nma)-NH2

    CAS:
    <p>Dnp-P-Cha-G-Cys(Me)-HA-K(Nma)-NH2 is a fluorogenic probe for MMP-1 and MMP-9 detection, releasing fluorescent Nma upon cleavage (Ex/Em: 340/440 nm).</p>
    Fórmula:C49H68N14O12S
    Forma y color:Solid
    Peso molecular:1077.22
  • Tilpisertib fosmecarbil TFA

    CAS:
    Tilpisertib fosmecarbil TFA, the TFA salt form of Tilpisertib, acts as an inhibitor of serine/threonine kinases. This compound also exhibits anti-inflammatory activity.
    Fórmula:C37H37ClF3N8O9P
    Forma y color:Solid
    Peso molecular:861.16