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Proteasas / Proteasoma

Proteasas / Proteasoma

Los inhibidores de proteasas y proteasomas son compuestos que bloquean la actividad de las proteasas y del proteasoma, que están involucrados en la degradación y renovación de proteínas. Estos inhibidores son vitales para estudiar la regulación de la homeostasis proteica, el control del ciclo celular y la apoptosis. Los inhibidores de proteasas y proteasomas también se utilizan en el tratamiento de enfermedades como el cáncer, donde la degradación anormal de proteínas desempeña un papel en la progresión de la enfermedad. Al inhibir las proteasas o el proteasoma, estos compuestos pueden inducir la muerte celular en células cancerosas y son herramientas esenciales tanto en la investigación básica como en el desarrollo terapéutico. En CymitQuimica, ofrecemos una amplia gama de inhibidores de proteasas y proteasomas de alta calidad para apoyar su investigación en bioquímica, biología celular y desarrollo de fármacos.

Subcategorías de "Proteasas / Proteasoma"

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Se han encontrado 1039 productos de "Proteasas / Proteasoma"

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  • NQ301
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    NQ301

    CAS:
    <p>NQ301, an antithrombotic agent, inhibits collagen-challenged rabbit platelet aggregation (IC50: 10 mg/mL).</p>
    Fórmula:C18H12ClNO3
    Pureza:99.74% - 99.76%
    Forma y color:Solid
    Peso molecular:325.75

    Ref: TM-T3757

  • Raltegravir
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    Raltegravir

    CAS:
    <p>Raltegravir (MK-0518) is a pyrrolidinone derivative and HIV INTEGRASE INHIBITOR that is used in combination with other ANTI-HIV AGENTS for the treatment of HIV</p>
    Fórmula:C20H21FN6O5
    Pureza:99.86% - >99.99%
    Forma y color:Solid
    Peso molecular:444.42

    Ref: TM-T2239L

  • 2-CHLOROMETHYL-1,1-DIOXO-1,2-DIHYDRO-1λ*6*-BENZO[D]ISOTHIAZOL-3-ONE
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    2-CHLOROMETHYL-1,1-DIOXO-1,2-DIHYDRO-1λ*6*-BENZO[D]ISOTHIAZOL-3-ONE

    CAS:
    <p>2-CHLOROMETHYL-1,1-DIOXO-1,2-DIHYDRO-1LAMBDA*6*-BENZO[D]ISOTHIAZOL-3-ONE targets the Neutrophil elastase (human).</p>
    Fórmula:C8H6ClNO3S
    Pureza:97.28%
    Forma y color:Solid
    Peso molecular:231.66

    Ref: TM-T8602

  • AF 399
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    AF 399

    CAS:
    <p>AF 399 is a CCR4 antagonist. It reverses the tumor-promoting environment.</p>
    Fórmula:C12H17N3O3S
    Pureza:99.83%
    Forma y color:Solid
    Peso molecular:283.35

    Ref: TM-T23646

  • Asunaprevir
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    Asunaprevir

    CAS:
    Asunaprevir (BMS-650032) is an effective hepatitis C virus (HCV) NS3 protease inhibitor.
    Fórmula:C35H46ClN5O9S
    Pureza:99.34% - 99.8%
    Forma y color:Solid
    Peso molecular:748.29

    Ref: TM-T4474

  • Alvelestat
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    Alvelestat

    CAS:
    <p>Alvelestat (AZD9668) is an orally bioavailable, selective and reversible inhibitor of human neutrophil elastase (NE), with potential anti-inflammatory activity.</p>
    Fórmula:C25H22F3N5O4S
    Pureza:98% - >99.99%
    Forma y color:Solid
    Peso molecular:545.53

    Ref: TM-T3107

  • Patamostat
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    Patamostat

    CAS:
    <p>Patamostat (E-3123) inhibits trypsin, plasmin, and thrombin; may reduce acute pancreatitis progression. IC50: trypsin 39 nM, plasmin 950 nM, thrombin 1.9 μM.</p>
    Fórmula:C20H20N4O4S
    Forma y color:Solid
    Peso molecular:412.46

    Ref: TM-T9670

  • Dabigatran Etexilate Mesylate
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    Dabigatran Etexilate Mesylate

    CAS:
    <p>Dabigatran Etexilate Mesylate (BIBR 1048MS) is the orally active prodrug of dabigatran. Dabigatran is a reversible and selective, direct thrombin inhibitor.</p>
    Fórmula:C34H41N7O5·CH4O3S
    Pureza:99.91%
    Forma y color:Solid
    Peso molecular:723.84

    Ref: TM-T5133

  • PSI-6130
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    PSI-6130

    CAS:
    <p>PSI-6130 (R 1656) is a potent and selective HCV NS5B polymerase inhibitor. PSI-6130 inhibits HCV replication with a mean IC50 of 0.6 μM.</p>
    Fórmula:C10H14FN3O4
    Pureza:98.63% - 99.79%
    Forma y color:Solid
    Peso molecular:259.23

    Ref: TM-T7607

  • Ximelagatran
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    Ximelagatran

    CAS:
    <p>Ximelagatran, oral direct thrombin inhibitor, transforms to active melagatran in body.</p>
    Fórmula:C24H35N5O5
    Pureza:95.48% - 99.60%
    Forma y color:Solid
    Peso molecular:473.57

    Ref: TM-T17265

  • SU 4942
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    SU 4942

    CAS:
    <p>SU-4942 is a modulator of tyrosine kinase signaling.</p>
    Fórmula:C15H10BrNO
    Pureza:99% - 99.32%
    Forma y color:Solid
    Peso molecular:300.15

    Ref: TM-T3567

  • STK16-IN-1
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    STK16-IN-1

    CAS:
    <p>STK16-IN-1 is an inhibitor of STK16 kinase (IC50: 295 nM).</p>
    Fórmula:C17H12FN3O
    Pureza:99.52%
    Forma y color:Solid
    Peso molecular:293.3

    Ref: TM-T16944

  • Boc-Asp(OMe)-fluoromethyl ketone
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    Boc-Asp(OMe)-fluoromethyl ketone

    CAS:
    <p>Boc-Asp(OMe)-FMK is a broad-spectrum caspase inhibitor that blocks Fas-mediated processes without affecting IL-8 chemotaxis.</p>
    Fórmula:C11H18FNO5
    Pureza:≥98%
    Forma y color:Solid
    Peso molecular:263.26

    Ref: TM-T39308

  • PSI-6206
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    PSI-6206

    CAS:
    <p>PSI-6206 (RO 2433) (RO2433) is a selective HCV RNA polymerase inhibitor.</p>
    Fórmula:C10H13FN2O5
    Pureza:98% - 99.79%
    Forma y color:Solid
    Peso molecular:260.22

    Ref: TM-T2117

  • Velpatasvir
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    Velpatasvir

    CAS:
    <p>Velpatasvir (GS-5816), also known as GS-5816, is a potent and selective Hepatitis C virus NS5A inhibitor.</p>
    Fórmula:C49H54N8O8
    Pureza:99.17% - 99.83%
    Forma y color:Solid
    Peso molecular:883

    Ref: TM-T3334

  • Fostemsavir
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    Fostemsavir

    CAS:
    Fostemsavir (BMS-663068) is an HIV-1 attachment inhibitor in development for the treatment of HIV-1 infection.
    Fórmula:C25H26N7O8P
    Pureza:98.95%
    Forma y color:Solid
    Peso molecular:583.49

    Ref: TM-T3523

  • S 3304
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    S 3304

    CAS:
    <p>S 3304 is a novel matrix metalloproteinases inhibitor which is specific for MMP-2 and MMP-9.</p>
    Fórmula:C24H20N2O4S2
    Pureza:98.09%
    Forma y color:Solid
    Peso molecular:464.56

    Ref: TM-T16966

  • Ivachtin
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    Ivachtin

    CAS:
    <p>Ivachtin (Caspase-3 Inhibitor VII) is a nonpeptide, noncompetitive and reversibl caspase-3 inhibitor(IC50 = 23 nM) and is a modest inhibitor of the remaining</p>
    Fórmula:C20H21N3O7S
    Pureza:99.74%
    Forma y color:Solid
    Peso molecular:447.46

    Ref: TM-T11696

  • Darunavir Ethanolate
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    Darunavir Ethanolate

    CAS:
    <p>Darunavir Ethanolate (UIC 94017) is an HIV PROTEASE INHIBITOR that is used in the treatment of AIDS and HIV INFECTIONS.</p>
    Fórmula:C29H43N3O8S
    Pureza:99.84% - 99.86%
    Forma y color:Solid
    Peso molecular:593.74

    Ref: TM-T3335

  • Chlorcyclizine
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    Chlorcyclizine

    CAS:
    <p>CHLORCYCLIZINE is a histamine H1 antagonist and a potent hepatitis C virus (HCV) entry inhibitor.</p>
    Fórmula:C18H21ClN2
    Pureza:98.75%
    Forma y color:Solid
    Peso molecular:300.83

    Ref: TM-T9717