Proteasas / Proteasoma
Los inhibidores de proteasas y proteasomas son compuestos que bloquean la actividad de las proteasas y del proteasoma, que están involucrados en la degradación y renovación de proteínas. Estos inhibidores son vitales para estudiar la regulación de la homeostasis proteica, el control del ciclo celular y la apoptosis. Los inhibidores de proteasas y proteasomas también se utilizan en el tratamiento de enfermedades como el cáncer, donde la degradación anormal de proteínas desempeña un papel en la progresión de la enfermedad. Al inhibir las proteasas o el proteasoma, estos compuestos pueden inducir la muerte celular en células cancerosas y son herramientas esenciales tanto en la investigación básica como en el desarrollo terapéutico. En CymitQuimica, ofrecemos una amplia gama de inhibidores de proteasas y proteasomas de alta calidad para apoyar su investigación en bioquímica, biología celular y desarrollo de fármacos.
Subcategorías de "Proteasas / Proteasoma"
- Acetil-CoA Carboxilasa(35 productos)
- Cisteína proteasa(96 productos)
- DPP-4(20 productos)
- Glutaminasa(40 productos)
- Proteasa del VIH(451 productos)
- PAI-1(25 productos)
- Inhibidores de la proteasa(50 productos)
- Receptor activado por proteasa(53 productos)
- Proteasoma(94 productos)
- Serina proteasa(49 productos)
- p97(14 productos)
Mostrar 3 subcategorías más
Se han encontrado 1039 productos de "Proteasas / Proteasoma"
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L-689502
CAS:<p>L-689502 is a potent HIV-l protease inhibitor (IC50: 1 nM).</p>Fórmula:C39H51N3O7Pureza:98%Forma y color:SolidPeso molecular:673.84MK-0674
CAS:<p>MK-0674 is a cathepsin K inhibitor (IC50: 0.4 nM) that inhibits Cat B, Cat F, Cat L, and Cat S for metabolism-related diseases.</p>Fórmula:C26H27F6N3O2Pureza:97.3% - 99.91%Forma y color:SolidPeso molecular:527.5Filibuvir
CAS:<p>Filibuvir (PF-00868554) inhibits HCV polymerase genotypes 1a/1b, EC50s 59 nM.</p>Fórmula:C29H37N5O3Pureza:99.28% - >99.99%Forma y color:SolidPeso molecular:503.64γ-Glu-Tyr
CAS:<p>gamma-Glu-Tyr (gamma-Glutamyltyrosine) is a kokumi peptide against dipeptidyl peptidase-IV (DPP-IV) and is used in the study of diabetes mellitus.</p>Fórmula:C14H18N2O6Pureza:98.92%Forma y color:SolidPeso molecular:310.3PDDC inhibitor
CAS:<p>PDDC inhibitor (Phenyl (R)-(1-(3-(3,4-dimethoxyphenyl)-2,6-dimethylimidazo[1,2-b]pyridazin-8-yl)pyrrolidin-3-yl)carbamate) is an nSMase2 inhibitor.</p>Fórmula:C27H29N5O4Pureza:96.09% - 99.39%Forma y color:SolidPeso molecular:487.55Nesbuvir
CAS:<p>Nesbuvir: HCV NS5B polymerase inhibitor, IC50 9 nM against HCV 1b replicon in liver cancer cells.</p>Fórmula:C22H23FN2O5SPureza:99.99%Forma y color:SolidPeso molecular:446.49ZED-1227
CAS:<p>ZED-1227 (TAK-227) is a TG2 inhibitor with anticancer activity that blocks inflammation-induced TG2 expression and activation for the treatment of Celiac Diseas</p>Fórmula:C26H36N6O6Pureza:99.04%Forma y color:SolidPeso molecular:528.6HIV-1 inhibitor-54
CAS:<p>HIV-1 inhibitor-54: potent anti-HIV (EC50: 32 nM), targets WT HIV-1 IIIB in MT-4 cells for infection research.</p>Fórmula:C27H30N6O4SPureza:98.05% - 99.44%Forma y color:SoildPeso molecular:534.63Ac-YVAD-AOM
CAS:<p>Ac-YVAD-AOM is a selective and potent caspase-1 inhibitor showing antitumor activity and potential analgesic activity.</p>Fórmula:C33H42N4O10Pureza:98%Forma y color:SolidPeso molecular:654.71Aderamastat
CAS:<p>Aderamastat (FP-025) is an orally active matrix metalloproteinase 12 (MMP-12) inhibitor indicated for the study of allergic asthma, COPD and pulmonary fibrosis.</p>Fórmula:C21H18N2O4SPureza:99.35%Forma y color:SolidPeso molecular:394.44BMS-212122
CAS:<p>BMS-212122 inhibits MTP, reduces lipids and plaque in animal tests.</p>Fórmula:C43H36F6N4O2Pureza:99.18%Forma y color:SolidPeso molecular:754.76Collagen proline hydroxylase inhibitor-1
CAS:<p>Collagen proline hydroxylase inhibitor-1 具有抗纤维增生活性。</p>Fórmula:C24H21N5O4Pureza:99.62%Forma y color:SolidPeso molecular:443.45VBY-825
CAS:<p>VBY-825 is a reversible inhibitor of cathepsin with high potency against cathepsins B, L, S and V.</p>Fórmula:C23H29F4N3O5SPureza:99.91%Forma y color:SolidPeso molecular:535.55Anti-infective agent 10
CAS:<p>Anti-infective agent 10 (Compound Example 30) is an ns5b polymerase inhibitor that functions as an anti-HCV agent.</p>Fórmula:C26H25N3O7SForma y color:SolidPeso molecular:523.56Freselestat quarterhydrate
<p>ONO-6818 quarterhydrate: oral neutrophil elastase inhibitor, Ki 12.2 nM; >100x less effective on other proteases; strong anti-inflammatory.</p>Fórmula:C23H30N6O5Forma y color:SolidPeso molecular:457.03PNU-248686A
CAS:<p>PNU-248686A is an inhibitor of matrix metalloproteinase (MMP).</p>Fórmula:C22H18ClNaO5S2Pureza:98%Forma y color:SolidPeso molecular:484.95Antiplatelet agent 3
CAS:<p>Antiplatelet agent 3 (Compound K-10) is a compound with antiplatelet aggregation activity, exhibiting IC50 values of 2.55, 3.22, and 2.09 mg/mL for platelet aggregation induced by ADP, AA, and COL, respectively. It holds potential for research in cardiovascular diseases.</p>Fórmula:C38H32N2O5Forma y color:SolidPeso molecular:596.671RO5461111
CAS:<p>RO5461111: Oral Cathepsin S inhibitor, IC50 of 0.4 nM (human) & 0.5 nM (mouse), reduces T/B cell activation, treats lung inflammation & lupus nephritis.</p>Fórmula:C27H24F6N4O4SForma y color:SolidPeso molecular:614.56Faldaprevir
CAS:Faldaprevir is an orally effective, selective, non-covalent HCV NS3/4A protease inhibitor with high inhibitory activity against HCV 1a and 1b genotype.Fórmula:C40H49BrN6O9SPureza:99.04% - 99.19%Forma y color:SolidPeso molecular:869.82Plodicitinib
CAS:<p>Plodicitinib is an inhibitor of Janus tyrosine kinase 3/TEC family kinase, exhibiting anti-inflammatory properties.</p>Fórmula:C19H22FN7O2Forma y color:SolidPeso molecular:399.422
