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Proteasas / Proteasoma

Proteasas / Proteasoma

Los inhibidores de proteasas y proteasomas son compuestos que bloquean la actividad de las proteasas y del proteasoma, que están involucrados en la degradación y renovación de proteínas. Estos inhibidores son vitales para estudiar la regulación de la homeostasis proteica, el control del ciclo celular y la apoptosis. Los inhibidores de proteasas y proteasomas también se utilizan en el tratamiento de enfermedades como el cáncer, donde la degradación anormal de proteínas desempeña un papel en la progresión de la enfermedad. Al inhibir las proteasas o el proteasoma, estos compuestos pueden inducir la muerte celular en células cancerosas y son herramientas esenciales tanto en la investigación básica como en el desarrollo terapéutico. En CymitQuimica, ofrecemos una amplia gama de inhibidores de proteasas y proteasomas de alta calidad para apoyar su investigación en bioquímica, biología celular y desarrollo de fármacos.

Subcategorías de "Proteasas / Proteasoma"

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Se han encontrado 1094 productos de "Proteasas / Proteasoma"

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  • LY 3000328

    CAS:
    LY 3000328 (Cathepsin S inhibitor) is a selective inhibitor of cathepsin S.Cost-effective and quality-assured.
    Fórmula:C25H29FN4O5
    Pureza:97.83% - 99.54%
    Forma y color:Solid
    Peso molecular:484.52
  • Patamostat

    CAS:
    Patamostat (E-3123) inhibits trypsin, plasmin, and thrombin; may reduce acute pancreatitis progression. IC50: trypsin 39 nM, plasmin 950 nM, thrombin 1.9 μM.
    Fórmula:C20H20N4O4S
    Forma y color:Solid
    Peso molecular:412.46
  • Efegatran

    CAS:
    <p>Efegatran is a hematologic agent and platelet aggregation inhibitor.</p>
    Fórmula:C21H32N6O3
    Forma y color:Solid
    Peso molecular:416.52
  • Rolipram

    CAS:
    Rolipram (SB 95952) is a phosphodiesterase 4 inhibitor with antidepressant properties.
    Fórmula:C16H21NO3
    Pureza:99.22% - >99.99%
    Forma y color:Solid
    Peso molecular:275.34
  • Bemnifosbuvir

    CAS:
    Bemnifosbuvir (AT-511) is a novel phosphoramidate prodrug of 2'-fluoro-2'-C-methylguanosine-5'-monophosphate that has potent in vitro activity against HCV.
    Fórmula:C24H33FN7O7P
    Pureza:99.35% - 99.54%
    Forma y color:Solid
    Peso molecular:581.53
  • Daclatasvir dihydrochloride

    CAS:
    Daclatasvir dihydrochloride is an oral antiviral that treats chronic hepatitis C by inhibiting HCV's NS5A; rare liver enzyme elevation, seldom causes jaundice.
    Fórmula:C40H52Cl2N8O6
    Pureza:99.67%
    Forma y color:Solid
    Peso molecular:811.8
  • CA-074 methyl ester

    CAS:
    CA-074 methyl ester (Cathepsin B Inhibitor IV) is a selective inhibitor of Cathepsin B (IC50=36.3 nM). neuroprotective effect. High-Quality, Low-Cost!
    Fórmula:C19H31N3O6
    Pureza:97.26% - 99.58%
    Forma y color:Solid
    Peso molecular:397.47
  • Raltegravir

    CAS:
    <p>Raltegravir (MK-0518) is a pyrrolidinone derivative and HIV INTEGRASE INHIBITOR that is used in combination with other ANTI-HIV AGENTS for the treatment of HIV</p>
    Fórmula:C20H21FN6O5
    Pureza:99.86% - >99.99%
    Forma y color:Solid
    Peso molecular:444.42
  • 2-CHLOROMETHYL-1,1-DIOXO-1,2-DIHYDRO-1λ*6*-BENZO[D]ISOTHIAZOL-3-ONE

    CAS:
    2-CHLOROMETHYL-1,1-DIOXO-1,2-DIHYDRO-1LAMBDA*6*-BENZO[D]ISOTHIAZOL-3-ONE targets the Neutrophil elastase (human).
    Fórmula:C8H6ClNO3S
    Pureza:97.28%
    Forma y color:Solid
    Peso molecular:231.66
  • Bortezomib-pinanediol

    CAS:
    Bortezomib-pinanediol is a proteasome inhibitor. is a prodrug of Bortezomib.
    Fórmula:C29H39BN4O4
    Pureza:97.5%
    Forma y color:Yellow Solid
    Peso molecular:518.46
  • Delavirdine mesylate

    CAS:
    Delavirdine mesylate (BHAP-U 90152 (mesylate)) is a non-nucleoside reverse transcriptase inhibitor (NNRTI).
    Fórmula:C23H32N6O6S2
    Pureza:99.99%
    Forma y color:Light Brown Solid
    Peso molecular:552.67
  • Coblopasvir

    CAS:
    Coblopasvir is a pan-genotypic non-structural protein 5A (NS5A) inhibitor. It can be used to study chronic hepatitis C virus infection.
    Fórmula:C41H50N8O8
    Pureza:99.33%
    Forma y color:Solid
    Peso molecular:782.88
  • Letermovir

    CAS:
    Letermovir (AIC246) (AIC246) is a novel anti-CMV compound (EC50: about 5 nM in fibroblast cells). It targets the pUL56 subunit of the viral terminase complex.
    Fórmula:C29H28F4N4O4
    Pureza:99.85% - 99.87%
    Forma y color:Solid
    Peso molecular:572.55
  • Obefazimod

    CAS:
    <p>Obefazimod (ABX-464) is a potent anti-HIV agent. ABX464 inhibits HIV-1 replication in stimulated peripheral blood mononuclear cells (PBMCs).</p>
    Fórmula:C16H10ClF3N2O
    Pureza:99.86%
    Forma y color:Solid
    Peso molecular:338.71
  • KKI-5 acetate(97145-43-2 free base)


    KKI-5 acetate: Serine protease inhibitor, targets kallikrein/plasmin, potential anticancer and angioedema therapy.
    Fórmula:C37H59N11O11
    Pureza:99.44%
    Forma y color:Solid
    Peso molecular:833.95
  • Belnacasan

    CAS:
    Belnacasan (VX-765) is an orally active IL-converting enzyme/caspase-1 inhibitor.
    Fórmula:C24H33ClN4O6
    Pureza:96.53% - 99.5%
    Forma y color:Solid
    Peso molecular:508.99
  • Daclatasvir

    CAS:
    Daclatasvir (EBP 883/BMS-790052) is a potent HCV NS5A inhibitor with EC50 9-50 pM across various genotypes. Phase 3.
    Fórmula:C40H50N8O6
    Pureza:99.81% - 99.99%
    Forma y color:Solid
    Peso molecular:738.88
  • Dabigatran Etexilate Mesylate

    CAS:
    Dabigatran Etexilate Mesylate (BIBR 1048MS) is the orally active prodrug of dabigatran. Dabigatran is a reversible and selective, direct thrombin inhibitor.
    Fórmula:C34H41N7O5·CH4O3S
    Pureza:99.91%
    Forma y color:Solid
    Peso molecular:723.84
  • PTACH

    CAS:
    PTACH (Cpd 51) (NCH-51) is a SAHA-based inhibitor of human HDAC. It can potently inhibit the growth of various human Y cells (EC50: 1 to 10 μM).
    Fórmula:C20H26N2O2S2
    Pureza:87.44% - 99.74%
    Forma y color:Solid
    Peso molecular:390.56
  • Ximelagatran

    CAS:
    Ximelagatran, oral direct thrombin inhibitor, transforms to active melagatran in body.
    Fórmula:C24H35N5O5
    Pureza:95.48% - 99.60%
    Forma y color:Solid
    Peso molecular:473.57