Proteasas / Proteasoma
Los inhibidores de proteasas y proteasomas son compuestos que bloquean la actividad de las proteasas y del proteasoma, que están involucrados en la degradación y renovación de proteínas. Estos inhibidores son vitales para estudiar la regulación de la homeostasis proteica, el control del ciclo celular y la apoptosis. Los inhibidores de proteasas y proteasomas también se utilizan en el tratamiento de enfermedades como el cáncer, donde la degradación anormal de proteínas desempeña un papel en la progresión de la enfermedad. Al inhibir las proteasas o el proteasoma, estos compuestos pueden inducir la muerte celular en células cancerosas y son herramientas esenciales tanto en la investigación básica como en el desarrollo terapéutico. En CymitQuimica, ofrecemos una amplia gama de inhibidores de proteasas y proteasomas de alta calidad para apoyar su investigación en bioquímica, biología celular y desarrollo de fármacos.
Subcategorías de "Proteasas / Proteasoma"
- Acetil-CoA Carboxilasa(36 productos)
- Cisteína proteasa(110 productos)
- DPP-4(24 productos)
- Glutaminasa(44 productos)
- Proteasa del VIH(498 productos)
- PAI-1(26 productos)
- Inhibidores de la proteasa(50 productos)
- Receptor activado por proteasa(54 productos)
- Proteasoma(90 productos)
- Serina proteasa(51 productos)
- p97(15 productos)
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Se han encontrado 1011 productos de "Proteasas / Proteasoma"
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Thrombin Inhibitor 2
CAS:Thrombin Inhibitor 2 is a small molecule direct thrombin inhibitor. Thrombin Inhibitor 2 has antithrombotic activity.Fórmula:C19H16ClF3N6O2Pureza:98%Forma y color:SolidPeso molecular:452.82Alvelestat tosylate
CAS:Alvelestat can inhibit neutrophil elastase (NE), which acts an important role in NET formation.Fórmula:C32H30F3N5O7S2Pureza:98%Forma y color:SolidPeso molecular:717.73DPP-4-IN-2
CAS:DPP-4-IN-2, analog of Alogliptin with 79 nM IC50, is a research tool for diabetes.Fórmula:C18H18N6OForma y color:SolidPeso molecular:334.38Tyrosinase-IN-8
Tyrosinase-IN-8, a potent inhibitor of tyrosinase, demonstrates an inhibitory concentration (IC 50) value of 1.6 µM and exhibits low cytotoxicity whileFórmula:C16H12O4Forma y color:SolidPeso molecular:268.26SQ 32602
CAS:SQ 32602 is a cathepsin E inhibitor.Fórmula:C32H52N3O7PForma y color:SolidPeso molecular:621.74SJA6017
CAS:SJA6017: inhibits calpain-1/2, cathepsins B/L; prevents apoptosis, protects spinal cord, boosts function. IC50s: 7.5-78 nM.Fórmula:C17H25FN2O4SPureza:98%Forma y color:SolidPeso molecular:372.45CP-471474
CAS:MMP inhibitor with IC50: MMP-2 (0.7 nM), MMP-13 (0.9 nM), MMP-9 (13 nM), MMP-3 (16 nM), MMP-1 (1170 nM); reduces heart dilation post-infarct.Fórmula:C16H17FN2O5SPureza:98%Forma y color:SolidPeso molecular:368.38Sheng Gelieting
CAS:CGT-8012 inhibits DP-IV enzyme, aiding type II diabetes research, with an IC50 of 87 nM.Fórmula:C17H16F6N4OForma y color:SolidPeso molecular:406.33Tec-IN-21
CAS:Tec-IN-21 is an inhibitor of Tec kinase, it also blocks unconventional secretion of fibroblast growth factor 2 (FGF2).Fórmula:C16H15ClN4O2SPureza:98%Forma y color:SolidPeso molecular:362.83Cysteine Protease inhibitor hydrochloride
CAS:Cysteine Protease inhibitor hydrochloride is a cysteine protease inhibitor.Fórmula:C18H15ClN4OPureza:98%Forma y color:SolidPeso molecular:338.79JNJ-10329670
CAS:JNJ 10329670 is a highly potent (Ki of approximately 30 nM), nonpeptidic, noncovalent inhibitor of human cathepsin S with immunosuppressive activity.Fórmula:C30H34ClF3N6O3SForma y color:SolidPeso molecular:651.14HCV-IN-33
CAS:HCV-IN-33 (Compound (S)-3i) is an inhibitor of HCV entry.Fórmula:C31H36ClN5Forma y color:SolidPeso molecular:514.1Gü2602
CAS:Gü2602 inhibits the cathepsin K zymogen autocatalytic activation that is a potent, reversible inhibitor of cathepsin K (CatK) with a Ki of 0.013 nM for matureFórmula:C16H22N4O3Forma y color:SolidPeso molecular:318.37Tyrosinase-IN-3
CAS:Tyrosinase-IN-3 inhibits melanin production; potential for skin whitening and food preservation.Fórmula:C21H23NO5Forma y color:SolidPeso molecular:369.41Anticancer agent 82
CAS:Anticancer agent 82, a FiVe1 derivative, selectively targets VIM in cancer cells to disrupt mitosis, with improved oral bioavailability.Fórmula:C19H18Cl2N4OForma y color:SolidPeso molecular:389.28Tyrosinase-IN-6
CAS:Tyrosinase-IN-6 (4B) is a potent tyrosinase inhibitor (IC50=3.80 μM) with good antioxidant activity.Fórmula:C24H31N3O2Forma y color:SolidPeso molecular:393.52Alicapistat
CAS:Alicapistat (ABT-957) is a human calpains 1 and 2 inhibitor. It can potentially be used to treat Alzheimer's disease (AD).Fórmula:C25H27N3O4Pureza:98%Forma y color:SolidPeso molecular:433.5VEL-0230
CAS:VEL-0230 (NC-2300) is a cathespin K inhibitor boosting bone growth and reducing loss, targeting bone diseases and developed by Velcura Therapeutics.Fórmula:C14H24NNaO5Forma y color:SolidPeso molecular:309.33PK44 phosphate
CAS:PK44 phosphate is a potent inhibitor of dipeptidyl peptidase IV (DPP-IV) (IC50: 15.8 nM).Fórmula:C17H19F5N7O5PForma y color:SolidPeso molecular:527.349BAY8040
CAS:BAY8040 is a potent selective human neutrophilic elastase inhibitor with excellent potency and selectivity with promising pharmacokinetic characteristics.Fórmula:C21H16F3N5O2Forma y color:SolidPeso molecular:427.38
