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Receptor de opioides

Receptor de opioides

Los receptores opioides son un grupo de receptores acoplados a proteínas G que median los efectos de los opioides endógenos y exógenos. Estos receptores desempeñan un papel central en la modulación del dolor, la regulación del estado de ánimo y los comportamientos adictivos. Los agonistas y antagonistas de los receptores opioides se utilizan ampliamente en el manejo del dolor y el tratamiento de adicciones, así como en la investigación de trastornos neurológicos y psiquiátricos. En CymitQuimica, ofrecemos una selección integral de moduladores de receptores opioides de alta calidad para apoyar su investigación en neurobiología, manejo del dolor y terapia de adicciones.

Se han encontrado 296 productos de "Receptor de opioides"

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  • Trimebutine maleate

    CAS:
    <p>Trimebutine maleate (Polibutin) is a weak mu-opioid agonist and has antimuscarinic effects.</p>
    Fórmula:C26H33NO9
    Pureza:99.76% - 99.98%
    Forma y color:White Solid
    Peso molecular:503.55
  • ZT 52656A hydrochloride

    CAS:
    <p>ZT 52656A is a selective agonist of kappa opioid, and used for the prevention or alleviation of pain in the eye.</p>
    Fórmula:C19H26ClF3N2O
    Pureza:98.78%
    Forma y color:Solid
    Peso molecular:390.87
  • Meptazinol hydrochloride

    CAS:
    <p>Meptazinol hydrochloride (Meptazinol HCl) , a unique centrally opioid analgesic, is used as a narcotic antagonist with analgesic properties.</p>
    Fórmula:C15H23NO·HCl
    Pureza:99.75%
    Forma y color:White Solid
    Peso molecular:269.81
  • CP 866087

    CAS:
    <p>CP 866087 is an opioid receptor antagonist for the study of female sexual dysfunction.</p>
    Fórmula:C24H30N2O3S
    Pureza:99.22% - 99.74%
    Forma y color:Solid
    Peso molecular:426.57
  • BTRX-335140

    CAS:
    <p>BTRX-335140 (CYM-53093) is a potent and selective orally active κ-opioid receptor (KOR) antagonist with antagonistic activity.Cost-effective and quality-assured.</p>
    Fórmula:C25H32FN5O2
    Pureza:98% - 99.89%
    Forma y color:Solid
    Peso molecular:453.55
  • Apitegromab

    CAS:
    <p>Apitegromab (SRK-015) is a new myostatin inhibitor, an antibody targeting myostatin precursor, which can be used to study neuromuscular diseases including</p>
    Pureza:95% - 97.59% (SDS-PAGE); 99.78% (SEC-HPLC)
    Forma y color:Liquid
  • Moguisteine

    CAS:
    <p>Moguisteine (BBR-2173) is a new-type peripheral non-narcotic antitussive drug.</p>
    Fórmula:C16H21NO5S
    Pureza:99.98%
    Forma y color:Solid
    Peso molecular:339.41
  • Matrine

    CAS:
    <p>Matrine (Vegard), an alkaloid isolated from the Sophora genus, acts as a kappa opioid receptor agonist.</p>
    Fórmula:C15H24N2O
    Pureza:97.16% - >99.99%
    Forma y color:Solid
    Peso molecular:248.36
  • Sinomenine hydrochloride

    CAS:
    <p>Sinomenine hydrochloride (Kukoline hydrochloride) is extracted from Sinomenium Acutum Rehderett Wilson.</p>
    Fórmula:C19H24ClNO4
    Pureza:99.43%
    Forma y color:Solid
    Peso molecular:365.851
  • Alvimopan

    CAS:
    <p>Alvimopan is a potent opioid antagonist targeting gut receptors to reverse opioid effects on motility.</p>
    Fórmula:C25H32N2O4
    Pureza:99.47% - 99.78%
    Forma y color:Solid
    Peso molecular:424.53
  • Loperamide hydrochloride

    CAS:
    <p>Loperamide hydrochloride (ADL 2-1294) is a synthetic, piperidine derivative and opioid agonist with antidiarrheal activity.</p>
    Fórmula:C29H34Cl2N2O2
    Pureza:99.91% - >99.99%
    Forma y color:Crystals Practically Insoluble In Water
    Peso molecular:513.50
  • Naltrexone hydrochloride

    CAS:
    <p>Naltrexone hydrochloride (Naltrexone HCl) is a synthetic opioid antagonist used in the prevention of relapse of opiate addiction and alcoholism.</p>
    Fórmula:C20H24ClNO4
    Pureza:98.72% - 99.65%
    Forma y color:White Crystalline Powder
    Peso molecular:377.862
  • Samidorphan HCl

    CAS:
    <p>Samidorphan HCl is an orally active and highly potent modulator of the opioid system that binds to μ‐opioid, κ‐opioid, and delta-opioid receptors.</p>
    Fórmula:C21H27ClN2O4
    Pureza:96.79% - 97.85%
    Forma y color:Soild
    Peso molecular:406.9
  • LY2940094

    CAS:
    <p>LY2940094 (LY-2940094) decreases ethanol self-administration in animal models.</p>
    Fórmula:C22H23ClF2N4O2S
    Pureza:99.4%
    Forma y color:Solid
    Peso molecular:480.96
  • DPDPE

    CAS:
    <p>DPDPE is selective δ-opioid receptor agonist peptide.</p>
    Fórmula:C30H39N5O7S2
    Pureza:98%
    Forma y color:Solid
    Peso molecular:645.79
  • ICI 174,864

    CAS:
    <p>Selective δ opioid antagonist. Exhibits partial agonist in vitro activity at δ receptors at high concentrations.</p>
    Fórmula:C38H53N5O7
    Pureza:98%
    Forma y color:White Solid
    Peso molecular:691.87
  • Neurotransmitter Receptor Compound Library


    <p>A unique collection of 1513 neurotransmitter receptor compounds, can be used for HTS and HCS screening;</p>
    Forma y color:Odour Solid
  • Biphalin TFA

    CAS:
    <p>Biphalin TFA is an opioid peptide analog that penetrates the blood-brain barrier (BBB) and encompasses two active enkephalin pharmacophores.</p>
    Fórmula:C46H56N10O10·xC2HF3O2
    Pureza:98%
    Forma y color:Solid
    Peso molecular:909.00 (free base)
  • β-Endorphin, equine TFA


    <p>β-Endorphin, equine TFA, an endogenous opioid peptide, demonstrates high affinity binding to μ/δ opioid receptors and possesses analgesic properties [1] [2] [3</p>
    Fórmula:C156H249F3N42O46S
    Forma y color:Solid
    Peso molecular:3537.96
  • Dermorphin

    CAS:
    <p>Dermorphin is agonist of μ-opioid receptor (MOR) agonist.</p>
    Fórmula:C40H50N8O10
    Pureza:98.82%
    Forma y color:Solid
    Peso molecular:802.87