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Receptor de glucagón

Receptor de glucagón

Los receptores de glucagón son GPCR que median los efectos del glucagón, una hormona involucrada en la regulación de la homeostasis de la glucosa al promover la descomposición del glucógeno y la liberación de glucosa desde el hígado. Estos receptores son cruciales en la gestión de los niveles de azúcar en sangre y son de particular interés en el estudio de la diabetes y los trastornos metabólicos. Los antagonistas de los receptores de glucagón se están explorando como posibles tratamientos para la hiperglucemia en la diabetes tipo 2. En CymitQuimica, ofrecemos una variedad de moduladores de receptores de glucagón de alta calidad para apoyar su investigación en endocrinología, diabetes y regulación metabólica.

Se han encontrado 164 productos de "Receptor de glucagón"

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  • Glucagon (1-29), bovine, human, porcine hydrochloride

    CAS:
    <p>Glucagon (1-29), bovine, human, porcine hydrochloride is a peptide hormone, produced by pancreatic α-cells. Glucagon increases HNF4α phosphorylation.</p>
    Fórmula:C153H225N43O49S·ClH
    Pureza:95.65% - 98.03%
    Forma y color:Solid
    Peso molecular:3519.21
  • Tirzepatide monosodium salt


    <p>Tirzepatide sodium salt (LY3298176 sodium salt) is a GIP and GLP-1 receptor agonist with neuroprotective activity and can be used to treat obesity.</p>
    Fórmula:C225H347N48O68Na
    Pureza:99.69%
    Forma y color:Soild
    Peso molecular:4835.51
  • Avexitide acetate

    CAS:
    <p>Avexitide acetate (exendin 9-39) is a potent glucagon-like peptide 1 receptor (GLP-1R) antagonist for the study of post-obesity hypoglycemia.</p>
    Fórmula:C155H246N40O53S
    Pureza:96.64% - 98.65%
    Forma y color:Solid
    Peso molecular:3549.91
  • Crotedumab

    CAS:
    <p>Crotedumab (REGN1193) is a humanized antibody targeting GCGR, which reduces fasting blood glucose and improves glucose tolerance, used in diabetes research.</p>
    Pureza:>95%
    Forma y color:Liquid
  • Retatrutide

    CAS:
    <p>Retatrutide (LY3437943) is a triple agonist of GCGR, GIPR and GLP-1R that can be used to study obesity.</p>
    Fórmula:C221H342N46O68
    Pureza:98.31%
    Forma y color:Solid
    Peso molecular:4732.09
  • PF-06882961

    CAS:
    <p>PF-06882961 is an orally bioavailable glucagon-like peptide-1 receptor (GLP-1R) agonist.</p>
    Fórmula:C31H30FN5O4
    Pureza:98.06% - 99.54%
    Forma y color:Solid
    Peso molecular:555.6
  • Volagidemab

    CAS:
    <p>Anti-CD34 Antibody is a CHO-expressed humanized monoclonal antibody targeting CD34, which can be used for the study of neurological and cardiovascular diseases.</p>
    Pureza:97.8% (SDS-PAGE); 98% (SEC-HPLC) - 97.8% (SDS-PAGE); 98% (SEC-HPLC)
    Forma y color:Liquid
  • Retatrutide sodium salt


    <p>Retatrutide sodium salt is a glucagon receptor and glucagon-like peptide-1 receptor agonist for the study of type 2 diabetes mellitus.</p>
    Pureza:99.97%
    Forma y color:Soild
  • VU0453379

    CAS:
    <p>VU0453379 is a highly selective and central nervous system penetrant positive allosteric modulator of glucagon-like peptide-1R (EC50: 1.3 μM).</p>
    Fórmula:C26H34N4O2
    Pureza:98%
    Forma y color:Solid
    Peso molecular:434.57
  • GLP-1R Antagonist 1

    CAS:
    <p>GLP-1R Antagonist 1 is an orally active, CNS penetrant and non-competitive glucagon-like peptide 1 receptor (GLP-1R) antagonist (IC50: 650 nM).</p>
    Fórmula:C16H11ClF6N4O2
    Pureza:99.84%
    Forma y color:Solid
    Peso molecular:440.73
  • GLP-1 receptor agonist 4

    CAS:
    <p>GLP-1 receptor agonist 4 targets GLP-1R, EC50 64.5 nM, potential diabetes treatment research.</p>
    Fórmula:C51H44Cl2N4O6
    Pureza:98%
    Forma y color:Solid
    Peso molecular:879.82
  • HAEGTFTSD

    CAS:
    <p>HAEGTFTSD is GLP-1's initial segment; GLP-1 (7-36) amide, tied to food intake, stems from preproglucagon in L-cells.</p>
    Fórmula:C40H57N11O17
    Pureza:98%
    Forma y color:Solid
    Peso molecular:963.94
  • Tirzepatide

    CAS:
    <p>Tirzepatide (LY-3298176) is a dual glucose-dependent polypeptide (GIP) (EC50=0.042 nM) and glucagon-like peptide-1 (GLP-1) (EC50=0.086 nM) receptor agonist.</p>
    Fórmula:C225H348N48O68
    Pureza:99.52% - 99.99%
    Forma y color:Solid
    Peso molecular:4813.45
  • Glucagon-like peptide 1 (1-37), human

    CAS:
    <p>Human GLP-1 (1-37) is a potent GLP-1 receptor agonist without impact on rat food intake or insulin secretion.</p>
    Fórmula:C186H275N51O59
    Pureza:98%
    Forma y color:Solid
    Peso molecular:4169.48
  • Cinnamtannin A2

    CAS:
    <p>Cinnamtannin A2, a tetrameric procyanidin, boosts GLP-1, insulin, CRH expression, and has antioxidant, anti-diabetic, nephroprotective properties.</p>
    Fórmula:C60H50O24
    Forma y color:Solid
    Peso molecular:1155.02
  • (S, R)-LSN 3318839

    CAS:
    <p>(S,R)-LSN 3318839 enhances GLP-1R, shows strong blood sugar lowering in animals, works with sitagliptin.</p>
    Fórmula:C26H23Cl2N3O2
    Pureza:99.57%
    Forma y color:Soild
    Peso molecular:480.39
  • Tirzepatide hydrochloride


    <p>Tirzepatide HCl is a dual GIP and GLP-1 receptor agonist.</p>
    Fórmula:C225H349N48O68Cl
    Pureza:98%
    Forma y color:Solid
    Peso molecular:4849.91
  • GLP-1 moiety from Dulaglutide


    <p>GLP-1 moiety from Dulaglutide is a 31-amino acid fragment of Dulaglutide which is a glucagon-like peptide 1 receptor (GLP-1) agonist.</p>
    Fórmula:C149H221N37O49
    Pureza:98%
    Forma y color:Solid
    Peso molecular:3314.62
  • V-0219 hydrochloride


    <p>V-0219 hydrochloride: oral GLP-1R PAM for obesity-linked diabetes study.</p>
    Fórmula:C20H26ClF3N4O2
    Pureza:99.97%
    Forma y color:Soild
    Peso molecular:446.89
  • GLP-1 (9-36) amide

    CAS:
    <p>GLP-1 (9-36) amide is an antagonist at the human GLP-1 receptor.</p>
    Fórmula:C140H214N36O43
    Pureza:97%
    Forma y color:Solid
    Peso molecular:3089.41