
Receptor de dopamina
Los receptores de dopamina son un grupo de receptores acoplados a proteínas G (GPCR) que responden al neurotransmisor dopamina, jugando un papel clave en la regulación del movimiento, la motivación, la recompensa y varias funciones cognitivas. Estos receptores se dividen en familias similares a D1 y D2, cada una con funciones y perfiles farmacológicos distintos. Los moduladores de los receptores de dopamina se estudian ampliamente por sus aplicaciones en el tratamiento de la enfermedad de Parkinson, la esquizofrenia, la adicción y otros trastornos neuropsiquiátricos. En CymitQuimica, ofrecemos una amplia gama de moduladores de receptores de dopamina de alta calidad para apoyar su investigación en neurociencia, salud mental y señalización GPCR.
Se han encontrado 443 productos de "Receptor de dopamina"
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BP 897
CAS:BP 897: potent selective dopamine D3 agonist, weak D2 antagonist. Ki: 0.92 nM (D3), 61 nM (D2), low affinity at D1/D4.Fórmula:C26H31N3O2Pureza:99.44%Forma y color:SolidPeso molecular:417.54Ref: TM-T9100
1mg80,00€5mg162,00€10mg227,00€25mg379,00€50mg540,00€100mg730,00€200mg938,00€1mL*10mM (DMSO)177,00€Rotigotine-
CAS:Rotigotine (N-0923) is a non-ergot dopamine receptor agonist used in the therapy of Parkinson disease and restless leg syndrome.Fórmula:C19H25NOSPureza:98.08% - 99.59%Forma y color:SolidPeso molecular:315.47Ref: TM-T6647
5mg52,00€10mg78,00€25mg145,00€50mg255,00€100mg378,00€200mg552,00€500mg868,00€1mL*10mM (DMSO)55,00€Perospirone
CAS:Perospirone (Lullan) is an antagonist of serotonin 5HT2A receptors and dopamine D2 receptors.Fórmula:C23H30N4O2SPureza:99.23%Forma y color:White PowderPeso molecular:426.57carfenazine
CAS:<p>carfenazine targets the Dopamine receptor and is used for schizophrenia research.</p>Fórmula:C24H31N3O2SPureza:98.06%Forma y color:SolidPeso molecular:425.59Sonepiprazole hydrochloride
CAS:Sonepiprazole HCl is a a selective dopamine D4 antagonist.Fórmula:C21H28ClN3O3SForma y color:SolidPeso molecular:437.98SK609
CAS:SK609: selective dopamine D3 agonist; enhances impaired paw function, corrects asymmetry in hemiparkinson rats.Fórmula:C10H14ClNForma y color:SolidPeso molecular:183.68Nuciferine
CAS:Nuciferine ((-)-Nuciferine) is an alkaloid found within the plants Nymphaea caerulea and Nelumbo nucifera.Fórmula:C19H21NO2Pureza:98.76% - 99.79%Forma y color:SolidPeso molecular:295.38Raclopride
CAS:Raclopride is a selective antagonist of dopamine D2/D3 receptor.Fórmula:C15H20Cl2N2O3Pureza:99.17%Forma y color:SolidPeso molecular:347.24Haloperidol lactate
CAS:Haloperidol lactate: a potent antipsychotic for acute/chronic schizophrenia and polyarousal syndrome research.Fórmula:C24H29ClFNO5Forma y color:SolidPeso molecular:465.95L-DOPA methyl ester (hydrochloride)
CAS:<p>L-DOPA methyl ester (LDME) is an agonist of dopamine D1 receptor.</p>Fórmula:C10H14ClNO4Pureza:98.69% - 99.81%Forma y color:White SolidPeso molecular:247.675Tetrahydropalmatine hydrochloride
CAS:Tetrahydropalmatine HCl (Gindarine) is a muscle relaxant alkaloid from Corydalis plants.Fórmula:C21H26ClNO4Pureza:98% - 99.59%Forma y color:SolidPeso molecular:391.888Zuclopenthixol dihydrochloride
CAS:Zuclopenthixol dihydrochloride is an D1 and D2 dopamine receptors antagonist.Fórmula:C22H27Cl3N2OSPureza:98%Forma y color:SolidPeso molecular:473.89AHN 1-055 hydrochloride
CAS:AHN 1-055 hydrochloride (3α-Bis-(4-fluorophenyl) Methoxytropane hydrochloride) is an inhibitor of dopamine transporter (DAT) and dopamine uptake(IC50 = 71 nM).Fórmula:C21H24ClF2NOPureza:99.89%Forma y color:SolidPeso molecular:379.87Ref: TM-T39429
2mg35,00€5mg52,00€10mg80,00€25mg137,00€50mg202,00€100mg311,00€200mg467,00€1mL*10mM (DMSO)52,00€Clebopride
CAS:Clebopride is antidopaminergic. Clebopride also has an effect of antiemetic.Fórmula:C20H24ClN3O2Forma y color:SolidPeso molecular:373.88L-745870 hydrochloride
CAS:L-745870 hydrochloride has excellent brain penetration. L-745870 hydrochloride is a high-affinity, selective and orally active human dopamine D4 receptorFórmula:C18H20Cl2N4Pureza:97.36%Forma y color:SolidPeso molecular:363.28Ref: TM-T11799
5mg40,00€10mg65,00€25mg111,00€50mg178,00€100mg259,00€200mg374,00€1mL*10mM (DMSO)34,00€Vanoxerine dihydrochloride
CAS:Vanoxerine dihydrochloride (GBR-12909 dihydrochloride) is a potent inhibitor that blocks dopamine uptake (IC50 : 1-51 nM)Fórmula:C28H34Cl2F2N2OPureza:98.16% - 98.35%Forma y color:White SolidPeso molecular:523.49Domperidone monomaleate
CAS:Domperidone monomaleate, a selective oral dopamine-2 antagonist, aids gastric motility and has antiemetic properties.Fórmula:C26H28ClN5O6Forma y color:SolidPeso molecular:541.98Mesdopetam
CAS:Mesdopetam (IRL790), a D3 antagonist, has Ki=90 nM, IC50=9.8 μM, stabilizes psychomotors, used in Parkinson's research.Fórmula:C12H18FNO3SForma y color:SolidPeso molecular:275.34Metergoline
CAS:Metergoline (Methergoline) is a dopamine agonist and serotonin antagonist.Fórmula:C25H29N3O2Pureza:99.83% - 99.97%Forma y color:SolidPeso molecular:403.52Bromopride hydrochloride
CAS:Bromopride HCl: Salt of a D2 blocker used for upper GI disorders, like dyspepsia and emesis.Fórmula:C14H23BrClN3O2Forma y color:SolidPeso molecular:380.71
