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Receptor de dopamina

Receptor de dopamina

Los receptores de dopamina son un grupo de receptores acoplados a proteínas G (GPCR) que responden al neurotransmisor dopamina, jugando un papel clave en la regulación del movimiento, la motivación, la recompensa y varias funciones cognitivas. Estos receptores se dividen en familias similares a D1 y D2, cada una con funciones y perfiles farmacológicos distintos. Los moduladores de los receptores de dopamina se estudian ampliamente por sus aplicaciones en el tratamiento de la enfermedad de Parkinson, la esquizofrenia, la adicción y otros trastornos neuropsiquiátricos. En CymitQuimica, ofrecemos una amplia gama de moduladores de receptores de dopamina de alta calidad para apoyar su investigación en neurociencia, salud mental y señalización GPCR.

Se han encontrado 443 productos de "Receptor de dopamina"

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  • BP 897

    CAS:
    BP 897: potent selective dopamine D3 agonist, weak D2 antagonist. Ki: 0.92 nM (D3), 61 nM (D2), low affinity at D1/D4.
    Fórmula:C26H31N3O2
    Pureza:99.44%
    Forma y color:Solid
    Peso molecular:417.54

    Ref: TM-T9100

    1mg
    80,00€
    5mg
    162,00€
    10mg
    227,00€
    25mg
    379,00€
    50mg
    540,00€
    100mg
    730,00€
    200mg
    938,00€
    1mL*10mM (DMSO)
    177,00€
  • Rotigotine-

    CAS:
    Rotigotine (N-0923) is a non-ergot dopamine receptor agonist used in the therapy of Parkinson disease and restless leg syndrome.
    Fórmula:C19H25NOS
    Pureza:98.08% - 99.59%
    Forma y color:Solid
    Peso molecular:315.47

    Ref: TM-T6647

    5mg
    52,00€
    10mg
    78,00€
    25mg
    145,00€
    50mg
    255,00€
    100mg
    378,00€
    200mg
    552,00€
    500mg
    868,00€
    1mL*10mM (DMSO)
    55,00€
  • Perospirone

    CAS:
    Perospirone (Lullan) is an antagonist of serotonin 5HT2A receptors and dopamine D2 receptors.
    Fórmula:C23H30N4O2S
    Pureza:99.23%
    Forma y color:White Powder
    Peso molecular:426.57

    Ref: TM-T4576

    10mg
    50,00€
    25mg
    87,00€
    50mg
    140,00€
    100mg
    234,00€
    200mg
    325,00€
    1mL*10mM (DMSO)
    35,00€
  • carfenazine

    CAS:
    <p>carfenazine targets the Dopamine receptor and is used for schizophrenia research.</p>
    Fórmula:C24H31N3O2S
    Pureza:98.06%
    Forma y color:Solid
    Peso molecular:425.59

    Ref: TM-T9827

    1mg
    92,00€
    5mg
    183,00€
    10mg
    274,00€
    25mg
    472,00€
    50mg
    A consultar
  • Sonepiprazole hydrochloride

    CAS:
    Sonepiprazole HCl is a a selective dopamine D4 antagonist.
    Fórmula:C21H28ClN3O3S
    Forma y color:Solid
    Peso molecular:437.98

    Ref: TM-T70262

    25mg
    1.586,00€
    50mg
    2.072,00€
    100mg
    2.660,00€
  • SK609

    CAS:
    SK609: selective dopamine D3 agonist; enhances impaired paw function, corrects asymmetry in hemiparkinson rats.
    Fórmula:C10H14ClN
    Forma y color:Solid
    Peso molecular:183.68

    Ref: TM-T70618

    25mg
    1.444,00€
    50mg
    1.882,00€
    100mg
    2.375,00€
  • Nuciferine

    CAS:
    Nuciferine ((-)-Nuciferine) is an alkaloid found within the plants Nymphaea caerulea and Nelumbo nucifera.
    Fórmula:C19H21NO2
    Pureza:98.76% - 99.79%
    Forma y color:Solid
    Peso molecular:295.38

    Ref: TM-T3369

    5mg
    47,00€
    10mg
    60,00€
    25mg
    119,00€
    50mg
    170,00€
    100mg
    255,00€
    500mg
    622,00€
    1mL*10mM (DMSO)
    50,00€
  • Raclopride

    CAS:
    Raclopride is a selective antagonist of dopamine D2/D3 receptor.
    Fórmula:C15H20Cl2N2O3
    Pureza:99.17%
    Forma y color:Solid
    Peso molecular:347.24

    Ref: TM-T7635

    5mg
    49,00€
    10mg
    67,00€
    25mg
    124,00€
    50mg
    208,00€
    100mg
    314,00€
    1mL*10mM (DMSO)
    55,00€
  • Haloperidol lactate

    CAS:
    Haloperidol lactate: a potent antipsychotic for acute/chronic schizophrenia and polyarousal syndrome research.
    Fórmula:C24H29ClFNO5
    Forma y color:Solid
    Peso molecular:465.95

    Ref: TM-T62975

    25mg
    1.444,00€
    50mg
    1.882,00€
    100mg
    2.375,00€
  • L-DOPA methyl ester (hydrochloride)

    CAS:
    <p>L-DOPA methyl ester (LDME) is an agonist of dopamine D1 receptor.</p>
    Fórmula:C10H14ClNO4
    Pureza:98.69% - 99.81%
    Forma y color:White Solid
    Peso molecular:247.675

    Ref: TM-T7654

    100mg
    52,00€
    500mg
    130,00€
    1mL*10mM (DMSO)
    37,00€
  • Tetrahydropalmatine hydrochloride

    CAS:
    Tetrahydropalmatine HCl (Gindarine) is a muscle relaxant alkaloid from Corydalis plants.
    Fórmula:C21H26ClNO4
    Pureza:98% - 99.59%
    Forma y color:Solid
    Peso molecular:391.888

    Ref: TM-T2917

    25mg
    40,00€
    50mg
    51,00€
    100mg
    74,00€
    200mg
    97,00€
  • Zuclopenthixol dihydrochloride

    CAS:
    Zuclopenthixol dihydrochloride is an D1 and D2 dopamine receptors antagonist.
    Fórmula:C22H27Cl3N2OS
    Pureza:98%
    Forma y color:Solid
    Peso molecular:473.89

    Ref: TM-T4117L2

    25mg
    1.444,00€
    50mg
    1.882,00€
    100mg
    2.375,00€
  • AHN 1-055 hydrochloride

    CAS:
    AHN 1-055 hydrochloride (3α-Bis-(4-fluorophenyl) Methoxytropane hydrochloride) is an inhibitor of dopamine transporter (DAT) and dopamine uptake(IC50 = 71 nM).
    Fórmula:C21H24ClF2NO
    Pureza:99.89%
    Forma y color:Solid
    Peso molecular:379.87

    Ref: TM-T39429

    2mg
    35,00€
    5mg
    52,00€
    10mg
    80,00€
    25mg
    137,00€
    50mg
    202,00€
    100mg
    311,00€
    200mg
    467,00€
    1mL*10mM (DMSO)
    52,00€
  • Clebopride

    CAS:
    Clebopride is antidopaminergic. Clebopride also has an effect of antiemetic.
    Fórmula:C20H24ClN3O2
    Forma y color:Solid
    Peso molecular:373.88

    Ref: TM-T7569L

    25mg
    1.444,00€
    50mg
    1.882,00€
    100mg
    2.375,00€
  • L-745870 hydrochloride

    CAS:
    L-745870 hydrochloride has excellent brain penetration. L-745870 hydrochloride is a high-affinity, selective and orally active human dopamine D4 receptor
    Fórmula:C18H20Cl2N4
    Pureza:97.36%
    Forma y color:Solid
    Peso molecular:363.28

    Ref: TM-T11799

    5mg
    40,00€
    10mg
    65,00€
    25mg
    111,00€
    50mg
    178,00€
    100mg
    259,00€
    200mg
    374,00€
    1mL*10mM (DMSO)
    34,00€
  • Vanoxerine dihydrochloride

    CAS:
    Vanoxerine dihydrochloride (GBR-12909 dihydrochloride) is a potent inhibitor that blocks dopamine uptake (IC50 : 1-51 nM)
    Fórmula:C28H34Cl2F2N2O
    Pureza:98.16% - 98.35%
    Forma y color:White Solid
    Peso molecular:523.49

    Ref: TM-T7153

    10mg
    52,00€
    25mg
    86,00€
    50mg
    120,00€
    100mg
    170,00€
    1mL*10mM (DMSO)
    37,00€
  • Domperidone monomaleate

    CAS:
    Domperidone monomaleate, a selective oral dopamine-2 antagonist, aids gastric motility and has antiemetic properties.
    Fórmula:C26H28ClN5O6
    Forma y color:Solid
    Peso molecular:541.98

    Ref: TM-T63819

    25mg
    1.444,00€
    50mg
    1.882,00€
    100mg
    2.375,00€
  • Mesdopetam

    CAS:
    Mesdopetam (IRL790), a D3 antagonist, has Ki=90 nM, IC50=9.8 μM, stabilizes psychomotors, used in Parkinson's research.
    Fórmula:C12H18FNO3S
    Forma y color:Solid
    Peso molecular:275.34

    Ref: TM-T38828

    5mg
    922,00€
  • Metergoline

    CAS:
    Metergoline (Methergoline) is a dopamine agonist and serotonin antagonist.
    Fórmula:C25H29N3O2
    Pureza:99.83% - 99.97%
    Forma y color:Solid
    Peso molecular:403.52

    Ref: TM-T4008

    10mg
    34,00€
    25mg
    A consultar
    50mg
    A consultar
    1mL*10mM (DMSO)
    34,00€
  • Bromopride hydrochloride

    CAS:
    Bromopride HCl: Salt of a D2 blocker used for upper GI disorders, like dyspepsia and emesis.
    Fórmula:C14H23BrClN3O2
    Forma y color:Solid
    Peso molecular:380.71

    Ref: TM-T69152

    25mg
    1.444,00€
    50mg
    1.882,00€
    100mg
    2.375,00€