
Receptor de dopamina
Los receptores de dopamina son un grupo de receptores acoplados a proteínas G (GPCR) que responden al neurotransmisor dopamina, jugando un papel clave en la regulación del movimiento, la motivación, la recompensa y varias funciones cognitivas. Estos receptores se dividen en familias similares a D1 y D2, cada una con funciones y perfiles farmacológicos distintos. Los moduladores de los receptores de dopamina se estudian ampliamente por sus aplicaciones en el tratamiento de la enfermedad de Parkinson, la esquizofrenia, la adicción y otros trastornos neuropsiquiátricos. En CymitQuimica, ofrecemos una amplia gama de moduladores de receptores de dopamina de alta calidad para apoyar su investigación en neurociencia, salud mental y señalización GPCR.
Se han encontrado 443 productos de "Receptor de dopamina"
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Nomifensine
CAS:Nomifensine ((±)-Nomifensin) is a norepinephrine-dopamine reuptake inhibitor that prevents dopamine reuptake into synaptosomes.Fórmula:C16H18N2Pureza:99.83% - ≥95%Forma y color:SolidPeso molecular:238.33Tavapadon
CAS:Tavapadon (CVL-751) is an orally active and highly selective dopamine D1/D5 receptor partial agonist.Fórmula:C19H16F3N3O3Pureza:99.33% - 99.8%Forma y color:SolidPeso molecular:391.34Ref: TM-T16999
1mg81,00€5mg170,00€10mg274,00€25mg502,00€50mg705,00€100mg938,00€1mL*10mM (DMSO)188,00€L-745870 hydrochloride
CAS:L-745870 hydrochloride has excellent brain penetration. L-745870 hydrochloride is a high-affinity, selective and orally active human dopamine D4 receptorFórmula:C18H20Cl2N4Pureza:97.36%Forma y color:SolidPeso molecular:363.28Ref: TM-T11799
5mg40,00€10mg65,00€25mg111,00€50mg178,00€100mg259,00€200mg374,00€1mL*10mM (DMSO)34,00€Ansofaxine hydrochloride
CAS:Ansofaxine hydrochloride (LY03005) is a serotonin-norepinephrine-dopamine reuptake inhibitor (IC50s: 723, 763 and 491 nM, respectively).Fórmula:C24H32ClNO3Pureza:99.57% - 99.77%Forma y color:SolidPeso molecular:417.97FAUC-365
CAS:FAUC-365 is a D3 dopamine receptor agonist.Fórmula:C23H25Cl2N3OSPureza:99.62%Forma y color:SolidPeso molecular:462.44Ref: TM-T21667
1mg52,00€5mg111,00€10mg169,00€25mg323,00€50mg512,00€100mg740,00€500mg1.539,00€1mL*10mM (DMSO)123,00€Haloperidol lactate
CAS:Haloperidol lactate: a potent antipsychotic for acute/chronic schizophrenia and polyarousal syndrome research.Fórmula:C24H29ClFNO5Forma y color:SolidPeso molecular:465.95Clebopride
CAS:Clebopride is antidopaminergic. Clebopride also has an effect of antiemetic.Fórmula:C20H24ClN3O2Forma y color:SolidPeso molecular:373.88Mesdopetam hemitartrate
CAS:Mesdopetam hemitartrate antagonizes dopamine D3 receptor (Ki=90 nM; IC50=9.8 μM) and stabilizes psychomotor function.Fórmula:C28H42F2N2O12S2Pureza:99.98%Forma y color:SolidPeso molecular:700.77Lurasidone hydrochloride
CAS:Lurasidone HCl: Atypical antipsychotic, treats schizophrenia & bipolar, affects dopamine, serotonin & adrenergic receptors.Fórmula:C28H36N4O2S·HClPureza:99.51%Forma y color:SolidPeso molecular:529.14Ref: TM-T1735
5mg42,00€10mg63,00€25mg80,00€50mg96,00€100mg144,00€200mg225,00€500mg472,00€1mL*10mM (DMSO)A consultarGBR 12935 dihydrochloride
CAS:GBR 12935 dihydrochloride (GBR 12935) can induce the increase of the extracellular levels of dopamine to basal levels.Fórmula:C28H36Cl2N2OPureza:99.09% - ≥95%Forma y color:SolidPeso molecular:487.5Loxapine
CAS:Loxapine, a dibenzoxazepine antipsychotic, treats schizophrenia by blocking D2/D4 and serotonin receptors. Related to clozapine.Fórmula:C18H18ClN3OPureza:99.88%Forma y color:Pale Yellowish Crystals From Petroleum Ether SolidPeso molecular:327.81Tetrahydropalmatine hydrochloride
CAS:Tetrahydropalmatine HCl (Gindarine) is a muscle relaxant alkaloid from Corydalis plants.Fórmula:C21H26ClNO4Pureza:98% - 99.59%Forma y color:SolidPeso molecular:391.888Lurasidone
CAS:Lurasidone (SM-13496) is an antagonist of both dopamine D2 and 5-HT7(IC50=1.68 and 0.495 nM, respectively).It also a partial agonist of 5-HT1A receptor(IC50 : 6Fórmula:C28H36N4O2SPureza:99.78% - 99.91%Forma y color:SolidPeso molecular:492.68Azaperone
CAS:Azaperone, a sedative and antiemetic veterinary tranquilizer, belongs to pyridinylpiperazine and butyrophenone classes.Fórmula:C19H22FN3OPureza:98.73%Forma y color:White Or Off-White CrystallinePeso molecular:327.4Metergoline
CAS:Metergoline (Methergoline) is a dopamine agonist and serotonin antagonist.Fórmula:C25H29N3O2Pureza:99.83% - 99.97%Forma y color:SolidPeso molecular:403.52Sertindole
CAS:<p>Sertindole, atypical antipsychotic, targets D2, 5-HT1D, 5-HT2A, 5-HT2C receptors (Kds: 2.7, 20, 0.14, 6 nM).</p>Fórmula:C24H26ClFN4OPureza:99.87% - 99.92%Forma y color:Off-White To Pale Yellow SolidPeso molecular:440.94Clebopride malate
CAS:Clebopride malate is a dopamine antagonist drug Used to treat functional gastrointestinal disorders such as nausea or vomiting.Fórmula:C24H30ClN3O7Pureza:99.52%Forma y color:SolidPeso molecular:507.96Flupentixol dihydrochloride
CAS:Flupentixol dihydrochloride is used in therapy of schizophrenia as well as in anxiolytic and depressive disorders.Fórmula:C23H27Cl2F3N2OSPureza:98.76% - >99.99%Forma y color:White Or Off-White SolidPeso molecular:507.43Carmoxirole (free base)
CAS:Carmoxirole: a dopamine D2 agonist, reduces pre-load/afterload, aids heart failure, lowers blood pressure by inhibiting noradrenaline release.Fórmula:C24H26N2O2Forma y color:SolidPeso molecular:374.48D-tetrahydropalmatine
CAS:D-Tetrahydropalmatine inhibits OCT1, reducing MCT uptake and hepatocyte damage in MDCK-hOCT1 cells and rat livers.Fórmula:C21H25NO4Pureza:99.34%Forma y color:SolidPeso molecular:355.43Ref: TM-T4S0779
2mg44,00€5mg64,00€10mg97,00€25mg182,00€50mg273,00€100mg393,00€200mg558,00€1mL*10mM (DMSO)65,00€
