
Receptor de dopamina
Los receptores de dopamina son un grupo de receptores acoplados a proteínas G (GPCR) que responden al neurotransmisor dopamina, jugando un papel clave en la regulación del movimiento, la motivación, la recompensa y varias funciones cognitivas. Estos receptores se dividen en familias similares a D1 y D2, cada una con funciones y perfiles farmacológicos distintos. Los moduladores de los receptores de dopamina se estudian ampliamente por sus aplicaciones en el tratamiento de la enfermedad de Parkinson, la esquizofrenia, la adicción y otros trastornos neuropsiquiátricos. En CymitQuimica, ofrecemos una amplia gama de moduladores de receptores de dopamina de alta calidad para apoyar su investigación en neurociencia, salud mental y señalización GPCR.
Se han encontrado 443 productos de "Receptor de dopamina"
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Rotundine
CAS:Rotundine (Gindarine) (L-tetrahydropalmatine, L-THP) is a selective dopamine D1 receptor antagonist with IC50 of 166 nM.Fórmula:C21H25NO4Pureza:99.8% - 99.91%Forma y color:Off-White SolidPeso molecular:355.43FAUC-365
CAS:FAUC-365 is a D3 dopamine receptor agonist.Fórmula:C23H25Cl2N3OSPureza:99.62%Forma y color:SolidPeso molecular:462.44Ref: TM-T21667
1mg52,00€5mg111,00€10mg169,00€25mg323,00€50mg512,00€100mg740,00€500mg1.539,00€1mL*10mM (DMSO)123,00€Haloperidol lactate
CAS:Haloperidol lactate: a potent antipsychotic for acute/chronic schizophrenia and polyarousal syndrome research.Fórmula:C24H29ClFNO5Forma y color:SolidPeso molecular:465.95Piribedil
CAS:Piribedil (Trivastan) is a dopamine D2 agonist, used in the treatment of Parkinson's disease.Fórmula:C16H18N4O2Pureza:99.79% - 99.82%Forma y color:SolidPeso molecular:298.34Tetrahydropalmatine hydrochloride
CAS:Tetrahydropalmatine HCl (Gindarine) is a muscle relaxant alkaloid from Corydalis plants.Fórmula:C21H26ClNO4Pureza:98% - 99.59%Forma y color:SolidPeso molecular:391.888Metergoline
CAS:Metergoline (Methergoline) is a dopamine agonist and serotonin antagonist.Fórmula:C25H29N3O2Pureza:99.83% - 99.97%Forma y color:SolidPeso molecular:403.52SKF38393 hydrobromide
CAS:SKF38393 hydrobromide is the salt form of SKF38393.a dopamine D1 receptor agonist that increases the expression of Shati/Nat8L mRNA in the NAc of mice;Fórmula:C16H18BrNO2Pureza:98.99%Forma y color:SolidPeso molecular:336.22Bromopride hydrochloride
CAS:Bromopride HCl: Salt of a D2 blocker used for upper GI disorders, like dyspepsia and emesis.Fórmula:C14H23BrClN3O2Forma y color:SolidPeso molecular:380.71Carmoxirole (free base)
CAS:Carmoxirole: a dopamine D2 agonist, reduces pre-load/afterload, aids heart failure, lowers blood pressure by inhibiting noradrenaline release.Fórmula:C24H26N2O2Forma y color:SolidPeso molecular:374.48Lurasidone
CAS:Lurasidone (SM-13496) is an antagonist of both dopamine D2 and 5-HT7(IC50=1.68 and 0.495 nM, respectively).It also a partial agonist of 5-HT1A receptor(IC50 : 6Fórmula:C28H36N4O2SPureza:99.78% - 99.91%Forma y color:SolidPeso molecular:492.68Dasotraline
CAS:Dasotraline: a triple reuptake inhibitor targeting DA, NE, and 5-HT with IC50 values of 4, 6, 11 nM. Possible new antidepressant class.Fórmula:C16H15Cl2NForma y color:SolidPeso molecular:292.2Perospirone
CAS:Perospirone (Lullan) is an antagonist of serotonin 5HT2A receptors and dopamine D2 receptors.Fórmula:C23H30N4O2SPureza:99.23%Forma y color:White PowderPeso molecular:426.57Clebopride
CAS:Clebopride is antidopaminergic. Clebopride also has an effect of antiemetic.Fórmula:C20H24ClN3O2Forma y color:SolidPeso molecular:373.88PD 168568
CAS:PD 168568: Oral DRD4 antagonist, selective over D2/D3, K_i - 8.8 nM. Used in GBM research.Fórmula:C22H27N3OForma y color:SolidPeso molecular:349.47Alizapride
CAS:Alizapride is an antagonist of dopamine receptor. Alizapride can be used in human digestive disorders which is a potent antiemetic [1] [3].Fórmula:C16H21N5O2Forma y color:SolidPeso molecular:315.37JNJ-37822681
CAS:JNJ-37822681 is a novel, highly selective dopamine D₂ receptor antagonist characterized by a rapid dissociation rate from the dopamine D₂ receptor.Fórmula:C17H17F5N4Pureza:99.84%Forma y color:SolidPeso molecular:372.34Domperidone monomaleate
CAS:Domperidone monomaleate, a selective oral dopamine-2 antagonist, aids gastric motility and has antiemetic properties.Fórmula:C26H28ClN5O6Forma y color:SolidPeso molecular:541.98Tiapride
CAS:Tiapride, an atypical neuroleptic, is a selective dopamine D2-receptor antagonist with varying IC50 values for D1-D4.Fórmula:C15H24N2O4SForma y color:SolidPeso molecular:328.43Rotigotine Hydrochloride
CAS:<p>Rotigotine HCl, D3-preferential dopamine agonist, is 50x stronger than quinpirole in anti-Parkinson's efficacy.</p>Fórmula:C19H26ClNOSPureza:99.53% - 99.56%Forma y color:Almost White To White Crystalline PowderPeso molecular:351.93BP 897
CAS:BP 897: potent selective dopamine D3 agonist, weak D2 antagonist. Ki: 0.92 nM (D3), 61 nM (D2), low affinity at D1/D4.Fórmula:C26H31N3O2Pureza:99.44%Forma y color:SolidPeso molecular:417.54Ref: TM-T9100
1mg80,00€5mg162,00€10mg227,00€25mg379,00€50mg540,00€100mg730,00€200mg938,00€1mL*10mM (DMSO)177,00€
