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Receptor de dopamina

Receptor de dopamina

Los receptores de dopamina son un grupo de receptores acoplados a proteínas G (GPCR) que responden al neurotransmisor dopamina, jugando un papel clave en la regulación del movimiento, la motivación, la recompensa y varias funciones cognitivas. Estos receptores se dividen en familias similares a D1 y D2, cada una con funciones y perfiles farmacológicos distintos. Los moduladores de los receptores de dopamina se estudian ampliamente por sus aplicaciones en el tratamiento de la enfermedad de Parkinson, la esquizofrenia, la adicción y otros trastornos neuropsiquiátricos. En CymitQuimica, ofrecemos una amplia gama de moduladores de receptores de dopamina de alta calidad para apoyar su investigación en neurociencia, salud mental y señalización GPCR.

Se han encontrado 445 productos de "Receptor de dopamina"

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  • MOR agonist-3


    MOR agonist-3 (Compound 84) is a dual D3R/MOR antagonist with K i values of 382 nM and 55.2 nM, respectively.
    Forma y color:Odour Solid

    Ref: TM-T81763

    5mg
    A consultar
    50mg
    A consultar
  • Amisulpride hydrochloride

    CAS:
    Amisulpride is an antagonist of 5-HT7 receptor and dopamine D2 and D3 receptors. It modulates beta 2- arresting signaling and increases neurite outgrowth.
    Fórmula:C17H28ClN3O4S
    Forma y color:Solid
    Peso molecular:405.94

    Ref: TM-T0811L

    25mg
    1.369,00€
  • Dopamine D2 receptor agonist-2

    CAS:

    Dopamine D2 receptor agonist-2 (Dopamine D2 Receptor) is a ligand targeting the dopamine D2 receptor.

    Fórmula:C25H31Cl2N5OS
    Pureza:98.93%
    Forma y color:Soild
    Peso molecular:520.52

    Ref: TM-T60075

    1mg
    38,00€
    5mg
    71,00€
    10mg
    90,00€
    25mg
    148,00€
    50mg
    210,00€
    100mg
    314,00€
    200mg
    452,00€
  • 7-Hydroxy-PIPAT maleate

    CAS:
    7-Hydroxy-PIPAT maleate is a D3R agonist.
    Fórmula:C16H22INO
    Forma y color:Solid
    Peso molecular:371.262

    Ref: TM-T38188

    10mg
    130,00€
    50mg
    513,00€
  • A 77636 hydrochloride

    CAS:
    A 77636 hydrochloride is a potent, orally active, selective and long acting dopamine D1 receptor agonist (pKi=7.40; Ki=39.8 nM).
    Fórmula:C20H28ClNO3
    Pureza:99.57%
    Forma y color:Solid
    Peso molecular:365.89

    Ref: TM-T21782

    1mg
    90,00€
    5mg
    205,00€
    10mg
    299,00€
    25mg
    505,00€
    50mg
    710,00€
  • ADTN hydrobromide

    CAS:

    ADTN hydrobromide (6,7-ADTN) is a dopamine receptor agonist (EC50s = 3.5 and 0.65 μM in rat striatal and nucleus accumbens homogenates, respectively).

    Fórmula:C10H14BrNO2
    Forma y color:Solid
    Peso molecular:260.13

    Ref: TM-T37150

    5mg
    139,00€
    25mg
    610,00€
    50mg
    1.064,00€
  • MOR agonist-2


    Compound 46, designated as MOR agonist-2, serves as a D3R antagonist and a MOR agonist with respective K i values of 7.26 nM and 564 nM.
    Fórmula:C37H47Cl2N5O3
    Pureza:98%
    Forma y color:Solid
    Peso molecular:680.71

    Ref: TM-T79547

    5mg
    A consultar
    50mg
    A consultar
  • LE 300

    CAS:
    LE 300 represents a structurally novel type of antagonists acting preferentially at the dopamine D(1)/D(5)receptors and the serotonin 5-HT(2A)receptor.
    Fórmula:C20H22N2
    Pureza:97.91% - 98.79%
    Forma y color:Solid
    Peso molecular:290.4

    Ref: TM-T22921

    1mg
    93,00€
    5mg
    197,00€
    10mg
    294,00€
    25mg
    492,00€
    50mg
    700,00€
    100mg
    954,00€
    500mg
    1.908,00€
  • PF-4363467

    CAS:
    PF-4363467 is a dopamine D3/D2 receptor antagonist that reduces opioid-seeking behavior without the side effects associated with D2 receptors. It has a Ki value of 3.1 nM for D3R and 692 nM for D2R.
    Fórmula:C22H30N2O3S
    Forma y color:Solid
    Peso molecular:402.55

    Ref: TM-T203495

    10mg
    A consultar
    50mg
    A consultar
  • Preclamol hydrochloride

    CAS:
    Preclamol hydrochloride: selective dopamine agonist with research potential in schizophrenia.
    Fórmula:C14H22ClNO
    Forma y color:Solid
    Peso molecular:255.78

    Ref: TM-T73684

    2mg
    34,00€
  • Cabergoline

    CAS:

    Cabergoline (FCE-21336), an ergot-derived dopamine D2-like agonist, targets D2/D3/5-HT2B, normalizes prolactin, controls pituitary tumors.

    Fórmula:C26H37N5O2
    Pureza:97.69% - 99.86%
    Forma y color:White Crystalline Solid
    Peso molecular:451.6

    Ref: TM-T14853

    1mg
    40,00€
    5mg
    85,00€
    10mg
    119,00€
    25mg
    230,00€
    50mg
    426,00€
    100mg
    627,00€
  • O-2172

    CAS:
    O-2172 is a carbocyclic analogue serving as an inhibitor of dopamine transporter (DAT), exhibiting IC50 values of 47 nM for DAT and 7000 nM for the serotonin transporter (SERT).
    Fórmula:C14H16Cl2O2
    Forma y color:Solid
    Peso molecular:287.18

    Ref: TM-T203629

    10mg
    A consultar
    50mg
    A consultar
  • Haloperidol D4

    CAS:
    Haloperidol D4 is deuterium-labeled haloperidol.
    Fórmula:C21H23ClFNO2
    Pureza:98%
    Forma y color:Solid
    Peso molecular:379.89

    Ref: TM-T11535

    1mg
    750,00€
  • ADTN

    CAS:
    ADTN is an agonist of the dopamine receptor.
    Fórmula:C10H13NO2
    Pureza:98%
    Forma y color:Solid
    Peso molecular:179.22

    Ref: TM-T23643

    5mg
    A consultar
  • (R)-Preclamol hydrochloride

    CAS:
    (R)-Preclamol HCl is a dopamine agonist stimulating both auto and postsynaptic receptors.
    Fórmula:C14H22ClNO
    Forma y color:Solid
    Peso molecular:255.78

    Ref: TM-T73685

    2mg
    34,00€
  • Secretoneurin, rat

    CAS:
    Secretoneurin, rat, a 33-amino acid polypeptide, is generated by proteolytic processing of secretogranin II (SgII).
    Fórmula:C159H252N40O58
    Pureza:98%
    Forma y color:Solid
    Peso molecular:3651.95

    Ref: TM-TP1597

    100mg
    A consultar
    500mg
    A consultar
  • Fluphenazine free base

    CAS:
    Flufenazine: antipsychotic for schizophrenia, blocks dopamine D2 receptors, reduces hallucinations and delusions.
    Fórmula:C22H26F3N3OS
    Forma y color:Solid
    Peso molecular:437.52

    Ref: TM-T0068L2

    25mg
    1.369,00€
  • Quinelorane

    CAS:
    Quinelorane is dextrorotary isomer.
    Fórmula:C14H22N4
    Forma y color:Solid
    Peso molecular:246.35

    Ref: TM-T34226

    25mg
    A consultar
    50mg
    A consultar
    100mg
    A consultar
  • N-0500 HCl

    CAS:
    N-0500 HCl, a potent DA receptor agonist, displaces [3H]DP_x005f_x0002_5,6-ADTN with an IC50 of 3nM.
    Fórmula:C15H22ClNO2
    Pureza:98.85% - 99.54%
    Forma y color:Solid
    Peso molecular:283.79

    Ref: TM-T60107

    5mg
    35,00€
    10mg
    55,00€
    1mL*10mM (DMSO)
    A consultar
  • Adrogolide HCl

    CAS:
    Adrogolide Hydrochloride is a selective dopamine receptor D1 agonist.
    Fórmula:C22H26ClNO4S
    Forma y color:Solid
    Peso molecular:435.96

    Ref: TM-T29674

    25mg
    2.043,00€
    50mg
    2.682,00€
    100mg
    3.600,00€