
Receptor de dopamina
Los receptores de dopamina son un grupo de receptores acoplados a proteínas G (GPCR) que responden al neurotransmisor dopamina, jugando un papel clave en la regulación del movimiento, la motivación, la recompensa y varias funciones cognitivas. Estos receptores se dividen en familias similares a D1 y D2, cada una con funciones y perfiles farmacológicos distintos. Los moduladores de los receptores de dopamina se estudian ampliamente por sus aplicaciones en el tratamiento de la enfermedad de Parkinson, la esquizofrenia, la adicción y otros trastornos neuropsiquiátricos. En CymitQuimica, ofrecemos una amplia gama de moduladores de receptores de dopamina de alta calidad para apoyar su investigación en neurociencia, salud mental y señalización GPCR.
Se han encontrado 445 productos de "Receptor de dopamina"
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MOR agonist-3
MOR agonist-3 (Compound 84) is a dual D3R/MOR antagonist with K i values of 382 nM and 55.2 nM, respectively.Forma y color:Odour SolidAmisulpride hydrochloride
CAS:Amisulpride is an antagonist of 5-HT7 receptor and dopamine D2 and D3 receptors. It modulates beta 2- arresting signaling and increases neurite outgrowth.Fórmula:C17H28ClN3O4SForma y color:SolidPeso molecular:405.94Dopamine D2 receptor agonist-2
CAS:Dopamine D2 receptor agonist-2 (Dopamine D2 Receptor) is a ligand targeting the dopamine D2 receptor.
Fórmula:C25H31Cl2N5OSPureza:98.93%Forma y color:SoildPeso molecular:520.527-Hydroxy-PIPAT maleate
CAS:7-Hydroxy-PIPAT maleate is a D3R agonist.Fórmula:C16H22INOForma y color:SolidPeso molecular:371.262A 77636 hydrochloride
CAS:A 77636 hydrochloride is a potent, orally active, selective and long acting dopamine D1 receptor agonist (pKi=7.40; Ki=39.8 nM).Fórmula:C20H28ClNO3Pureza:99.57%Forma y color:SolidPeso molecular:365.89ADTN hydrobromide
CAS:ADTN hydrobromide (6,7-ADTN) is a dopamine receptor agonist (EC50s = 3.5 and 0.65 μM in rat striatal and nucleus accumbens homogenates, respectively).
Fórmula:C10H14BrNO2Forma y color:SolidPeso molecular:260.13MOR agonist-2
Compound 46, designated as MOR agonist-2, serves as a D3R antagonist and a MOR agonist with respective K i values of 7.26 nM and 564 nM.Fórmula:C37H47Cl2N5O3Pureza:98%Forma y color:SolidPeso molecular:680.71LE 300
CAS:LE 300 represents a structurally novel type of antagonists acting preferentially at the dopamine D(1)/D(5)receptors and the serotonin 5-HT(2A)receptor.Fórmula:C20H22N2Pureza:97.91% - 98.79%Forma y color:SolidPeso molecular:290.4PF-4363467
CAS:PF-4363467 is a dopamine D3/D2 receptor antagonist that reduces opioid-seeking behavior without the side effects associated with D2 receptors. It has a Ki value of 3.1 nM for D3R and 692 nM for D2R.Fórmula:C22H30N2O3SForma y color:SolidPeso molecular:402.55Preclamol hydrochloride
CAS:Preclamol hydrochloride: selective dopamine agonist with research potential in schizophrenia.Fórmula:C14H22ClNOForma y color:SolidPeso molecular:255.78Cabergoline
CAS:Cabergoline (FCE-21336), an ergot-derived dopamine D2-like agonist, targets D2/D3/5-HT2B, normalizes prolactin, controls pituitary tumors.
Fórmula:C26H37N5O2Pureza:97.69% - 99.86%Forma y color:White Crystalline SolidPeso molecular:451.6O-2172
CAS:O-2172 is a carbocyclic analogue serving as an inhibitor of dopamine transporter (DAT), exhibiting IC50 values of 47 nM for DAT and 7000 nM for the serotonin transporter (SERT).Fórmula:C14H16Cl2O2Forma y color:SolidPeso molecular:287.18Haloperidol D4
CAS:Haloperidol D4 is deuterium-labeled haloperidol.Fórmula:C21H23ClFNO2Pureza:98%Forma y color:SolidPeso molecular:379.89ADTN
CAS:ADTN is an agonist of the dopamine receptor.Fórmula:C10H13NO2Pureza:98%Forma y color:SolidPeso molecular:179.22(R)-Preclamol hydrochloride
CAS:(R)-Preclamol HCl is a dopamine agonist stimulating both auto and postsynaptic receptors.Fórmula:C14H22ClNOForma y color:SolidPeso molecular:255.78Secretoneurin, rat
CAS:Secretoneurin, rat, a 33-amino acid polypeptide, is generated by proteolytic processing of secretogranin II (SgII).Fórmula:C159H252N40O58Pureza:98%Forma y color:SolidPeso molecular:3651.95Fluphenazine free base
CAS:Flufenazine: antipsychotic for schizophrenia, blocks dopamine D2 receptors, reduces hallucinations and delusions.Fórmula:C22H26F3N3OSForma y color:SolidPeso molecular:437.52Quinelorane
CAS:Quinelorane is dextrorotary isomer.Fórmula:C14H22N4Forma y color:SolidPeso molecular:246.35N-0500 HCl
CAS:N-0500 HCl, a potent DA receptor agonist, displaces [3H]DP_x005f_x0002_5,6-ADTN with an IC50 of 3nM.Fórmula:C15H22ClNO2Pureza:98.85% - 99.54%Forma y color:SolidPeso molecular:283.79Adrogolide HCl
CAS:Adrogolide Hydrochloride is a selective dopamine receptor D1 agonist.Fórmula:C22H26ClNO4SForma y color:SolidPeso molecular:435.96

