
Receptor de dopamina
Los receptores de dopamina son un grupo de receptores acoplados a proteínas G (GPCR) que responden al neurotransmisor dopamina, jugando un papel clave en la regulación del movimiento, la motivación, la recompensa y varias funciones cognitivas. Estos receptores se dividen en familias similares a D1 y D2, cada una con funciones y perfiles farmacológicos distintos. Los moduladores de los receptores de dopamina se estudian ampliamente por sus aplicaciones en el tratamiento de la enfermedad de Parkinson, la esquizofrenia, la adicción y otros trastornos neuropsiquiátricos. En CymitQuimica, ofrecemos una amplia gama de moduladores de receptores de dopamina de alta calidad para apoyar su investigación en neurociencia, salud mental y señalización GPCR.
Se han encontrado 407 productos de "Receptor de dopamina"
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D3R ligand 1
<p>D3R Ligand 1 (compound 23b) is a potent, selective antagonist of the dopamine D3 receptor (Ki=66 nM), incorporating a THPB template.</p>Fórmula:C27H37NO5Pureza:98%Forma y color:SolidPeso molecular:455.59ADTN
CAS:<p>ADTN is an agonist of the dopamine receptor.</p>Fórmula:C10H13NO2Pureza:98%Forma y color:SolidPeso molecular:179.22Cabergoline
CAS:<p>Cabergoline (FCE-21336), an ergot-derived dopamine D2-like agonist, targets D2/D3/5-HT2B, normalizes prolactin, controls pituitary tumors.</p>Fórmula:C26H37N5O2Pureza:97.69% - 99.86%Forma y color:White Crystalline SolidPeso molecular:451.6A 77636 hydrochloride
CAS:<p>A 77636 hydrochloride is a potent, orally active, selective and long acting dopamine D1 receptor agonist (pKi=7.40; Ki=39.8 nM).</p>Fórmula:C20H28ClNO3Pureza:99.57%Forma y color:SolidPeso molecular:365.89O-2172
CAS:<p>O-2172 is a carbocyclic analogue serving as an inhibitor of dopamine transporter (DAT), exhibiting IC50 values of 47 nM for DAT and 7000 nM for the serotonin transporter (SERT).</p>Fórmula:C14H16Cl2O2Forma y color:SolidPeso molecular:287.18(R)-Preclamol hydrochloride
CAS:<p>(R)-Preclamol HCl is a dopamine agonist stimulating both auto and postsynaptic receptors.</p>Fórmula:C14H22ClNOForma y color:SolidPeso molecular:255.78Haloperidol D4
CAS:<p>Haloperidol D4 is deuterium-labeled haloperidol.</p>Fórmula:C21H23ClFNO2Pureza:98%Forma y color:SolidPeso molecular:379.89Preclamol hydrochloride
CAS:<p>Preclamol hydrochloride: selective dopamine agonist with research potential in schizophrenia.</p>Fórmula:C14H22ClNOForma y color:SolidPeso molecular:255.78Secretoneurin, rat
CAS:<p>Secretoneurin, rat, a 33-amino acid polypeptide, is generated by proteolytic processing of secretogranin II (SgII).</p>Fórmula:C159H252N40O58Pureza:98%Forma y color:SolidPeso molecular:3651.95Fluphenazine free base
CAS:<p>Flufenazine: antipsychotic for schizophrenia, blocks dopamine D2 receptors, reduces hallucinations and delusions.</p>Fórmula:C22H26F3N3OSForma y color:SolidPeso molecular:437.52Adrogolide HCl
CAS:<p>Adrogolide Hydrochloride is a selective dopamine receptor D1 agonist.</p>Fórmula:C22H26ClNO4SForma y color:SolidPeso molecular:435.96N-0500 HCl
CAS:<p>N-0500 HCl, a potent DA receptor agonist, displaces [3H]DP_x005f_x0002_5,6-ADTN with an IC50 of 3nM.</p>Fórmula:C15H22ClNO2Pureza:98.85% - 99.54%Forma y color:SolidPeso molecular:283.79(-)-GSK598809 hydrochloride
CAS:<p>(-)-GSK598809 hydrochloride, a DRD3 selective antagonist, may correct reward deficits in substance dependence.</p>Fórmula:C22H24ClF4N5OSPureza:98.36%Forma y color:SoildPeso molecular:517.97Quinelorane
CAS:<p>Quinelorane is dextrorotary isomer.</p>Fórmula:C14H22N4Forma y color:SolidPeso molecular:246.35PF-4363467
CAS:<p>PF-4363467 is a dopamine D3/D2 receptor antagonist that reduces opioid-seeking behavior without the side effects associated with D2 receptors. It has a Ki value of 3.1 nM for D3R and 692 nM for D2R.</p>Fórmula:C22H30N2O3SForma y color:SolidPeso molecular:402.55D3R/MOR antagonist 2
<p>Compound 121, a D3R/MOR antagonist with K i values of 361 nM and 85.2 nM for D3R and MOR respectively, has the potential for analgesic effects through MOR</p>Fórmula:C25H31ClN2OPureza:98%Forma y color:SolidPeso molecular:410.98ST-836 hydrochloride
CAS:<p>ST-836 hydrochloride is a dopamine receptor ligand; Antiparkinsonian agent .</p>Fórmula:C23H35ClN4OSPureza:98%Forma y color:SolidPeso molecular:451.07cis-(Z)-Flupentixol dihydrochloride
CAS:<p>cis-(Z)-Flupentixol dihydrochloride (Emergil) is a dopamine receptor antagonist.</p>Fórmula:C23H27Cl2F3N2OSPureza:98.07%Forma y color:SolidPeso molecular:507.44Haloperidol (D4')
CAS:<p>Haloperidol D4' is deuterium-labeled haloperidol. Haloperidol is a dopamine D2 receptor antagonist.</p>Fórmula:C21H23ClFNO2Pureza:98%Forma y color:SolidPeso molecular:379.89Eticlopride hydrochloride
CAS:<p>Eticlopride, an antipsychotic, is a Selective dopamine D2/D3 receptor antagonist (Ki: 0.5/0.16 nM).</p>Fórmula:C17H25ClN2O3·HClPureza:98%Forma y color:SolidPeso molecular:377.31

