
Receptor de dopamina
Los receptores de dopamina son un grupo de receptores acoplados a proteínas G (GPCR) que responden al neurotransmisor dopamina, jugando un papel clave en la regulación del movimiento, la motivación, la recompensa y varias funciones cognitivas. Estos receptores se dividen en familias similares a D1 y D2, cada una con funciones y perfiles farmacológicos distintos. Los moduladores de los receptores de dopamina se estudian ampliamente por sus aplicaciones en el tratamiento de la enfermedad de Parkinson, la esquizofrenia, la adicción y otros trastornos neuropsiquiátricos. En CymitQuimica, ofrecemos una amplia gama de moduladores de receptores de dopamina de alta calidad para apoyar su investigación en neurociencia, salud mental y señalización GPCR.
Se han encontrado 445 productos de "Receptor de dopamina"
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Opromazine hydrochloride
CAS:Opromazine hydrochloride, a phenothiazine antipsychotic, blocks brain dopamine receptors to treat schizophrenia and psychosis.Fórmula:C17H20Cl2N2OSPureza:98.03%Forma y color:SolidPeso molecular:371.32Ref: TM-T50054
1mg38,00€5mg82,00€10mg111,00€25mg182,00€50mg269,00€100mg389,00€200mg555,00€1mL*10mM (DMSO)94,00€WAY-100635 Monomaleate
CAS:WAY-100635 maleate is a selective 5-hydroxytryptamine 1A receptor antagonist with an IC50 value of 0.91 nM and a Ki value of 0.39 nM.Fórmula:C25H34N4O2·C4H4O4Pureza:98.44% - 99.46%Forma y color:SolidPeso molecular:538.64Ref: TM-T2631
2mg43,00€5mg63,00€10mg89,00€25mg170,00€50mg315,00€100mg470,00€200mg680,00€500mg1.054,00€1mL*10mM (DMSO)74,00€Thozalinone
CAS:Thozalinone is a psychostimulant agent inducing the release of norepinephrine and dopamine.Fórmula:C11H12N2O2Pureza:99.68%Forma y color:SolidPeso molecular:204.23Nomifensine maleate
CAS:Nomifensine maleate (Nomifensine (maleate)) is a selective inhibitor of dopamine uptake. Nomifensine maleate is used in adult attention deficit disorder.
Fórmula:C20H22N2O4Pureza:98.46%Forma y color:SolidPeso molecular:354.4GBR 12935
CAS:GBR-12935: selective dopamine inhibitor, used in Parkinson's research.Fórmula:C28H34N2OForma y color:SolidPeso molecular:414.58Alizapride hydrochloride
CAS:Alizapride hydrochloride (Alizapride HCl) is a dopamine receptor antagonist used for the treatment of nausea and vomiting.Fórmula:C16H21N5O2·HClPureza:99.35% - 99.48%Forma y color:CoaPeso molecular:351.83Raclopride tartrate
CAS:Raclopride is a selective antagonist on D2 dopamine receptor ( D2 Ki: 1.8 nm, D3 Ki: 3.5 nm, D4 Ki: 2400, D1 Ki: 18000 nM).Fórmula:C19H26Cl2N2O9Forma y color:SolidPeso molecular:497.32Bisacodyl
CAS:Bisacodyl (Fenilaxan) is a diphenylmethane stimulant laxative used for the treatment of constipation and for bowel evacuation.Fórmula:C22H19NO4Pureza:99.45% - 99.78%Forma y color:Smaller Than 50 Microns Predominate White To Off-White Crystalline PowderPeso molecular:361.39Raclopride
CAS:Raclopride is a selective antagonist of dopamine D2/D3 receptor.Fórmula:C15H20Cl2N2O3Pureza:99.17%Forma y color:SolidPeso molecular:347.24BisfluoroModafinil
CAS:CRL-40940 is a selective dopaminergic reuptake inhibitorFórmula:C15H13F2NO2SPureza:99.19%Forma y color:SolidPeso molecular:309.339-FLUORENOL
CAS:9-FLUORENOL is a dopamine reuptake inhibitor with IC50 of 9 μM, and a major metabolite of a compound developed as a wakefulness-promoting agent.Fórmula:C13H10OPureza:99.98%Forma y color:Off-White Crystalline PowderPeso molecular:182.22Butyrophenone
CAS:Butyrophenone (NSC-8463) is a chemical compound. Some of its derivatives are used to treat various psychiatric disorders.Fórmula:C10H12OPureza:99.84%Forma y color:Colourless To Yellow LiquidPeso molecular:148.23-CPMT
CAS:3-CPMT (FC-1) is a dopamine uptake inhibitor and a potent long-acting antihistaminic agent.Fórmula:C21H25Cl2NOPureza:99.03%Forma y color:SolidPeso molecular:378.33NGB 2904
CAS:NGB 2904 is a potent and selective antagonist of dopamine D3 receptor. NGB2904 potently antagonizes mitogenesis stimulated by quinpirole (IC50 = 6.8 nM).Fórmula:C28H29Cl2N3OPureza:98.79%Forma y color:SolidPeso molecular:494.46Ref: TM-T28167
2mg38,00€5mg55,00€10mg86,00€25mg155,00€50mg264,00€100mg374,00€500mgA consultar1mL*10mM (DMSO)72,00€ML417
CAS:ML417 is a selective and brain penetrant agonist of D3 Dopamine (EC50 : 38 nM).Fórmula:C22H25N3O3Pureza:98.4% - 99.42%Forma y color:SolidPeso molecular:379.45Dimethocaine
CAS:Dimethocaine (Larocaine) is a local anesthetic which also effects on the central nervous system acting as dopamine-reuptake-inhibitor.Fórmula:C16H26N2O2Pureza:99.52%Forma y color:SolidPeso molecular:278.39(S)-Amisulpride
CAS:(S)-Amisulpride ((S) Amisulpride) (Esamisulpride) is a potent dopamine D2/D3 receptor antagonist.Fórmula:C17H27N3O4SPureza:98.38%Forma y color:SolidPeso molecular:369.48Ref: TM-T26375
1mg34,00€5mg84,00€10mg123,00€25mg225,00€50mg358,00€100mg485,00€200mg622,00€1mL*10mM (DMSO)94,00€(+)-PD 128907 hydrochloride
CAS:(+)-PD 128907 hydrochloride is an agonist of D3 dopamine receptor .
Fórmula:C14H20ClNO3Pureza:97.76%Forma y color:SolidPeso molecular:285.77GSK163090
CAS:GSK163090 is a specific and orally active 5-HT1A/B/D receptor antagonist (pKis: 9.4/8.5/9.7, and 6.3/6.7 for 5-HT1A/B/D, and dopamine D2/D3).Fórmula:C25H29N5OPureza:99.2%Forma y color:SolidPeso molecular:415.53Ref: TM-TQ0311
1mg34,00€2mg49,00€5mg75,00€10mg118,00€25mgA consultar50mgA consultar1mL*10mM (DMSO)82,00€OS-3-106
CAS:OS-3-106 is a novel arylamide phenylpiperazines, as partial agonists at the D3R in the adenylyl cyclase inhibition assay.Fórmula:C25H30N4O2SPureza:99.4% - 99.57%Forma y color:SolidPeso molecular:450.6
