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Receptor de dopamina

Receptor de dopamina

Los receptores de dopamina son un grupo de receptores acoplados a proteínas G (GPCR) que responden al neurotransmisor dopamina, jugando un papel clave en la regulación del movimiento, la motivación, la recompensa y varias funciones cognitivas. Estos receptores se dividen en familias similares a D1 y D2, cada una con funciones y perfiles farmacológicos distintos. Los moduladores de los receptores de dopamina se estudian ampliamente por sus aplicaciones en el tratamiento de la enfermedad de Parkinson, la esquizofrenia, la adicción y otros trastornos neuropsiquiátricos. En CymitQuimica, ofrecemos una amplia gama de moduladores de receptores de dopamina de alta calidad para apoyar su investigación en neurociencia, salud mental y señalización GPCR.

Se han encontrado 407 productos de "Receptor de dopamina"

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  • Bisacodyl

    CAS:
    <p>Bisacodyl (Fenilaxan) is a diphenylmethane stimulant laxative used for the treatment of constipation and for bowel evacuation.</p>
    Fórmula:C22H19NO4
    Pureza:99.45% - 99.78%
    Forma y color:Smaller Than 50 Microns Predominate White To Off-White Crystalline Powder
    Peso molecular:361.39
  • BisfluoroModafinil

    CAS:
    <p>CRL-40940 is a selective dopaminergic reuptake inhibitor</p>
    Fórmula:C15H13F2NO2S
    Pureza:99.19%
    Forma y color:Solid
    Peso molecular:309.33
  • (S)-Amisulpride

    CAS:
    <p>(S)-Amisulpride ((S) Amisulpride) (Esamisulpride) is a potent dopamine D2/D3 receptor antagonist.</p>
    Fórmula:C17H27N3O4S
    Pureza:98.38%
    Forma y color:Solid
    Peso molecular:369.48
  • WAY-100635 Monomaleate

    CAS:
    <p>WAY-100635 maleate is a selective 5-hydroxytryptamine 1A receptor antagonist with an IC50 value of 0.91 nM and a Ki value of 0.39 nM.</p>
    Fórmula:C25H34N4O2·C4H4O4
    Pureza:98.44% - 99.46%
    Forma y color:Solid
    Peso molecular:538.64
  • (+)-PD 128907 hydrochloride

    CAS:
    <p>(+)-PD 128907 hydrochloride is an agonist of D3 dopamine receptor .</p>
    Fórmula:C14H20ClNO3
    Pureza:97.76%
    Forma y color:Solid
    Peso molecular:285.77
  • Butyrophenone

    CAS:
    <p>Butyrophenone (NSC-8463) is a chemical compound. Some of its derivatives are used to treat various psychiatric disorders.</p>
    Fórmula:C10H12O
    Pureza:99.84%
    Forma y color:Colourless To Yellow Liquid
    Peso molecular:148.2
  • 9-FLUORENOL

    CAS:
    <p>9-FLUORENOL is a dopamine reuptake inhibitor with IC50 of 9 μM, and a major metabolite of a compound developed as a wakefulness-promoting agent.</p>
    Fórmula:C13H10O
    Pureza:99.98%
    Forma y color:Off-White Crystalline Powder
    Peso molecular:182.22
  • NGB 2904

    CAS:
    <p>NGB 2904 is a potent and selective antagonist of dopamine D3 receptor. NGB2904 potently antagonizes mitogenesis stimulated by quinpirole (IC50 = 6.8 nM).</p>
    Fórmula:C28H29Cl2N3O
    Pureza:98.79%
    Forma y color:Solid
    Peso molecular:494.46
  • Glaucine

    CAS:
    <p>Glaucine: antitussive, antioxidative, antiviral, may fight arthritis, boosts IL-10, hinders breast cancer cell spread by inhibiting MMP-9 and NF-κB.</p>
    Fórmula:C21H25NO4
    Pureza:99.42% - 99.56%
    Forma y color:Solid
    Peso molecular:355.43
  • DOPEXAMINE

    CAS:
    <p>Dopexamine is a dopaminergic agonist</p>
    Fórmula:C22H32N2O2
    Pureza:99.42%
    Forma y color:Solid
    Peso molecular:356.5
  • ML417

    CAS:
    <p>ML417 is a selective and brain penetrant agonist of D3 Dopamine (EC50 : 38 nM).</p>
    Fórmula:C22H25N3O3
    Pureza:98.4% - 99.42%
    Forma y color:Solid
    Peso molecular:379.45
  • 3-CPMT

    CAS:
    <p>3-CPMT (FC-1) is a dopamine uptake inhibitor and a potent long-acting antihistaminic agent.</p>
    Fórmula:C21H25Cl2NO
    Pureza:99.03%
    Forma y color:Solid
    Peso molecular:378.33
  • Dimethocaine

    CAS:
    <p>Dimethocaine (Larocaine) is a local anesthetic which also effects on the central nervous system acting as dopamine-reuptake-inhibitor.</p>
    Fórmula:C16H26N2O2
    Pureza:99.52%
    Forma y color:Solid
    Peso molecular:278.39
  • GSK163090

    CAS:
    <p>GSK163090 is a specific and orally active 5-HT1A/B/D receptor antagonist (pKis: 9.4/8.5/9.7, and 6.3/6.7 for 5-HT1A/B/D, and dopamine D2/D3).</p>
    Fórmula:C25H29N5O
    Pureza:99.2%
    Forma y color:Solid
    Peso molecular:415.53
  • Nomifensine

    CAS:
    <p>Nomifensine ((±)-Nomifensin) is a norepinephrine-dopamine reuptake inhibitor that prevents dopamine reuptake into synaptosomes.</p>
    Fórmula:C16H18N2
    Pureza:99.83% - ≥95%
    Forma y color:Solid
    Peso molecular:238.33
  • Propionylpromazine hydrochloride

    CAS:
    <p>Propionylpromazine hydrochloride (Propiopromazine hydrochloride) is a dopamine receptor D2 (DRD2) antagonist.</p>
    Fórmula:C20H25ClN2OS
    Pureza:99.17%
    Forma y color:Solid
    Peso molecular:376.94
  • SKF-83566

    CAS:
    <p>SKF-83566: Blood-brain permeable, orally active D1 dopamine antagonist; weaker 5-HT2 antagonist, Ki=11 nM.</p>
    Fórmula:C17H18BrNO
    Pureza:95.00% - 99.82%
    Forma y color:Solid
    Peso molecular:332.23
  • Fluoroclebopride

    CAS:
    <p>Fluoroclebopride is a dopamine (DA) D2 receptor ligand.</p>
    Fórmula:C20H23ClFN3O2
    Pureza:99.68% - 99.91%
    Forma y color:Solid
    Peso molecular:391.87
  • Decynium 22

    CAS:
    <p>Decynium 22 is a plasma membrane monoamine transporter (PMAT) inhibitor</p>
    Fórmula:C23H23IN2
    Pureza:99.92%
    Forma y color:Dark Red Crystals
    Peso molecular:454.35
  • AHN 1-055 hydrochloride

    CAS:
    <p>AHN 1-055 hydrochloride (3α-Bis-(4-fluorophenyl) Methoxytropane hydrochloride) is an inhibitor of dopamine transporter (DAT) and dopamine uptake(IC50 = 71 nM).</p>
    Fórmula:C21H24ClF2NO
    Pureza:99.89%
    Forma y color:Solid
    Peso molecular:379.87