
Receptor de dopamina
Los receptores de dopamina son un grupo de receptores acoplados a proteínas G (GPCR) que responden al neurotransmisor dopamina, jugando un papel clave en la regulación del movimiento, la motivación, la recompensa y varias funciones cognitivas. Estos receptores se dividen en familias similares a D1 y D2, cada una con funciones y perfiles farmacológicos distintos. Los moduladores de los receptores de dopamina se estudian ampliamente por sus aplicaciones en el tratamiento de la enfermedad de Parkinson, la esquizofrenia, la adicción y otros trastornos neuropsiquiátricos. En CymitQuimica, ofrecemos una amplia gama de moduladores de receptores de dopamina de alta calidad para apoyar su investigación en neurociencia, salud mental y señalización GPCR.
Se han encontrado 445 productos de "Receptor de dopamina"
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Nomifensine
CAS:Nomifensine ((±)-Nomifensin) is a norepinephrine-dopamine reuptake inhibitor that prevents dopamine reuptake into synaptosomes.Fórmula:C16H18N2Pureza:99.83% - ≥95%Forma y color:SolidPeso molecular:238.33Propionylpromazine hydrochloride
CAS:Propionylpromazine hydrochloride (Propiopromazine hydrochloride) is a dopamine receptor D2 (DRD2) antagonist.Fórmula:C20H25ClN2OSPureza:99.17%Forma y color:SolidPeso molecular:376.94Perospirone
CAS:Perospirone (Lullan) is an antagonist of serotonin 5HT2A receptors and dopamine D2 receptors.Fórmula:C23H30N4O2SPureza:99.23%Forma y color:White PowderPeso molecular:426.57Decynium 22
CAS:Decynium 22 is a plasma membrane monoamine transporter (PMAT) inhibitorFórmula:C23H23IN2Pureza:99.92%Forma y color:Dark Red CrystalsPeso molecular:454.35Cariprazine
CAS:Cariprazine (RGH-188) is a novel antipsychotic drug candidate that exhibits high affinity for the D3 (Ki=0.085 nM) and D2 (Ki=0.49 nM) receptors, and moderateFórmula:C21H32Cl2N4OPureza:99.68% - 99.87%Forma y color:SolidPeso molecular:427.41Ref: TM-T4577
1mg49,00€5mg92,00€10mg145,00€25mg281,00€50mg394,00€100mg550,00€200mg780,00€1mL*10mM (DMSO)103,00€GSK 789472 hydrochloride
CAS:GSK 789472 hydrochloride is both a dopamine D3 receptor antagonist and a D2 partial agonist.Fórmula:C15H22ClN3OPureza:99.89%Forma y color:SolidPeso molecular:295.81L-745870 trihydrochloride
CAS:L-745870 trihydrochloride is a highly potent and selective D4 dopamine receptor antagonist.Fórmula:C18H22Cl4N4Pureza:97.52%Forma y color:SolidPeso molecular:436.21Bromopride hydrochloride
CAS:Bromopride HCl: Salt of a D2 blocker used for upper GI disorders, like dyspepsia and emesis.Fórmula:C14H23BrClN3O2Forma y color:SolidPeso molecular:380.71Rimcazole
CAS:Rimcazole is a sigma receptor antagonist. It also binds to the dopamine transporter and inhibiting dopamine uptake.Fórmula:C21H27N3Pureza:98%Forma y color:SolidPeso molecular:321.46WAY-100635 Monomaleate
CAS:WAY-100635 maleate is a selective 5-hydroxytryptamine 1A receptor antagonist with an IC50 value of 0.91 nM and a Ki value of 0.39 nM.Fórmula:C25H34N4O2·C4H4O4Pureza:98.44% - 99.46%Forma y color:SolidPeso molecular:538.64Ref: TM-T2631
2mg43,00€5mg63,00€10mg89,00€25mg170,00€50mg315,00€100mg470,00€200mg680,00€500mg1.054,00€1mL*10mM (DMSO)74,00€Ocaperidone
CAS:Ocaperidona (Ocaperidone (Ocaperidona)), a very high affinity dopamine D2 antagonist.Fórmula:C24H25FN4O2Pureza:99.33%Forma y color:SolidPeso molecular:420.48carfenazine
CAS:carfenazine targets the Dopamine receptor and is used for schizophrenia research.Fórmula:C24H31N3O2SPureza:98.06%Forma y color:SolidPeso molecular:425.59Pimozide
CAS:Pimozide: antipsychotic that blocks type 2 dopamine, alpha-adrenergic, and 5-HT2 receptors, reducing tics and delusions.Fórmula:C28H29F2N3OPureza:99.63% - >99.99%Forma y color:SolidPeso molecular:461.55Rotigotine-
CAS:Rotigotine (N-0923) is a non-ergot dopamine receptor agonist used in the therapy of Parkinson disease and restless leg syndrome.Fórmula:C19H25NOSPureza:98.08% - 99.59%Forma y color:SolidPeso molecular:315.47Ref: TM-T6647
5mg50,00€10mg73,00€25mg138,00€50mg241,00€100mg358,00€200mg523,00€500mg822,00€1mL*10mM (DMSO)52,00€Pergolide mesylate
CAS:Pergolide mesylate (LY127809), a dopamine agonist for Parkinson's and hyperprolactinemia, was withdrawn for heart valve risk.Fórmula:C20H30N2O3S2Pureza:99.70%Forma y color:White To Off-White SolidPeso molecular:410.59Rotundine
CAS:Rotundine (Gindarine) (L-tetrahydropalmatine, L-THP) is a selective dopamine D1 receptor antagonist with IC50 of 166 nM.Fórmula:C21H25NO4Pureza:99.8% - 99.91%Forma y color:Off-White SolidPeso molecular:355.43SKF38393 hydrobromide
CAS:SKF38393 hydrobromide is the salt form of SKF38393.a dopamine D1 receptor agonist that increases the expression of Shati/Nat8L mRNA in the NAc of mice;Fórmula:C16H18BrNO2Pureza:98.99%Forma y color:SolidPeso molecular:336.22Thozalinone
CAS:Thozalinone is a psychostimulant agent inducing the release of norepinephrine and dopamine.Fórmula:C11H12N2O2Pureza:99.68%Forma y color:SolidPeso molecular:204.23Alizapride
CAS:Alizapride is an antagonist of dopamine receptor. Alizapride can be used in human digestive disorders which is a potent antiemetic [1] [3].Fórmula:C16H21N5O2Forma y color:SolidPeso molecular:315.37Rotigotine Hydrochloride
CAS:Rotigotine HCl, D3-preferential dopamine agonist, is 50x stronger than quinpirole in anti-Parkinson's efficacy.
Fórmula:C19H26ClNOSPureza:99.53% - 99.56%Forma y color:Almost White To White Crystalline PowderPeso molecular:351.93
