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Receptor de dopamina

Receptor de dopamina

Los receptores de dopamina son un grupo de receptores acoplados a proteínas G (GPCR) que responden al neurotransmisor dopamina, jugando un papel clave en la regulación del movimiento, la motivación, la recompensa y varias funciones cognitivas. Estos receptores se dividen en familias similares a D1 y D2, cada una con funciones y perfiles farmacológicos distintos. Los moduladores de los receptores de dopamina se estudian ampliamente por sus aplicaciones en el tratamiento de la enfermedad de Parkinson, la esquizofrenia, la adicción y otros trastornos neuropsiquiátricos. En CymitQuimica, ofrecemos una amplia gama de moduladores de receptores de dopamina de alta calidad para apoyar su investigación en neurociencia, salud mental y señalización GPCR.

Se han encontrado 445 productos de "Receptor de dopamina"

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  • Nomifensine

    CAS:
    Nomifensine ((±)-Nomifensin) is a norepinephrine-dopamine reuptake inhibitor that prevents dopamine reuptake into synaptosomes.
    Fórmula:C16H18N2
    Pureza:99.83% - ≥95%
    Forma y color:Solid
    Peso molecular:238.33

    Ref: TM-T7308

    10mg
    35,00€
    25mg
    49,00€
    50mg
    70,00€
    100mg
    104,00€
    1mL*10mM (DMSO)
    35,00€
  • Propionylpromazine hydrochloride

    CAS:
    Propionylpromazine hydrochloride (Propiopromazine hydrochloride) is a dopamine receptor D2 (DRD2) antagonist.
    Fórmula:C20H25ClN2OS
    Pureza:99.17%
    Forma y color:Solid
    Peso molecular:376.94

    Ref: TM-T9228

    1mg
    35,00€
    5mg
    77,00€
    10mg
    113,00€
    25mg
    177,00€
    50mg
    266,00€
    1mL*10mM (DMSO)
    87,00€
  • Perospirone

    CAS:
    Perospirone (Lullan) is an antagonist of serotonin 5HT2A receptors and dopamine D2 receptors.
    Fórmula:C23H30N4O2S
    Pureza:99.23%
    Forma y color:White Powder
    Peso molecular:426.57

    Ref: TM-T4576

    10mg
    48,00€
    25mg
    82,00€
    50mg
    133,00€
    100mg
    221,00€
    200mg
    309,00€
    1mL*10mM (DMSO)
    34,00€
  • Decynium 22

    CAS:
    Decynium 22 is a plasma membrane monoamine transporter (PMAT) inhibitor
    Fórmula:C23H23IN2
    Pureza:99.92%
    Forma y color:Dark Red Crystals
    Peso molecular:454.35

    Ref: TM-T22714

    50mg
    33,00€
    1mL*10mM (DMSO)
    39,00€
  • Cariprazine

    CAS:
    Cariprazine (RGH-188) is a novel antipsychotic drug candidate that exhibits high affinity for the D3 (Ki=0.085 nM) and D2 (Ki=0.49 nM) receptors, and moderate
    Fórmula:C21H32Cl2N4O
    Pureza:99.68% - 99.87%
    Forma y color:Solid
    Peso molecular:427.41

    Ref: TM-T4577

    1mg
    49,00€
    5mg
    92,00€
    10mg
    145,00€
    25mg
    281,00€
    50mg
    394,00€
    100mg
    550,00€
    200mg
    780,00€
    1mL*10mM (DMSO)
    103,00€
  • GSK 789472 hydrochloride

    CAS:
    GSK 789472 hydrochloride is both a dopamine D3 receptor antagonist and a D2 partial agonist.
    Fórmula:C15H22ClN3O
    Pureza:99.89%
    Forma y color:Solid
    Peso molecular:295.81

    Ref: TM-T22817

    2mg
    42,00€
    5mg
    64,00€
    10mg
    96,00€
    25mg
    170,00€
    50mg
    245,00€
    100mg
    371,00€
    200mg
    494,00€
  • L-745870 trihydrochloride

    CAS:
    L-745870 trihydrochloride is a highly potent and selective D4 dopamine receptor antagonist.
    Fórmula:C18H22Cl4N4
    Pureza:97.52%
    Forma y color:Solid
    Peso molecular:436.21

    Ref: TM-T22904

    1mg
    46,00€
    5mg
    93,00€
    10mg
    118,00€
    25mg
    263,00€
    50mg
    376,00€
    100mg
    532,00€
    200mg
    705,00€
  • Bromopride hydrochloride

    CAS:
    Bromopride HCl: Salt of a D2 blocker used for upper GI disorders, like dyspepsia and emesis.
    Fórmula:C14H23BrClN3O2
    Forma y color:Solid
    Peso molecular:380.71

    Ref: TM-T69152

    25mg
    1.369,00€
    50mg
    1.783,00€
    100mg
    2.250,00€
  • Rimcazole

    CAS:
    Rimcazole is a sigma receptor antagonist. It also binds to the dopamine transporter and inhibiting dopamine uptake.
    Fórmula:C21H27N3
    Pureza:98%
    Forma y color:Solid
    Peso molecular:321.46

    Ref: TM-T24712

    25mg
    1.369,00€
    50mg
    1.783,00€
    100mg
    2.250,00€
  • WAY-100635 Monomaleate

    CAS:
    WAY-100635 maleate is a selective 5-hydroxytryptamine 1A receptor antagonist with an IC50 value of 0.91 nM and a Ki value of 0.39 nM.
    Fórmula:C25H34N4O2·C4H4O4
    Pureza:98.44% - 99.46%
    Forma y color:Solid
    Peso molecular:538.64

    Ref: TM-T2631

    2mg
    43,00€
    5mg
    63,00€
    10mg
    89,00€
    25mg
    170,00€
    50mg
    315,00€
    100mg
    470,00€
    200mg
    680,00€
    500mg
    1.054,00€
    1mL*10mM (DMSO)
    74,00€
  • Ocaperidone

    CAS:
    Ocaperidona (Ocaperidone (Ocaperidona)), a very high affinity dopamine D2 antagonist.
    Fórmula:C24H25FN4O2
    Pureza:99.33%
    Forma y color:Solid
    Peso molecular:420.48

    Ref: TM-T3497

    1mg
    44,00€
    5mg
    93,00€
    10mg
    113,00€
    25mg
    200,00€
    50mg
    334,00€
    100mg
    485,00€
    1mL*10mM (DMSO)
    92,00€
  • carfenazine

    CAS:
    carfenazine targets the Dopamine receptor and is used for schizophrenia research.
    Fórmula:C24H31N3O2S
    Pureza:98.06%
    Forma y color:Solid
    Peso molecular:425.59

    Ref: TM-T9827

    1mg
    96,00€
    5mg
    173,00€
    10mg
    260,00€
    25mg
    447,00€
    50mg
    A consultar
  • Pimozide

    CAS:
    Pimozide: antipsychotic that blocks type 2 dopamine, alpha-adrenergic, and 5-HT2 receptors, reducing tics and delusions.
    Fórmula:C28H29F2N3O
    Pureza:99.63% - >99.99%
    Forma y color:Solid
    Peso molecular:461.55

    Ref: TM-T2546

    25mg
    34,00€
    50mg
    49,00€
    1mL*10mM (DMSO)
    50,00€
  • Rotigotine-

    CAS:
    Rotigotine (N-0923) is a non-ergot dopamine receptor agonist used in the therapy of Parkinson disease and restless leg syndrome.
    Fórmula:C19H25NOS
    Pureza:98.08% - 99.59%
    Forma y color:Solid
    Peso molecular:315.47

    Ref: TM-T6647

    5mg
    50,00€
    10mg
    73,00€
    25mg
    138,00€
    50mg
    241,00€
    100mg
    358,00€
    200mg
    523,00€
    500mg
    822,00€
    1mL*10mM (DMSO)
    52,00€
  • Pergolide mesylate

    CAS:
    Pergolide mesylate (LY127809), a dopamine agonist for Parkinson's and hyperprolactinemia, was withdrawn for heart valve risk.
    Fórmula:C20H30N2O3S2
    Pureza:99.70%
    Forma y color:White To Off-White Solid
    Peso molecular:410.59

    Ref: TM-T2226

    5mg
    49,00€
    10mg
    70,00€
    25mg
    109,00€
    50mg
    168,00€
    1mL*10mM (DMSO)
    54,00€
  • Rotundine

    CAS:
    Rotundine (Gindarine) (L-tetrahydropalmatine, L-THP) is a selective dopamine D1 receptor antagonist with IC50 of 166 nM.
    Fórmula:C21H25NO4
    Pureza:99.8% - 99.91%
    Forma y color:Off-White Solid
    Peso molecular:355.43

    Ref: TM-T6648

    1g
    145,00€
    50mg
    37,00€
    100mg
    52,00€
    500mg
    97,00€
  • SKF38393 hydrobromide

    CAS:
    SKF38393 hydrobromide is the salt form of SKF38393.a dopamine D1 receptor agonist that increases the expression of Shati/Nat8L mRNA in the NAc of mice;
    Fórmula:C16H18BrNO2
    Pureza:98.99%
    Forma y color:Solid
    Peso molecular:336.22

    Ref: TM-T23359

    1mg
    49,00€
    5mg
    90,00€
    10mg
    129,00€
    25mg
    253,00€
    50mg
    373,00€
    100mg
    546,00€
    200mg
    783,00€
  • Thozalinone

    CAS:
    Thozalinone is a psychostimulant agent inducing the release of norepinephrine and dopamine.
    Fórmula:C11H12N2O2
    Pureza:99.68%
    Forma y color:Solid
    Peso molecular:204.23

    Ref: TM-T19893

    10mg
    40,00€
    25mg
    66,00€
    50mg
    88,00€
    100mg
    133,00€
    200mg
    192,00€
    1mL*10mM (DMSO)
    33,00€
  • Alizapride

    CAS:
    Alizapride is an antagonist of dopamine receptor. Alizapride can be used in human digestive disorders which is a potent antiemetic [1] [3].
    Fórmula:C16H21N5O2
    Forma y color:Solid
    Peso molecular:315.37

    Ref: TM-T60813

    25mg
    1.369,00€
    50mg
    1.783,00€
    100mg
    2.250,00€
  • Rotigotine Hydrochloride

    CAS:

    Rotigotine HCl, D3-preferential dopamine agonist, is 50x stronger than quinpirole in anti-Parkinson's efficacy.

    Fórmula:C19H26ClNOS
    Pureza:99.53% - 99.56%
    Forma y color:Almost White To White Crystalline Powder
    Peso molecular:351.93

    Ref: TM-T21446

    5mg
    44,00€
    10mg
    59,00€
    25mg
    96,00€
    50mg
    116,00€
    100mg
    159,00€
    200mg
    227,00€