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Receptor de adenosina

Receptor de adenosina

Los receptores de adenosina son una clase de GPCR que responden al nucleósido endógeno adenosina. Estos receptores están involucrados en la regulación de diversos procesos fisiológicos, incluidos la función cardiovascular, los ciclos sueño-vigilia y las respuestas inmunitarias. Los moduladores de los receptores de adenosina tienen un potencial terapéutico en el tratamiento de afecciones como las arritmias cardíacas, la inflamación y las enfermedades neurodegenerativas. En CymitQuimica, ofrecemos una selección de moduladores de receptores de adenosina de alta calidad para apoyar su investigación en biología cardiovascular, neurociencia e inmunología.

Se han encontrado 242 productos de "Receptor de adenosina"

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  • CGS 15943

    CAS:
    <p>CGS 15943 is an orally bioavailable non-xanthine antagonist of Adenosine Receptor.</p>
    Fórmula:C13H8ClN5O
    Pureza:97.4%
    Forma y color:Solid
    Peso molecular:285.69
  • YT 146

    CAS:
    <p>YT 146 is a biochemical.</p>
    Fórmula:C18H25N5O4
    Pureza:98.81% - 99.25%
    Forma y color:Solid
    Peso molecular:375.42
  • N6-Ethyladenosine

    CAS:
    <p>N6-Ethyladenosine is an adenosine derivative, acts as an agonist of Adenosine receptor(hA1AR and hA3AR with Kis of 4.9 and 4.7 nM , respectively).</p>
    Fórmula:C12H17N5O4
    Pureza:99.96%
    Forma y color:Solid
    Peso molecular:295.29
  • Adenosine 5'-monophosphate monohydrate

    CAS:
    <p>Adenosine 5'-monophosphate monohydrate (5'-AMP) , also known as 5'-adenylic acid, is a nucleotide that is used as a monomer in RNA.</p>
    Fórmula:C10H14N5O7P·H2O
    Pureza:97.68% - 98.49%
    Forma y color:White Powder
    Peso molecular:365.24
  • Acefylline

    CAS:
    <p>Acefylline (Theophylline-7-acetic acid), a stimulant drug of the xanthine chemical class, acts as an adenosine receptor antagonist.</p>
    Fórmula:C9H10N4O4
    Pureza:99.57%
    Forma y color:White Crystalline Solid
    Peso molecular:238.2
  • Amp579 TFA


    <p>Amp579 TFA is a novel adenosine A1/A2a receptor agonist that induces acute and delayed preconditioning against myocardial shock in vivo.</p>
    Fórmula:C24H29ClF3N5O5S
    Pureza:96.56%
    Forma y color:Soild
    Peso molecular:592.03
  • Theophylline

    CAS:
    <p>Theophylline (1,3-Dimethylxanthine) is a methyl xanthine derivative from tea with diuretic, smooth muscle relaxant, bronchial dilation, cardiac and central</p>
    Fórmula:C7H8N4O2
    Pureza:99.65% - 99.98%
    Forma y color:White Solid Powder
    Peso molecular:180.16
  • AB928

    CAS:
    <p>AB928 is an orally bioavailable, selective dual adenosine receptor (A2aR/A2bR) antagonist. It has immunomodulatory activity[1].</p>
    Fórmula:C23H22N8O
    Pureza:98.09% - >99.99%
    Forma y color:Solid
    Peso molecular:426.47
  • Pamabrom

    CAS:
    <p>Pamabrom is a diuretic for premenstrual and menstrual bloating, swelling, and fullness.</p>
    Fórmula:C11H18BrN5O3
    Pureza:99.84% - >99.99%
    Forma y color:Coa
    Peso molecular:348.2
  • N6-Cyclohexyladenosine

    CAS:
    <p>N6-Cyclohexyladenosine (CHA) is a selective agonist of A1 receptor with EC50 of 8.2 Nm.</p>
    Fórmula:C16H23N5O4
    Pureza:99.84% - 99.98%
    Forma y color:Solid
    Peso molecular:349.38
  • DPTN dihydrochloride

    CAS:
    <p>DPTN dihydrochloride is a potent and selective A3AR antagonist with Ki values of 1.65, 9.61 and 8.53 nM in human, mouse and rat, respectively.</p>
    Fórmula:C22H20Cl2N4OS
    Pureza:99.95%
    Forma y color:Soild
    Peso molecular:459.39
  • Pentoxifylline

    CAS:
    <p>Pentoxifylline (PTX) stimulates cytokines, inhibits phosphodiesterase, enhances blood flow, and increases cell flexibility.</p>
    Fórmula:C13H18N4O3
    Pureza:99.26% - 99.93%
    Forma y color:Solid
    Peso molecular:278.31
  • Aminophylline

    CAS:
    <p>Aminophylline (Phyllocontin) is a competitive nonselective phosphodiesterase inhibitor giving a bronchodilatory effect.</p>
    Fórmula:C7H8O2·C2H8N2
    Pureza:99.31%
    Forma y color:White Or Slightly Yellowish Granules Or Powder Solid
    Peso molecular:420.43
  • Quercetin-3'-o-phosphate TEA


    <p>Quercetin-3'-o-phosphate TEA (Quercetin 3'-phosphate TEA) is an adenosine A receptor antagonist that can be used to prevent and treat metabolic disorders.</p>
    Fórmula:C21H26NO10P
    Pureza:95.63%
    Forma y color:Soild
    Peso molecular:483.41
  • Ticlopidine hydrochloride

    CAS:
    <p>Ticlopidine hydrochloride (Ticlodix) is an effective inhibitor of platelet aggregation commonly used in the placement of STENTS in CORONARY ARTERIES.</p>
    Fórmula:C14H15Cl2NS
    Pureza:99.85% - >99.99%
    Forma y color:White Powder
    Peso molecular:300.25
  • Theophylline monohydrate

    CAS:
    <p>Theophylline monohydrate (Quibron) appears to inhibit phosphodiesterase and prostaglandin production, regulate calcium flux and intracellular calcium</p>
    Fórmula:C7H8N4O2·H2O
    Pureza:99.78%
    Forma y color:Solid
    Peso molecular:198.18
  • Doxofylline

    CAS:
    <p>Doxofylline (Doxophylline) is a methylxanthine derivative with the presence of a dioxolane group in position 7.</p>
    Fórmula:C11H14N4O4
    Pureza:99.958% - >99.99%
    Forma y color:Solid
    Peso molecular:266.25
  • Adenosine A1 receptor activator T62

    CAS:
    <p>Adenosine A1 receptor activator T62 is an allosteric enhancer of adenosine A1 receptor, and it produces antinociception in animal models of acute pain and also</p>
    Fórmula:C15H14ClNOS
    Pureza:97.83%
    Forma y color:Solid
    Peso molecular:291.8
  • Diphylline

    CAS:
    <p>Diphylline is a bronchodilator with mild vasodilator and diuretic properties, used for asthma, bronchitis, and emphysema.</p>
    Fórmula:C10H14N4O4
    Pureza:98.54%
    Forma y color:Crystals From Alcohol Solid
    Peso molecular:254.24
  • Danshenol B


    <p>Danshenol B is a natural product that can be used as a reference standard.</p>
    Fórmula:C22H26O4
    Forma y color:Solid
    Peso molecular:354.446