Inhibidores
Los inhibidores son moléculas que se unen a enzimas, receptores u otras proteínas para reducir o bloquear su actividad biológica. Estos compuestos se utilizan ampliamente en la investigación para estudiar vías biológicas, comprender los mecanismos de las enfermedades y desarrollar fármacos terapéuticos. Los inhibidores desempeñan un papel crucial en el tratamiento de diversas enfermedades, incluyendo el cáncer, las enfermedades cardiovasculares y las infecciones. En CymitQuimica, ofrecemos una amplia gama de inhibidores de alta calidad para apoyar su investigación en bioquímica, biología celular y desarrollo farmacéutico.
Subcategorías de "Inhibidores"
- Angiogénesis(2.715 productos)
- Apoptosis(6.164 productos)
- Ciclo celular / Checkpoint(4.727 productos)
- Cromatina / Epigenética(2.400 productos)
- Señalización citoesquelética(1.492 productos)
- Daño al ADN / Reparación del ADN(2.928 productos)
- Endocrinología / Hormonas(3.653 productos)
- Enzima(3.661 productos)
- GPCR / proteína G(8.861 productos)
- Inmunología e inflamación(3.801 productos)
- Virus de la gripe(299 productos)
- Señalización JAK / STAT(412 productos)
- Señalización MAPK(1.239 productos)
- Transportador de membrana / canal de iones(2.979 productos)
- Metabolismo(10.029 productos)
- Microbiología / Virología(7.445 productos)
- Neurociencia(10.281 productos)
- Otros inhibidores(36.478 productos)
- Reducción de oxidación(44 productos)
- Señalización PI3K / Akt / mTOR(1.443 productos)
- Proteasas / Proteasoma(1.695 productos)
- Células madre y Derivados(829 productos)
- Tirosina quinasa / adaptadores(2.035 productos)
- Ubiquitinación(1.693 productos)
Mostrar 16 subcategorías más
Se han encontrado 66676 productos de "Inhibidores"
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L 734217
CAS:L 734217 is an antagonist of the fibrinogen receptor.Fórmula:C18H31N3O4Pureza:98%Forma y color:SolidPeso molecular:353.46JTP-117968
CAS:JTP-117968: Non-steroidal SGRM, glucocorticoid receptor modulator, IC50 = 6.8 nM, offers better inhibitory/activatory balance.Fórmula:C31H31F3N2O2Forma y color:SolidPeso molecular:520.59Pareptide monohydrochloride
CAS:Pareptide monohydrochloride is a metabolically stable analog of melatonin inhibitor (MIF).Fórmula:C14H27ClN4O3Pureza:98%Forma y color:SolidPeso molecular:334.84L 668411
CAS:L 668411, the 2,3-ditritiated methyl ester of L 659699, inhibits HMG-CoA synthase.Fórmula:C19H30O5Pureza:98%Forma y color:SolidPeso molecular:338.44SGK1-IN-3
SGK1-IN-3: Potent oral inhibitor of SGK1, may target osteoarthritis.Fórmula:C23H20Cl2N6O3SForma y color:SolidPeso molecular:531.41MI-1851
CAS:<p>MI-1851 is a potent peptidomimetic inhibitor. MI-1851could prevent proteolytic processing of the S protein from SARSCoV-2 by endogenous furin in HEK293 cells.</p>Fórmula:C34H53N15O6Forma y color:SolidPeso molecular:767.88BMS-986143
CAS:BMS-986143: oral BTK inhibitor, IC50=0.26 nM, potential for autoimmune research, also targets TEC, BLK, BMX, TXK, YES1, ITK.Fórmula:C31H24Cl2N4O4Forma y color:SolidPeso molecular:587.45YKL-04-085
CAS:<p>YKL-04-085 inhibits viral translation effectively, with strong antiviral action at much lower doses than those affecting host-cell growth.</p>Fórmula:C30H29N5O2Forma y color:SolidPeso molecular:491.6PptT-IN-1
PptT-IN-1, a potent PptT inhibitor (IC50: 2.8 μM), shows promise for tuberculosis research.Fórmula:C18H29N5O2Forma y color:SolidPeso molecular:347.46LA-810
CAS:LA-810 is a nitrous oxide donor.Fórmula:C15H25N5O7SForma y color:SolidPeso molecular:419.45Trk-IN-8
<p>Trk-IN-8: TRK inhibitor with IC50 of 0.42 nM (TRKA), 0.89 nM (TRKA-G595R), 1.5 nM (TRKC-G623R).</p>Fórmula:C18H16F2N6O2Forma y color:SolidPeso molecular:386.36BI-207524
CAS:BI-207524 is a novel NS5B Thumb Pocket 1 Inhibitor with Improved Potency for the Potential Treatment of Chronic Hepatitis C Virus Infection.Fórmula:C35H36ClN5O5Forma y color:SolidPeso molecular:642.14BI-4916
CAS:BI-4916 is a phosphoglycerate dehydrogenase (PHGDH) inhibitor that inhibits SSP and reduces cancer cell migration.Fórmula:C23H24Cl2N2O6SPureza:98.55%Forma y color:SolidPeso molecular:527.42RN941
CAS:RN941 is a highly potent Bruton's tyrosine kinase (BTK) inhibitor.Fórmula:C34H34FN7O5Pureza:98%Forma y color:SolidPeso molecular:639.68Anticancer agent 26
Anticancer agent 26 is a promising candidate for cancer therapy and deserves further development.Fórmula:C28H33NO5Forma y color:SolidPeso molecular:463.57RORγt/DHODH-IN-1
CAS:RORγt/DHODH-IN-1 (compound (R)-14d) is a potent, orally active dual inhibitor of RORγt (IC50: 0.083 μM) and DHODH (IC50: 0.172 μM), which exhibits significantFórmula:C24H26ClF6N3O3SForma y color:SolidPeso molecular:585.99VEGFR-2-IN-25
CAS:VEGFR-2-IN-25 (compound 5d) is a potent inhibitor of VEGFR-2 (IC50: 12.1 nM).Fórmula:C24H22N6O2Forma y color:SolidPeso molecular:426.47BW-10
CAS:<p>BW-10 potently inhibits bombesin evoked release of gastrointestinal hormones in vitro and in vivo.</p>Fórmula:C57H72N14O8Forma y color:SolidPeso molecular:1081.27Antimalarial agent 7
Antimalarial agent 7 is a potent and effective inhibitor of PfATP4. Antimalarial agent 7 has potential for the study of the human plasmodium falciparum.Fórmula:C23H22F2N4O3Forma y color:SolidPeso molecular:440.44HIV-1 inhibitor-40
HIV-1 inhibitor-40 (4ab) is a potent NNRTI (EC50: 1.9 nM), non-toxic in vivo, and a sensitive CYP inhibitor.Fórmula:C25H18N6O2Forma y color:SolidPeso molecular:434.45Squalestatin 3
CAS:Squalestatin 3 is an inhibitor of squalene synthase.Fórmula:C25H30O13Pureza:98%Forma y color:SolidPeso molecular:538.5Dicetrorelix pamoate
CAS:Cetrorelix pamoate is a synthetic decapeptide that acts as a GnRH antagonist, inhibiting the release of LH and FSH from the pituitary.Fórmula:C163H200Cl2N34O34Forma y color:SolidPeso molecular:3250.49SARS-CoV-2-IN-6
SARS-CoV-2-IN-6 is an inhibitor of SARS-CoV-2 3CLpro with the IC 50 value of 73 nM.Fórmula:C17H13ClN2O2Forma y color:SolidPeso molecular:312.75IAA65
CAS:<p>IAA65 is a potent inhibitor of T-type calcium channels, exhibiting an IC50 value of 18.9 μM, and holds potential for use in epilepsy research [1].</p>Fórmula:C16H13F6NO2Forma y color:SolidPeso molecular:365.27PI3Kβ-IN-1
CAS:PI3Kβ-IN-1 is a selective, orally active PI3Kβ inhibitor (IC50: 2 nM).Fórmula:C25H14F2N8Forma y color:SolidPeso molecular:464.43TMX-4113
<p>TMX-4113 has potential to be used in cancer that is a phosphodiesterase 6D(PDE6D) and casein kinase 1α(CK1α) degrader [1].</p>Fórmula:C12H12N4O2S2Forma y color:SolidPeso molecular:308.38ent-8-iso-15(S)-Prostaglandin F2α
CAS:Isoprostanes are produced by the non-enzymatic, free radical peroxidation of phospholipid-esterified arachidonic acid.Fórmula:C20H34O5Forma y color:SolidPeso molecular:354.48TAI-95
CAS:TAI-95 is an inhibitor of highly expressed cancer protein 1 (Hec1).Fórmula:C24H23N5O3S2Forma y color:SolidPeso molecular:493.60IL-17 modulator 5
CAS:IL-17 modulator 5 is a IL-17 inhibitor, with an IC 50 of 1 nM .Fórmula:C28H23F6N9O2Forma y color:SolidPeso molecular:631.53PDE4B/7A-IN-1
CAS:5-HT1A antagonist; Ki=8nM, Kb=0.04nM. PDE4B IC50=80.4μM; PDE7A IC50=151.3μM. Good biofilm penetration, stable, anticognitive, antidepressant.Fórmula:C25H35N3O3Forma y color:SolidPeso molecular:425.56HIV-1 inhibitor-52
CAS:HIV-1 inhibitor-52: potent, broad-spectrum with EC50s 1.6-6.4 nM against various HIV-1 strains.Fórmula:C46H72FNO5SForma y color:SolidPeso molecular:770.13Anti-inflammatory agent 16
Compound 14 is a peptidomimetic that significantly lowers TNFα, NO, CD40, and CD86, showcasing strong anti-inflammatory effects.Fórmula:C21H23N5O3Forma y color:SolidPeso molecular:393.44MB-07344 sodium
"MB-07344 sodium is a TR-β agonist with a 2.17 nM Ki, boosts Atorvastatin's cholesterol-lowering effects in various animals."Fórmula:C19H25NaO5PPureza:98%Forma y color:SolidPeso molecular:387.36MMSET-IN-1
CAS:MMSET-IN-1 is an inhibitor of multiple myeloma SET domain (MMSET, aka NSD2/WHSC1) .Fórmula:C18H29N7O5Pureza:98%Forma y color:SolidPeso molecular:423.4716(R)-Iloprost
CAS:<p>Iloprost, a potent prostacyclin analog, binds IP & EP1 receptors (Ki 11 nM), contains 16(S/R) isomers, and inhibits platelets (IC50 65 nM).</p>Fórmula:C22H32O4Forma y color:SolidPeso molecular:360.49HIV-1 inhibitor-14
<p>HIV-1 inhibitor-14: potent, broad HIV-1 RT inhibitor. IC50=0.14μM. Effective against wild-type and resistant strains, EC50=5.79-28.3nM.</p>Fórmula:C29H32N6O4SForma y color:SolidPeso molecular:560.67PRMT5-IN-19
PRMT5-IN-19 is a potent, selective PRMT5 inhibitor with IC50 of 23.9 nM and 47 nM, showing anti-cancer activity by inducing apoptosis.Fórmula:C25H24N4OForma y color:SolidPeso molecular:396.48GNE-431
CAS:GNE-431: potent, selective noncovalent Btk inhibitor, IC50=3.2 nM; effective against C481R, T474I, T474M mutants, may counter ibrutinib resistance.Fórmula:C30H32N10O2Forma y color:SolidPeso molecular:564.64XR8-69
<p>XR8-69 is a SARS-CoV-2 PLpro inhibitor. XR8-69 has a low micromolar antiviral effect in SARS-CoV-2 infected human cells.</p>Fórmula:C26H30N4O2SForma y color:SolidPeso molecular:462.61FGFR4-IN-10
FGFR4-IN-10 (compound 5a) is a potent, selective FGFR4 inhibitor with IC50 of 70.7 nM, sparing FGFR1-3.Fórmula:C20H19F3N6O3Forma y color:SolidPeso molecular:448.4DS69910557
DS69910557: potent hPTHR1 antagonist, IC50 0.08 μM, oral, for hyperparathyroidism & osteoporosis research.Fórmula:C32H33Cl2FN4O3Forma y color:SolidPeso molecular:611.53KCa2 channel modulator 2
Compound 2q is a potent, subtype-selective K/Ca 2 modulator, effective on human K Ca 2.3 and rat K Ca 2.2a with EC50s of 0.60 μM and 0.64 μM.Fórmula:C16H15ClFN5Forma y color:SolidPeso molecular:331.78SB 258741 hydrochloride
SB 258741 hydrochloride is a potent antagonist of the 5-HT 7 receptor, designed specifically for studying schizophrenia [1].Fórmula:C19H31ClN2O2SForma y color:SolidPeso molecular:386.98Kallikrein-IN-1
CAS:Kallikrein-IN-1 (Formula A) is an inhibitor of the kinin-releasing enzyme Kallikrein.Fórmula:C28H26FN5O4Forma y color:SolidPeso molecular:515.54Irinotecan Carboxylate Sodium Salt
CAS:Irinotecan Carboxylate Sodium Salt is a DNA topoisomerase inhibitor.Fórmula:C33H39N4NaO7Forma y color:SolidPeso molecular:626.68Cav 3.2 inhibitor 1
<p>Cav 3.2 inhibitor 1 targets T-type calcium channels, weakly binds D2 receptors, and aids physical and visceral pain research.</p>Fórmula:C32H39N3OForma y color:SolidPeso molecular:481.67BMS-066
CAS:BMS-066 is an IKKβ/Tyk2 pseudokinase inhibitor. With IC50s of 9 nM and 72 nM, respectively.Fórmula:C19H21N7O2Pureza:98%Forma y color:SolidPeso molecular:379.42AKT-IN-10
CAS:AKT-IN-10, a potent AKT inhibitor, has potential for breast and prostate cancer research, impacting cell growth and survival pathways.Fórmula:C26H34ClN5O2Forma y color:SolidPeso molecular:484.03AZ14145845
AZ14145845 is an in vivo potent and highly selective type I1/2 Mer/Axl bispecific kinase inhibitor.Fórmula:C32H35N9OForma y color:SolidPeso molecular:561.68LY 245769
CAS:LY 245769 is an inhibitor of leukotriene E4 (LTE4).Fórmula:C25H33F3N8OSPureza:98%Forma y color:SolidPeso molecular:550.64OM-153
CAS:OM-153 blocks tankyrase 1 (IC50: 13 nM) and 2 (IC50: 2 nM), stifling WNT signaling and COLO 320DM cell growth.Fórmula:C28H24FN7O2Forma y color:SolidPeso molecular:509.53FPDT
FPDT combats glioblastoma by inhibiting the AKT pathway; IC50: >100 μM (astrocytes), 45-68 μM (GBM cells).Fórmula:C16H12FNO2SForma y color:SolidPeso molecular:301.34LY3130481
CAS:LY3130481: TARP γ-8 dependent AMPA receptor blocker; selectively targets AMPA/TARP γ-8 with 65 nM IC50.Fórmula:C19H18N4O3SForma y color:SolidPeso molecular:382.44PARP1/BRD4-IN-2
PARP1/BRD4-IN-2, a potent inhibitor of PARP1 and BRD4, halts cell cycle, triggers apoptosis, and has antitumor effects on TNBC.Fórmula:C25H20N4O4Forma y color:SolidPeso molecular:440.45LAF-153
CAS:LAF-153 is a reversible Methionine Aminopeptidase‑2 (MetAP-2) Inhibitor.Fórmula:C18H32N2O7Forma y color:SolidPeso molecular:388.46MEIS-IN-2
MEIS-IN-2 is an inhibitor of MEIS1. MEIS-IN-2 can be used in studies of cardiac regeneration and haematopoietic stem cell (HSC) regulation.Fórmula:C23H21ClN2O4Forma y color:SolidPeso molecular:424.88NS2B/NS3-IN-4
CAS:<p>Compound 34e inhibits DENV2/ZIKV proteases; IC50: 0.69 µM (DENV2), 1.04 µM (ZIKV).</p>Fórmula:C15H11NO4Forma y color:SolidPeso molecular:269.25LolCDE-IN-2
CAS:<p>LolCDE-IN-2 is a potent Lol protein (LolCDE) inhibitor. LolCDE-IN-2 shows antibacterial activity with a MIC of 2 μg/ml against E. coli MG1655 [1].</p>Fórmula:C22H17N5OPureza:98%Forma y color:SolidPeso molecular:367.40Revamilast sodium
CAS:Revamilast sodium, also known as GRC4039 sodium, is a phosphodiesterase IV inhibitor for potentially treating of asthma and rheumatoid arthritisFórmula:C18H8Cl2F2N3NaO4Forma y color:SolidPeso molecular:462.17PARP10/15-IN-2
CAS:PARP10/15-IN-2 (Compound 8h) blocks PARP10/15, has IC50s: 0.15μM/0.37μM, cell-permeable, prevents apoptosis.Fórmula:C15H11FN2O3Forma y color:SolidPeso molecular:286.26MRGPRX1 agonist 4
Potent, oral MRGPRX1 agonist 4 modulates receptor positively (EC50: 0.1 μM) and reduces mice's thermal allergy response.Fórmula:C23H17Cl2F3N2O2SForma y color:SolidPeso molecular:513.36MB-7133
CAS:MB-7133 is an inhibitor of DNA synthesis.Fórmula:C17H21N4O8PPureza:98%Forma y color:SolidPeso molecular:440.34SP4206
CAS:SP4206 is an interaction inhibitor of IL-2/IL-2Rα (IL-2 and IL-2Rα with Kd of 70 nM and 10 nM,respectively)Fórmula:C30H37Cl2N7O6Pureza:98%Forma y color:SolidPeso molecular:662.56sEH inhibitor-4
Compound B15: potent sEH inhibitor (0.03 nm), reduces inflammation & pain.Fórmula:C27H28Cl2N4O3Forma y color:SolidPeso molecular:527.44Dyrk1A-IN-1
Dyrk1A-IN-1 is a triple inhibitor of Dyrk1A kinase activity, aggregation of tau and α-syn oligomers, with an IC50 value of 119 nM for Dyrk1A kinase.Fórmula:C23H20N4O3SForma y color:SolidPeso molecular:432.49J-104118
CAS:J-104118 potentially inhibits squalene synthase.Fórmula:C28H26Cl2FNO5Pureza:98%Forma y color:SolidPeso molecular:546.41LSD1/2-IN-3
LSD1/2-IN-3 selectively inhibits LSD1 (Ki 11 nM) over LSD2 (Ki 7 μM), and hinders tumor stem cell proliferation.Fórmula:C9H8BrF2NForma y color:SolidPeso molecular:248.07SB-612111
CAS:SB-612111: potent ORL-1 antagonist, Ki=0.33 nM; μ-, κ-, δ-receptor Ki=57.6, 160.5, 2109 nM; blocks nociceptin's pain effect.Fórmula:C24H29Cl2NOForma y color:SolidPeso molecular:418.40Anti-MRSA agent 6
Anti-MRSA agent 6 (compound 3q6) is a potent anti-methicillin-resistant Staphylococcus aureus (anti-MRSA) agent with low cytoxicity for MCF-7, A549 cells [1].Fórmula:C16H11F2N3Forma y color:SolidPeso molecular:283.28AM-9514
CAS:AM-9514: a potent Glucokinase activator with strong in vitro results, good pharmacokinetics, and efficacy in diabetes.Fórmula:C18H25N5O4Forma y color:SolidPeso molecular:375.42SSTR5 antagonist 2 TFA
CAS:Potent, oral SSTR5 antagonist 2 TFA may treat type 2 diabetes.Fórmula:C34H36F4N2O7Pureza:98%Forma y color:SolidPeso molecular:660.65mPGES-1-IN-1
MPGES-1, potential anti-inflammatory drug target, has IC50 of 0.03 μM with mPGES-1-IN-1.Fórmula:C21H14N4O2SForma y color:SolidPeso molecular:386.43AMG-548 dihydrochloride
AMG-548 dihydrochloride, an oral p38α inhibitor (Ki: 0.5 nM), selectively targets p38β, γ, δ, inhibits TNFα (IC50: 3 nM), and suppresses Wnt signaling.Fórmula:C29H29Cl2N5OForma y color:SolidPeso molecular:534.48BM635 mesylate (1493762-74-5 free base)
BM635 mesylate is an MmpL3 inhibitor with outstanding anti-mycobacterial activity (MIC50: 0.12 μM against M. tuberculosis H37Rv).Fórmula:C26H33FN2O4SPureza:98%Forma y color:SolidPeso molecular:488.61Kahweol Acetate
CAS:Kahweol Acetate, a semi-synthetic coffee bean derivative, inhibits osteoclasts, cancer cells, DNA damage, and oxidative stress.Fórmula:C22H28O4Forma y color:SolidPeso molecular:356.46Daeatal
CAS:Dynorphin A ethylamide (1-9), the opioid activities were examined in the bioassays.Fórmula:C56H93N19O10Pureza:98%Forma y color:SolidPeso molecular:1192.46OncoFAP
CAS:<p>OncoFAP is an ultra-high affinity fibroblast activating protein (FAP) ligand with potential tumour targeting.</p>Fórmula:C21H19F2N5O5Pureza:99.77%Forma y color:SolidPeso molecular:459.40Casuarinin
CAS:<p>Casuarinin, an ellagitannin found in pomegranates and certain Casuarina/Stachyurus plants, is a carbonic anhydrase inhibitor and astringent.</p>Fórmula:C41H28O26Forma y color:SolidPeso molecular:936.65RET-IN-1
CAS:RET-IN-1 is a RET kinase inhibitor (IC50s: 1 nM, 7 nM, and 101 nM for RET (WT), RET (V804M) , and RET (G810R), respectively).Fórmula:C29H31N9O3Pureza:98%Forma y color:SolidPeso molecular:553.61MK-7445
CAS:MK-7445 is a conformationally constrained inhibitor of non-nucleoside reverse transcriptase.Fórmula:C21H13Cl2N7OForma y color:SolidPeso molecular:450.28MRTX849 acid
CAS:MRTX849 acid, used to make PROTAC LC-2, effectively degrades KRAS G12C at 0.25-0.76 μM DC50.Fórmula:C34H37ClFN7O4Forma y color:SolidPeso molecular:662.16BMS-986120
CAS:BMS-986120: Oral, reversible PAR4 antagonist. IC50: 9.5 nM (human), 2.1 nM (monkey). Potent, selective antiplatelet.Fórmula:C23H23N5O5S2Forma y color:SolidPeso molecular:513.59WIN 66306
CAS:WIN 66306: Cyclic heptapeptide, blocks NK1/NK2 receptors, inhibits substance P-triggered contractions in guinea pig ileum.Fórmula:C41H52N8O9Forma y color:SolidPeso molecular:800.9RMS-07
CAS:RMS-07, a covalent MPS1/TTK inhibitor, has an IC50 of 13.1 nM, targeting a kinase hinge cysteine.Fórmula:C35H40N8O2Forma y color:SolidPeso molecular:604.74BCL6-IN-9
CAS:BCL6-IN-9 (compound 1) is a potent inhibitor of B-cell lymphoma 6 protein (BCL6) (IC50: 3.9 nM) and can be used to study cancer.Fórmula:C22H18ClF2N5O2Forma y color:SolidPeso molecular:457.86GSK945237
CAS:<p>GSK945237 is a type IIA topoisomerase inhibitor, effective on Gram-positive and negative bacteria, with favorable pharmacokinetics and in vivo efficacy.</p>Fórmula:C24H26FN5O3Forma y color:SolidPeso molecular:451.49BI 224436
CAS:BI 224436 is an inhibitor of HIV-1 noncatalytic site integrase. With EC50 values of less than 15 nM against different HIV-1 laboratory strains.Fórmula:C27H26N2O4Forma y color:SolidPeso molecular:442.51Barixibat
CAS:Barixibat is a bile acid transport inhibitor.Fórmula:C42H55N5O8Forma y color:SolidPeso molecular:757.91Scytonemin
CAS:Scytonemin, a cyanobacterial pigment, inhibits cancer cell growth by decreasing Plk1 activity, especially effective on U266 myeloma cells.Fórmula:C36H20N2O4Forma y color:SolidPeso molecular:544.55Antioxidant agent-8
<p>Antioxidant agent-8, an oral Aβ 1-42 inhibitor, reduces fibril aggregation & promotes disaggregation; it's neuroprotective & BBB permeable.</p>Fórmula:C13H12O5Forma y color:SolidPeso molecular:248.23STA 2
CAS:STA 2 is an analogue of TXA2, a thromboxane receptor in the colonic epithelium.Fórmula:C21H34O3SForma y color:SolidPeso molecular:366.56JBJ-09-063
CAS:JBJ-09-063: EGFR inhibitor, IC50s 0.147-0.396 nM for various mutants; hinders EGFR/Akt/ERK1/2 phosphorylation; targets TKI-sensitive/resistant lung cancer.Fórmula:C31H29FN4O3SForma y color:SolidPeso molecular:556.65Nurr1 agonist 1
Nurr1 agonist 1 is an inverse agonist tool for the neuroprotective transcription factor Nurr1 which is an appealing target to treat neurodegenerative diseases.Fórmula:C16H14N2O2Forma y color:SolidPeso molecular:266.29Onfasprodil
CAS:Onfasprodil, NR2B inhibitor & GABA regulator, potential for Alzheimer's research. (Patent CN111481543A)Fórmula:C20H23FN2O3Forma y color:SolidPeso molecular:358.41Fonadelpar
CAS:Fonadelpar is an agonist of PPARδ. It also is used in the research of neuroparalytic keratopathy.Fórmula:C25H23F3N2O4SPureza:98%Forma y color:SolidPeso molecular:504.52Nedocromil sodium
CAS:Nedocromil sodium is a pharmacologic stabilizer of mast cells, has been shown to normalize cytokine levels and attenuate cardiac remodeling.Fórmula:C19H17NNaO7Pureza:98%Forma y color:SolidPeso molecular:394.335SB 243213 dihydrochloride
CAS:SB 243213 dihydrochloride is an orally active, selective and high-affinity antagonist of 5-hydroxytryptamine (5-HT)2C receptor(pKi of 9.37 and a pKb of 9.8 forFórmula:C22H21Cl2F3N4O2Pureza:98%Forma y color:SolidPeso molecular:501.33PPARγ agonist 2
PPARγ agonist 2 is a highly effective compound that acts as a partial agonist for PPARγ.Fórmula:C24H20O5Forma y color:SolidPeso molecular:388.41Nrf2 activator-2
Compound O15, an Osthole derivative, is a potent Nrf2 agonist with an EC50 of 2.9 μM; it inhibits Keap1-Nrf2 binding and Nrf2 ubiquitination.Fórmula:C20H17BrO3Forma y color:SolidPeso molecular:385.25BRD5631
CAS:BRD5631 is an autophagy enhancer, enhances autophagy through an mTOR-independent pathway.Fórmula:C30H35N3O4Pureza:98%Forma y color:SolidPeso molecular:501.62
