Inhibidores
Los inhibidores son moléculas que se unen a enzimas, receptores u otras proteínas para reducir o bloquear su actividad biológica. Estos compuestos se utilizan ampliamente en la investigación para estudiar vías biológicas, comprender los mecanismos de las enfermedades y desarrollar fármacos terapéuticos. Los inhibidores desempeñan un papel crucial en el tratamiento de diversas enfermedades, incluyendo el cáncer, las enfermedades cardiovasculares y las infecciones. En CymitQuimica, ofrecemos una amplia gama de inhibidores de alta calidad para apoyar su investigación en bioquímica, biología celular y desarrollo farmacéutico.
Subcategorías de "Inhibidores"
- Angiogénesis(2.687 productos)
- Apoptosis(6.097 productos)
- Ciclo celular / Checkpoint(4.691 productos)
- Cromatina / Epigenética(2.376 productos)
- Señalización citoesquelética(1.472 productos)
- Daño al ADN / Reparación del ADN(2.921 productos)
- Endocrinología / Hormonas(3.611 productos)
- Enzima(3.655 productos)
- GPCR / proteína G(8.755 productos)
- Inmunología e inflamación(3.765 productos)
- Virus de la gripe(298 productos)
- Señalización JAK / STAT(407 productos)
- Señalización MAPK(1.230 productos)
- Transportador de membrana / canal de iones(2.947 productos)
- Metabolismo(9.940 productos)
- Microbiología / Virología(7.347 productos)
- Neurociencia(10.240 productos)
- Otros inhibidores(36.533 productos)
- Reducción de oxidación(43 productos)
- Señalización PI3K / Akt / mTOR(1.437 productos)
- Proteasas / Proteasoma(1.675 productos)
- Células madre y Derivados(830 productos)
- Tirosina quinasa / adaptadores(2.028 productos)
- Ubiquitinación(1.682 productos)
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Se han encontrado 66582 productos de "Inhibidores"
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Ep vinyl quinidine
CAS:3-Epiquinine is a Quinidine stereoisomer, used in malaria, antiarrhythmic, inhibits P450db, and blocks K+ channels, IC50: 19.9 μM.Fórmula:C20H24N2O2Forma y color:SolidPeso molecular:324.429(S),10(S),13(S)-TriHOME
CAS:9(S),10(S),13(S)-TriHOME is an oxylipin derived from linoleic acid. It has been detected in beer and in bronchoalveolar lavage fluid (BALF) from female smokers.Fórmula:C18H34O5Forma y color:SolidPeso molecular:330.46IMP-321
CAS:IMP-321 is a soluble dimeric recombinant form of LAG-3 and first-in-class antigen presenting cell activator.Fórmula:C56H78N18O14SForma y color:SolidPeso molecular:1259.4GSK852
GSK852 is a potent, second bromodomain (BD2)-selective, bromo and extra-terminal domain (BET) inhibitor with pIC50 of 7.9.Fórmula:C24H26N2O4Forma y color:SolidPeso molecular:406.47LH secretion antagonist 1
CAS:LH secretion antagonist 1 is an antagonist of luteinizing hormone secretion with analgesic activity.Fórmula:C18H24ClNO2Pureza:98%Forma y color:SolidPeso molecular:321.84Samuraciclib hydrochloride hydrate
Samuraciclib (CT7001) is a potent oral CDK7 inhibitor (IC50: 41 nM) with anti-breast cancer properties.Fórmula:C22H35ClN6O3Forma y color:SolidPeso molecular:521.7Anti-Trypanosoma cruzi agent-2
Compd 3b: anti-trypanosomal, IC50 0.51 μM (NINOA), 3.06 μM (INC-5), also combats T. gondii.Fórmula:C17H10ClNO5Forma y color:SolidPeso molecular:343.72PARP10/15-IN-1
PARP10/15-IN-1 (compound 8l) is a dual PARP10 and PARP15 inhibitor with IC50s of 160 nM and 370 nM, respectively. It can be used in cancer research[1].Fórmula:C13H10N2O3SForma y color:SolidPeso molecular:274.3CDK8-IN-11 hydrochloride
CDK8-IN-11 HCl: potent, selective CDK8 inhibitor (IC50: 46 nM), blocks WNT/β-catenin pathway, used in colon cancer research.Fórmula:C19H16ClF3N4O2Forma y color:SolidPeso molecular:424.8Hit 1
<p>Hit 1 is an activator of insulin-degrading enzymes (IDE) (EC50: 5.5 μM) and reduces glucose-stimulated insulin secretion.</p>Fórmula:C22H24N4O3S2Forma y color:SolidPeso molecular:456.58RS 2135
CAS:RS 2135 is a novel class I antiarrhythmic agent to inhibit ischemia-induced ventricular arrhythmias.Fórmula:C18H21ClN2O2Pureza:98%Forma y color:SolidPeso molecular:332.83DSP-1053 benzenesulfonate
CAS:DSP-1053: Benzylpiperidine-based, potent SERT inhibitor (Ki=1.02nM), partial 5-HT1A receptor agonist (Ki=5.05nM), antidepressant.Fórmula:C32H38BrNO7SForma y color:SolidPeso molecular:660.62SC13
CAS:SC13, a novel mitragynine analog, exhibits low-efficacy agonism at Mu opioid receptors and provides antinociception while minimizing adverse effects.Fórmula:C26H30N2O5Forma y color:SolidPeso molecular:450.53Antifungal agent 11
<p>Antifungal agent 11 has a good antifungal effect.</p>Fórmula:C21H19F2N7O3S2Forma y color:SolidPeso molecular:519.55SPR7
SPR7 is a potent and selective rhodesain inhibitor (Ki: 0.51 nM). SPR7 exhibited antiparasitic effects against T. b. brucei (EC50: 1.65 μM).Fórmula:C30H32ClN3O3Forma y color:SolidPeso molecular:518.05Antifungal agent 13
CAS:Antifungal agent 13 demonstrates significant antifungal activity against Sclerotinia sclerotiorum, achieving an EC50 of 1.25 mg/L.Fórmula:C21H16ClF3N4OForma y color:SolidPeso molecular:432.83SARS-CoV-2 nsp14-IN-2
<p>SARS-CoV-2 nsp14-IN-2: Strong Nsp14 methyltransferase inhibitor (IC50: 0.09 μM), potential for COVID-19 research.</p>Fórmula:C21H21N5O5SForma y color:SolidPeso molecular:455.49Antibacterial agent 99
CAS:Compound 7b (Antibacterial agent 99) is an effective agent with antibacterial, antifungal properties and no haemolytic activity.Fórmula:C27H27BrN2Forma y color:SolidPeso molecular:459.42Spliceostatin A
CAS:<p>Spliceostatin A is an anticancer agent and splicing inhibitor that induces apoptosis by inducing cell cycle arrest in the G1 and G2/M phases.</p>Fórmula:C28H43NO8Pureza:94.66%Forma y color:SolidPeso molecular:521.643Galectin-8-IN-1
Galectin-8-IN-1 selectively binds galectin-8N with 48 μM affinity, 15x more than galectin-3.Fórmula:C16H18N2O6Forma y color:SolidPeso molecular:334.32TH-6
TH-6, a potent HDAC inhibitor (IC50: HDAC1-0.115, 2-0.135, 3-0.242, 6-0.138, 8-2.120 μM), blocks cell migration, invasion, and has anti-tumor properties.Fórmula:C22H24FN3O5Forma y color:SolidPeso molecular:429.44H 218-54
CAS:H 218-54 is a renin inhibitor.Fórmula:C37H56N2O5SForma y color:SolidPeso molecular:640.92MDL-27788
CAS:<p>MDL-27788 is a tricyclic inhibitor.</p>Fórmula:C24H26N2O5SForma y color:SolidPeso molecular:454.54L-365260 hemihydrate
L-365260 hemihydrate: selective oral CCK-B/gastrin blocker, Ki=1.9/2.0 nM, competes with guinea pig receptors.Fórmula:C24H24N4O3Forma y color:SolidPeso molecular:407.47Carumonam Sodium
CAS:Carumonam Sodium is a monobactam, penicillin-binding protein inhibitor. It is used as antibacterials.Fórmula:C12H12N6Na2O10S2Pureza:98%Forma y color:SolidPeso molecular:510.37RORγt/DHODH-IN-3
<p>RORγt/DHODH-IN-3 (compound (S)-14d) is a potent, orally active dual inhibitor of RORγt (IC50: 0.098 μM) and DHODH (IC50: 0.432 μM).RORγt/DHODH-IN-1 has</p>Fórmula:C24H26ClF6N3O3SForma y color:SolidPeso molecular:585.99GLPG0492 (R enantiomer)
CAS:GLPG0492 R enantiomer is the R enantiomer of GLPG-0492, a novel selective androgen receptor modulator.Fórmula:C19H14F3N3O3Forma y color:SolidPeso molecular:389.33FGFR1 inhibitor-6
FGFR1 inhibitor-6, IC50: 16.31 nM, blocks cell cycle at pro-G1/G2/M and induces apoptosis.Fórmula:C27H19N5O4S2Forma y color:SolidPeso molecular:541.6CDK7/12-IN-1
CAS:CDK7/12-IN-1 is a selective CDK7 (IC50: 3 nM) and CDK12 (IC50: 277 nM) inhibitor, effective against tumor growth.Fórmula:C25H34N8OForma y color:SolidPeso molecular:462.59Danavorexton
CAS:Danavorexton is an orexin receptor agonist.Fórmula:C21H32N2O5SForma y color:SolidPeso molecular:424.55Gabaculine HCl
CAS:<p>Gabaculine, an irreversible GABA-T inhibitor (Ki: 2.9 μM), impacts plastid development and affects DPOR/GluTR levels.</p>Fórmula:C7H10ClNO2Forma y color:SolidPeso molecular:175.61Topo I-IN-1
<p>Topo I-IN-1 (14d) is a powerful Topo I inhibitor with antitumor effects and DNA intercalation, inducing apoptosis.</p>Fórmula:C20H14BrN3O2Forma y color:SolidPeso molecular:408.25PDE4B/7A-IN-1
CAS:5-HT1A antagonist; Ki=8nM, Kb=0.04nM. PDE4B IC50=80.4μM; PDE7A IC50=151.3μM. Good biofilm penetration, stable, anticognitive, antidepressant.Fórmula:C25H35N3O3Forma y color:SolidPeso molecular:425.56PRMT5-IN-1 hydrochloride
PRMT5 IN-1 hydrochloride is a potent PRMT5 inhibitor (IC50: 11 nM), forms covalent adduct with C449, and converts to an aldehyde in vivo.Fórmula:C19H20Cl2N4O5Forma y color:SolidPeso molecular:455.29Elocalcitol
CAS:Elocalcitol is a calcitriol analog for inhibition of prostate cell growth.Fórmula:C29H43FO2Forma y color:SolidPeso molecular:442.65Retelliptine
CAS:Retelliptine, a DNA topoisomerase II inhibitor, is used potentially for the treatment of cancer.Fórmula:C25H32N4OPureza:98%Forma y color:SolidPeso molecular:404.55AZ-3
CAS:AZ-3 is a potent and selective JAK1 inhibitor (IC50: 34 nM).Fórmula:C20H28FN7Pureza:98%Forma y color:SolidPeso molecular:385.48Cathepsin C-IN-5
CAS:<p>Cathepsin C-IN-5 (SF38) is a potent, oral Cathepsin C blocker with an IC50 of 59.9 nM; less active against Cat L/S/B/K; has anti-inflammatory effects.</p>Fórmula:C21H17ClN6OSForma y color:SolidPeso molecular:436.92Tubulin inhibitor 17
Compound 3b inhibits tubulin polymerization, IC50 12.38 µM, with anticancer properties and promotes cell apoptosis.Fórmula:C17H16N2OForma y color:SolidPeso molecular:264.32MCTR1
CAS:MCTR1, a pro-resolving mediator derived from DHA, promotes tissue repair and reduces inflammation by enhancing phagocytosis and decreasing eicosanoids.Fórmula:C32H47N3O9SForma y color:SolidPeso molecular:649.8U92016A hydrochloride
CAS:U92016A hydrochloride: potent, orally active 5-HT1A agonist, metabolically stable, high intrinsic activity, Ki=0.2 nM.Fórmula:C19H26ClN3Forma y color:SolidPeso molecular:331.89Nnc 09-0026
CAS:Nnc 09-0026 is a neuronal calcium channel blockerFórmula:C25H35Cl2F3N2OForma y color:SolidPeso molecular:507.46BRD4-BD1/2-IN-2
CAS:BRD4-BD1/2-IN-2 inhibits BRD4 BD1/BD2 with IC50 <300 nM/<0.5 nM (WO2021233371A1).Fórmula:C30H33N5O4Forma y color:SolidPeso molecular:527.61NPEC-caged-(S)-3,4-DCPG
CAS:mGlu8a agonistFórmula:C19H16N2O10Pureza:98%Forma y color:SolidPeso molecular:432.34LSD1/ER-IN-1
LSD1/ER-IN-1 inhibits ER & LSD1 (IC50: 1.55 μM), and fights MCF-7 breast cancer (IC50: 8.79 μM).Fórmula:C23H18FNO6SForma y color:SolidPeso molecular:455.46CV 5975
CAS:CV 5975 is a nonsulfhydryl ACE inhibitor that was investigated for use in hypertension and heart failure.Fórmula:C22H31N3O5SForma y color:SolidPeso molecular:449.5620S Proteasome-IN-4
CAS:<p>20S Proteasome-IN-4: brain-penetrant, parasite-specific, oral, inhibits T.b. brucei proteasome (IC50: 6.3nM), for HAT research.</p>Fórmula:C20H18ClF2N3O3Forma y color:SolidPeso molecular:421.83α-Glucosidase-IN-17
CAS:α-Glucosidase-IN-17 (Compound 12B) is a potent and orally active inhibitor of α-glucosidase, demonstrating antidiabetic activity with an inhibitoryFórmula:C30H27NO2SForma y color:SolidPeso molecular:465.61Anticancer agent 79
<p>Anticancer agent 79 (3d) has potent activity against breast cancer, with cytotoxic effects on T47-D, IC50=13.64±0.26μM.</p>Fórmula:C20H12F3NO5Forma y color:SolidPeso molecular:403.31HBV-IN-11
CAS:HBV-IN-11 is a potent inhibitor of HBsAg secretion (EC50: 0.46 μM).Fórmula:C21H24ClNO6Forma y color:SolidPeso molecular:421.87Valopicitabine dihydrochloride
CAS:Valopicitabine, a NS5B inhibitor, is used potentially for the treatment of HCV infection.Fórmula:C15H25ClN4O6Forma y color:SolidPeso molecular:392.84DC41SMe
CAS:<p>DC41SMe, a DC1 derivative and CC-1065 analogue, targets cancer with 18-25 pM IC50 against Ramos, Namalwa, HL60/s cells.</p>Fórmula:C38H36ClN5O4S2Pureza:98%Forma y color:SolidPeso molecular:726.31NA 382
CAS:NA 382 is a staurosporine derivative that inhibits multidrug resistance.Fórmula:C31H28N4O6Forma y color:SolidPeso molecular:552.58SARS-CoV-2-IN-22
CAS:<p>SARS-CoV-2-IN-22 is a SARS-CoV-2 pseudovirus inhibitor (IC50: 16.96 μM).</p>Fórmula:C27H24N2O3SForma y color:SolidPeso molecular:456.56J-104871
CAS:<p>J-104871 (UNII-6137X5QNJF) is an FTase inhibitor that inhibits tumor growth in nude mice transplanted with activated H-ras-transformed NIH3T3 cells.</p>Fórmula:C38H32N2O12Pureza:98%Forma y color:SolidPeso molecular:708.67Zanapezil fumarate
CAS:Zanapezil is an acetylcholinesterase (AChE) inhibitor. Zanapezil increases choline acetyltransferase activity in cultured rat septal cholinergic neurons.Fórmula:C29H36N2O5Forma y color:SolidPeso molecular:492.61SHP2-IN-9
<p>SHP2-IN-9: Potent SHP2 inhibitor, IC50=1.174 μM, 85x SHP1 selectivity, crosses blood-brain barrier, hampers cancer growth.</p>Fórmula:C20H20FN3O2SForma y color:SolidPeso molecular:385.46AFP464 free base
CAS:AFP464 (NSC710464) free base is an active HIF-1α inhibitor (IC50: 0.25 μM) and a potent aryl hydrocarbon receptor (AhR) activator.Fórmula:C22H23F3N4O3Pureza:98%Forma y color:SolidPeso molecular:448.44AZD-3409
CAS:AZD-3409 is a more potent prenyl transferase inhibitor than lonafarnib with varied IC(50) in cells, acting on gefitinib-resistant breast cancer.Fórmula:C34H41FN4O4S2Forma y color:SolidPeso molecular:652.847(Z),11(Z)-Nonacosadiene
CAS:7(Z),11(Z)-Nonacosadiene, a female fly pheromone, spurs male courtship; it's a C29 diene made by a female-specific elongase.Fórmula:C29H56Forma y color:SolidPeso molecular:404.75Unoprostone
CAS:Unoprostone is a prostaglandin F2α analogs (PGAs), and reduces intraocular pressure and is used topically for glaucoma or ocular hypertension.Fórmula:C22H38O5Pureza:98%Forma y color:SolidPeso molecular:382.53LY3325656
CAS:LY3325656, a GPR142 agonist with anti-diabetic properties, progresses to phase 1 trials for Type 2 diabetes.Fórmula:C21H23F3N6O2Forma y color:SolidPeso molecular:448.44UCN-02
CAS:UCN-02 (7-epi-Hydroxystaurosporine) is a PKC inhibitor produced by Streptomyces N-126 strain, which inhibits PKA.Fórmula:C28H26N4O4Pureza:98%Forma y color:SolidPeso molecular:482.53KPH2f
CAS:KPH2f: dual URAT1/GLUT9 inhibitor, orally active, IC50: 0.24μM (URAT1), 9.37μM (GLUT9), minimal OAT1/ABCG2 impact.Fórmula:C24H16N3NaO2SForma y color:SolidPeso molecular:433.46AChE/BACE1/GSK3β-IN-1
AChE/BACE1/GSK3β-IN-1 is an orally active, blood-brain barrier-transparent, moderately bioavailable triple inhibitor of AChE/BACE1/GSK3β.Fórmula:C26H27FN2O4Forma y color:SolidPeso molecular:450.5Topoisomerase II inhibitor 6
Topoisomerase II inhibitor 6, a potent tryptanthrin derivative, blocks G2 phase in CCRF-CEM cells, induces DNA breaks, and may be used for cancer research.Fórmula:C19H18N4O2Forma y color:SolidPeso molecular:334.37Antifungal agent 27
<p>Antifungal agent 27 shows moderate action against MRSA, weak against C. albicans, with MICs of 8 μg/mL and 32 μg/mL, respectively.</p>Fórmula:C18H23N5OSForma y color:SolidPeso molecular:357.47IRAK4-IN-15
CAS:IRAK4-IN-15: selective IRAK4 inhibitor, IC50 0.002 μM, good PK, low clearance, synergizes with Acalabrutinib in MyD88/CD79 mutant ABC-DLBCL.Fórmula:C25H29FN10Forma y color:SolidPeso molecular:488.56B-3852
CAS:B-3852 is a Bradykinin inhibitor.Fórmula:C55H74F3N15O11Forma y color:SolidPeso molecular:1178.27PF-00446687
CAS:PF-00446687 is a selective agonist of melanocortin-4 receptor (MC4R) (EC50 of 12 ± 1 nM).Fórmula:C28H36F2N2O2Pureza:98%Forma y color:SolidPeso molecular:470.59Pegcantratinib
CAS:Pegcantratinib is a tropomyosin receptor kinase inhibitor for treatment for inherited CYLD defective skin tumours.Fórmula:C32H28N4O7Forma y color:SolidPeso molecular:580.59α-Glucosidase-IN-13
α-Glucosidase-IN-13 is an inhibitor of α-glucosidase (IC50: 5.69 μM).Fórmula:C25H28N4O3S2Forma y color:SolidPeso molecular:496.64hTrkA-IN-2
<p>hTrkA-IN-2 is a selective hTrkA metamorphosis inhibitor (IC50: 3.9 nM).</p>Fórmula:C24H22F3N5O3Forma y color:SolidPeso molecular:485.46D-Cl-amidine hydrochloride
D-Cl-amidine hydrochloride is a potent and highly selective inhibitor of PAD1. It exhibits excellent tolerance and does not induce significant toxicity [1].Fórmula:C14H20Cl2N4O2Forma y color:SolidPeso molecular:347.24WS-898
<p>WS-898 boosts paclitaxel efficacy in resistant cells by inhibiting ABCB1; IC50: SW620/Ad300 - 5.0 nM, KB-C2 - 3.67 nM, HEK293/ABCB1 - 3.68 nM.</p>Fórmula:C33H25N7OSForma y color:SolidPeso molecular:567.66RXR antagonist 2
RXR antagonist 2 is a potent antagonist of RXR (Ki: 0.391 μM, Kd: 0.281 μM). RXR antagonist 2 has shown research potential for RXR-related diseases.Fórmula:C29H35F3N2O3Forma y color:SolidPeso molecular:516.6Tubulin inhibitor 19
Tubulin inhibitor 19 (9b), a potent indole chalcone, strongly blocks tubulin, valuable in cancer studies.Fórmula:C21H23NO5Forma y color:SolidPeso molecular:369.41Freselestat quarterhydrate
ONO-6818 quarterhydrate: oral neutrophil elastase inhibitor, Ki 12.2 nM; >100x less effective on other proteases; strong anti-inflammatory.Fórmula:C23H30N6O5Forma y color:SolidPeso molecular:457.03A1-Phytoprostane-I
CAS:A1-Phytoprostane-I: cyclopentenone from α-linolenic acid in plants, induces gene expression & increases phytoalexin synthesis.Fórmula:C18H28O4Forma y color:SolidPeso molecular:308.41VVD-118313
CAS:VVD-118313 (5a) is a potent JAK1 inhibitor targeting allosteric cysteine, blocking cytokine signaling for cancer research.Fórmula:C19H22Cl2N2O3SForma y color:SolidPeso molecular:429.36PF-9404C
CAS:PF-9404C: S-S diastereoisomer, beta-blocker with vasodilation, boosts cyclic GMP in rat aorta cells from 3 to 53 pmol/mg protein.Fórmula:C16H25N3O9Pureza:98%Forma y color:SolidPeso molecular:403.38FTO-IN-4
CAS:FTO-IN-4 is a potent and selective inhibitor of adiposity and obesity-associated protein (FTO).Fórmula:C22H16Cl2N6O6Forma y color:SolidPeso molecular:531.31CLK1/4-IN-1
CLK1/4-IN-1 inhibits Clk1/4 (IC50: 9.7/6.6 nM), curbing T24 cell growth (GI50: 1.1 μM). Potential cancer research tool.Fórmula:C18H14ClNO4SForma y color:SolidPeso molecular:375.83VEGFR-2-IN-16
VEGFR-2-IN-16 (Compound 15b) is a potent inhibitor of VEGFR-2 (IC50: 86.36 nM) that exhibits antitumour effects.Fórmula:C21H13Cl2N3O2Forma y color:SolidPeso molecular:410.25Bilanafos
CAS:Bilanafos is an agent of Anti-Bacterial.Fórmula:C11H22N3O6PPureza:98%Forma y color:SolidPeso molecular:323.28Antitubercular agent-15
Antitubercular agent-15 (5n): low toxicity, fights M. tuberculosis strains; MIC90 values range 0.73-18.8 μg/mL.Fórmula:C21H29FN2Forma y color:SolidPeso molecular:328.47ALK-IN-23
ALK-IN-23 inhibits ALK (IC50: 1.6-0.71 nM), hinders cancer cell spread, forms colonies in vitro, and reduces tumors in mice with low toxicity.Fórmula:C26H29ClN8O3SForma y color:SolidPeso molecular:569.08CXN37378
CAS:CXN37378, aka NAP, is a potent MOR-selective antagonist with no official name yet, termed per MedKoo Nomenclature.Fórmula:C27H31N3O4Forma y color:SolidPeso molecular:461.55KRAS G12D inhibitor 1
CAS:KRAS G12D inhibitor 1 (example 243) is an inhibitor of KRAS G12D with an IC 50 of 0.8 nM for KRAS G12D-mediated ERK phosphorylation [1].Fórmula:C33H32F2N6O2Forma y color:SolidPeso molecular:582.64(+)-Cevimeline hydrochloride hemihydrate
(+)-Cevimeline HCl hemihydrate is a muscarinic agonist for dry mouth in Sjogren's with rapid absorption, differing metabolism in species.Fórmula:C10H19ClNO1·5SPureza:98%Forma y color:SolidPeso molecular:244.78MRS2279 diammonium
CAS:<p>MRS2279 diammonium, a P2Y1 antagonist with K i 2.5 nM, IC 50 51.6 nM, blocks ADP-induced platelet aggregation, pK b 8.05.</p>Fórmula:C13H24ClN7O8P2Forma y color:SolidPeso molecular:503.77CDK/HDAC-IN-1
<p>CDK/HDAC-IN-1 inhibits CDK2/4/6 & HDAC6 with IC50s: 60.9, 276, 27.2, and 128.6 nM respectively.</p>Fórmula:C20H18N4O4Forma y color:SolidPeso molecular:378.38Anticancer agent 65
CAS:Anticancer agent 65: Effective on A549 cells, IC50 1.07 μM, halts S phase, triggers apoptosis, elevates p53/p21, causes ROS and MMP collapse.Fórmula:C36H63NO5Forma y color:SolidPeso molecular:589.89JAK3/BTK-IN-4
CAS:JAK3/BTK-IN-4, a dual inhibitor for JAK3/BTK, shows synergy in autoimmune disease treatment. (Patent WO2021147953A1, compound 003)Fórmula:C21H25ClN8OForma y color:SolidPeso molecular:440.93Brostallicin HCl
CAS:Brostallicin, a synthetic MGB, inhibits DNA replication in cancer cells, inducing cell death, effective against MMR-defective tumors.Fórmula:C30H36BrClN12O5Forma y color:SolidPeso molecular:760.04Idraparinux Na
CAS:Idraparinux Na is an Antithrombotic, Indirect, Selective, Synthetic Factor Xa InhibitorFórmula:C38H55Na9O49S7Forma y color:SolidPeso molecular:1727.14Ladirubicin
CAS:Ladirubicin, as an anthracyclines analog is the leading compound of alkylcyclines.Fórmula:C29H31NO11SForma y color:SolidPeso molecular:601.62A 74273
CAS:<p>A 74273, a nonpeptidic and renin inhibitor, may be used to treat cardiovascular diseases due to renin inhibition.</p>Fórmula:C44H74N4O8Pureza:98%Forma y color:SolidPeso molecular:787.08HDAC6/HSP90-IN-2
<p>HDAC6/HSP90-IN-2, a cancer research chemical, inhibits HDAC6 & Hsp90 with IC50s of 105.7 & 61 nM.</p>Fórmula:C19H22N2O5Forma y color:SolidPeso molecular:358.39
