Inhibidores
Los inhibidores son moléculas que se unen a enzimas, receptores u otras proteínas para reducir o bloquear su actividad biológica. Estos compuestos se utilizan ampliamente en la investigación para estudiar vías biológicas, comprender los mecanismos de las enfermedades y desarrollar fármacos terapéuticos. Los inhibidores desempeñan un papel crucial en el tratamiento de diversas enfermedades, incluyendo el cáncer, las enfermedades cardiovasculares y las infecciones. En CymitQuimica, ofrecemos una amplia gama de inhibidores de alta calidad para apoyar su investigación en bioquímica, biología celular y desarrollo farmacéutico.
Subcategorías de "Inhibidores"
- Angiogénesis(2.524 productos)
- Apoptosis(5.793 productos)
- Ciclo celular / Checkpoint(4.452 productos)
- Cromatina / Epigenética(2.242 productos)
- Señalización citoesquelética(1.382 productos)
- Daño al ADN / Reparación del ADN(2.826 productos)
- Endocrinología / Hormonas(3.507 productos)
- Enzima(3.640 productos)
- GPCR / proteína G(8.333 productos)
- Inmunología e inflamación(3.527 productos)
- Virus de la gripe(296 productos)
- Señalización JAK / STAT(404 productos)
- Señalización MAPK(1.203 productos)
- Transportador de membrana / canal de iones(2.792 productos)
- Metabolismo(9.449 productos)
- Microbiología / Virología(6.981 productos)
- Neurociencia(9.926 productos)
- Otros inhibidores(37.921 productos)
- Reducción de oxidación(41 productos)
- Señalización PI3K / Akt / mTOR(1.400 productos)
- Proteasas / Proteasoma(1.597 productos)
- Células madre y Derivados(830 productos)
- Tirosina quinasa / adaptadores(2.015 productos)
- Ubiquitinación(1.650 productos)
Mostrar 16 subcategorías más
Se han encontrado 66639 productos de "Inhibidores"
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Mesulergine hydrochloride
CAS:<p>5-HT2A and 2C receptor antagonist</p>Fórmula:C18H27ClN4O2SPureza:98%Forma y color:SolidPeso molecular:398.95AAK1-IN-2 TFA
<p>AAK1-IN-2 TFA (compound (S)-31) is a selective and potent AAK1 inhibitor (IC50: 5.8 nM) that can cross the blood-brain barrier.</p>Fórmula:C24H22F6N4O4Forma y color:SolidPeso molecular:544.45AChE/BChE-IN-1
<p>AChE/BChE-IN-1: dual AChE/BChE inhibitor, IC50 of 1.06 nM/7.3 nM, crosses blood-brain barrier, with antioxidant properties for Alzheimer's research.</p>Fórmula:C32H35ClN6O3Forma y color:SolidPeso molecular:587.11LY 215840
CAS:<p>5-HT2/5-HT7 receptor antagonist</p>Fórmula:C24H33N3O2Pureza:98%Forma y color:SolidPeso molecular:395.54JBJ-02-112-05
CAS:<p>JBJ-02-112-05 is a potent, mutant-selective, allosteric and orally active inhibitor of EGFR with an IC 50 of 15 nM for EGFR L858R/T790M [1].</p>Fórmula:C27H20N4O2SPureza:98%Forma y color:SolidPeso molecular:464.54ATX inhibitor 22
<p>ATX inhibitor 22 is a novel inhibitor of ATX (autotaxin) (IC50: 218.9 μM) that lacks inhibitory activity against LPAR1.</p>Fórmula:C19H17Cl3F2N2O4SForma y color:SolidPeso molecular:513.77C.I. Pigment Red 60
CAS:<p>C.I. Pigment Red 60 is a bright, scarlet, semi-transparent red pigment.</p>Fórmula:C17H9N2Na3O9S2Pureza:98%Forma y color:SolidPeso molecular:518.35ML-SI1
CAS:<p>ML-SI1, a racemic mixture of diastereoisomers, is a TRPML inhibitor and acts on TRPML1 (IC50: 15 μM).</p>Fórmula:C23H26Cl2N2O3Forma y color:SolidPeso molecular:449.37IRAK4-IN-12
<p>IRAK4-IN-12 (compound 37) is a potent inhibitor of IRAK4 (IC50: 0.015 μM) with cellular pIRAK4 potency (IC50: 0.5 μM).</p>Fórmula:C24H31FN8OForma y color:SolidPeso molecular:466.55Pim-1 kinase inhibitor 3
CAS:<p>Pim-1 kinase inhibitor 3 (Compound H5) is a potent inhibitor of Pim-1 kinase, demonstrating an inhibitory concentration (IC50) of 35.13 nM [1].</p>Fórmula:C20H25N3O2Forma y color:SolidPeso molecular:339.43Arverapamil
CAS:<p>Arverapamil is a chiral metabolite of Verapamil.</p>Fórmula:C26H36N2O4Forma y color:SolidPeso molecular:440.58Dopamine D3 receptor antagonist-2
<p>Dopamine D3 receptor antagonist-2 is a dopamine D3 receptor selective (Ki=2.16 nM) or multi-targeting dual ligand that shows potential effects in CNS disorders.</p>Fórmula:C23H27Cl2N3O3Forma y color:SolidPeso molecular:464.38MI-1851
CAS:<p>MI-1851 is a potent peptidomimetic inhibitor. MI-1851could prevent proteolytic processing of the S protein from SARSCoV-2 by endogenous furin in HEK293 cells.</p>Fórmula:C34H53N15O6Forma y color:SolidPeso molecular:767.88MEIS-IN-2
<p>MEIS-IN-2 is an inhibitor of MEIS1. MEIS-IN-2 can be used in studies of cardiac regeneration and haematopoietic stem cell (HSC) regulation.</p>Fórmula:C23H21ClN2O4Forma y color:SolidPeso molecular:424.88DC41
CAS:<p>DC41 is a CC-1065-based cancer drug, an antibody-linked DNA alkylator.</p>Fórmula:C37H34ClN5O4SPureza:98%Forma y color:SolidPeso molecular:680.22AChE/PDE4-IN-1
<p>AChE/PDE4-IN-1, compound 12c, dual inhibitor; IC50: 0.28μM for AChE, 1.88μM for PDE4D, may reduce Alzheimer's neuroinflammation.</p>Fórmula:C23H28N2O3Forma y color:SolidPeso molecular:380.48Dinordrin
CAS:<p>Dinordrin is an implantation inhibitor and hormone.</p>Fórmula:C27H36O4Pureza:98%Forma y color:SolidPeso molecular:424.57Topoisomerase II inhibitor 5
<p>Topoisomerase II inhibitor 5 (Compound E24) is a DNAtopoisomerase II inhibitor with anticancer effects.</p>Fórmula:C26H27N5O4Forma y color:SolidPeso molecular:473.52Demethoxyviridin
CAS:<p>Demethoxyviridin inhibits mammalian Ptdlns 3-kinase (p110) and is antifungal.</p>Fórmula:C19H14O5Pureza:98%Forma y color:SolidPeso molecular:322.31Refametinib R enantiomer
CAS:<p>Refametinib R enantiomer (RDEA119 R enantiomer) is an MEK inhibitor with an EC50 of 2.0-15 nM.Refametinib (R enantiomer) has anticancer activity and can be used</p>Fórmula:C19H20F3IN2O5SPureza:99.86%Forma y color:SolidPeso molecular:572.34(±)-J 113397
CAS:<p>(±)-J-113397 is a potent and selective non-peptidyl ORL1 receptor antagonist (K(i): cloned human ORL1=1.8 nM).</p>Fórmula:C24H37N3O2Forma y color:SolidPeso molecular:399.57NTPDase-IN-3
CAS:<p>NTPDase-IN-3 inhibits NTPDase1/2/3/8 (IC50: 0.21/1.07/0.38/0.05 μM), useful for cancer and thrombosis research.</p>Fórmula:C22H24ClN3OS2Forma y color:SolidPeso molecular:446.03IT-066 HCl
CAS:<p>IT-066 HCl is a histamine H2 receptor antagonist.</p>Fórmula:C19H25ClN4O3Forma y color:SolidPeso molecular:392.88Implitapide
CAS:<p>Implitapide is an inhibitor of microsomal triglyceride transfer protein (MTP).</p>Fórmula:C35H37N3O2Pureza:98%Forma y color:SolidPeso molecular:531.69Indoluidin E
<p>Indoluidin E selectively inhibits DHODH and has an inhibitory effect on cancer cell growth.</p>Fórmula:C28H30N4O2Forma y color:SolidPeso molecular:454.56Kinamycin B
CAS:<p>Kinamycin B is an antibacterial agent with anticancer activity.</p>Fórmula:C20H16N2O8Pureza:98%Forma y color:SolidPeso molecular:412.35SARS-CoV-2-IN-6
<p>SARS-CoV-2-IN-6 is an inhibitor of SARS-CoV-2 3CLpro with the IC 50 value of 73 nM.</p>Fórmula:C17H13ClN2O2Forma y color:SolidPeso molecular:312.75Minnelide free acid
CAS:<p>Minnelide treats pancreatic cancer, hinders androgen-related prostate growth, shrinks tumors, and improves survival.</p>Fórmula:C21H27O10PForma y color:SolidPeso molecular:470.41GYKI-53784
CAS:<p>GYKI-53784 (LY 303070) is an effective selective AMPA receptor antagonist.</p>Fórmula:C19H20N4O3Forma y color:SolidPeso molecular:352.39JH295 hydrate
<p>JH295 hydrate: potent, irreversible Nek2 inhibitor (IC50 = 770 nM), selective, doesn't target Cdk1, Aurora B or Plk1.</p>Fórmula:C18H18N4O3Forma y color:SolidPeso molecular:338.36Lp-PLA2-IN-10
<p>Lp-PLA2-IN-10, a potent Lp-PLA2 inhibitor, may research neurodegenerative and cardiovascular diseases.</p>Fórmula:C21H15F5N4O4Forma y color:SolidPeso molecular:482.36(rel)-AR234960
CAS:(rel)-AR234960 is an active relative configuration of AR234960. AR234960 is a non-peptide agonist of MAS.Fórmula:C27H30FN5O5SForma y color:SolidPeso molecular:555.63HCV-IN-38
<p>Potent oral HCV inhibitor HCV-IN-38 has 15 nM EC50, 431 SI, high efficacy, and low toxicity.</p>Fórmula:C22H24ClF3N4O4Forma y color:SolidPeso molecular:500.9KUSC-5037
<p>KUSC-5037 inhibits HIF-1 (IC50 = 1.2 μM) and mitochondrial complex V/FoF1ATP synthase.</p>Fórmula:C18H17F3N6O2Forma y color:SolidPeso molecular:406.13651AChE-IN-8
<p>AChE-IN-8 (Compound 19), potent acetylcholinesterase blocker; IC50 = 1.95 μM; potential Alzheimer's treatment.</p>Fórmula:C20H22N4O2SForma y color:SolidPeso molecular:382.48AZD0424
CAS:<p>AZD0424: oral Src/Abl kinase inhibitor; potential anticancer; induces apoptosis, cell cycle arrest in lymphoma.</p>Fórmula:C25H29ClN6O5Pureza:98%Forma y color:SolidPeso molecular:528.99Antibiotic MA 144M2
CAS:<p>Antibiotic MA 144M2, an anthracycline glycoside, targets gram-positive bacteria and tumors, derived from Streptomyces and aclacinomycin A conversion.</p>Fórmula:C42H55NO16Forma y color:SolidPeso molecular:829.88(S)-ZG197
<p>(S)-ZG197 is a compound that acts as a highly selective activator of the Staphylococcus aureus Caseinolytic Protease P (Sa ClpP), demonstrating efficacy at a</p>Fórmula:C28H35F3N4O3Forma y color:SolidPeso molecular:532.6AR antagonist 4
<p>AR antagonist 4 (Compound 67-b) is an orally active androgen receptor (AR) antagonist that acts on wild-type AR (IC50: 246.6 nM).</p>Fórmula:C29H36N4OForma y color:SolidPeso molecular:456.62Musettamycin
CAS:<p>Musettamycin triggers erythroid differentiation in blood cells, acts like anthracycline antibiotics, but only inhibits gram-positive bacteria.</p>Fórmula:C36H45NO14Forma y color:SolidPeso molecular:715.74AMD-7049
CAS:<p>AMD-7049 is a biochemical.</p>Fórmula:C25H39N5Forma y color:SolidPeso molecular:409.61CCT369260
CAS:<p>CCT369260 (compound 1), an orally active inhibitor targeting B-cell lymphoma 6 (BCL6), demonstrates anti-tumor efficacy with an IC50 value of 520 nM [1].</p>Fórmula:C24H31ClF2N6O2Forma y color:SolidPeso molecular:508.99Wikstrol A
CAS:<p>Wikstrol A: antifungal, anti-mitotic, anti-HIV agent with various IC50/MDC values (67.8-131 µM) and deforms P. oryzae mycelia.</p>Fórmula:C30H22O10Forma y color:SolidPeso molecular:542.49B-3852
CAS:<p>B-3852 is a Bradykinin inhibitor.</p>Fórmula:C55H74F3N15O11Forma y color:SolidPeso molecular:1178.27Flusoxolol
CAS:<p>Flusoxolol is a beta-adrenoceptor partial agonist.</p>Fórmula:C22H30FNO4Forma y color:SolidPeso molecular:391.48HDAC-IN-27
<p>HDAC-IN-27 is a potent and orally active inhibitor of HDAC Class I (0.43 nM - 3.01 nM for HDAC1-3).</p>Fórmula:C20H22N4O2Forma y color:SolidPeso molecular:350.41BAY-364
CAS:<p>BAY-364 (BAY-299N) functions as an inhibitor targeting the second bromine domain in TAF1, demonstrating inhibitory effects on TAF1 in Kasumi-1 cells, CD34+</p>Fórmula:C23H19N3O4Forma y color:SolidPeso molecular:401.417(Z),11(Z)-Nonacosadiene
CAS:<p>7(Z),11(Z)-Nonacosadiene, a female fly pheromone, spurs male courtship; it's a C29 diene made by a female-specific elongase.</p>Fórmula:C29H56Forma y color:SolidPeso molecular:404.75DNA Gyrase-IN-1
<p>DNA Gyrase-IN-1: potent, selective promoter inhibitor. IC50: 2.6 μM, inhibits Mtb, MIC: 0.49 μM. Useful for tuberculosis research.</p>Fórmula:C24H24FN7O6Forma y color:SolidPeso molecular:525.49EBI-907
CAS:<p>EBI-907 is a potent, oral B-RafV600E inhibitor with an IC50 of 4.9 nM, over 10x stronger than Vemurafenib, and effective against key cancer kinases.</p>Fórmula:C23H21ClF2N4O3SForma y color:SolidPeso molecular:506.95G-479
CAS:<p>G-479, a potent MEK inhibitor and improved analogue of GDC-0623, has distributed polarity enhancing bioactivity.</p>Fórmula:C16H15FIN5O4Forma y color:SolidPeso molecular:487.22Py-MPB-amino-C3-PBD
CAS:<p>Py-MPB-amino-C3-PBD is a cytotoxic agent comprised non-alkylating group,with antimicrobial activity.</p>Fórmula:C41H44N8O6Pureza:98%Forma y color:SolidPeso molecular:744.84Methyl Streptonigrin
CAS:<p>Methyl Streptonigrin is an ABCG2 transporter function inhibitor.</p>Fórmula:C26H24N4O8Pureza:98%Forma y color:SolidPeso molecular:520.49GSK 366
CAS:GSK 366 is a potent kynurenine-3-monooxygenase (KMO) inhibitor (IC50s: 0.7 nM and 2.3 nM for P. fluorescens-KMO and human KMO).Fórmula:C17H16ClN3O4Pureza:98%Forma y color:SolidPeso molecular:361.78FTI-2628
CAS:<p>FTI-2628 is a novel inhibitor of protein farnesyltransferase (FT), inhibiting the growth of P. falciparum in red blood cells and suppressing parasitemia.</p>Fórmula:C31H34N4O3SForma y color:SolidPeso molecular:542.69PF-06726304 acetate
CAS:<p>PF-06726304 acetate is a selective inhibitor of EZH2, with robust antitumor growth activity.</p>Fórmula:C24H25Cl2N3O5Pureza:98%Forma y color:SolidPeso molecular:506.38Human carbonic anhydrase II-IN-2
<p>Compound R-13, a potent inhibitor of hCA I/II/IV/IX with K i s of 60.7, 320.7, 2298, and 35.2 nM.</p>Fórmula:C20H25N3O4SForma y color:SolidPeso molecular:403.5hCAIX/XII-IN-5
<p>Coumarin 9a: Selective inhibitor of hCA IX/XII (Ki 93.3/85.7 nM), blocks cancer cell growth, and induces apoptosis.</p>Fórmula:C18H13NO3Forma y color:SolidPeso molecular:291.3IDO1-IN-13
<p>IDO1-IN-13 is a potent IDO1 inhibitor (IC50: 61.6 nM, EC50: 30 nM in HeLa) that reduces kyn/trp ratio by 51% in SK-OV-3 tumors.</p>Fórmula:C20H16BrN5O2SForma y color:SolidPeso molecular:470.34E-3030 free acid
CAS:<p>E-3030 free acid, a PPAR agonist, lowers blood glucose, triglycerides, and insulin; boosts adiponectin; reduces apo C-III; and raises lipoprotein lipase.</p>Fórmula:C22H23ClFNO5Pureza:98%Forma y color:SolidPeso molecular:435.87Teslexivir hydrochloride
CAS:<p>Teslexivir (BTA074) HCl inhibits HPV 6/11 by blocking E1-E2 protein interaction, vital for DNA replication. Used in condyloma research.</p>Fórmula:C35H37BrClN3O4Forma y color:SolidPeso molecular:679.04PD-149163
CAS:<p>PD-149163: brain-penetrating, selective NTR1 agonist; shows pro-cognitive, anti-psychotic, anxiolytic effects.</p>Fórmula:C42H71N9O6Forma y color:SolidPeso molecular:798.07P7170
CAS:<p>P7170 is an anti-cancer agent active as an mTORC1/C2 and activin receptor-like kinase 1 (ALK1) inhibitor.</p>Fórmula:C21H16F3N9Forma y color:SolidPeso molecular:451.42Carmegliptin dihydrochloride
CAS:<p>Carmegliptin dihydrochloride (RG-1579, RO4876904) is a salt of Camegliptin, a DPP-4 inhibitor for type 2 diabetes.</p>Fórmula:C20H30Cl2FN3O3Forma y color:SolidPeso molecular:450.38SB 243213 hydrochloride
CAS:<p>SB 243213 hydrochloride is an orally active, selective and high-affinity antagonist of 5-hydroxytryptamine (5-HT)2C receptor(pKi of 9.37 and a pKb of 9.8).It</p>Fórmula:C22H20ClF3N4O2Pureza:98%Forma y color:SolidPeso molecular:464.87PF-00446687
CAS:<p>PF-00446687 is a selective agonist of melanocortin-4 receptor (MC4R) (EC50 of 12 ± 1 nM).</p>Fórmula:C28H36F2N2O2Pureza:98%Forma y color:SolidPeso molecular:470.59RdRP-IN-4
<p>RdRP-IN-4, an oral arylbenzohydrazide, inhibits influenza A/B by targeting PB1 of RdRP, with EC50s of 53 nM (H1N1) and 20 nM (Flu B), and aids infected mice.</p>Fórmula:C17H17Br2N3O2Forma y color:SolidPeso molecular:455.14Ivaltinostat formic
<p>Ivaltinostat (CG-200745) is an oral panHDAC inhibitor, inducing apoptosis and enhancing cancer drug sensitivity.</p>Fórmula:C25H35N3O6Forma y color:SolidPeso molecular:473.56Azaphilone-9
CAS:<p>AZA-9 inhibits cancer growth by blocking HuR-ARE RNA binding; IC50=1.2μM.</p>Fórmula:C21H23BrO5Forma y color:SolidPeso molecular:435.31NCI-006
CAS:<p>NCI-006, an LDH inhibitor, slows tumor growth and enhances pyruvate's role in mitochondrial metabolism.</p>Fórmula:C31H24F2N4O4S3Forma y color:SolidPeso molecular:650.74Uprosertib hydrochloride
CAS:<p>Uprosertib hydrochloride is a potent and selective inhibitor of pan-Akt (IC50: 180/328/38 nM for Akt1/Akt2/Akt3, respectively).</p>Fórmula:C18H17Cl3F2N4O2Pureza:98%Forma y color:SolidPeso molecular:465.71Galidesivir
CAS:<p>Galidesivir (BCX4430) is an antiviral compound that inhibits viral RNA-dependent RNA polymerase (RdRp) activity and reduces lung infections in infected animals.</p>Fórmula:C11H15N5O3Pureza:96.73% - 99.13%Forma y color:SolidPeso molecular:265.27Mal-PEG4-VA-PBD
CAS:<p>Mal-PEG4-VA-PBD is a drug-linker conjugate for Antibody-Drug Conjugates (ADCs), comprising the antitumor antibiotic Pyrrolobenzodiazepine (PBD), connected</p>Fórmula:C68H79N9O17Pureza:98%Forma y color:SolidPeso molecular:1294.41Meclocycline
CAS:<p>Meclocycline: a tetracycline antibiotic, inhibits LDH, reduces cell toxicity from mutant huntingtin, doesn't change protein levels in PC12 cells.</p>Fórmula:C22H21ClN2O8Forma y color:SolidPeso molecular:476.86MV061194
CAS:<p>MV061194 is a potent and selective cathepsin K (Cat K) inhibitor.</p>Fórmula:C28H37N5O4SForma y color:SolidPeso molecular:539.69PqsR-IN-2
<p>PqsR-IN-2, potent PqsR inhibitor, curbs Pseudomonas aeruginosa communication, reduces pyocyanin, with low toxicity.</p>Fórmula:C18H20ClN3OSForma y color:SolidPeso molecular:361.89HIV-1 inhibitor-18
<p>HIV-1 inhibitor-18 blocks HIV-1 capsid, effective on NL4-3 strain (EC50: 5.14 μM), slightly toxic (MT-4CC50>9.51).</p>Fórmula:C27H31N3O6SForma y color:SolidPeso molecular:525.62Antileishmanial agent-4
<p>Antileishmanial agent-4, a ribonucleoside analogue, functions as an antileishmanial agent [1].</p>Fórmula:C17H18N4O4Forma y color:SolidPeso molecular:342.35Stauprimide
CAS:<p>Stauprimide inhibits MYC by blocking NME2, reducing MYC transcription in ESCs.</p>Fórmula:C35H28N4O5Pureza:98%Forma y color:SolidPeso molecular:584.62p38-α MAPK-IN-5
CAS:<p>p38-α MAPK-IN-5: potent p38α inhibitor, IC50s: 0.1 nM (α), 0.2 nM (β), 944 nM (γ), 4100 nM (δ); anti-inflammatory, promising for asthma/COPD research.</p>Fórmula:C37H49N11O2Forma y color:SolidPeso molecular:679.86NF-κB-IN-4
<p>NF-κB-IN-4 (compound 17) is a potent inhibitor of NF-κB pathway which can cross blood brain barrier (BBB).</p>Fórmula:C18H15FN4OForma y color:SolidPeso molecular:322.34Desacetylravidomycin
CAS:<p>Desacetylravidomycin is a new inhibitor of IL-4 signal transduction, produced by Streptomyces sp. WK-6326.</p>Fórmula:C29H31NO8Forma y color:SolidPeso molecular:521.56Bcl-2-IN-7
<p>Bcl-2-IN-7 inhibits Bcl-2, encourages apoptosis in cancer cells, and has anti-tumor activity with various IC50 values.</p>Fórmula:C24H22N4O5S2Forma y color:SolidPeso molecular:510.59Tenellin
CAS:<p>Tenellin is a fungal metabolite that inhibits Mg2+-, Ca2+-, and Na+/K+-ATPase activities in erythrocytes. Tenellin is cytotoxic to Sf9 and Sf21 insect cells.</p>Fórmula:C21H23NO5Forma y color:SolidPeso molecular:369.41Antitumor agent-65
CAS:<p>Antitumor agent-65 (Compound 5) is an analogue/derivative of (-)-cleistenolide. Antitumor agent-65 has potential in cancer research.</p>Fórmula:C18H17NO10Forma y color:SolidPeso molecular:407.33LL-Z 1640-4
CAS:A signal-specific JNK/p38 pathway and TAK 1 inhibitorFórmula:C19H24O7Pureza:98%Forma y color:SolidPeso molecular:364.39HIF-1/2α-IN-1
<p>HIF-1/2α-IN-1, an orally active compound, functions as an inhibitor of HIF-2α.</p>Fórmula:C17H16N6O4Forma y color:SolidPeso molecular:368.35BET-IN-1
<p>BET-IN-1 is a potent inhibitor of BET, exhibiting good brain permeability and a reasonable metabolic stability.</p>Fórmula:C23H24ClFN4O3SForma y color:SolidPeso molecular:490.98GGTI-2154 hydrochloride
CAS:<p>GGTI-2154 hydrochloride: selective GGTase I inhibitor, IC50 21 nM, used in cancer research.</p>Fórmula:C24H29ClN4O3Forma y color:SolidPeso molecular:456.97ATR-IN-7
CAS:<p>ATR-IN-7 is a potent inhibitor of ATR.</p>Fórmula:C21H22FN7OForma y color:SolidPeso molecular:407.44PDE4B-IN-3
<p>PDE4B-IN-3 is a potent inhibitor of PDE4B (IC50: 0.94 μM) and exhibits anti-inflammatory effects.</p>Fórmula:C30H35N3O4S2Forma y color:SolidPeso molecular:565.75Coleon-U-quinone
CAS:<p>Coleon-U-quinone, a P-gp inhibitor, reduces cancer cell viability and enhances Doxorubicin sensitivity in resistant cells.</p>Fórmula:C20H24O5Forma y color:SolidPeso molecular:344.4PF-06795071
CAS:<p>PF-06795071 is an effective and selective covalent inhibitor of MAGL (IC50: 3 nM).</p>Fórmula:C18H17F4N3O3Pureza:98%Forma y color:SolidPeso molecular:399.34844-TFM
<p>844-TFM, a NBTI DNA gyrase blocker, IC50: 1.5 μM, kills Mycobacterium abscessus.</p>Fórmula:C24H25F3N4O2Forma y color:SolidPeso molecular:458.48SHR2415
<p>SHR2415: Potent, selective ERK1/2 inhibitor, oral; ERK1 IC50: 2.8 nM, ERK2 IC50: 5.9 nM; effective in Colo205 (IC50: 44.6 nM), for cancer research.</p>Fórmula:C23H22ClN7O2Forma y color:SolidPeso molecular:463.92AMG-315
CAS:<p>AMG-315: Chiral AEA analogue, potent CB1 agonist (Ki 7.8 nM, EC50 0.6 nM), stable against hydrolyzing/oxidative enzymes.</p>Fórmula:C24H41NO2Forma y color:SolidPeso molecular:375.59EBOV-GP-IN-1
<p>EBOV-GP-IN-1 (Compound 28) is a potent inhibitor of Ebola entry, acting on the Ebola virus envelope glycoprotein (EBOV-GP) (IC50: 0.05 μM).</p>Fórmula:C25H40ClN3O2Forma y color:SolidPeso molecular:450.06Kalafungin
CAS:<p>Kalafungin inhibits various fungi, yeasts, protozoa, and gram-positive bacteria, less so for gram-negative bacteria.</p>Fórmula:C16H12O6Forma y color:SolidPeso molecular:300.26Belotecan
CAS:<p>Belotecan (CKD-602) inhibits DNA topoisomerase I, blocks cell cycle, induces apoptosis, and is a camptothecin-derived anticancer agent.</p>Fórmula:C25H27N3O4Forma y color:SolidPeso molecular:433.5A2A receptor antagonist 2
<p>A2A receptor antagonist 2 is a highly selective and potent antagonist of the adenosine A2Areceptor (IC50: 8.3 nM).</p>Fórmula:C25H28FN7O3Forma y color:SolidPeso molecular:493.53
