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Inhibidores

Inhibidores

Los inhibidores son moléculas que se unen a enzimas, receptores u otras proteínas para reducir o bloquear su actividad biológica. Estos compuestos se utilizan ampliamente en la investigación para estudiar vías biológicas, comprender los mecanismos de las enfermedades y desarrollar fármacos terapéuticos. Los inhibidores desempeñan un papel crucial en el tratamiento de diversas enfermedades, incluyendo el cáncer, las enfermedades cardiovasculares y las infecciones. En CymitQuimica, ofrecemos una amplia gama de inhibidores de alta calidad para apoyar su investigación en bioquímica, biología celular y desarrollo farmacéutico.

Subcategorías de "Inhibidores"

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Se han encontrado 66641 productos de "Inhibidores"

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  • Venetoclax N-oxide

    CAS:
    <p>Venetoclax N-oxide is a byproduct of potent, oral Bcl-2 inhibitor Venetoclax (ABT-199/GDC-0199) with Ki &lt;0.01 nM.</p>
    Fórmula:C45H50ClN7O8S
    Forma y color:Solid
    Peso molecular:884.44
  • Z16078526

    CAS:
    <p>Z16078526 promotes Ucp1, p38 MAPK, lipolysis, thermogenic genes, and mitochondrial activity in mouse brown adipocytes.</p>
    Fórmula:C18H17N3O4S
    Pureza:98.93%
    Forma y color:Solid
    Peso molecular:371.41
  • spisulosine

    CAS:
    <p>spisulosine is a natural product for research related to life sciences. The catalog number is T9664 and the CAS number is 196497-48-0.</p>
    Fórmula:C18H39NO
    Forma y color:Solid
    Peso molecular:285.516
  • Antitumor agent-103


    <p>Antitumor Agent-103 (compound 24l) induces apoptosis and possesses antiproliferative and anti-colony formation properties.</p>
    Fórmula:C36H36N8O9S2
    Pureza:98%
    Forma y color:Solid
    Peso molecular:788.85
  • 3-Hydroxy-12-oleanene-23,28-dioic acid

    CAS:
    <p>3-Hydroxy-12-oleanene-23,28-dioic acid is a natural product for research related to life sciences.</p>
    Fórmula:C30H46O5
    Pureza:98%
    Forma y color:Solid
    Peso molecular:486.68
  • IC 86621

    CAS:
    <p>IC 86621: DNA-PK ATP-competitive inhibitor, IC50 120 nM, enhances DSB antitumor effects, EC50 68 µM for repair.</p>
    Fórmula:C12H15NO3
    Pureza:99.68%
    Forma y color:Solid
    Peso molecular:221.25
  • 6-Hydroxykaempferol 3-Rutinoside -6-glucoside

    CAS:
    <p>6-Hydroxykaempferol 3-Rutinoside -6-glucoside is a natural product of Chrysactinia, Asteraceae.</p>
    Fórmula:C33H40O21
    Pureza:98%
    Forma y color:Solid
    Peso molecular:772.66
  • Isosativanone

    CAS:
    <p>Isosativanone is a natural product for research related to life sciences. The catalog number is TN5543 and the CAS number is 82829-55-8.</p>
    Fórmula:C17H16O5
    Pureza:98%
    Forma y color:Solid
    Peso molecular:300.31
  • Kushenol C

    CAS:
    <p>Kushenol C: Antioxidant, SGLT2 inhibitor, fights S. aureus &amp; S. mutans, may prevent/treat Alzheimer's by inhibiting BACE1 (IC50 5.45μM).</p>
    Fórmula:C25H26O7
    Pureza:98%
    Forma y color:Solid
    Peso molecular:438.47
  • Hellebrin

    CAS:
    <p>Cytotoxic and antiproliferative effects of Hellebrin on breast and lung cancer cells.</p>
    Fórmula:C36H52O15
    Forma y color:Solid
    Peso molecular:724.79
  • Kijimicin

    CAS:
    <p>Kijimicin is a polyether antibiotic and human immunodeficiency virus inhibitor in acutely and chronically infected cells.</p>
    Fórmula:C37H64O11
    Pureza:98%
    Forma y color:Solid
    Peso molecular:684.90
  • MVL5

    CAS:
    <p>MVL5, a non-degradable multivalent cationic lipid, serves as a highly efficient vector for both DNA and siRNA [1].</p>
    Fórmula:C59H116Cl5N7O4
    Forma y color:Solid
    Peso molecular:1164.86
  • Upidosin

    CAS:
    <p>Upidosin (SB-216469), a uroselective α1 blocker: Ki α1a=0.34 nM, α1b=3.9 nM, α1d=1.5 nM, α2=33.3 nM.</p>
    Fórmula:C31H33N3O4
    Pureza:99.66%
    Forma y color:Solid
    Peso molecular:511.61
  • HO-PEG24-CH2COOH


    <p>HO-PEG24-CH2COOH is a PEG-based linker for PROTACs which joins two essential ligands, crucial for forming PROTAC molecules.</p>
    Fórmula:C50H100O27
    Pureza:98%
    Forma y color:Solid
    Peso molecular:1133.31
  • PC Biotin-PEG3-NHS ester

    CAS:
    <p>PC Biotin-PEG3-NHS ester: A cleavable 3-PEG unit ADC linker for antibody-drug conjugate synthesis.</p>
    Fórmula:C36H52N6O15S
    Pureza:98%
    Forma y color:Solid
    Peso molecular:840.89
  • Destruxin B2

    CAS:
    <p>Destruxin B2, found in M. anisopliae, has antiviral, insecticidal properties, inhibits HBsAg (IC50=1.3 μM), and is toxic to Sf9 cells (ECIS50=92 μM).</p>
    Fórmula:C29H49N5O7
    Forma y color:Solid
    Peso molecular:579.739
  • β-Peltoboykinolic acid

    CAS:
    <p>Beta-Peltoboykinolic acid inhibits PTP1B (IC50: 5.2±0.5 µM) and shows cytotoxicity.</p>
    Fórmula:C30H48O3
    Pureza:98%
    Forma y color:Solid
    Peso molecular:456.7
  • Isofistularin-3


    <p>Isofistularin-3: DNA demethylating, induces cancer cell cycle arrest, TRAIL sensitization, ADC cytotoxin, DNMT1 inhibitor, IC50 13.5 μM.</p>
    Fórmula:C31H30Br6N4O11
    Pureza:98%
    Forma y color:Solid
    Peso molecular:1114.01
  • Salvicine


    <p>Salvicine is a useful organic compound for research related to life sciences and the catalog number is T125239.</p>
    Fórmula:C20H26O4
    Forma y color:Solid
    Peso molecular:330.424
  • m-Acetotoluide

    CAS:
    <p>m-Acetotoluide is a bioactive chemical.</p>
    Fórmula:C9H11NO
    Pureza:98%
    Forma y color:Physical Description White Solid (Ntp 1992)
    Peso molecular:149.19