Inhibidores
Los inhibidores son moléculas que se unen a enzimas, receptores u otras proteínas para reducir o bloquear su actividad biológica. Estos compuestos se utilizan ampliamente en la investigación para estudiar vías biológicas, comprender los mecanismos de las enfermedades y desarrollar fármacos terapéuticos. Los inhibidores desempeñan un papel crucial en el tratamiento de diversas enfermedades, incluyendo el cáncer, las enfermedades cardiovasculares y las infecciones. En CymitQuimica, ofrecemos una amplia gama de inhibidores de alta calidad para apoyar su investigación en bioquímica, biología celular y desarrollo farmacéutico.
Subcategorías de "Inhibidores"
- Angiogénesis(2.687 productos)
- Apoptosis(6.097 productos)
- Ciclo celular / Checkpoint(4.691 productos)
- Cromatina / Epigenética(2.376 productos)
- Señalización citoesquelética(1.472 productos)
- Daño al ADN / Reparación del ADN(2.921 productos)
- Endocrinología / Hormonas(3.611 productos)
- Enzima(3.655 productos)
- GPCR / proteína G(8.755 productos)
- Inmunología e inflamación(3.765 productos)
- Virus de la gripe(298 productos)
- Señalización JAK / STAT(407 productos)
- Señalización MAPK(1.230 productos)
- Transportador de membrana / canal de iones(2.947 productos)
- Metabolismo(9.940 productos)
- Microbiología / Virología(7.347 productos)
- Neurociencia(10.240 productos)
- Otros inhibidores(36.533 productos)
- Reducción de oxidación(43 productos)
- Señalización PI3K / Akt / mTOR(1.437 productos)
- Proteasas / Proteasoma(1.675 productos)
- Células madre y Derivados(830 productos)
- Tirosina quinasa / adaptadores(2.028 productos)
- Ubiquitinación(1.682 productos)
Mostrar 16 subcategorías más
Se han encontrado 66582 productos de "Inhibidores"
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PPO-IN-1
PPO-IN-1 is a potent inhibitor of protoporphyrinogen IX oxidase (PPO) (Ki: 2.5 nM).Fórmula:C18H10F3N3O4SForma y color:SolidPeso molecular:421.359-cis-β-Carotene
CAS:9-cis-β-Carotene, a precursor of retinal, is cleaved by beta-carotene oxygenase 1 (BCMO1) to produce 9-cis-retinal.Fórmula:C40H56Pureza:98%Forma y color:SolidPeso molecular:536.87Antifungal agent 40
<p>Antifungal agent 40 blocks C. albicans CYP51 in pocket II, hindering lanosterol demethylase and biofilm growth.</p>Fórmula:C22H20Cl2N4SeForma y color:SolidPeso molecular:490.29SP-471
SP-471 is a potent inhibitor of dengue virus (DENV) protease (IC50: 18 μM) and inhibits the inter- and intramolecular protease processes of DENV.Fórmula:C33H26BrN5Forma y color:SolidPeso molecular:572.5PEN-866
CAS:PEN-866, a conjugate of HSP90i and SN-38, may control early NSCLC tumor growth.Fórmula:C49H49N7O9Forma y color:SolidPeso molecular:879.95SLN124
<p>SLN124, a GalNAc-siRNA targeting TMPRSS6, may normalize iron balance by restoring ferroregulation.</p>Forma y color:SolidFXIa-IN-6
CAS:<p>FXIa-IN-6: Potent, selective FXIa inhibitor (Ki=0.3 nM); strong PK with high oral bioavailability, low clearance preclinically.</p>Fórmula:C31H29ClF2N4O4Forma y color:SolidPeso molecular:595.04Glutaminyl cyclases-IN-1
<p>Glutaminyl cyclase inhibitor IsoQC-IN-1: IC50=12 nM for QC, 73 nM for isoQC; blocks CD47/SIRPα; boosts THP-1, U937 macrophage phagocytosis.</p>Fórmula:C25H30N6O2SForma y color:SolidPeso molecular:478.61LpxC-IN-10
CAS:LpxC-IN-10 is a selective LpxC inhibitor with an MIC of 0.5 μg/mL against E. coli and K. pneumoniae and is capable of being used to study bacterial infections.Fórmula:C30H31N5O3Forma y color:SolidPeso molecular:509.6Annonin VI
CAS:Annonin VI is a natural inhibitor of NADH:ubiquinone oxidoreductase.Fórmula:C37H66O7Forma y color:SolidPeso molecular:622.92M826
<p>M826, a non-peptide, potent, selective, and reversible caspase-3 inhibitor, exhibits an IC50 of 0.005 μM and demonstrates strong anti-apoptotic activity in</p>Fórmula:C28H45N7O6Pureza:98%Forma y color:SolidPeso molecular:575.7VEGFR-2-IN-11
<p>VEGFR-2-IN-11 is a potent inhibitor of VEGFR-2 (IC50: 60.27 nM) with an IC50 value of 60.27 nM, which induces apoptosis and has anticancer activity.</p>Fórmula:C29H22BrN5SForma y color:SolidPeso molecular:552.49Glucosylceramide synthase-IN-3
Glucosylceramide synthase-IN-3 (BZ1) is a potent, brain-accessible, oral GCS inhibitor with a 16 nM IC50, relevant for Gaucher's disease study.Fórmula:C21H20FN3O3Forma y color:SolidPeso molecular:381.4JBJ-02-112-05
CAS:JBJ-02-112-05 is a potent, mutant-selective, allosteric and orally active inhibitor of EGFR with an IC 50 of 15 nM for EGFR L858R/T790M [1].Fórmula:C27H20N4O2SPureza:98%Forma y color:SolidPeso molecular:464.54FNDR-20123
FNDR-20123: First safe, effective anti-malarial HDAC inhibitor for Plasmodium (IC50: 31 nM) & human HDACs, with nanomolar potency across several subtypes.Fórmula:C21H24ClN5O2Forma y color:SolidPeso molecular:413.9NNC-11-1585
CAS:NNC-11-1585 is an M(1) and M(2) muscarinic acetylcholine receptor (mAChR) agonist.Fórmula:C18H19N3OSForma y color:SolidPeso molecular:325.43Aurora B inhibitor 1
CAS:<p>Aurora B inhibitor 1 is an Aurora B (Aurora-1) inhibitor (Ki <0.010 uM) with potential anticancer activity for cancer research.</p>Fórmula:C25H26ClF2N7O2Pureza:98.37%Forma y color:SolidPeso molecular:529.97AGN-204396
CAS:AGN-204396 is an antagonist that selectively blocks the activity of prostamides (prostaglandin-ethanolamides).Fórmula:C32H44FN3O4Forma y color:SolidPeso molecular:553.71Tonapofylline
CAS:Tonapofylline, orally active, selectively blocks A1 adenosine receptor (Ki: 7.4 nM), used in heart failure research.Fórmula:C22H32N4O4Pureza:98.57%Forma y color:SolidPeso molecular:416.51Amrubicin HCl
CAS:Amrubicin (SM-5887), an anthracycline, treats lung cancer by inhibiting DNA replication and topoisomerase II, with less cardiac toxicity.Fórmula:C25H25NO9Forma y color:SolidPeso molecular:483.47PF-07054894
CAS:PF-07054894: potent CCR6 antagonist, targets GPCR, for inflammatory bowel disease research.Fórmula:C24H30N6O4Forma y color:SolidPeso molecular:466.53KAG-308
CAS:KAG-308: selective EP4 agonist; Ki: 2.57 nM, EC50: 17 nM; suppresses colitis, promotes mucosal healing, inhibits TNF-α.Fórmula:C24H30F2N4O3Pureza:98%Forma y color:SolidPeso molecular:460.52KRAS G12C inhibitor 37
CAS:KRAS G12C inhibitor 37 targets a key signaling protein, showing promise for cancer research involving KRAS G12C.Fórmula:C35H39F3N8O2Forma y color:SolidPeso molecular:660.73HDAC/HSP90-IN-4
HDAC/HSP90-IN-4 inhibits HDAC (20 IC50=194nM, 26 IC50=360nM) & HSP90α (20 IC50=153nM, 26 IC50=77nM), affects cancer cell survival and invasion.Fórmula:C20H23N3O6Forma y color:SolidPeso molecular:401.15869Cdc7-IN-11
CAS:Cdc7-IN-11 is a potent inhibitor of Cdc7 (IC50 ≤ 1 nM) and can be used in the study of proliferative diseases.Fórmula:C20H22F2N4O2SForma y color:SolidPeso molecular:420.48Teslexivir hydrochloride
CAS:Teslexivir (BTA074) HCl inhibits HPV 6/11 by blocking E1-E2 protein interaction, vital for DNA replication. Used in condyloma research.Fórmula:C35H37BrClN3O4Forma y color:SolidPeso molecular:679.04Antioxidant agent-3
Antioxidant agent-3 shows strong DPPH and ABTS+ radical scavenging (IC50: 26.58, 30.31 μM). Boosts ROS, SOD, GSH; lowers LDH in H2O2-exposed HepG2 cells.Fórmula:C18H14O8Forma y color:SolidPeso molecular:358.3WM382
CAS:<p>WM382, a potent dual PMIX/X inhibitor, has IC50s of 1.4 nM/0.03 nM and effective against various malaria stages.</p>Fórmula:C29H36N4O4Forma y color:SolidPeso molecular:504.62Gemilukast
CAS:<p>Gemilukast (ONO-6950) is a cysteinyl leukotriene 1 and 2 receptor inhibitor that inhibits bronchoconstriction and is used in the treatment of asthma.</p>Fórmula:C36H37F2NO5Pureza:98.27% - 99.5%Forma y color:SolidPeso molecular:601.68FXIa-IN-9
CAS:FXIa-IN-9, a potent FXIa inhibitor (K i : human 0.17 nM, rabbit 0.5 nM), forms hydrogen bonds and has anticoagulant properties.Fórmula:C23H18Cl2F3N9O2Forma y color:SolidPeso molecular:580.35Oxythiamine diphosphate ammonium
<p>Oxythiamin diphosphate ammonium is a potent inhibitor of transketolase (TK).</p>Forma y color:Solidγ-secretase modulator 5
Compound 22d is a GSM that crosses the blood-brain barrier, inhibits Aβ42 production (IC50: 60 nM), and may help study Alzheimer's.Forma y color:SolidBACE1-IN-8
<p>BACE1-IN-8 is a potent inhibitor of BACE1 (β-site APP lyase 1) (IC50: 3.9 μM).</p>Fórmula:C29H45N5O7Forma y color:SolidPeso molecular:575.7RF9 hydrochloride
<p>RF9 hydrochloride is a potent and selective Neuropeptide FF receptor antagonist that acts on hNPFF1R (Ki: 58 nM) and hNPFF2R (Ki: 7 nM).</p>Fórmula:C26H39ClN6O3Forma y color:SolidPeso molecular:519.08Vibegron
CAS:Vibegron (MK-4618) is an effective and selective Beta 3 adrenergic receptor agonist, used to treat overactive bladder (OAB).Fórmula:C26H28N4O3Forma y color:SolidPeso molecular:444.53GSK699
CAS:<p>GSK699 is a potent, cell penetrant PCAF/GCN5 PROTAC.</p>Fórmula:C45H51BrN8O7Forma y color:SolidPeso molecular:895.84VHL Ligand 8
CAS:VHL Ligand 8, a VHL ligand essential for synthesizing ARD-266, acts as a highly potent VHL E3 ligase-based androgen receptor (AR) PROTAC degrader.Fórmula:C23H29N3O6Pureza:98%Forma y color:SolidPeso molecular:443.49L 767679
CAS:L 767679 is an antagonist of the fibrinogen receptors.Fórmula:C20H24N4O4Pureza:98%Forma y color:SolidPeso molecular:384.43NAZ2329
CAS:NAZ2329: Cell-permeable, targets R5 RPTPs, inhibits hPTPRZ1 (IC50=7.5 μM) & hPTPRG (IC50=4.8 μM), hampers glioblastoma growth, affects stem cell traits.Fórmula:C21H18F3NO4S3Forma y color:SoildPeso molecular:501.56RET-IN-1
CAS:RET-IN-1 is a RET kinase inhibitor (IC50s: 1 nM, 7 nM, and 101 nM for RET (WT), RET (V804M) , and RET (G810R), respectively).Fórmula:C29H31N9O3Pureza:98%Forma y color:SolidPeso molecular:553.61FGFR1 inhibitor-6
FGFR1 inhibitor-6, IC50: 16.31 nM, blocks cell cycle at pro-G1/G2/M and induces apoptosis.Fórmula:C27H19N5O4S2Forma y color:SolidPeso molecular:541.6PptT-IN-3
PptT-IN-3 (5p), an inhibitor of PptT in Mycobacterium tuberculosis, IC50=3.5μM, is key for TB research.Fórmula:C16H27N5O3SForma y color:SolidPeso molecular:369.48HPK1-IN-16
CAS:HPK1-IN-16, a potent HPK1 inhibitor, useful for cancer research and treatment.Fórmula:C28H27FN4OForma y color:SolidPeso molecular:454.54RBM10-8
CAS:RBM10-8 irreversibly inhibits human sphingosine-1- phosphate lyase (hS1PL) while behaving also as an enzyme substrate.Fórmula:C17H36NO5PForma y color:SolidPeso molecular:365.45Dexnebivolol
CAS:Dexnebivolol (R67138), a ß-adrenergic antagonist, is Nebivolol's enantiomer with β1 blocking and vasodilation properties.Fórmula:C22H25F2NO4Forma y color:SolidPeso molecular:405.43AP5
CAS:<p>AP5: GPR40 agonist, positive allosteric modulator; rat hIP1 EC50: 0.49 nM.</p>Fórmula:C28H28FNO4Pureza:98%Forma y color:SolidPeso molecular:461.52A25822B
CAS:A25822B is an antifungal agent.Fórmula:C28H45NOPureza:98%Forma y color:SolidPeso molecular:411.66PF1070A
CAS:PF1070A is a natural cyclic tetrapeptide HDAC Inhibitor through the inhibition of PfHDAC1 catalytic activity, potently inducing the synthesis of metallothioneinFórmula:C31H44N4O6Forma y color:SolidPeso molecular:568.7Pralatrexate, (R)-
CAS:Pralatrexate is a high-affinity DHFR inhibitor targeting RFC-1, used in cancer treatment and immunosuppression.Fórmula:C23H23N7O5Pureza:98%Forma y color:SolidPeso molecular:477.47LolCDE-IN-2
CAS:<p>LolCDE-IN-2 is a potent Lol protein (LolCDE) inhibitor. LolCDE-IN-2 shows antibacterial activity with a MIC of 2 μg/ml against E. coli MG1655 [1].</p>Fórmula:C22H17N5OPureza:98%Forma y color:SolidPeso molecular:367.40Fostriecin (free base)
CAS:Fostriecin inhibits PP2A/PP4 (IC50s = 3.2/3 nM), weakly affects topoisomerase II/PP1 (IC50s = 40/131 μM), doesn't inhibit PP2B, and may modify epigenetics.Fórmula:C19H27O9PForma y color:SolidPeso molecular:430.39SM-433 hydrochloride
SM-433 hydrochloride, a Smac mimetic & IAP inhibitor, binds XIAP BIR3; potent IC50 <1 μM. (Patent WO2008128171A2)Fórmula:C32H44ClN5O4Forma y color:SolidPeso molecular:598.18(Z)-Lanoconazole
<p>(Z)-Lanoconazole, an imidazole antifungal for dermatophytosis and onychomycosis, inhibits fungal ergosterol production.</p>Fórmula:C14H10ClN3S2Forma y color:SolidPeso molecular:319.83Hypothemycin
CAS:Hypothemycin, a fungal polyketide, inhibits multiple kinases (VEGFR, MEK, FLT-3, PDGFR, ERK) with Kis ranging from 10 nM to 2.4 μM.Fórmula:C19H22O8Pureza:98%Forma y color:SolidPeso molecular:378.37Dyrk1A/α-synuclein-IN-2
<p>Dyrk1A/α-synuclein-IN-2 (Compound b20) is a dual inhibitor of Dyrk1A and α-synuclein aggregation that acts on α-synuclein (IC50: 7.8 μM).</p>Fórmula:C21H16N4O4SForma y color:SolidPeso molecular:420.44ODN 21158
CAS:<p>ODN 21158 is a potent, non-cytotoxic inhibitor of G-modified TLR3 and TLR9. ODN 21158 dose-dependently inhibits IFN-α secretion.</p>Forma y color:SolidZLWT-37
ZLWT-37: Oral CDK inhibitor, CDK9 IC50=0.002 µM, CDK2 IC50=0.054 µM; halts HCT116 cells at G2/M, induces apoptosis.Fórmula:C26H30ClN5OForma y color:SolidPeso molecular:464FMK-MEA
CAS:FMK-MEA is a potent and selective p90 Ribosomal S6 Kinase (RSK) inhibitor.Fórmula:C21H26FN5O2Pureza:98%Forma y color:SolidPeso molecular:399.46AKT-IN-11
AKT-IN-11 is one of the most potent antibacterial agents against human hepatocellular carcinoma Bel-7402 cell line (IC50: 1.15 μM).Fórmula:C27H27ClF3NO4Forma y color:SolidPeso molecular:521.96Imolamine hydrochloride
CAS:Imolamine hydrochloride is a blood platelet aggregation antagonist.Fórmula:C14H21ClN4OForma y color:SolidPeso molecular:296.80MALT1-IN-5
CAS:MALT1-IN-5 is a potent inhibitor of the MALT1 protease and can be used in cancer research.Fórmula:C17H17ClF2N6O3Forma y color:SolidPeso molecular:426.80LT-850-166
LT-850-166 is a potent inhibitor of FLT3 and has shown efficacy in overcoming a wide range of FLT3 mutations.Fórmula:C30H29Cl2N7OForma y color:SolidPeso molecular:574.5ONL-1204
CAS:ONL-1204 is a small molecule, CD95 antigen inhibitor (Fas inhibitor) being developed by ONL Therapeutics for the treatment of retinal detachment.Fórmula:C71H100N18O16Forma y color:SolidPeso molecular:1461.66BMS-748730
CAS:BMS-748730, also known as 4′-Hydroxy Dasatinib, is a Dasatinib metabolite.Fórmula:C22H26ClN7O3SForma y color:SolidPeso molecular:504.01Tubulin inhibitor 14
Tubulin inhibitor 14 blocks NQO2 and microtubule formation, disrupts blood vessels, and may target tumors; IC50 of 1.0 μM.Fórmula:C15H9F2NOForma y color:SolidPeso molecular:257.23Detajmium
CAS:Detajmium is an anti-arrhythmia compound. It is an Na(+)-channel-blocking drug with an extremely long recovery from use-dependent sodium channel block.Fórmula:C27H42N3O3Pureza:98%Forma y color:SolidPeso molecular:456.64GENZ-882706
CAS:<p>GENZ-882706 is a potent colony stimulating factor-1 receptor (CSF-1R) Inhibitor.</p>Fórmula:C26H25N5O3Pureza:98%Forma y color:SolidPeso molecular:455.51ROS1-IN-1
<p>ROS1-IN-1, a potent ROS1 kinase inhibitor, has an IC50 of 0.097 μM.</p>Fórmula:C17H15ClN6SForma y color:SolidPeso molecular:370.86GPBAR1-IN-3
CAS:GPBAR1-IN-3 (Compound 14) is both a selective agonist for GPBAR1, with an EC50 value of 0.17 μM, and an antagonist for CysLT1R [1].Fórmula:C21H23NO2Forma y color:SolidPeso molecular:321.41TRPC5-IN-4
CAS:<p>TRPC5-IN-4: Potent, safe inhibitor; IC50 14.07 nM (TRPC5), 65 nM (TRPC4); non-toxic to liver/kidney cells; for CKD research.</p>Fórmula:C18H11ClF4N4O3Forma y color:SolidPeso molecular:442.75Iloprost
CAS:Iloprost (Ciloprost) is an inhibitor of platelet aggregation and vasodilatation used in the study of cardiovascular disease.Fórmula:C22H32O4Forma y color:Colorless OilPeso molecular:360.49LAS195319
CAS:LAS195319 is a potent and selective inhaled PI3Kδ Inhibitor (IC50 = 0.5 nM) for the Treatment of Respiratory Diseases.Fórmula:C29H26N10O3SForma y color:SolidPeso molecular:594.65EP-7041 HCl
CAS:EP-7041 is a novel, potent, and selective Factor XIa inhibitor.Fórmula:C19H27ClN4O4Forma y color:SolidPeso molecular:410.89Elongation factor P-IN-1
EFP-IN-1: potent β-lysine derivative, inhibits EFP, slows E. coli growth.Fórmula:C14H31N3O2Forma y color:SolidPeso molecular:273.41Hypoglycemic agent 1
CAS:Hypoglycemic agent 1 has an action for lowering blood sugar. It acts as a therapeutic and/or prophylactic agent for diabetes.Fórmula:C25H24FN5O4Pureza:98%Forma y color:SolidPeso molecular:477.49Aurora/LIM kinase-IN-1
Aurora/LIM kinase-IN-1 (Compound F114) is a dual inhibitor targeting aurora and lim kinases, potentially useful in GBM cancer treatment efforts.Fórmula:C16H20N6OForma y color:SolidPeso molecular:312.37Topoisomerase I/II inhibitor 2
<p>Compound 1a inhibits Topoisomerase I/II, shrinks mouse liver tumors, IC50: 6.83/9.82 μM for LM9/Huh7 cells.</p>Fórmula:C19H16N2O4Forma y color:SolidPeso molecular:336.34SCH 563705
CAS:SCH 563705 is a CXCR2 and CXCR1 antagonist used in the study of acute respiratory syndrome, chronic obstructive pulmonary disease, and inflammation.Fórmula:C23H27N3O5Pureza:98.03%Forma y color:SolidPeso molecular:425.48Carbodine
CAS:Carbodine is an antiviral targeting CTP synthetase, effective against influenza A0/PR-8/34 and A2/Aichi/2/68.Fórmula:C10H15N3O4Pureza:98%Forma y color:SolidPeso molecular:241.24MSA-2 dimer
CAS:MSA-2 dimer: selective oral non-nucleotide STING agonist, Kd=145 μM, long-term antitumor effect, non-covalent, higher permeability.Fórmula:C29H28O8S2Forma y color:SolidPeso molecular:568.66PAT-347
CAS:PAT-347 is a potent inhibitor of Autotaxin, an enzyme linked to cell survival and diseases like cancer and fibrosis.Fórmula:C28H21ClF2N2O3SForma y color:SolidPeso molecular:538.99CAII-IN-1
CAII-IN-1 (3n) is a selective bovine CA-II inhibitor with 10.3 μM IC50, used in carbonic anhydrase disorder studies.Fórmula:C19H21FN4SForma y color:SolidPeso molecular:356.46WW437
WW437 is a histone deacetylase (HDAC) inhibitor that exhibits potent anti-breast cancer activity both in vitro and in vivo.Fórmula:C23H27N5O4Forma y color:SolidPeso molecular:437.49Carbonic anhydrase inhibitor 3
Carbonic anhydrase inhibitor 3 (compound 11g) is an inhibitor of carbonic anhydrase II that reduces the intraocular pressure in glaucomatous rabbits [1].Fórmula:C15H17N3O3SForma y color:SolidPeso molecular:319.38CL656
CAS:<p>CL656 is a stimulator of interferon genes (STING) activator.</p>Fórmula:C20H21F2N9O9P2S2Pureza:98%Forma y color:SolidPeso molecular:695.51cis-RdRP-IN-5
Cis-RdRP-IN-5 is an effective inhibitor of the influenza virus RNA-dependent RNA polymerase (RdRP), employed in influenza virus research.Fórmula:C23H21N3O5Forma y color:SolidPeso molecular:419.43RS 61756-007
CAS:RS 61756-007 is a selective thromboxane receptor (TP) agonist.Fórmula:C23H28O5Pureza:98%Forma y color:SolidPeso molecular:384.47Carbonic anhydrase inhibitor 4
<p>CA inhibitor 4, photoprobe; targets hCA I-XIV; Ki: 640-1166 nM.</p>Fórmula:C21H18N2O4SForma y color:SolidPeso molecular:394.44MB-07344 sodium
"MB-07344 sodium is a TR-β agonist with a 2.17 nM Ki, boosts Atorvastatin's cholesterol-lowering effects in various animals."Fórmula:C19H25NaO5PPureza:98%Forma y color:SolidPeso molecular:387.36NLRP3-IN-8
CAS:NLRP3-IN-8, orally active inflammasome blocker, IC50 of 1.23μM, stable (t1/2 = 138.63min), non-toxic (IC50 >100μM).Fórmula:C23H20N2O6Forma y color:SolidPeso molecular:420.41Epothilone E
CAS:<p>Epothilone E, a derivative of epothilone, functions by inhibiting microtubule protein activity, thereby halting cell division and exhibiting anti-tumor</p>Fórmula:C26H39NO7SForma y color:SolidPeso molecular:509.66KP 10614
CAS:KP 10614 is a new prostacyclin analog that inhibits platelet-polymorphonuclear leukocyte interaction.Fórmula:C23H32O4Forma y color:SolidPeso molecular:372.50LSD1-IN-19
LSD1-IN-19 is a potent, selective LSD1 inhibitor with Ki of 0.108 μM and 72h IC50 values of 0.17-0.40 μM.Fórmula:C33H42N6O2Forma y color:SolidPeso molecular:554.73GNE-203
CAS:<p>GNE-203 is a Met inhibitor.</p>Fórmula:C30H29Cl2F3N8O3Forma y color:SolidPeso molecular:677.50TPI-287
CAS:TPI 287: synthetic taxane; may halt cancer by stabilizing microtubules, blocking cell division, inducing apoptosis.Fórmula:C46H63NO15Forma y color:SolidPeso molecular:869.99ATP synthase inhibitor 2
CAS:<p>ATP synthase inhibitor 2 blocks P. aeruginosa ATP synthase; IC50=10 μg/mL, fully inhibits at 128 μg/mL.</p>Fórmula:C21H22N2O3SForma y color:SolidPeso molecular:382.48Calcipotriol Impurity C
CAS:<p>Calcipotriol Impurity C is the impurity of Calcipotriol. Calcipotriol is a VDR-like receptors ligand.</p>Fórmula:C27H40O3Pureza:98%Forma y color:SolidPeso molecular:412.614ACHN-975 TFA
CAS:<p>ACHN-975 TFA is a selective LpxC inhibitor with a subnanomolar inhibitory. It is against a wide range of gram-negative bacterias with low MIC values (≤1 μg/mL).</p>Fórmula:C22H24F3N3O6Pureza:98%Forma y color:SolidPeso molecular:483.4377(RS)-AMPA monohydrate
CAS:(RS)-AMPA monohydrate, potent glutamate analogue, selectively activates L-glutamic acid without affecting kainic acid or NMDA receptors.Fórmula:C7H12N2O5Forma y color:SolidPeso molecular:204.182BCL6-IN-9
CAS:<p>BCL6-IN-9 (compound 1) is a potent inhibitor of B-cell lymphoma 6 protein (BCL6) (IC50: 3.9 nM) and can be used to study cancer.</p>Fórmula:C22H18ClF2N5O2Forma y color:SolidPeso molecular:457.86SR 33805 oxalate
CAS:Ca2+ channel antagonistFórmula:C34H42N2O9SPureza:98%Forma y color:SolidPeso molecular:654.77Cathepsin C-IN-5
CAS:<p>Cathepsin C-IN-5 (SF38) is a potent, oral Cathepsin C blocker with an IC50 of 59.9 nM; less active against Cat L/S/B/K; has anti-inflammatory effects.</p>Fórmula:C21H17ClN6OSForma y color:SolidPeso molecular:436.92GSK 366
CAS:GSK 366 is a potent kynurenine-3-monooxygenase (KMO) inhibitor (IC50s: 0.7 nM and 2.3 nM for P. fluorescens-KMO and human KMO).Fórmula:C17H16ClN3O4Pureza:98%Forma y color:SolidPeso molecular:361.78T-Type calcium channel inhibitor 2
Compound 6g inhibits T-type Ca channels (IC50: Cav3.1-31μM, Cav3.2-83μM), cytotoxic to A549 (IC50: 5μM) & HCT-116 cells (IC50: 6.4μM).Fórmula:C36H39FN4OSForma y color:SolidPeso molecular:594.78OICR-9429-N-C2-NH2
CAS:OICR-9429-N-C2-NH2, a ligand for WDR5, intermediate 2, serves as a crucial compound in the synthesis of PROTACs.Fórmula:C31H38F3N7O2Forma y color:SolidPeso molecular:597.687Salacinol
CAS:Salacinol is a naturally occurring alpha-glucosidase inhibitor isolated from an Ayurvedic traditional medicine Salacia reticulata.Fórmula:C9H18O9S2Forma y color:SolidPeso molecular:334.37HBV-IN-11
CAS:HBV-IN-11 is a potent inhibitor of HBsAg secretion (EC50: 0.46 μM).Fórmula:C21H24ClNO6Forma y color:SolidPeso molecular:421.87Hymenidin
CAS:Hymenidin, isolated from the Okinawan sponge Hymeniacidon sp., is a 5-hydroxytryptaminergic receptor antagonist and voltage-gated potassium channel inhibitor.Fórmula:C11H12BrN5OPureza:96.85% - 99.52%Forma y color:SolidPeso molecular:310.15PF-06305591 dihydrate
PF-06305591 dihydrate is a potent and highly selective voltage gated sodium channel NaV1.8 blocker (IC 50 = 15 nM) with an excellent preclinical in vitro ADMEFórmula:C15H26N4O3Forma y color:SolidPeso molecular:310.39J-104118
CAS:J-104118 potentially inhibits squalene synthase.Fórmula:C28H26Cl2FNO5Pureza:98%Forma y color:SolidPeso molecular:546.41USP7-IN-10
CAS:<p>USP7-IN-10 is a potent inhibitor of ubiquitin-specific protease 7 (USP7), exhibiting an inhibition concentration half-maximal (IC50) value of 13.39 nM.</p>Fórmula:C26H29ClN4O3SForma y color:SolidPeso molecular:513.05BM635 mesylate (1493762-74-5 free base)
BM635 mesylate is an MmpL3 inhibitor with outstanding anti-mycobacterial activity (MIC50: 0.12 μM against M. tuberculosis H37Rv).Fórmula:C26H33FN2O4SPureza:98%Forma y color:SolidPeso molecular:488.61NUCC-555
CAS:NUCC-555 is a first-in-class antagonist of activin. It opens a completely new approach to inhibiting the activity of TGF-beta receptor superfamily members.Fórmula:C25H25N5O3Pureza:98%Forma y color:SolidPeso molecular:443.5Antibacterial agent 78
<p>Antibacterial agent 78 (compound 30) is an antibacterial agent with improved cytotoxicity profile[1].</p>Fórmula:C16H23N3S2Forma y color:SolidPeso molecular:321.5(S)-Butaprost free acid
CAS:(S)-Butaprost (free acid) is a potent and highly selective EP2 receptor agonist[1].Fórmula:C23H38O5Forma y color:SolidPeso molecular:394.54Anti-Influenza agent 3
Compound 11h: Potent, low-toxicity anti-influenza, inhibits M2 ion channels. EC50: 3.29μM (H3N2), 2.45μM (H1N1).Fórmula:C16H22ClNOSForma y color:SolidPeso molecular:311.87C5aR-IN-3
CAS:C5aR-IN-3, a potent C5aR inhibitor, may treat autoimmune and inflammatory diseases.Fórmula:C36H40FN5O3Forma y color:SolidPeso molecular:609.73Steroid sulfatase/17β-HSD1-IN-3
Steroid sulfatase/17β-HSD1-IN-3 (compound 19) is a dual inhibitor of steroid sulfatase (STS) and 17β-hydroxysteroid dehydrogenase type 1 (17β HSD1).Fórmula:C19H17ClN2O5SForma y color:SolidPeso molecular:420.87PI3K-IN-37
CAS:PI3K-IN-37 inhibits PI3K α/β/δ (IC50: 6/8/4 nM) and mTOR (IC50: 4 nM).Fórmula:C25H26N6O2Forma y color:SolidPeso molecular:442.51BRD-7880
CAS:BRD-7880 is a potent and highly specific inhibitor of aurora kinases B and C.Fórmula:C32H38N4O7Forma y color:SolidPeso molecular:590.67Cenicriviroc Sulfone
CAS:Cenicriviroc Sulfone, a Cenicriviroc derivative, inhibits CCR2/CCR5 to block HIV entry into cells.Fórmula:C41H52N4O5SForma y color:SolidPeso molecular:712.94IRE1α kinase-IN-5
<p>IRE1α kinase-IN-5 (compound 7) is a potent inhibitor of IRE1α (Ki: 98 nM) and is an ATP-competitive ligand for IRE1α.</p>Fórmula:C28H30N6O3SForma y color:SolidPeso molecular:530.64Anti-ToCV agent 1
Anti-ToCV agent 1 can be used as a potential anti-ToCV drug.Fórmula:C22H19FN2O5SForma y color:SolidPeso molecular:442.46Chitin synthase inhibitor 7
Compound 9c, a chitin synthase inhibitor, has an IC50 of 0.37 nM and is useful for studying fungal infections.Fórmula:C24H25N3O5Forma y color:SolidPeso molecular:435.47Cilazaprilat
CAS:Cilazaprilat is the active metabolite of cilazapril, a pyridazine angiotensin-converting enzyme (ACE) inhibitor with antihypertensive activity.Fórmula:C20H27N3O5Forma y color:SolidPeso molecular:389.45PI3K-IN-35
CAS:<p>PI3K-IN-35 (6l) selectively inhibits PI3K-α, β, δ (IC50: 13.98, 7.22, 10.94 μM), blocks G2/M phase, induces apoptosis, and is useful in leukemia research.</p>Fórmula:C25H23N7O2Forma y color:SolidPeso molecular:453.5sEH inhibitor-1
<p>TCPU (sEH inhibitor-1) is a potent oral human sEH blocker with IC50s of 0.4 nM (human) and 5.3 nM (mouse).</p>Forma y color:SolidCDK9-IN-13
<p>CDK9-IN-13 is a potent and selective CDK inhibitor (IC50<3 nM). CDK9-IN-13 has a very short half-life in rodents.</p>Fórmula:C27H35N5O2Forma y color:SolidPeso molecular:461.6CYP11B1-IN-2
<p>CYP11B1-IN-2 selectively inhibits human and rat CYP11B1 (IC50: 9/25 nM) orally to research cortisol-related diseases.</p>Forma y color:SolidAntifungal agent 28
<p>Antifungal 28 disrupts Candida, hits fluconazole-resistant strains, and inhibits biofilms.</p>Fórmula:C22H29N5OSForma y color:SolidPeso molecular:411.56TAS05567
CAS:TAS05567 is a potent, highly selective, and ATP-competitive Syk inhibitor (IC50: 0.37 nM).Fórmula:C21H29N9O2Pureza:98%Forma y color:SolidPeso molecular:439.51L5-DA
<p>L5-DA, a G-quadruplex ligand, stabilizes G4s in HeLa cells, induces apoptosis, and is cytotoxic with an IC50 of 4.3 μM.</p>Fórmula:C32H34N6O2Forma y color:SolidPeso molecular:534.65COX-2/NO-IN-1
COX-2/NO-IN-1: oral iNOS & NO blocker (IC50=3.52μM), COX-2 supressor, anti-inflammatory, protects kidneys.Fórmula:C15H15NO3Forma y color:SolidPeso molecular:257.28Henagliflozin
CAS:Henagliflozin (SHR3824): an oral, selective SGLT2 inhibitor, weak on SGLT1.Fórmula:C22H24ClFO7Forma y color:SolidPeso molecular:454.87Akt/NF-κB/JNK-IN-1
Akt/NF-κB/JNK-IN-1 (Compound 2i) is an inhibitor of Akt, NF-κB and JNK signalling pathways.Akt/NF-κB/JNK-IN-1 exhibits an inhibitory effect on nitric oxideFórmula:C22H22N2O6Forma y color:SolidPeso molecular:410.42PDE4B/7A-IN-1
CAS:5-HT1A antagonist; Ki=8nM, Kb=0.04nM. PDE4B IC50=80.4μM; PDE7A IC50=151.3μM. Good biofilm penetration, stable, anticognitive, antidepressant.Fórmula:C25H35N3O3Forma y color:SolidPeso molecular:425.56NLRP3-IN-4
NLRP3-IN-4 is an effective, oral NLRP3 inflammasome inhibitor with potent anti-inflammatory effects on colitis.Fórmula:C22H22N2O5Forma y color:SolidPeso molecular:394.42AVE-1330A sodium
CAS:AVE-1330A sodium is a beta-Lactamase inhibitor.Fórmula:C7H10N3NaO6SForma y color:SolidPeso molecular:287.23Anticancer agent 143
CAS:Anticancer Agent 143 (Compound 369), a potent dual inhibitor targeting PTPN2 and PTP1B, exhibits IC50 values below 2.5 nM.Fórmula:C19H15BrF2N3O6PS2Pureza:98%Forma y color:SolidPeso molecular:594.34Ibafloxacine
CAS:Ibafloxacine (R835) is a fluoroquinolone antibiotic that is used exclusively in veterinary applications and shows zero good bacteriostatic effect againstFórmula:C15H14FNO3Pureza:97.67%Forma y color:SolidPeso molecular:275.27GRPR antagonist-2
GRPR antagonist-2 blocks GRPR, kills some cancer cells, effective on HGC-27 (IC50: 0.77 μM) & Pan02 (IC50: 2.5 μM).Fórmula:C28H32F3N5O4Forma y color:SolidPeso molecular:559.58Gepotidacin hydrochloride
CAS:Gepotidacin (GSK-2140944) is a potent DNA topoisomerase inhibitor, a novel antibacterial efficacious against various anaerobes.Fórmula:C24H29ClN6O3Forma y color:SolidPeso molecular:484.98Factor B-IN-3
CAS:Factor B-IN-3 is a potent inhibitor of complement factor B. Factor B-IN-3 can be used to study inflammatory and immune-related diseases.Fórmula:C24H29N3O4Forma y color:SolidPeso molecular:423.5(±)-ANAP hydrochloride (1185251-08-4 free base)
(±)-ANAP hydrochloride is the amino acid analog of prodan. It can be used as a fluorescent probes and enhance environmental sensitivity.Fórmula:C15H17ClN2O3Pureza:98%Forma y color:SolidPeso molecular:308.76PF-446687
CAS:PF-446687 is a highly selective MC4 receptor (MC4R) agonist.Fórmula:C28H37ClF2N2O2Forma y color:SolidPeso molecular:507.06MEIS-IN-1
CAS:<p>MEIS-IN-1 is a potent MEIS inhibitor that induces the expansion of hematopoietic stem cells in mice and humans.</p>Fórmula:C24H21F3N2O4Forma y color:SolidPeso molecular:458.43Chitin synthase inhibitor 1
Potent, selective CHS inhibitor with 0.12 mM IC50; effective against drug-resistant fungi.Fórmula:C22H20ClN3O3Forma y color:SolidPeso molecular:409.87SMCypI C31
SMCypIC31, a non-peptide cyclophilin inhibitor, blocks PPIase at 0.1 μM IC50 and fights various HCV genotypes (EC50: 1.20-7.76 μM).Fórmula:C27H30N4O2SForma y color:SolidPeso molecular:474.62Pociredir
CAS:Pociredir (FTX-6058), a potent EED inhibitor (KD=0.163 nM), may help in SCD research.Fórmula:C22H18FN5O2Forma y color:SolidPeso molecular:403.41Atiratecan
CAS:Atiratecan (TP300), a CH0793076-based camptothecin prodrug, combats BCRP+/- tumors; doesn't affect AChE.Fórmula:C31H34N6O6Pureza:98%Forma y color:SolidPeso molecular:586.64Hit 1
<p>Hit 1 is an activator of insulin-degrading enzymes (IDE) (EC50: 5.5 μM) and reduces glucose-stimulated insulin secretion.</p>Fórmula:C22H24N4O3S2Forma y color:SolidPeso molecular:456.58CEP-7055
CAS:CEP-18770: oral proteasome inhibitor; blocks NF-kappaB; may cause cancer cell apoptosis; less toxic than bortezomib in normal cells.Fórmula:C32H35N3O4Forma y color:SolidPeso molecular:525.64HDAC-IN-9
HDAC-IN-9, a dual tubulin/HDAC inhibitor, impedes A549 cell invasion/migration and shows strong anti-tumor/angiogenic effects.Fórmula:C33H38N2O4Forma y color:SolidPeso molecular:526.67SphK1-IN-1
<p>SphK1-IN-1: SphK1 ATPase inhibitor, IC50=2.48 μM, potential for cancer research.</p>Fórmula:C22H22N6O2Forma y color:SolidPeso molecular:402.45Metoquizine
CAS:Metoquizine is an anticholinergic compound. It is a muscarinic acetylcholine receptor antagonist that has been used to treat ulcers.Fórmula:C22H27N5OPureza:98%Forma y color:SolidPeso molecular:377.485-Iminodaunorubicin hydrochloride
CAS:<p>5-Iminodaunorubicin HCl: quinone-modified anthracycline with antitumor properties, induces DNA breaks in cancer cells.</p>Fórmula:C27H31ClN2O9Forma y color:SolidPeso molecular:563.00Riminkefon
CAS:<p>Riminkefon is a kappa opioid receptor agonist .</p>Fórmula:C38H57N7O6Forma y color:SolidPeso molecular:707.9Fipravirimat
CAS:Fipravirimat is a potent inhibitor of HIV-1 with potential applications in HIV and AIDS research.Fórmula:C43H67FN2O4SForma y color:SolidPeso molecular:727.07Samuraciclib hydrochloride hydrate
Samuraciclib (CT7001) is a potent oral CDK7 inhibitor (IC50: 41 nM) with anti-breast cancer properties.Fórmula:C22H35ClN6O3Forma y color:SolidPeso molecular:521.7AChE-IN-11
AChE-IN-11 aids Alzheimer's research, has neuroprotection/antioxidant properties (ORAC=2.5), and acts on AChE, MAO-B, BACE1 with IC50 values of 7.9-9.9 μM.Fórmula:C18H28N2O4Forma y color:SolidPeso molecular:336.43CDK7/12-IN-1
CAS:CDK7/12-IN-1 is a selective CDK7 (IC50: 3 nM) and CDK12 (IC50: 277 nM) inhibitor, effective against tumor growth.Fórmula:C25H34N8OForma y color:SolidPeso molecular:462.59FGFR4-IN-4
CAS:FGFR4-IN-4 is a FGFR4 inhibitor with anti-tumor activity.Fórmula:C28H32Cl2N6O5Pureza:98%Forma y color:SolidPeso molecular:603.5STAT3-IN-8
CAS:<p>"STAT3-IN-8 (compound H172) is a potent inhibitor of STAT3 with potential applications in cancer research [1]."</p>Fórmula:C19H7F7N2O3Pureza:98%Forma y color:SolidPeso molecular:444.26D-473
CAS:<p>D-473 is a novel orally active triple reuptake inhibitor targeting dopamine, serotonin and norepinephrine transporters.</p>Fórmula:C26H27F2NO3Forma y color:SolidPeso molecular:439.49GnRH-R antagonist 1
CAS:Compound 21a: Oral GnRH-R antagonist, IC50=0.57 nM, potent against prostate cancer/prevents LH surges.Fórmula:C31H28F5N7O6SPureza:98%Forma y color:SolidPeso molecular:721.65α-Amylase-IN-1
CAS:α-Amylase-IN-1 is an α-Amylase inhibitor (IC50: 0.5509 μM).Fórmula:C18H18N2O3Pureza:99.92%Forma y color:SoildPeso molecular:310.35NR1H4 activator 1
CAS:NR1H4 activator 1 is a potent and selective agonist of Famesoid X Receptor (FXR).Fórmula:C34H53NO7SPureza:98%Forma y color:SolidPeso molecular:619.85ZBH-1205
CAS:<p>ZBH-1205, a camptothecin derivative, shows strong antitumor effects via apoptosis, outperforming cpt-11 and sn38 in topoisomerase-1 inhibition.</p>Fórmula:C29H31N3O8Forma y color:SolidPeso molecular:549.57CJ-887
CAS:<p>CJ-887 is a STAT3 inhibitor.</p>Fórmula:C34H45N6O10PForma y color:SolidPeso molecular:728.73BIIE-0246 HCl
CAS:BIIE-0246: A potent, non-peptide Y2 receptor antagonist; >650-fold more selective than Y1, Y4, Y5.Fórmula:C49H59Cl2N11O6Forma y color:SolidPeso molecular:968.97PF-06648671
CAS:<p>PF-06648671 is a γ-secretase modulator for the treatment of neurodegenerative and/or neurological disorders.</p>Fórmula:C25H23ClF4N4O3Pureza:98%Forma y color:SolidPeso molecular:538.92NOS-IN-2
NOS-IN-2: potent, selective imidamide NOS inhibitor, IC50=20μM for iNOS, spares eNOS, low toxicity, useful in inflammation research.Fórmula:C18H20F3N3O2Forma y color:SolidPeso molecular:367.3715(R)-Lipoxin A4
CAS:<p>Lipid-derived lipoxins are produced at the site of vascular and mucosal inflammation where they down-regulate polymorphonuclear leukocyte recruitment and</p>Fórmula:C20H32O5Forma y color:SolidPeso molecular:352.47LAF-153
CAS:LAF-153 is a reversible Methionine Aminopeptidase‑2 (MetAP-2) Inhibitor.Fórmula:C18H32N2O7Forma y color:SolidPeso molecular:388.46Dehatrine
CAS:Dehatrine: alkaloid from Beilschmiedia madang, inhibits Plasmodium falciparum K1 growth.Fórmula:C37H38N2O6Forma y color:SolidPeso molecular:606.71EGFR/HER2-IN-7
EGFR/HER2-IN-7: Potent, selective dual inhibitor for MCF-7 cancer; IC50: EGFR 0.18μM, HER2 0.146μM, DHFR 0.907μM.Fórmula:C19H21N3O2SForma y color:SolidPeso molecular:355.45Anticancer agent 29
<p>Compound E/Z-6f, anticancer, IC50: CDK2 (0.054 μM), CDK1 (0.127 μM), CDK4 (0.129 μM), CDK6 (0.396 μM).</p>Fórmula:C22H15ClFNOForma y color:SolidPeso molecular:363.81SS-RJW100
SS-RJW100 is an enantiomer of RJW100 targeting LRH-1, SF-1, enhances Tif2 interaction, and disrupts LRH-1 networks with lowered stability.Fórmula:C28H34OForma y color:SolidPeso molecular:386.57FNC-TP trisodium
<p>FNC-TP trisodium, active intracellular FNC form, inhibits NRTI, fights HIV, HBV, and HCV.</p>Fórmula:C9H11FN6Na3O13P3Forma y color:SolidPeso molecular:592.11RGB-286638
CAS:RGB-286638 inhibits multiple CDKs and GSK-3β, TAK1, Jak2, MEK1 with IC50s as low as 1-54 nM.Fórmula:C29H37Cl2N7O4Forma y color:SolidPeso molecular:618.55c-Met/HDAC-IN-2
CAS:Potent dual c-Met/HDAC inhibitor, IC50: HDAC1 5.4 nM, c-Met 18.49 nM; anti-cancer, induces apoptosis, G2/M arrest in HCT-116.Fórmula:C34H33N5O7Forma y color:SolidPeso molecular:623.66CAII-IN-2
CAII-IN-2 (3g): potent, selective CA-II inhibitor; IC50-12.1 μM for bovine CA-II; valuable in CA-related disorder research.Fórmula:C18H19BrN4SForma y color:SolidPeso molecular:403.34STA 2
CAS:STA 2 is an analogue of TXA2, a thromboxane receptor in the colonic epithelium.Fórmula:C21H34O3SForma y color:SolidPeso molecular:366.56FAK-IN-3
<p>FAK-IN-3 inhibits FAK, reduces PA-1 cell migration/invasion, and tumor growth, with no major side effects.</p>Fórmula:C28H28N6O4Forma y color:SolidPeso molecular:512.56LasR-IN-1
LasR-IN-1 (9g) strongly inhibits LasR, potent vs E. coli, with a 28.13 μM MIC against P. aeruginosa.Fórmula:C23H21N3O2Forma y color:SolidPeso molecular:371.43DWN-12088 HCl
CAS:DWN-12088 HCl is the salt form of DWN-12088 Free Base, an orally administered small molecule prolyl-tRNA synthetase (PRS) inhibitorFórmula:C15H21Cl4N3OForma y color:SolidPeso molecular:401.15Symplostatin 1
CAS:<p>Symplostatin 1 is a dolastatin 10 analog from the marine cyanobacterium Symploca hydnoides.</p>Fórmula:C43H70N6O6SForma y color:SolidPeso molecular:799.12Tubulin polymerization-IN-32
Tubulin polymerization-IN-32: a cancer cell growth inhibitor used for research in cancers like lymphoma.Fórmula:C29H30N2O7Forma y color:SolidPeso molecular:518.56FAAH/MAGL-IN-3
<p>FAAH/MAGL-IN-3 irreversibly inhibits FAAH (IC50: 179 nM) & MAGL (IC50: 759 nM) with low PAMPA permeability.</p>Fórmula:C21H25N3O6SForma y color:SolidPeso molecular:447.5CRS-3123
CAS:CRS-3123, a methionyl-tRNA synthetase inhibitor, is used potentially for the treatment of enteric infections.Fórmula:C19H19Br2N3O2SPureza:98%Forma y color:SolidPeso molecular:513.25KUS121
CAS:KUS121: VCP ATPase activity inhibitor (IC50=330 nM), protects cells from ER stress, assists in cerebral ischemia, and preserves vision in retinitis pigmentosa.Fórmula:C22H17FN4NaO3SForma y color:SolidPeso molecular:459.4522-HDHA
CAS:22-HDHA is an oxidation product of docosahexaenoic acid .Fórmula:C22H32O3Forma y color:SolidPeso molecular:344.49GAT564
GAT564, an allosteric CB1R modulator, shows EC50s of 87 nM (cAMP) & 320 nM (β-arrestin2) and lowers IOP effectively in glaucoma mice.Fórmula:C20H16N2O2SForma y color:SolidPeso molecular:348.42YM158 free base
CAS:YM158 free base is a potent and selective antagonist of TXA2 and LTD4 receptor (pA2s: about 8.81 and 8.87).Fórmula:C32H33ClN6O5S2Pureza:98%Forma y color:SolidPeso molecular:681.22Fasitibant
CAS:<p>Fasitibant is a potent and selective nonpeptide kinin B2 receptor antagonist.</p>Fórmula:C36H49Cl2N6O6SForma y color:SolidPeso molecular:764.78Antitumor agent-77
<p>Antitumor agent-77 suppresses cancer cell growth, migration, induces apoptosis, and hinders EMT.</p>Fórmula:C7H11F3N2O5PtForma y color:SolidPeso molecular:455.25MSX-3 free acid
CAS:MSX-3 free acid is an A2A adenosine receptor antagonist and a prodrug of MSX-2.Fórmula:C21H23N4O7PForma y color:SolidPeso molecular:474.40RET-IN-7
CAS:RET-IN-7 exhibits strong inhibitory effects against RET kinase in vitro and shows significant efficacy in treating RET-driven tumor xenografts in mice throughFórmula:C22H24ClFN6O2Forma y color:SolidPeso molecular:458.92DS89002333
<p>DS89002333: oral PRKACA inhibitor with 0.3 nM IC50, effective against FL-HCC with DNAJB1-PRKACA fusion in xenografts.</p>Fórmula:C22H20ClF2N3O3Forma y color:SolidPeso molecular:447.86Myxothiazol
CAS:Myxothiazol blocks mitochondrial complex III and triggers SESN2, a gene important for stress response.Fórmula:C25H33N3O3S2Forma y color:SolidPeso molecular:487.68
