Inhibidores
Los inhibidores son moléculas que se unen a enzimas, receptores u otras proteínas para reducir o bloquear su actividad biológica. Estos compuestos se utilizan ampliamente en la investigación para estudiar vías biológicas, comprender los mecanismos de las enfermedades y desarrollar fármacos terapéuticos. Los inhibidores desempeñan un papel crucial en el tratamiento de diversas enfermedades, incluyendo el cáncer, las enfermedades cardiovasculares y las infecciones. En CymitQuimica, ofrecemos una amplia gama de inhibidores de alta calidad para apoyar su investigación en bioquímica, biología celular y desarrollo farmacéutico.
Subcategorías de "Inhibidores"
- Angiogénesis(2.687 productos)
- Apoptosis(6.097 productos)
- Ciclo celular / Checkpoint(4.691 productos)
- Cromatina / Epigenética(2.376 productos)
- Señalización citoesquelética(1.472 productos)
- Daño al ADN / Reparación del ADN(2.921 productos)
- Endocrinología / Hormonas(3.611 productos)
- Enzima(3.655 productos)
- GPCR / proteína G(8.755 productos)
- Inmunología e inflamación(3.765 productos)
- Virus de la gripe(298 productos)
- Señalización JAK / STAT(407 productos)
- Señalización MAPK(1.230 productos)
- Transportador de membrana / canal de iones(2.947 productos)
- Metabolismo(9.940 productos)
- Microbiología / Virología(7.347 productos)
- Neurociencia(10.240 productos)
- Otros inhibidores(36.533 productos)
- Reducción de oxidación(43 productos)
- Señalización PI3K / Akt / mTOR(1.437 productos)
- Proteasas / Proteasoma(1.675 productos)
- Células madre y Derivados(830 productos)
- Tirosina quinasa / adaptadores(2.028 productos)
- Ubiquitinación(1.682 productos)
Mostrar 16 subcategorías más
Se han encontrado 66582 productos de "Inhibidores"
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ROPA
CAS:ROPA, a potent PKCalpha and PKCgamma activator, promotes tumor growth through PKC-activation.Fórmula:C28H32O6Pureza:98%Forma y color:SolidPeso molecular:464.55PF-06380101
CAS:PF-06380101, a potent auristatin analog and Dolastatin 10 derivative, shows strong anti-tumor activity and unique ADME attributes.Fórmula:C39H62N6O6SPureza:98%Forma y color:SolidPeso molecular:743.01Bcl-2-IN-8
Bcl-2-IN-8: potent, hinders cell growth/migration, induces apoptosis, promising in triple-negative breast cancer research.Fórmula:C36H44O6Forma y color:SolidPeso molecular:572.73Antimalarial agent 3
Antimalarial agent 3 has a potent IC50 of 0.035 μM against Plasmodium and high selectivity for mammalian cells.Fórmula:C15H16BrN3O2Forma y color:SolidPeso molecular:350.21Thiomuscimol hydrobromide
CAS:Thiomuscimol hydrobromide is an agonist of GABAA receptor.Fórmula:C4H6N2OSPureza:98%Forma y color:SolidPeso molecular:130.17GSK-2878175
CAS:GSK-2878175, a NS5B inhibitor, is used potentially for the treatment of HCV infection.Fórmula:C27H23BClFN2O6SPureza:98%Forma y color:SolidPeso molecular:568.81HER2-IN-9
<p>HER2-IN-9, an oral HER2 inhibitor (IC50: 0.03 μM), hinders growth and spread of HER2+ breast cancer.</p>Fórmula:C19H14BrF3N2OForma y color:SolidPeso molecular:423.23HIV-1 inhibitor-17
HIV-1 inhibitor-18 blocks HIV-1 capsid, acts on NL4-3 strain (EC50: 2.57 μM), has low cytotoxicity (MT-4 CC50: >8.55).Fórmula:C32H32N4O5SForma y color:SolidPeso molecular:584.69KRAS G12D inhibitor 3
CAS:KRAS G12D Inhibitor 3, a compound targeting the KRAS G12D mutation, demonstrates potent antitumor efficacy with an inhibitory concentration (IC50) of less thanFórmula:C34H31ClF3N5O2Forma y color:SolidPeso molecular:634.09PI4KIIIbeta-IN-11
CAS:PI4KIIIbeta-IN-11 is a PI4KIIIβ inhibitor (mean pIC50=9.1) that can be used to study diseases caused by RNA viruses and Plasmodium falciparum.Fórmula:C33H39N7O3Forma y color:SolidPeso molecular:581.71BMS-520
CAS:BMS-520: potent oral S1P1 agonist, effective in rat arthritis and mouse multiple sclerosis model.Fórmula:C23H17F3N4O4Forma y color:SolidPeso molecular:470.4UNC7467
CAS:UNC7467, potent IP6K2/1/6 inhibitor (4.9/8.9/1320 nM); lowers inositol pyrophosphates, minimal impact on other inositol phosphates; for obesity research.Fórmula:C20H13NO3Pureza:98.28% - 98.64%Forma y color:SoildPeso molecular:315.32Bulgecin A
CAS:Bulgecin A is an inhibitor of binuclear metallo-beta-lactamases and Lytic transglycosolase.Fórmula:C16H29N3O14S2Forma y color:SolidPeso molecular:551.54microRNA-21-IN-1
CAS:microRNA-21-IN-1: microRNA inhibitor, curbs HeLa/HCT-116 growth (IC50: 5.5/2.8 μM), induces HeLa apoptosis, elevates PTEN/EGR1/SLIT2, for cancer research.Fórmula:C30H37FN6O3Forma y color:SolidPeso molecular:548.65S1PR1 agonist 2
CAS:S1PR1 agonist 2 is potent for autoimmune research (from WO2021175225A1).Fórmula:C25H25N5O4Forma y color:SolidPeso molecular:459.50Purine phosphoribosyltransferase-IN-2
Purine PRTase-IN-2 inhibits Pf, Pv, Tbr PRT; Ki: 30, 20, 2 nM.Fórmula:C11H15N5Na4O10P2Forma y color:SolidPeso molecular:531.17P2X receptor-1
P2X receptor-1 is a potential inhibitor of P2X receptor for the treatment of pain and inflammation.Fórmula:C14H14ClN3O3S2Forma y color:SolidPeso molecular:371.86BACE1-IN-5
CAS:<p>BACE1-IN-5 inhibits BACE1 (IC50: 9.1 nM) & Aβ production (IC50: 0.82 nM), enhances hERG inhibition & P-gp efflux.</p>Fórmula:C18H16F5N5O2SPureza:98%Forma y color:SolidPeso molecular:461.41TLR7/8 agonist 7
CAS:<p>TLR7/8 agonist 7 activates immune cells, useful in ISAC synthesis and immunity research.</p>Fórmula:C26H37N7O2Forma y color:SolidPeso molecular:479.62T-3764518
CAS:T-3764518 is a novel and potent inhibitor of stearoyl coenzyme A desaturase (SCD)(IC50 of 4.7 nM).Fórmula:C20H17F6N5O2Pureza:98%Forma y color:SolidPeso molecular:473.37MLKL-IN-6
<p>MLKL-IN-6 (compound P28) is a mixed lineage kinase inhibitor that specifically targets the Mixed Lineage Kinase domain-like (MLKL) protein.</p>Fórmula:C20H18N4O5Pureza:98%Forma y color:SolidPeso molecular:394.38SOS1-IN-10
SOS1-IN-10 is a potent inhibitor of SOS1 that acts on KRAS G12C-SOS1 (IC50: 13 nM).Fórmula:C22H19F5N4OForma y color:SolidPeso molecular:450.4HBV-IN-19 TFA
CAS:<p>HBV-IN19 TFA suppresses HBsAg, hampers HBV infection, and aids in HBV research.</p>Fórmula:C26H31F3N2O8Forma y color:SolidPeso molecular:556.53COX-2/PI3K-IN-1
COX-2/PI3K-IN-1 (compound 5d) is a potent inhibitor of PI3K (IC50: 1.14 nM). COX-2/PI3K-IN-1 is a selective inhibitor of COX-2 (Ki: 3.24 nM).Fórmula:C19H14ClN5S2Forma y color:SolidPeso molecular:411.93Protease-Activated Receptor-1 antagonist 1
Compound 13 is a PAR-1 antagonist with a 3 nM IC50, useful for thrombosis and heart disease research.Fórmula:C25H24F2N2O3Forma y color:SolidPeso molecular:438.47PTP1B-IN-19
<p>PTP1B-IN-19, a benzimidazole, selectively inhibits protein tyrosine phosphatase 1B with a Ki of 23.3 μM, potential for type 2 diabetes research.</p>Fórmula:C26H19N3O4SForma y color:SolidPeso molecular:469.51Zalunfiban dihydrochloride
<p>Zalunfiban (RUC-4) is a potent αIIbβ3 platelet antagonist, IC50 45 nM, used in myocardial infarction research.</p>Fórmula:C16H20Cl2N8O2SForma y color:SolidPeso molecular:459.35(S)-3-Hydroxy Midostaurin
CAS:(S)-3-Hydroxy Midostaurin is a potent inhibitor of kinases(IC50 of <400 nM for 13 kinases (VEGFR-2, TRK-A, FLT3, et)).Fórmula:C35H30N4O5Pureza:98%Forma y color:SolidPeso molecular:586.64HDAC-IN-37
HDAC-IN-37 inhibits HDACs 1, 3, 8, & 6, induces histone acetylation, halts G1 to S phase, and triggers early apoptosis.Fórmula:C23H24ClN7OForma y color:SolidPeso molecular:449.94AD5075
CAS:<p>AD5075 is a bioactive chemical.</p>Fórmula:C22H20N2O5SForma y color:SolidPeso molecular:424.47KF26777
CAS:KF26777 is a potent and selective antagonist of adenosine A3 receptor.Fórmula:C16H16BrN5OPureza:98%Forma y color:SolidPeso molecular:374.23Casuarinin
CAS:<p>Casuarinin, an ellagitannin found in pomegranates and certain Casuarina/Stachyurus plants, is a carbonic anhydrase inhibitor and astringent.</p>Fórmula:C41H28O26Forma y color:SolidPeso molecular:936.655-HT6R/MAO-B modulator 1
5-HT6R/MAO-B modulator 1 blocks 5-HT6R and permanently inhibits MAO-B, protects glial cells, and reverses memory loss.Fórmula:C33H38N4O3SForma y color:SolidPeso molecular:570.74G-4120
CAS:G-4120 is a biochemical that has been shown to have a dose-dependent complete inhibition of arterial and venous thrombosis.Fórmula:C26H36N8O11SForma y color:SolidPeso molecular:668.68Cathepsin C-IN-3
Cathepsin C-IN-3 is a potent inhibitor of histone C (IC50: 61.79 nM) and also inhibits THP-1 cells (IC50: 101.5 nM) and U937 cells (IC50: 86.5 nM).Fórmula:C28H21F3N6OSForma y color:SolidPeso molecular:546.57Stauprimide
CAS:Stauprimide inhibits MYC by blocking NME2, reducing MYC transcription in ESCs.Fórmula:C35H28N4O5Pureza:98%Forma y color:SolidPeso molecular:584.62NNTA
CAS:<p>NNTA is a highly selective and potent activator of μ/κ-opioid heteromers.</p>Fórmula:C31H32N2O4Forma y color:SolidPeso molecular:496.60FR 901537
CAS:FR 901537 is a new aromatase inhibitor with antitumor effects.Fórmula:C23H29N3O6S2Pureza:98%Forma y color:SolidPeso molecular:507.62GABAA receptor agonist 1
Compound 3e, a potent GABAA agonist, targets GABA sites and has potential anti-depressive effects in mice.Fórmula:C20H30O3Forma y color:SolidPeso molecular:318.45Dual AChE-MAO B-IN-1
<p>Dual AChE-MAO B-IN-1: orally active CNS-permeable, safe, stable neuroprotective agent; AChE IC50=550 nM, MAO-B IC50=8.2 nM.</p>Fórmula:C23H25F2NO4Forma y color:SolidPeso molecular:417.45Salacinol
CAS:Salacinol is a naturally occurring alpha-glucosidase inhibitor isolated from an Ayurvedic traditional medicine Salacia reticulata.Fórmula:C9H18O9S2Forma y color:SolidPeso molecular:334.37EP4 receptor antagonist 2
CAS:EP4 receptor antagonist 2 (compound 2-13) is a potent agonist of the EP4 receptor (IC50: 7.8 nM) and has antitumour effects.Fórmula:C27H29N3O5Forma y color:SolidPeso molecular:475.54Domitroban
CAS:<p>Domitroban, also known as S-145, is a thromboxane (Tx) A2-receptor antagonist with partial agonistic activity in vascular smooth muscle.</p>Fórmula:C20H27NO4SForma y color:SolidPeso molecular:377.5Nomelidine
CAS:Nomelidine, the active N-demethylated metabolite of zimelidine, has been used as an antidepressant and analgesic.Fórmula:C15H15BrN2Pureza:98%Forma y color:SolidPeso molecular:303.20Topo I/COX-2-IN-1
Topo I/COX-2-IN-1: potent dual inhibitor; IC50 0.24μM (COX-2), 4.42μM (Topo I); anti-cancer; induces apoptosis, halts migration.Fórmula:C21H18ClFN2O3Forma y color:SolidPeso molecular:400.83HbF inducer-1
HbF inducer-1 is a fetal hemoglobin inducer which is orally bioavailable.Fórmula:C18H19N3O3Forma y color:SolidPeso molecular:325.36Lobaric acid
CAS:<p>Lobaric acid, from Stereocaulon lichen, has antioxidant and anticancer properties, inhibits PTP1B and 12(S)-LOX, and reduces TMV lesions in plants.</p>Fórmula:C25H28O8Forma y color:SolidPeso molecular:456.48T-Type calcium channel inhibitor 2
Compound 6g inhibits T-type Ca channels (IC50: Cav3.1-31μM, Cav3.2-83μM), cytotoxic to A549 (IC50: 5μM) & HCT-116 cells (IC50: 6.4μM).Fórmula:C36H39FN4OSForma y color:SolidPeso molecular:594.78VRT-18858
CAS:VRT-18858 is a metabolite of VX-740.Fórmula:C24H25N5O7Forma y color:SolidPeso molecular:495.48XP-524
CAS:XP-524: BET & EP300 inhibitor, suppresses KRAS tumors in vivo, targets PDAC, boosts immune response.Fórmula:C30H28N6O3SForma y color:SolidPeso molecular:552.65Pparδ agonist 5
Pparδ agonist 5 is a selective, orally active PPARδ agonist with an EC50 of 0.335 μM and better selectivity than GW0742.Fórmula:C23H21F3N2O2SForma y color:SolidPeso molecular:446.49Adecypenol
CAS:Adecypenol is a unique adenosine deaminase inhibitor. It shows effective inhibitory activity against calf intestinal adenosine deaminase.Fórmula:C12H16N4O4Pureza:98%Forma y color:SolidPeso molecular:280.28ONO-9780307
CAS:ONO-9780307 is a specific antagonist of LPA1 (lysophosphatidic acid receptor 1) (IC50: 2.7 nM).Fórmula:C30H35NO7Forma y color:SolidPeso molecular:521.6ONL-1204
CAS:ONL-1204 is a small molecule, CD95 antigen inhibitor (Fas inhibitor) being developed by ONL Therapeutics for the treatment of retinal detachment.Fórmula:C71H100N18O16Forma y color:SolidPeso molecular:1461.66ODN 21158
CAS:<p>ODN 21158 is a potent, non-cytotoxic inhibitor of G-modified TLR3 and TLR9. ODN 21158 dose-dependently inhibits IFN-α secretion.</p>Forma y color:SolidGLS1 Inhibitor-5
<p>GLS1 Inhibitor-5 (24y): Selective, oral glutaminase 1 inhibitor; IC50 68 nM; induces apoptosis; anti-tumor.</p>Forma y color:SolidCDK8-IN-5
CAS:CDK8-IN-5: potent CDK8 inhibitor, IC50=72 nM, boosts IL-10 by 43%, may aid inflammatory bowel disease research.Fórmula:C26H22N2O4Forma y color:SolidPeso molecular:426.46Ataprost
CAS:Ataprost (ONO 41483), an oral Carboprostacyclin analogue, is 2.6x more potent in inhibiting ADP-induced platelet aggregation and can relieve coronary spasm.Fórmula:C21H32O4Forma y color:SolidPeso molecular:348.48Protopine hydrochloride
CAS:Protopine inhibits thromboxane, lowers intracellular calcium, and reduces cell adhesion by altering adhesive factors.Fórmula:C20H20ClNO5Pureza:98%Forma y color:Prisms From Alc SolidPeso molecular:389.83JBJ-02-112-05
CAS:JBJ-02-112-05 is a potent, mutant-selective, allosteric and orally active inhibitor of EGFR with an IC 50 of 15 nM for EGFR L858R/T790M [1].Fórmula:C27H20N4O2SPureza:98%Forma y color:SolidPeso molecular:464.54NA 0346
CAS:NA 0346 is a derivative of SF 2370 that shows long lasting antihypertensive action as well as potent protein kinases inhibitory activity.Fórmula:C26H22N4O3Forma y color:SolidPeso molecular:438.48RBM10-8
CAS:RBM10-8 irreversibly inhibits human sphingosine-1- phosphate lyase (hS1PL) while behaving also as an enzyme substrate.Fórmula:C17H36NO5PForma y color:SolidPeso molecular:365.45Bometolol Hydrochloride
CAS:<p>Bometolol Hydrochloride is a beta-adrenergic blocking compound used for the treatment of cardiovascular disease.</p>Fórmula:C25H33ClN2O7Pureza:98%Forma y color:SolidPeso molecular:508.99γ-Secretase modulator 11 hydrochloride
CAS:<p>γ-Secretase modulator 11 hydrochloride is a potent, orally active γ-secretase modulator (IC50: 0.029 μM).</p>Fórmula:C28H23ClF2N4O2Forma y color:SolidPeso molecular:520.96VEGFR-2-IN-13
<p>VEGFR-2-IN-13 (Compound 19a) is a potent VEGFR-2 inhibitor (IC50: 3.4 nM). vEGFR-2-IN-13 arrests the HepG2 cell cycle in G2/M phase and induces apoptosis.</p>Fórmula:C24H18N6O2SForma y color:SolidPeso molecular:454.5Lavendomycin
CAS:Lavendomycin can be extracted from Streptomyces lavendulae and has active against Gram-positive bacteria.Fórmula:C29H50N10O8Forma y color:SolidPeso molecular:666.77MDK-3345
CAS:MDK-3345 is a reversible covalent inhibitor for Mcl-1.Fórmula:C36H34BN3O7Pureza:98%Forma y color:SolidPeso molecular:631.48DBCO-Sulfo-Link-biotin
CAS:DBCO-Sulfo-Link-biotin is a cleavable linker employed in the synthesis of antibody-drug conjugates (ADCs) [1].Fórmula:C31H35N5O7S2Pureza:98%Forma y color:SolidPeso molecular:653.77HG-12-6
CAS:HG-12-6 is a type II IRAK4 inhibitor, targeting its inactive form with an IC50 of 165 nM, and is used in autoimmunity and inflammation.Fórmula:C29H27F3N6O2SPureza:98%Forma y color:SolidPeso molecular:580.62(R)-BAY-899
(R)-BAY-899: R-isomer, selective LH-R antagonist, effective on hLH (IC50: 185 nM) and rLH (IC50: 46 nM), orally active.Fórmula:C25H19F2N5O2Forma y color:SolidPeso molecular:459.45EGFR-IN-58
EGFR-IN-58 is a potent, selective, ATP-competitive inhibitor of EGFR. EGFR-IN-58 exhibits significant cytotoxicity against melanoma, colon and blood cancers.Fórmula:C31H30FN7OForma y color:SolidPeso molecular:535.61Kaitocephalin
CAS:Kaitocephalin: naturally occurring, non-selective antagonist blocking glutamate receptors, made by Eupenicillium shearii fungus.Fórmula:C18H21Cl2N3O9Forma y color:SolidPeso molecular:494.28PD-1/PD-L1-IN-23
CAS:PD-1/PD-L1-IN-23: potent, oral PD-1/PD-L1 inhibitor; L7's ester prodrug; exhibits strong antitumor effects.Fórmula:C32H30BrCl2N3O6Forma y color:SolidPeso molecular:703.41CGS 22652
CAS:<p>CGS 22652 has thromboxane receptor antagonism combined with thromboxane synthase inhibition.</p>Fórmula:C22H29ClN2O4SForma y color:SolidPeso molecular:452.99Dicetrorelix pamoate
CAS:Cetrorelix pamoate is a synthetic decapeptide that acts as a GnRH antagonist, inhibiting the release of LH and FSH from the pituitary.Fórmula:C163H200Cl2N34O34Forma y color:SolidPeso molecular:3250.49TK-129
TK-129: Oral KDM5B inhibitor, IC50=44 nM, low-toxicity, cardioprotective, aids in heart disease research.Fórmula:C15H23N5O2Forma y color:SolidPeso molecular:305.38PKCiota-IN-1
CAS:<p>PKCiota-IN-1: Strong PKC-ι inhibitor (IC50=2.7 nM); also blocks PKC-α/ε (IC50s=45/450 nM).</p>Fórmula:C25H22FN5OForma y color:SolidPeso molecular:427.47GSK5852
GSK5852, an HCV NS5B inhibitor, has IC50 of 50 nM; potently fights HCV with EC50 of 3.0 nM for GT1a and 1.7 nM for GT1b.Fórmula:C27H27BF2N2O6SForma y color:SolidPeso molecular:556.39PARP-1/HDAC-IN-1
CAS:<p>PARP-1/HDAC-IN-1 is a PARP-1 and HDAC6 inhibitor with anticancer, antimigratory, and antiangiogenic activities and is used in tumor research.</p>Fórmula:C22H18N4O4Pureza:95.94%Forma y color:SolidPeso molecular:402.4Sekikaic Acid
CAS:Sekikaic acid, a phenolic lichen metabolite in H. obscurata, has antioxidant and antiviral properties, inhibiting MLL1-CBP.Fórmula:C22H26O8Forma y color:SolidPeso molecular:418.44OP-5244 sodium
OP-5244 sodium: potent oral CD73 inhibitor (IC50: 0.25 nM), potential in cancer research by hindering adenosine, reversing immunosuppression.Fórmula:C19H28ClN5NaO9PForma y color:SolidPeso molecular:559.87Rubropunctatin
CAS:Rubropunctatin is a monascus pigment with very potent cancer cell proliferation inhibitory effects.Fórmula:C21H23NO4Forma y color:SolidPeso molecular:353.41Nrf2 activator-6
CAS:Nrf2 activator-6, a tetrahydroisoquinoline, inhibits Kelch-Nrf2 at 5 nM IC50 (WO2021214470A1).Fórmula:C31H37ClFN5O5Forma y color:SolidPeso molecular:614.11Chitin synthase inhibitor 1
Potent, selective CHS inhibitor with 0.12 mM IC50; effective against drug-resistant fungi.Fórmula:C22H20ClN3O3Forma y color:SolidPeso molecular:409.87Beloranib
CAS:Beloranib is a fumagillin anticancer drug. Beloranib belongs to an angiogenesis inhibitor.Fórmula:C29H41NO6Pureza:98%Forma y color:SolidPeso molecular:499.64Beloxepin
CAS:Beloxepin is an oral dual selective inhibitor of serotonin and norepinephrine uptake.Fórmula:C19H21NO2Pureza:98%Forma y color:SolidPeso molecular:295.38CXCR4 probe 1
CAS:<p>CXCR4 probe 1, a specific PET tracer, targets CXCR4 with antagonist TN14003 (IC50: 6.9 nM), aiding in imaging CXCR4-related diseases and tumors.</p>Fórmula:C24H30FN5O4SForma y color:SolidPeso molecular:502.59CAII-IN-1
CAII-IN-1 (3n) is a selective bovine CA-II inhibitor with 10.3 μM IC50, used in carbonic anhydrase disorder studies.Fórmula:C19H21FN4SForma y color:SolidPeso molecular:356.46Calphostin I
CAS:Calphostins, from Cladosporium fungus, inhibit PKC. Notably, calphostin C is a potent biochemical tool.Fórmula:C44H38O15Forma y color:SolidPeso molecular:806.76Akt/NF-κB/JNK-IN-1
Akt/NF-κB/JNK-IN-1 (Compound 2i) is an inhibitor of Akt, NF-κB and JNK signalling pathways.Akt/NF-κB/JNK-IN-1 exhibits an inhibitory effect on nitric oxideFórmula:C22H22N2O6Forma y color:SolidPeso molecular:410.42Estrogen receptor antagonist 7
CAS:ER antagonist 7, compound 13, inhibits ERs, halts breast/ovarian cancer cell growth, has anticancer properties.Fórmula:C23H17N3O4Forma y color:SolidPeso molecular:399.4Pisiferic acid
CAS:<p>Pisiferic acid is a novel PP2C activator and an an antimicrobial diterpenoid</p>Fórmula:C20H28O3Forma y color:SolidPeso molecular:316.43Quinagolide hydrochloride
CAS:Quinagolide hydrochloride is a selective agonist of dopamine D2 receptor.Fórmula:C20H34ClN3O3SPureza:98%Forma y color:SolidPeso molecular:432.029(S)-HEPE
CAS:9(S)-HEPE is a monohydroxy fatty acid derived from EPA. The biological activity of 9(S)-HEPE has not been documented.Fórmula:C20H30O3Forma y color:SolidPeso molecular:318.45Unoprostone
CAS:Unoprostone is a prostaglandin F2α analogs (PGAs), and reduces intraocular pressure and is used topically for glaucoma or ocular hypertension.Fórmula:C22H38O5Pureza:98%Forma y color:SolidPeso molecular:382.53FPI-1465
CAS:<p>FPI-1465: Dual serine-β-lactamase & PBP inhibitor; IC50 PBP2=1.0 μg/mL; Kd CTX-M-15=0.011μM, OXA-48=5.3μM.</p>Fórmula:C11H18N4O7SForma y color:SolidPeso molecular:350.35AZD-4121 tert-butylammonium
CAS:AZD-4121 tert-butylammonium is an oral cholesterol absorption inhibitor targeting NPC1L1 for the treatment of dyslipidaemia.Fórmula:C40H50F2N4O7SForma y color:SolidPeso molecular:768.91RGT-068A
CAS:RGT-068A is a potent, selective and oral bioavailable MALT1 inhibitor .Fórmula:C17H16ClN9O2Forma y color:SolidPeso molecular:413.82TP-030-2
CAS:<p>TP-030-2 is a RIPK1 inhibitor (human K i =0.43 nM ; mouse IC 50 =100 nM) .</p>Fórmula:C23H21BrN4O3Forma y color:SolidPeso molecular:481.34Nrf2 activator-2
Compound O15, an Osthole derivative, is a potent Nrf2 agonist with an EC50 of 2.9 μM; it inhibits Keap1-Nrf2 binding and Nrf2 ubiquitination.Fórmula:C20H17BrO3Forma y color:SolidPeso molecular:385.25FT001
CAS:<p>FT001: Oral BET Bromodomain inhibitor, IC50=0.46μM, suppresses MYC, anti-cancer, effective in vitro/vivo.</p>Fórmula:C25H29N3O4SPureza:99.9%Forma y color:SolidPeso molecular:467.58Netupitant metabolite Monohydroxy Netupitant
CAS:Monohydroxy Netupitant is a highly selective antagonist of NK1 receptor, and is Netupitant metabolite.Fórmula:C30H32F6N4O2Pureza:98%Forma y color:SolidPeso molecular:594.59Chitin synthase inhibitor 5
Calpain Inhibitor-2, lipophilic, inhibits calpain; shows anti-proliferative effects on melanoma, PC-3 cells; blocks 80% DU-145 cell invasion.Fórmula:C23H22BrN3O5Forma y color:SolidPeso molecular:500.34(S)-Purvalanol B
CAS:<p>(S)-Purvalanol B is the S enantiomer of Purvalanol B. Purvalanol B is an inhibitor of cyclin-dependent kinase(CDK) .</p>Fórmula:C20H25ClN6O3Pureza:98%Forma y color:SolidPeso molecular:432.96-trans-12-epi-Leukotriene B4
CAS:<p>6-trans-12-epi-Leukotriene B4, a metabolite of arachidonic acid, serves as a potent anti-inflammatory agent.</p>Fórmula:C20H32O4Forma y color:SolidPeso molecular:336.47ZIKV-IN-5
ZIKV-IN-5 is an acid-stable, low cytotoxic anti-ZIKV agent with an EC50 value of 0.71 μM. ZIKV-IN-5 showed effective inhibition of ZIKV NS5 MTase activity.Fórmula:C36H45NO4SiForma y color:SolidPeso molecular:583.83OXS007417
OXS007417 induces AML cell differentiation at 48 nM EC50 and shows potent in vivo antitumor effects.Fórmula:C20H14F3N3OForma y color:SolidPeso molecular:369.34P-gp modulator 2
P-gp modulator 2 (Compound 27) is a potent competitive and metabotropic P-glycoprotein (P-gp) modulator.Fórmula:C22H20BrN3O4Forma y color:SolidPeso molecular:470.32SSR-182289A (Free)
CAS:SSR-182289A (Free) is a thrombin inhibitor.Fórmula:C30H33F2N5O4SPureza:98%Forma y color:SolidPeso molecular:597.68CD73-IN-7
CAS:<p>CD73-IN-7: potent inhibitor of CD73, blocks adenosine production to treat tumors.</p>Fórmula:C13H11ClN4O2Forma y color:SolidPeso molecular:290.7BMS-986034
CAS:<p>BMS-986034 is a GPR119 agonist.</p>Fórmula:C24H24Cl2N6O4Forma y color:SolidPeso molecular:531.39LL-Z 1640-4
CAS:A signal-specific JNK/p38 pathway and TAK 1 inhibitorFórmula:C19H24O7Pureza:98%Forma y color:SolidPeso molecular:364.39MraY-IN-1
MraY-IN-1 inhibits MraY (IC50: 140μM), fights E. coli K12, B. subtilis W23, P. fluorescens (MIC50: 7-46μg/ml), for antimicrobial research.Fórmula:C35H46N3O5Forma y color:SolidPeso molecular:588.76EED ligand 1
<p>EED ligand 1: potent PRC2 inhibitor targeting EED subunit.</p>Fórmula:C19H19FN8OForma y color:SolidPeso molecular:394.41HIF-2α-IN-7
CAS:HIF-2α-IN-7 is a hypoxia inducible factor 2α (HIF-2α) inhibitor.Fórmula:C18H9F6NO2Forma y color:SolidPeso molecular:385.26Antibacterial agent 76
Antibacterial agent 76 (compound 9) is a potent antibacterial agent.Fórmula:C23H27N3O2SForma y color:SolidPeso molecular:409.54PI3K-IN-29
CAS:<p>PI3K-IN-29: Strong PI3K block, inhibits Akt phosphorylation. IC50: U87MG 0.264µM, HeLa 2.04µM, HL60 1.14µM.</p>Fórmula:C27H22ClN7O3SForma y color:SolidPeso molecular:560.03Antifungal agent 38
<p>Antifungal agent 38, a heterocyclic disulfide, shrinks hyphae and damages cell membranes, causing leakage.</p>Fórmula:C8H12N2S2Forma y color:SolidPeso molecular:200.32Pim-1 kinase inhibitor 2
CAS:Compound 13, a potent Pim-1 inhibitor, induces apoptosis with potential for cancer research.Fórmula:C24H14N4O3Forma y color:SolidPeso molecular:406.39C108297
CAS:C108297: glucocorticoid modulator, combats diet obesity/inflammation, reduces appetite/lipid storage, boosts fat burn.Fórmula:C30H36FN3O4SPureza:98%Forma y color:SolidPeso molecular:553.69AKN-028 acetate
AKN-028 acetate: an oral TK inhibitor for AML research, targets FLT3 with IC50 of 6 nM, inhibits autophosphorylation, and induces apoptosis.Fórmula:C19H18N6O2Forma y color:SolidPeso molecular:362.39BRD50837
CAS:BRD50837 is a potent and selective inhibitor of Sonic Hedgehog (Shh).Fórmula:C26H32ClN3O6SPureza:98%Forma y color:SolidPeso molecular:550.07IACS-8779 disodium
CAS:IACS-8779 disodium: potent STING agonist, strong systemic anti-tumor effects, effective in melanoma model.Fórmula:C21H23N9Na2O10P2S2Forma y color:SolidPeso molecular:733.52JAK-IN-19
JAK-IN-19 inhibits JAK (pIC50: 7.2, 7.7), less so for VEGFR2 (7.0) and Aurora B (5.8).Fórmula:C26H36FN5O2Forma y color:SolidPeso molecular:469.59Geissoschizoline
CAS:Geissoschizoline inhibits human AChE/BChE (IC50: 20.40/10.21 µM) and has anti-inflammatory properties.Fórmula:C19H26N2OForma y color:SolidPeso molecular:298.42PCSK9-IN-17
CAS:<p>PCSK9-IN-17 is a PCSK9 inhibitor utilized in the research of cholesterol metabolism.</p>Fórmula:C16H19N5OSForma y color:SolidPeso molecular:329.42Turoctocog alfa
CAS:Turoctocog alfa: recombinant FVIII from CHO cells for hemophilia A study.Forma y color:SolidCRV431
CAS:CRV431 is a novel Pan-Cyclophilin Inhibitor, potently inhibiting all cyclophilin isoforms tested - A, B, D, and G (IC50 values ranged from 1-7 nM).Fórmula:C67H122N12O13Forma y color:SolidPeso molecular:1303.76MY-875
MY-875 inhibits microtubule formation, binds like colchicine (IC50: 0.92 μM), activates Hippo pathway, and induces apoptosis with anticancer properties.Fórmula:C21H25NO6Forma y color:SolidPeso molecular:387.43GZN39838
CAS:GZN39838, a natural Kv1.2 blocker, induces C-type inactivation without blocking the outer pore.Fórmula:C22H30O6Forma y color:SolidPeso molecular:390.47APJ receptor agonist 3
CAS:<p>APJ receptor agonist 3 is a highly effective and orally administerable agonist of the APJ receptor, demonstrating a potent EC50 value of 0.027 nM.</p>Fórmula:C26H29ClN4O5Forma y color:SolidPeso molecular:512.9818-Deoxyherboxidiene
CAS:<p>18-Deoxyherboxidiene (RQN-18690A) inhibits angiogenesis, targeting SF3b in U2 snRNP spliceosome, affects HUVEC, useful for cancer research.</p>Fórmula:C25H42O5Forma y color:SolidPeso molecular:422.6Cathepsin C-IN-4
Cathepsin C-IN-4 is a potent inhibitor (IC50: 65.6 nM) of histone C. Cathepsin C-IN-4 inhibits THP-1 cells (IC50: 203.4 nM) and U937 cells (IC50: 177.6 nM).Fórmula:C21H14ClF3N4SForma y color:SolidPeso molecular:446.88PD 113271
CAS:PD 113,271 is an analog of the fermentation products fostriecin with antitumor activity in vitro and in vivo.Fórmula:C19H27O10PPureza:98%Forma y color:SolidPeso molecular:446.39BAY-693
CAS:<p>BAY-693 is a ERK5 negative control agent with IC50 (ERK5) = 6400 nM. Its analog, BAY-885, is a potent and selective ERK5 (MAPK7) inhibitor with IC50 of 40 nM</p>Fórmula:C26H30F3N7O2Forma y color:SolidPeso molecular:529.56eIF4A3-IN-4
eIF4A3-IN-4 is a novel inhibitor of eIF4A (IC50: 8.6 μM).Fórmula:C24H20N2O5Forma y color:SolidPeso molecular:416.43(S)-Seco-Duocarmycin SA
CAS:(S)-Seco-Duocarmycin SA is a DNA alkylating agent and antibiotic with potent antitumor activity that can be used to synthesize ADC compounds.Fórmula:C25H24ClN3O7Pureza:98%Forma y color:SolidPeso molecular:513.93NAZ2329
CAS:NAZ2329: Cell-permeable, targets R5 RPTPs, inhibits hPTPRZ1 (IC50=7.5 μM) & hPTPRG (IC50=4.8 μM), hampers glioblastoma growth, affects stem cell traits.Fórmula:C21H18F3NO4S3Forma y color:SoildPeso molecular:501.56S39625
CAS:S39625 is a stable, potent topoisomerase I inhibitor with anticancer properties, resistant to efflux transporters, inducing gamma-H2AX at nanomolar levels.Fórmula:C25H22N2O5Pureza:98%Forma y color:SolidPeso molecular:430.45BRD4 Inhibitor-17
BRD4 Inhibitor-17: Potent with 0.33 μM IC50; modulates gene expression, may counter arsenic toxicity.Fórmula:C16H16FN3O3SForma y color:SolidPeso molecular:349.38Namitecan
CAS:Namitecan is an effective inhibitor of topoisomerase I. It has antitumor property.Fórmula:C23H22N4O5Pureza:98%Forma y color:SolidPeso molecular:434.44SARS-CoV-2 nsp3-IN-1
<p>Compound 15c selectively inhibits SARS-CoV-2 nsp3 Mac1 with IC50 of 6.1 μM.</p>Fórmula:C17H15N5O2Forma y color:SolidPeso molecular:321.33HMG499
CAS:HMG499 inhibits HMG-CoA reductase (IC50: 0.41μM), reduces statin-induced HMGCR, lowers cholesterol, and lessens atherosclerosis.Fórmula:C33H54O3Pureza:98%Forma y color:SolidPeso molecular:498.78Notch inhibitor 1
CAS:Notch inhibitor 1 blocks Notch 1/3 (IC50: 7.8/8.5 nM) and aids cancer research.Fórmula:C26H25F7N4O3Pureza:98%Forma y color:SolidPeso molecular:574.49SIK1 activator 1
CAS:SIK1 activator 1 boosts SIK1 phosphorylation, reduces type 2 diabetes hyperglycemia, and inhibits liver gluconeogenesis.Fórmula:C23H32O6Forma y color:SolidPeso molecular:404.50AY 17,605
CAS:AY 17,605 is an inhibitor of bovine heart and rat brain nucleoside-3',5'- monophosphate phosphodiesterase.Fórmula:C25H36O5Forma y color:SolidPeso molecular:416.55Falecalcitriol
CAS:<p>Falecalcitriol is an analog of calcitriol. It has a higher potency both in vivo and in vitro systems, which is longer duration of action in vivo.</p>Fórmula:C27H38F6O3Pureza:98%Forma y color:SolidPeso molecular:524.58Kendomycin
CAS:Kendomycin is a proteasome inhibitor and endothelin receptor antagonist. It induces apoptosis in lymphoma.Fórmula:C29H42O6Forma y color:SolidPeso molecular:486.64LSD1-IN-13 hydrochloride
CAS:<p>LSD1-IN-13 hydrochloride (7e) is an oral LSD1 inhibitor (IC50: 24.43 nM), promoting differentiation in AML cell lines.</p>Fórmula:C23H30ClN3O2SForma y color:SolidPeso molecular:448.02MtTMPK-IN-7
<p>MtTMPK-IN-7 inhibits MtbTMPK (IC50: 47 μM), active against M. brevis (MIC: 2.3-4.7 μM), useful for tuberculosis research.</p>Fórmula:C27H29ClN6O3Forma y color:SolidPeso molecular:521.015(S),6(R)-DiHETE
CAS:5(S),6(R)-DiHETE is a dihydroxy fatty acid from LTA4 hydrolysis and weak LTD4 agonist with ED50 of 1.3 μM for guinea pig ileum contraction.Fórmula:C20H32O4Forma y color:SolidPeso molecular:336.47ONO-AE1-329
CAS:<p>ONO-AE1-329 is a novel agonist of the prostaglandin PGE2 receptor EP4.</p>Fórmula:C22H30O6S2Forma y color:SolidPeso molecular:454.6Axl-IN-3
Axl-IN-3 is a selective, potent and orally active inhibitor of AXL kinase (IC50: 41.5 nM) and has a low inhibitory effect on other kinases.Fórmula:C24H25ClN6O2Forma y color:SolidPeso molecular:464.95Furaprevir
CAS:Furaprevir is an HCV NS3/4A InhibitorFórmula:C47H56N6O10SForma y color:SolidPeso molecular:897.05Antitubercular agent-13
Compound 3d: antitubercular, MIC 0.007 μg/mL vs MTB H37Rv, 1.851 μg/mL vs MDR-MTB 16833, metabolically unstable.Fórmula:C18H18N4O5Forma y color:SolidPeso molecular:370.36Pexacerfont
CAS:Pexacerfont (BMS-562086) is a selective antagonist of the corticotropin-releasing factor receptor (IC50: 6.1±0.6 nM for the human CRF1 receptor).Fórmula:C18H24N6OPureza:99.77%Forma y color:SolidPeso molecular:340.42Aurora B inhibitor 1
CAS:<p>Aurora B inhibitor 1 is an Aurora B (Aurora-1) inhibitor (Ki <0.010 uM) with potential anticancer activity for cancer research.</p>Fórmula:C25H26ClF2N7O2Pureza:98.37%Forma y color:SolidPeso molecular:529.97DGY-08-097
CAS:<p>DGY-08-097: potent HCV NS3 degrader, low resistance risk, strong inhibition in cells, DC50 of 50nM at 4h.</p>Fórmula:C60H76N10O14Forma y color:SolidPeso molecular:1161.3ATP synthase inhibitor 2
CAS:<p>ATP synthase inhibitor 2 blocks P. aeruginosa ATP synthase; IC50=10 μg/mL, fully inhibits at 128 μg/mL.</p>Fórmula:C21H22N2O3SForma y color:SolidPeso molecular:382.48PTP1B-IN-3 diammonium
PTP1B-IN-3 diammonium, an oral enzyme inhibitor, has potent antidiabetic and anticancer effects, with a 120 nM IC50.Fórmula:C12H13BrF2N3O3PForma y color:SolidPeso molecular:396.12DI-404
CAS:DI-404: Potent DCN1-UBC12 inhibitor, selectivity blocks cullin 3 neddylation, Kd=6.9 nM.Fórmula:C35H45ClN6O6SPureza:98%Forma y color:SolidPeso molecular:713.29HCV-IN-40
CAS:<p>HCV-IN-39 is a potent oral drug inhibiting HCV, effective on GT1a (EC50: 0.259μM), GT1b (EC50: 0.434μM), GT1b CES1 (EC50: 0.069μM) replicons.</p>Fórmula:C21H26BrFN3O9PForma y color:SolidPeso molecular:594.32DH376
CAS:<p>DH376 inhibits DAGLα in a time and dose dependent manner in mouse brain. DH376 shows picomolar activity.</p>Fórmula:C31H28F2N4O3Forma y color:SolidPeso molecular:542.58MIV-150
CAS:MIV-150 is a nonnucleoside inhibitor of reverse transcriptase (NNRT). MIV-150 also blocking HIV-1 and HIV-2 infections (EC50<1 nM against HIV-1/HIV-2MN).Fórmula:C19H17FN4O3Pureza:98%Forma y color:SolidPeso molecular:368.36ALK5-IN-7
CAS:ALK5-IN-7 inhibits ALK5, useful in TGF-β disease research like cancer, fibrosis, and autoimmune disorders. See WO2021129621A1.Fórmula:C26H28N4O3SForma y color:SolidPeso molecular:476.59IMR687
CAS:IMR687: a PDE9 inhibitor that could improve memory in Alzheimer's by slowing cGMP hydrolysis.Fórmula:C21H26N6O2Pureza:98%Forma y color:SolidPeso molecular:394.47FPDT
FPDT combats glioblastoma by inhibiting the AKT pathway; IC50: >100 μM (astrocytes), 45-68 μM (GBM cells).Fórmula:C16H12FNO2SForma y color:SolidPeso molecular:301.34MEIS-IN-3
MEIS-IN-3 is a potent inhibitor of MEIS.Fórmula:C25H26N2O4Forma y color:SolidPeso molecular:418.48Dyrk1A-IN-2
<p>Dyrk1A-IN-2 is a DYRK1A inhibitor (EC50: 37 nM). dyrk1A-IN-2 exhibits efficient promotion of human β-cell replication, as well as low cytotoxicity.</p>Fórmula:C27H32N6O4Forma y color:SolidPeso molecular:504.58HIV-1 inhibitor-13
<p>HIV-1 inhibitor-13: oral NNRTI, IC50=0.14μM for HIV-1 RT, effective on resistant strains (EC50=2.85-18nM).</p>Fórmula:C30H32N6O3Forma y color:SolidPeso molecular:524.61SMCypI C31
SMCypIC31, a non-peptide cyclophilin inhibitor, blocks PPIase at 0.1 μM IC50 and fights various HCV genotypes (EC50: 1.20-7.76 μM).Fórmula:C27H30N4O2SForma y color:SolidPeso molecular:474.62(2R,3S)-Azelaprag
CAS:(2R,3S)-N-(4-(2,6-dimethoxyphenyl)-5-(5-methylpyridin-3-yl)-4H-1,2,4-triazol-3-yl)-3-(5-methylpyrimidin-2-yl)butane-2-sulfonamide is an Apelin receptor agonistFórmula:C25H29N7O4SPureza:97.47% - >99.99%Forma y color:SoildPeso molecular:523.61Vps34-IN-3
Vps34-IN-3 is a potent, selective, and orally bioavailable inhibitor of VPS34 kinase .Fórmula:C14H20N4O2Forma y color:SolidPeso molecular:276.33MK-8970
MK-8970 is an acetal carbonate prodrug of raltegravir with enhanced colonic absorption.Fórmula:C25H29FN6O8Forma y color:SolidPeso molecular:560.54KU-32
CAS:<p>KU-32 is a novel and novobiocin-based Hsp90 inhibitor. It can protect against neuronal cell death.</p>Fórmula:C20H25NO8Pureza:98%Forma y color:SolidPeso molecular:407.41Antitumor agent-42
Antitumor agent-42 inhibits microtubule multimerisation and NO release, exhibiting anti-angiogenic, colony-forming and apoptosis-inducing effects.Fórmula:C24H19BrN2O8SForma y color:SolidPeso molecular:575.39Factor B-IN-4
CAS:Factor B-IN-4 is a potent inhibitor (IC50: 1 μM) of complement factor B. Factor B-IN-4 can be used to study inflammatory and immune-related diseases.Fórmula:C27H32N2O4Forma y color:SolidPeso molecular:448.55KP 10614
CAS:KP 10614 is a new prostacyclin analog that inhibits platelet-polymorphonuclear leukocyte interaction.Fórmula:C23H32O4Forma y color:SolidPeso molecular:372.50KRAS inhibitor-13
CAS:KRAS inhibitor-13 blocks KRAS G12C (IC50: 0.883 μM) and p-ERK in some cancer cells; promising for pancreatic, colorectal, lung cancer research.Fórmula:C25H19ClFN3O2SForma y color:SolidPeso molecular:479.95Epothilone E
CAS:<p>Epothilone E, a derivative of epothilone, functions by inhibiting microtubule protein activity, thereby halting cell division and exhibiting anti-tumor</p>Fórmula:C26H39NO7SForma y color:SolidPeso molecular:509.66MIF2-IN-1
MIF2-IN-1, potent inhibitor of MIF2 (IC50: 1μM), halts non-small cell lung cancer growth via MAPK pathway.Fórmula:C26H19F3N2O2SForma y color:SolidPeso molecular:480.5Antifungal agent 17
Antifungal agent 17 showed good antifungal activity against B. cinerea (EC50: 2.86 μg/mL).Fórmula:C18H16Br2O2Forma y color:SolidPeso molecular:424.13E-3030 free acid
CAS:<p>E-3030 free acid, a PPAR agonist, lowers blood glucose, triglycerides, and insulin; boosts adiponectin; reduces apo C-III; and raises lipoprotein lipase.</p>Fórmula:C22H23ClFNO5Pureza:98%Forma y color:SolidPeso molecular:435.87ZK 93426 hydrochloride
CAS:benzodiazepine receptor antagonist,competitiveFórmula:C18H21ClN2O3Pureza:98%Forma y color:SolidPeso molecular:348.82Arterolane
CAS:Arterolane is an antimalarial compound. For against P. falciparum Ro73 and W2, the IC50s are both 1.1 nM.Fórmula:C22H36N2O4Forma y color:SolidPeso molecular:392.53GLPG0492 (R enantiomer)
CAS:GLPG0492 R enantiomer is the R enantiomer of GLPG-0492, a novel selective androgen receptor modulator.Fórmula:C19H14F3N3O3Forma y color:SolidPeso molecular:389.33Hypothemycin
CAS:Hypothemycin, a fungal polyketide, inhibits multiple kinases (VEGFR, MEK, FLT-3, PDGFR, ERK) with Kis ranging from 10 nM to 2.4 μM.Fórmula:C19H22O8Pureza:98%Forma y color:SolidPeso molecular:378.37TAK-915
CAS:TAK-915: potent, brain-ready PDE2A inhibitor, 0.61 nM IC50, 4100x selectivity over PDE1A.Fórmula:C19H18F4N4O5Pureza:98%Forma y color:SolidPeso molecular:458.36P7170
CAS:<p>P7170 is an anti-cancer agent active as an mTORC1/C2 and activin receptor-like kinase 1 (ALK1) inhibitor.</p>Fórmula:C21H16F3N9Forma y color:SolidPeso molecular:451.42Idraparinux Na
CAS:Idraparinux Na is an Antithrombotic, Indirect, Selective, Synthetic Factor Xa InhibitorFórmula:C38H55Na9O49S7Forma y color:SolidPeso molecular:1727.14HBV-IN-24
<p>HBV-IN-24 inhibits HBV DNA, HBsAg, HBeAg (EC50: 0.6, 0.6, 4.6 nM), and has antiviral properties with neurotoxicity mitigation.</p>Fórmula:C23H27NO6Forma y color:SolidPeso molecular:413.46TAK-024
CAS:TAK-024 is an inhibitor of platelet(IC50s of 31, 79 and 51 nM in human, monkey and guinea pig, respectively).Fórmula:C27H34N10O6Pureza:98%Forma y color:SolidPeso molecular:594.62L2H2-6OTD
CAS:L2H2-6OTD is a telomerase inhibitor with G-quadruplex loops; IC50: 15 nM.Fórmula:C30H30N10O8Forma y color:SolidPeso molecular:658.62L 734217
CAS:L 734217 is an antagonist of the fibrinogen receptor.Fórmula:C18H31N3O4Pureza:98%Forma y color:SolidPeso molecular:353.46OP-2507
CAS:OP-2507, a prostacyclin agonist, is used potentially for the treatment of hepatic insufficiency and hypertension.Fórmula:C25H41NO4Pureza:98%Forma y color:SolidPeso molecular:419.6NMDA receptor antagonist-3
<p>NMDA antagonist-3: recovery rate 40% at 100 μM, low toxicity in SH-SY5Y, human stem cells.</p>Fórmula:C13H19N3O6Forma y color:SolidPeso molecular:313.31VU0463271 quarterhydrate
VU0463271 quarterhydrate is a potent KCC2 antagonist, with an IC 50 of 61 nM [1].Fórmula:C19H20N4O2S2Forma y color:SolidPeso molecular:387Canosimibe
CAS:Canosimibe is a cholesterol absorption inhibitorFórmula:C44H60FN3O10Forma y color:SolidPeso molecular:809.96
