Inhibidores
Los inhibidores son moléculas que se unen a enzimas, receptores u otras proteínas para reducir o bloquear su actividad biológica. Estos compuestos se utilizan ampliamente en la investigación para estudiar vías biológicas, comprender los mecanismos de las enfermedades y desarrollar fármacos terapéuticos. Los inhibidores desempeñan un papel crucial en el tratamiento de diversas enfermedades, incluyendo el cáncer, las enfermedades cardiovasculares y las infecciones. En CymitQuimica, ofrecemos una amplia gama de inhibidores de alta calidad para apoyar su investigación en bioquímica, biología celular y desarrollo farmacéutico.
Subcategorías de "Inhibidores"
- Angiogénesis(2.542 productos)
- Apoptosis(5.816 productos)
- Ciclo celular / Checkpoint(4.466 productos)
- Cromatina / Epigenética(2.252 productos)
- Señalización citoesquelética(1.381 productos)
- Daño al ADN / Reparación del ADN(2.830 productos)
- Endocrinología / Hormonas(3.518 productos)
- Enzima(3.640 productos)
- GPCR / proteína G(8.362 productos)
- Inmunología e inflamación(3.540 productos)
- Virus de la gripe(296 productos)
- Señalización JAK / STAT(405 productos)
- Señalización MAPK(1.201 productos)
- Transportador de membrana / canal de iones(2.809 productos)
- Metabolismo(9.462 productos)
- Microbiología / Virología(7.003 productos)
- Neurociencia(9.942 productos)
- Otros inhibidores(37.827 productos)
- Reducción de oxidación(40 productos)
- Señalización PI3K / Akt / mTOR(1.399 productos)
- Proteasas / Proteasoma(1.598 productos)
- Células madre y Derivados(830 productos)
- Tirosina quinasa / adaptadores(2.012 productos)
- Ubiquitinación(1.651 productos)
Mostrar 16 subcategorías más
Se han encontrado 66618 productos de "Inhibidores"
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Naltrindole
CAS:<p>Naltrindole is a delta opioid receptor antagonist.</p>Fórmula:C26H26N2O3Forma y color:SolidPeso molecular:414.5BRD7539
CAS:<p>BRD7539B: PfDHODH inhibitor, IC50 0.033μM; selective vs HsDHODH, IC50 >50μM.</p>Fórmula:C23H22FN3O2Pureza:98%Forma y color:SolidPeso molecular:391.44Antitumor agent-76
CAS:<p>Antitumor agent-76 is a water-soluble, orally active, rapid-release prodrug of Triptolide that exhibits anticancer effects.</p>Fórmula:C28H36ClNO10Forma y color:SolidPeso molecular:582.04Gamendazole
CAS:<p>Gamendazole is a novel drug candidate for male contraception. It has been shown to reduce fertility in male rats without affecting testosterone levels.</p>Fórmula:C18H11Cl2F3N2O2Pureza:98%Forma y color:SolidPeso molecular:415.19EP-7041 HCl
CAS:<p>EP-7041 is a novel, potent, and selective Factor XIa inhibitor.</p>Fórmula:C19H27ClN4O4Forma y color:SolidPeso molecular:410.89Topoisomerase I/II inhibitor 4
<p>Topoisomerase I/II inhibitor 4 halts cell growth and spread, induces apoptosis, and is used in liver cancer research.</p>Fórmula:C27H21N5O6Forma y color:SolidPeso molecular:511.49EGFR/HER2/DHFR-IN-1
<p>Potent EGFR/HER2/DHFR inhibitor for MCF-7 breast cancer; IC50: 0.153/0.108/0.291 μM; arrests G1/S phase, triggers apoptosis.</p>Fórmula:C14H11BrN4O2SForma y color:SolidPeso molecular:379.23Aurora/LIM kinase-IN-1
<p>Aurora/LIM kinase-IN-1 (Compound F114) is a dual inhibitor targeting aurora and lim kinases, potentially useful in GBM cancer treatment efforts.</p>Fórmula:C16H20N6OForma y color:SolidPeso molecular:312.37Norbinaltorphimine dihydrochloride
CAS:<p>Norbinaltorphimine dihydrochloride is a selective and potent κ opioid receptor antagonist that induces itch-associated responses in mice.</p>Fórmula:C40H45Cl2N3O6Pureza:98.17% - 99.88%Forma y color:SolidPeso molecular:734.71CXCR7 modulator 2
CAS:CXCR7 modulator 2 is a 7-type C-X-C chemokine receptor (CXCR7) modulator with a Ki of 13 nM.Fórmula:C29H42N6O3Forma y color:SolidPeso molecular:522.68AP5
CAS:<p>AP5: GPR40 agonist, positive allosteric modulator; rat hIP1 EC50: 0.49 nM.</p>Fórmula:C28H28FNO4Pureza:98%Forma y color:SolidPeso molecular:461.52A25822B
CAS:<p>A25822B is an antifungal agent.</p>Fórmula:C28H45NOPureza:98%Forma y color:SolidPeso molecular:411.66AChE/GSK-3β-IN-1
CAS:<p>AChE/GSK-3β-IN-1 is a potent dual AChE/GSK-3β inhibitor that crosses the blood-brain barrier and acts on hAChE (IC50: 1.2 nM), hBChE (IC50: 149.8 nM) and hGSK-</p>Fórmula:C31H35N7O3SForma y color:SolidPeso molecular:585.72AGN-204396
CAS:AGN-204396 is an antagonist that selectively blocks the activity of prostamides (prostaglandin-ethanolamides).Fórmula:C32H44FN3O4Forma y color:SolidPeso molecular:553.71EGFR-IN-18
<p>EGFR-IN-18 strongly inhibits L858R/T790M/C797S mutant EGFR (4.9 nM) and also targets wild-type EGFR (47 nM).</p>Fórmula:C33H28N6O3SForma y color:SolidPeso molecular:588.68NBD-10007
CAS:NBD-10007 is an inhibitor of HIV-1 entry.Fórmula:C20H25ClN4O3SPureza:98%Forma y color:SolidPeso molecular:436.96Cgs 25155
CAS:<p>Cgs 25155 is an orally active inhibitor of NEP 24.11.</p>Fórmula:C25H34N2O6SPureza:98%Forma y color:SolidPeso molecular:490.61BRD-7880
CAS:<p>BRD-7880 is a potent and highly specific inhibitor of aurora kinases B and C.</p>Fórmula:C32H38N4O7Forma y color:SolidPeso molecular:590.67Cenicriviroc Sulfone
CAS:<p>Cenicriviroc Sulfone, a Cenicriviroc derivative, inhibits CCR2/CCR5 to block HIV entry into cells.</p>Fórmula:C41H52N4O5SForma y color:SolidPeso molecular:712.94Saphenamycin
CAS:<p>Saphenamycin is an antibiotic from a strain of Streptomyces.</p>Fórmula:C23H18N2O5Pureza:98%Forma y color:SolidPeso molecular:402.40Carbodine
CAS:<p>Carbodine is an antiviral targeting CTP synthetase, effective against influenza A0/PR-8/34 and A2/Aichi/2/68.</p>Fórmula:C10H15N3O4Pureza:98%Forma y color:SolidPeso molecular:241.24K-14585
CAS:<p>K-14585 blocks PAR(2), reduces NFkappaB activity, and IL-8 response, but alone can boost IL-8.</p>Fórmula:C51H56Cl2N8O4Forma y color:SolidPeso molecular:915.95Epolactaene
CAS:<p>Epolactaene: neuritogenic, inhibits mammalian DNA polymerases & human DNA topoisomerase II.</p>Fórmula:C21H27NO6Forma y color:SolidPeso molecular:389.44DNA gyrase B-IN-1
<p>DNA gyrase B-IN-1, a potent inhibitor of P. aeruginosa DNA gyrase B, has IC50 of 2.2 μM with high affinity and stability.</p>Fórmula:C23H18ClF3N6O4SForma y color:SolidPeso molecular:566.94(3S,4R)-Tofacitinib
CAS:(3S,4R)-Tofacitinib is an less active enantiomer of Tofacitinib. Tofacitinib is a JAK3 inhibitor(IC50 : 1 nM).Fórmula:C16H20N6OPureza:98%Forma y color:SolidPeso molecular:312.37JAK2 JH2 binder-1
CAS:<p>JAK2 JH2 binder-1: potent, selective, Ki=37.1 nM, potential for studying myeloproliferative neoplasms.</p>Fórmula:C29H25N7O6SForma y color:SolidPeso molecular:599.62AZD-4121
CAS:<p>AZD-4121 is an oral cholesterol absorption inhibitor targeting NPC1L1 for the treatment of dyslipidaemia.</p>Fórmula:C36H39F2N3O7SForma y color:SolidPeso molecular:695.77GP-1681
CAS:<p>GP-1681, a G-protein coupled receptor (GPCR) agonist, is used potentially for the treatment of influenza infection.</p>Fórmula:C24H30NaO5Pureza:98%Forma y color:SolidPeso molecular:421.48hDDAH-1-IN-2 sulfate
<p>hDDAH-1-IN-2: selective oral hDDAH-1 inhibitor with low cell toxicity.</p>Fórmula:C8H24N4O10S2Forma y color:SolidPeso molecular:400.43DS89002333
<p>DS89002333: oral PRKACA inhibitor with 0.3 nM IC50, effective against FL-HCC with DNAJB1-PRKACA fusion in xenografts.</p>Fórmula:C22H20ClF2N3O3Forma y color:SolidPeso molecular:447.86LY 235959
CAS:<p>LY 235959 is a NMDA receptor antagonist.</p>Fórmula:C11H20NO5PPureza:98%Forma y color:SolidPeso molecular:277.25Anticancer agent 35
<p>Compound 10, a sulfonylurea, inhibits A549, A431, PACA2 cells with IC50s: 18.1, 4.0, 18.9 μg/mL.</p>Fórmula:C15H13N3O3S3Forma y color:SolidPeso molecular:379.48Barixibat
CAS:<p>Barixibat is a bile acid transport inhibitor.</p>Fórmula:C42H55N5O8Forma y color:SolidPeso molecular:757.91Quinagolide Free Base
CAS:<p>Quinagolide Free Base is a non-ergot dopamine D(2)-agonist.</p>Fórmula:C20H33N3O3SForma y color:SolidPeso molecular:395.56VEGFR-2-IN-10
<p>VEGFR-2-IN-10 has enhanced antiangiogenic potency against VEGFR2 phosphorylation induced by VEGF with an IC50 value of 0.7 μM and no cytotoxic effects.</p>Fórmula:C20H21N3O2Forma y color:SolidPeso molecular:335.4NDT-30805
<p>NDT-30805, a triazolopyridine, blocks IL-1β in PBMC (IC50: 0.013μM) & NLRP3 inflammasome, for inflammation research.</p>Fórmula:C23H22N6SForma y color:SolidPeso molecular:414.53C108297
CAS:<p>C108297: glucocorticoid modulator, combats diet obesity/inflammation, reduces appetite/lipid storage, boosts fat burn.</p>Fórmula:C30H36FN3O4SPureza:98%Forma y color:SolidPeso molecular:553.69RO5461111
CAS:<p>RO5461111: Oral Cathepsin S inhibitor, IC50 of 0.4 nM (human) & 0.5 nM (mouse), reduces T/B cell activation, treats lung inflammation & lupus nephritis.</p>Fórmula:C27H24F6N4O4SForma y color:SolidPeso molecular:614.56YK5
CAS:<p>YK5 is an allosteric inhibitor pocket of Hsp70 and represents a previously unknown chemical tool to investigate cellular mechanisms associated with Hsp70.</p>Fórmula:C18H24N8O3SPureza:98%Forma y color:SolidPeso molecular:432.50BTK-IN-15
<p>BTK-IN-15: Oral BTK inhibitor, IC50 0.7 nM, induces cancer cell apoptosis, selective with anti-tumor effects.</p>Fórmula:C28H24FN5O2Forma y color:SolidPeso molecular:481.52FGFR4-IN-7
<p>FGFR4-IN-7 is a covalent, reversible FGFR4 inhibitor (IC50: 0.42 μM) that blocks the FGFR4 signaling pathway, thereby inducing apoptosis.</p>Fórmula:C26H25Cl2N5O3Forma y color:SolidPeso molecular:526.41N-methyl Leukotriene C4
CAS:<p>N-methyl LTC4 is a stable synthetic analog of LTC4 and a selective CysLT2 agonist, useful in studying leukotriene pharmacology.</p>Fórmula:C31H49N3O9SForma y color:SolidPeso molecular:639.8LLS30
CAS:<p>LLS30 inhibits Gal-1, reduces its binding affinity, and may help treat advanced prostate cancer.</p>Fórmula:C34H33Cl4N5O3Forma y color:SolidPeso molecular:701.47Mu opioid receptor antagonist 3
<p>Potent, selective MOR antagonist (compound 26); crosses blood-brain barrier. Ki: 0.24 nM, EC50: 0.54 nM; for studying OUD.</p>Fórmula:C25H28N2O4SForma y color:SolidPeso molecular:452.57U92016A hydrochloride
CAS:<p>U92016A hydrochloride: potent, orally active 5-HT1A agonist, metabolically stable, high intrinsic activity, Ki=0.2 nM.</p>Fórmula:C19H26ClN3Forma y color:SolidPeso molecular:331.89GLP-1R agonist 8
CAS:<p>GLP-1R agonist 8 is a potent agonist of GLP-1R (EC50 < 2 nM).</p>Fórmula:C33H32N4O5Forma y color:SolidPeso molecular:564.63Adecypenol
CAS:<p>Adecypenol is a unique adenosine deaminase inhibitor. It shows effective inhibitory activity against calf intestinal adenosine deaminase.</p>Fórmula:C12H16N4O4Pureza:98%Forma y color:SolidPeso molecular:280.28Diospyrin
CAS:<p>Diospyrin is a plant product that has significant inhibitory effect on the growth of Leishmania donovani promastigotes.</p>Fórmula:C22H14O6Forma y color:SolidPeso molecular:374.34SH498
CAS:<p>SH498 is a novel Bmi-1-mediated anti-tumor agent with significant anti-proliferative effects.</p>Fórmula:C27H25F3N2O4Forma y color:SolidPeso molecular:498.49MB-07344 sodium
<p>"MB-07344 sodium is a TR-β agonist with a 2.17 nM Ki, boosts Atorvastatin's cholesterol-lowering effects in various animals."</p>Fórmula:C19H25NaO5PPureza:98%Forma y color:SolidPeso molecular:387.36Anticancer agent 29
<p>Compound E/Z-6f, anticancer, IC50: CDK2 (0.054 μM), CDK1 (0.127 μM), CDK4 (0.129 μM), CDK6 (0.396 μM).</p>Fórmula:C22H15ClFNOForma y color:SolidPeso molecular:363.81AN-12-H5
CAS:<p>AN-12-H5 is an anti-enteroviral compound that targets the replication process of PV and EV71 viruses.</p>Fórmula:C24H23N3O4S3Forma y color:SolidPeso molecular:513.65URAT1 inhibitor 2
<p>URAT1 inhibitor 2: oral URAT1/CYP blocker, IC50 of 1.36μM (URAT1), 16.97μM (CYP1A2), 5.22μM (CYP2C9); potential gout treatment.</p>Fórmula:C21H18BrN3O2SForma y color:SolidPeso molecular:456.36Ambrosin
CAS:<p>Ambrosin is a sesquiterpene lactone and a potent NF-κβ inhibitor. It is currently being studied as a potential lead drug for Alzheimer disease therapeutics.</p>Fórmula:C15H18O3Forma y color:SolidPeso molecular:246.3HBV-IN-11
CAS:<p>HBV-IN-11 is a potent inhibitor of HBsAg secretion (EC50: 0.46 μM).</p>Fórmula:C21H24ClNO6Forma y color:SolidPeso molecular:421.87Trk-IN-7
<p>Trk-IN-7 inhibits TRKA/B/C (IC50: 0.25-10 nM) & EML4-ALK (<15 nM), also targets various ALK mutations (IC50: 5-50 nM).</p>Fórmula:C18H17FN6O2Forma y color:SolidPeso molecular:368.36Epiderstatin
CAS:<p>Epiderstatin is isolated from Streptomyces pulveraceus subsp. epiderstagenes; inhibits mitogenic activity of epidermal growth factor.</p>Fórmula:C15H20N2O4Forma y color:SolidPeso molecular:292.3318-Deoxyherboxidiene
CAS:<p>18-Deoxyherboxidiene (RQN-18690A) inhibits angiogenesis, targeting SF3b in U2 snRNP spliceosome, affects HUVEC, useful for cancer research.</p>Fórmula:C25H42O5Forma y color:SolidPeso molecular:422.6Antibacterial agent 78
<p>Antibacterial agent 78 (compound 30) is an antibacterial agent with improved cytotoxicity profile[1].</p>Fórmula:C16H23N3S2Forma y color:SolidPeso molecular:321.5TGR5 Receptor Agonist 3
CAS:<p>TGR5 Receptor Agonist 3 is a GPBAR1 agonist with EC50 of 16.4 nM (hTGR5) & 209 nM (mTGR5), ensures gallbladder safety and reduces filling.</p>Fórmula:C29H27N3O6Forma y color:SolidPeso molecular:513.54ZK824859 hydrochloride
<p>ZK824859 hydrochloride: oral uPA inhibitor with IC50 of 79 nM (uPA), 1580 nM (tPA), 1330 nM (fibrin).</p>Fórmula:C23H23ClF2N2O4Forma y color:SolidPeso molecular:464.89Antiproliferative agent-4
<p>Antiproliferative agent-4 suppresses cancer cell growth with low toxicity, inhibits tumors in mice, and induces apoptosis in EC109 cells.</p>Fórmula:C29H35ClO8Forma y color:SolidPeso molecular:547.04Squalestatin 2
CAS:<p>Squalestatin 2 is an inhibitor of squalene synthase.</p>Fórmula:C33H44O13Pureza:98%Forma y color:SolidPeso molecular:648.69MtTMPK-IN-2
CAS:<p>MtTMPK-IN-2 inhibits M. tuberculosis TMPK (IC50: 1.1 μM), Mtb H37Rv (MIC: 12.5 μM), and is cytotoxic in MRC-5 cells (EC50: 6.1 μM).</p>Fórmula:C23H24ClN3O3Forma y color:SolidPeso molecular:425.91KMN-80
CAS:<p>KMN-80 is a potent, selective EP4 agonist with IC50 3 nM, spurring osteoblast differentiation, and showing in vivo bone repair efficacy.</p>Fórmula:C21H33NO4Forma y color:SolidPeso molecular:363.49CS-003 HCl
CAS:<p>CS-003 HCl is a TNRA - triple neurokinin receptor antagonist.</p>Fórmula:C34H39Cl3N2O6SForma y color:SolidPeso molecular:710.1FMK-MEA
CAS:<p>FMK-MEA is a potent and selective p90 Ribosomal S6 Kinase (RSK) inhibitor.</p>Fórmula:C21H26FN5O2Pureza:98%Forma y color:SolidPeso molecular:399.46(±)-HIP-B
CAS:<p>(±)-HIP-B is an excitatory amino acid transporter blocker.</p>Fórmula:C6H8N2O4Pureza:98%Forma y color:SolidPeso molecular:172.14DLK-IN-1
CAS:DLK-IN-1: Oral DLK (MAP3K12) inhibitor, Ki=3nM, effective in Alzheimer's model, CNS permeable, well-tolerated with sustained brain levels.Fórmula:C20H24F3N5O2Forma y color:SolidPeso molecular:423.43VEGFR-2-IN-11
<p>VEGFR-2-IN-11 is a potent inhibitor of VEGFR-2 (IC50: 60.27 nM) with an IC50 value of 60.27 nM, which induces apoptosis and has anticancer activity.</p>Fórmula:C29H22BrN5SForma y color:SolidPeso molecular:552.49TH-6
TH-6, a potent HDAC inhibitor (IC50: HDAC1-0.115, 2-0.135, 3-0.242, 6-0.138, 8-2.120 μM), blocks cell migration, invasion, and has anti-tumor properties.Fórmula:C22H24FN3O5Forma y color:SolidPeso molecular:429.44H 218-54
CAS:<p>H 218-54 is a renin inhibitor.</p>Fórmula:C37H56N2O5SForma y color:SolidPeso molecular:640.92Tubulin inhibitor 17
<p>Compound 3b inhibits tubulin polymerization, IC50 12.38 µM, with anticancer properties and promotes cell apoptosis.</p>Fórmula:C17H16N2OForma y color:SolidPeso molecular:264.32MS8815
CAS:<p>MS8815 is a selective EZH2 PROTAC degrader with IC50 of 8.6 nM, used in triple-negative breast cancer research.</p>Fórmula:C65H87N9O8SForma y color:SolidPeso molecular:1154.51L-365260 hemihydrate
<p>L-365260 hemihydrate: selective oral CCK-B/gastrin blocker, Ki=1.9/2.0 nM, competes with guinea pig receptors.</p>Fórmula:C24H24N4O3Forma y color:SolidPeso molecular:407.47Beloranib
CAS:<p>Beloranib is a fumagillin anticancer drug. Beloranib belongs to an angiogenesis inhibitor.</p>Fórmula:C29H41NO6Pureza:98%Forma y color:SolidPeso molecular:499.64Irinotecan Carboxylate Sodium Salt
CAS:<p>Irinotecan Carboxylate Sodium Salt is a DNA topoisomerase inhibitor.</p>Fórmula:C33H39N4NaO7Forma y color:SolidPeso molecular:626.68Tubulin polymerization-IN-8
CAS:<p>Compound IIc inhibits tubulin polymerization, arrests cell cycle at G2/M in HCT116 cells, IC50 12.7 μM, potential for cancer research.</p>Fórmula:C21H24N4O4SForma y color:SolidPeso molecular:428.5Tezosentan
CAS:<p>Tezosentan is an antagonist of the endothelin receptor (pA2s: 9.5, 7.7 for ETA and ETB receptors, respectively).</p>Fórmula:C27H27N9O6SPureza:98%Forma y color:SolidPeso molecular:605.63Pulvomycin
CAS:<p>Pulvomycin is a protein biosynthesis inhibitor preventing ternary complex formation between elongation factor Tu, GTP, and aminoacyl-tRNA.</p>Fórmula:C47H66O13Pureza:98%Forma y color:SolidPeso molecular:839.032Antiviral agent 7
<p>Antiviral agent 7 is a peptide-based coating that kills viruses.</p>Fórmula:C29H31F2N3O6Forma y color:SolidPeso molecular:555.57Fonadelpar
CAS:<p>Fonadelpar is an agonist of PPARδ. It also is used in the research of neuroparalytic keratopathy.</p>Fórmula:C25H23F3N2O4SPureza:98%Forma y color:SolidPeso molecular:504.52MtMetAP1-IN-1
<p>MtMetAP1-IN-1 is an inhibitor of methionine aminopeptidase 1 ( MetAP1 ). MtMetAP1-IN-1 shows antimycobacterial activity.</p>Fórmula:C15H10BrN5O2SForma y color:SolidPeso molecular:404.24DG013A
CAS:<p>DG013A inhibits ERAP1 & ERAP2 (IC50: 33 nM & 11 nM) to research autoimmune diseases & cancer.</p>Fórmula:C27H37N4O4PForma y color:SolidPeso molecular:512.58Anti-MRSA agent 2
CAS:<p>Anti-MRSA agent 2 inhibits MRSA at 0.098 μg/ml, with low toxicity and disrupts bacterial membranes and DNA.</p>Fórmula:C18H10Br2N2OForma y color:SolidPeso molecular:430.09Anti-inflammatory agent 6
<p>Anti-inflammatory agent 6 blocks IKKα/β, IκBα, and NF-κB p65 phosphorylation, key to controlling inflammation.</p>Fórmula:C22H20O12Forma y color:SolidPeso molecular:476.39GPR84 antagonist 3
CAS:<p>Potent GPR84 antagonist 3 (compound 42), pIC50 8.28, inhibits GTPγS, with good pharmacokinetics.</p>Fórmula:C29H27N5OForma y color:SolidPeso molecular:461.56MsbA-IN-5
<p>MsbA-IN-5 (compound 40) is a potent and highly selective inhibitor of MsbA (IC50: 2 nM). MsbA-IN-5 can be used in Gram-negative studies.</p>Fórmula:C23H19Cl2N5OForma y color:SolidPeso molecular:452.34Naltalimide
CAS:<p>Naltalimide: µ-opioid receptor partial agonist, improves bladder storage by affecting spinal cord reflex.</p>Fórmula:C28H28N2O5Pureza:98%Forma y color:SolidPeso molecular:472.53α5β1 integrin agonist-1
CAS:<p>α5β1 integrin agonist-1 is an α5β1 integrin agonist that selectively delivers 5-FU to tumour cells and induces tumour cell death.</p>Fórmula:C24H26FN5O9Forma y color:SolidPeso molecular:547.49BMS-986104 HCl
CAS:<p>BMS-986104 is a potent and selective S1P1 receptor modulator.</p>Fórmula:C22H36ClNOPureza:98%Forma y color:SolidPeso molecular:365.98DNA crosslinker 3 dihydrochloride
CAS:<p>Compound 1: a DNA minor groove binder with 1.4°C ΔTm; useful in cancer research.</p>Fórmula:C15H22Cl2N8OForma y color:SolidPeso molecular:401.29COX-2/NO-IN-1
<p>COX-2/NO-IN-1: oral iNOS & NO blocker (IC50=3.52μM), COX-2 supressor, anti-inflammatory, protects kidneys.</p>Fórmula:C15H15NO3Forma y color:SolidPeso molecular:257.28L5-DA
<p>L5-DA, a G-quadruplex ligand, stabilizes G4s in HeLa cells, induces apoptosis, and is cytotoxic with an IC50 of 4.3 μM.</p>Fórmula:C32H34N6O2Forma y color:SolidPeso molecular:534.65Anti-Aβ agent 1A
<p>Anti-Aβ agent 1A is a potent anti-amyloid-β agent.</p>Fórmula:C35H49NO4Forma y color:SolidPeso molecular:547.77GW-597901 cinnamate
CAS:<p>GW-597901 cinnamate is a long-acting beta(2)-agonist.</p>Fórmula:C34H46N2O8SForma y color:SolidPeso molecular:642.80DNA crosslinker 2 dihydrochloride
CAS:<p>Potent DNA crosslinker 2 binds minor groove, increases Tm by 1.2°C, and inhibits NCI-H460, A2780, MCF-7 cancer cells.</p>Fórmula:C15H22Cl2N8OForma y color:SolidPeso molecular:401.29RXR antagonist 2
<p>RXR antagonist 2 is a potent antagonist of RXR (Ki: 0.391 μM, Kd: 0.281 μM). RXR antagonist 2 has shown research potential for RXR-related diseases.</p>Fórmula:C29H35F3N2O3Forma y color:SolidPeso molecular:516.6TTA-P1
CAS:<p>TTA-P1: potent T-type calcium channel inhibitor; impacts neuron firing, hormone secretion, cell growth; potential in absence epilepsy research.</p>Fórmula:C19H27Cl2FN2OForma y color:SolidPeso molecular:389.33L 668411
CAS:L 668411, the 2,3-ditritiated methyl ester of L 659699, inhibits HMG-CoA synthase.Fórmula:C19H30O5Pureza:98%Forma y color:SolidPeso molecular:338.44CB2 receptor antagonist 1
CAS:<p>Compound 29 is a potent, CB2-selective antagonist/reverse agonist. Derivatives 23 & 24 offer antinociception; 24 activates cannabinoid/TRPV1 receptors.</p>Fórmula:C28H47NO3Forma y color:SolidPeso molecular:445.68Tubulin inhibitor 19
<p>Tubulin inhibitor 19 (9b), a potent indole chalcone, strongly blocks tubulin, valuable in cancer studies.</p>Fórmula:C21H23NO5Forma y color:SolidPeso molecular:369.41AMG-222 tosylate
CAS:<p>AMG-222 tosylate is a DPP-IV inhibitor in clinical development for type II diabetes.</p>Fórmula:C39H47N9O6SForma y color:SolidPeso molecular:769.91Oberadilol
CAS:<p>Oberadilol is a pyridazinone derivative with vasodilatory and beta-adrenergic blocking activities and type III phosphodiesterase inhibitory action</p>Fórmula:C25H30ClN5O3Forma y color:SolidPeso molecular:483.99Anti-MRSA agent 6
<p>Anti-MRSA agent 6 (compound 3q6) is a potent anti-methicillin-resistant Staphylococcus aureus (anti-MRSA) agent with low cytoxicity for MCF-7, A549 cells [1].</p>Fórmula:C16H11F2N3Forma y color:SolidPeso molecular:283.28LSD1/2-IN-3
<p>LSD1/2-IN-3 selectively inhibits LSD1 (Ki 11 nM) over LSD2 (Ki 7 μM), and hinders tumor stem cell proliferation.</p>Fórmula:C9H8BrF2NForma y color:SolidPeso molecular:248.07Saprisartan potassium
CAS:<p>Saprisartan potassium is an Angiotensin II Type 1 receptor antagonist and antihypertensive agent.</p>Fórmula:C25H21BrF3KN4O4SForma y color:SolidPeso molecular:649.52Gly-7-MAD-MDCPT
CAS:<p>Gly-7-MAD-MDCPT: anticancer Camptothecin with IC50 of 10-1000 nM against diverse cancers.</p>Fórmula:C24H22N4O7Forma y color:SolidPeso molecular:478.45JAK3-IN-13
<p>JAK3-IN-13: Oral JAK3 inhibitor, selective & potent. Acts on NK1, JNK2, JNK3, Tyk2. Anti-tumor. IC50: JNK3, 8 nM; Tyk2, 365 nM; JNK2, 2039 nM; NK1, 4728 nM.</p>Fórmula:C25H33ClN6O5Forma y color:SolidPeso molecular:533.02Neuraminidase-IN-11
<p>Neuraminidase-IN-11 (15e) inhibits H1N1 (IC50: 4.7nM), H5N1 (8.46nM), H5N8 viruses (1.5nM) selectively & potently.</p>Forma y color:SolidSC-435 mesylate
CAS:<p>SC-435 is an ileal apical sodium co-dependent bile acid transporter (ASBT). SC-435 inhibits plasma cholesterol.</p>Fórmula:C37H59N3O7S2Pureza:98%Forma y color:SolidPeso molecular:722.01SR121566A
CAS:SR121566A is a novel non-peptide antagonist of Glycoprotein IIb/IIIa (GP IIb-IIIa).Fórmula:C20H25N5O4SPureza:98%Forma y color:SolidPeso molecular:431.51Freselestat quarterhydrate
<p>ONO-6818 quarterhydrate: oral neutrophil elastase inhibitor, Ki 12.2 nM; >100x less effective on other proteases; strong anti-inflammatory.</p>Fórmula:C23H30N6O5Forma y color:SolidPeso molecular:457.03J-104132
CAS:<p>J-104132: potent human ETA/B antagonist; Ki: ETA=0.034nM, ETB=0.104nM; prevents ET-1 effects, ED50 i.v.=0.045mg/kg, p.o.=0.35mg/kg.</p>Fórmula:C31H33NO7Pureza:98%Forma y color:SolidPeso molecular:531.60G108
CAS:<p>G108 is an inhibitor of human cGAS and is used in the study of autoimmune diseases associated with human cGAS.</p>Fórmula:C16H14Cl2N4O2Pureza:99.13% - 99.75%Forma y color:SolidPeso molecular:365.21(RS)-AMPA
CAS:<p>(RS)-AMPA ((±)-AMPA) is a glutamate analog. (RS)-AMPA is an agonist of effective and selective excitatory neurotransmitter L-glutamic acid.</p>Fórmula:C7H10N2O4Pureza:98%Forma y color:SolidPeso molecular:186.17A1-Phytoprostane-I
CAS:<p>A1-Phytoprostane-I: cyclopentenone from α-linolenic acid in plants, induces gene expression & increases phytoalexin synthesis.</p>Fórmula:C18H28O4Forma y color:SolidPeso molecular:308.41SML-10-70-1
CAS:<p>SML-10-70-1 is a Novel Active Site Inhibitor of Oncogenic K-Ras G12C.</p>Fórmula:C25H42ClN7O13P2Forma y color:SolidPeso molecular:746.04Resolvin D1 methyl ester
CAS:<p>Resolvin D1, from docosahexaenoic acid via 15-/5-lipoxygenase, curbs acute inflammation; EC50 ~30 nM. Its methyl ester may enhance bioavailability.</p>Fórmula:C23H34O5Forma y color:SolidPeso molecular:390.51ABT 491 Hydrochloride
CAS:<p>ABT-491 hydrochloride is an active platelet activator receptor (PAF-R) antagonist with good selectivity and oral administration.</p>Fórmula:C28H23ClFN5O2Forma y color:SolidPeso molecular:515.97VVD-118313
CAS:<p>VVD-118313 (5a) is a potent JAK1 inhibitor targeting allosteric cysteine, blocking cytokine signaling for cancer research.</p>Fórmula:C19H22Cl2N2O3SForma y color:SolidPeso molecular:429.36PD 134922
CAS:PD 134922 is a HIV-1 protease inhibitors. Inactivation of the protease prevents infectious virion formation.Fórmula:C37H61N5O7SPureza:98%Forma y color:SolidPeso molecular:719.97NBTIs-IN-4
<p>NBTIs-IN-4, a broad-spectrum Gram-positive antibacterial, inhibits DNA rotamases/topoisomerase IV, with low resistance.</p>Fórmula:C22H24FN5O5SForma y color:SolidPeso molecular:489.52LXR agonist 2
<p>LXR agonist 2 is a potent agonist of the LXR (liver X receptor). LXR agonist 2 stabilises NCOA1 (coactivator), which in turn agonises the LXR.</p>Fórmula:C35H40ClN3O3Forma y color:SolidPeso molecular:586.16JBIR-22
CAS:<p>JBIR-22 is a natural inhibitor for protein−protein interaction of the homodimer of proteasome assembly factor 3.</p>Fórmula:C23H33NO6Forma y color:SolidPeso molecular:419.51Furametpyr
CAS:Furametpyr is a kind of low toxicity pesticides used to control plant diseases caused by various pathogenic microorganisms.Fórmula:C17H20ClN3O2Pureza:98%Forma y color:SolidPeso molecular:333.81CXCR2 antagonist 5
<p>CXCR2 antagonist 5 (compound 25) binds strongly (IC50=0.013μM) and mobilizes calcium (IC50=0.1μM).</p>Fórmula:C15H14F2N4O2SForma y color:SolidPeso molecular:352.36LSD1-IN-22
<p>LSD1-IN-22: potent LSD1 inhibitor, K_i 98 nM, curbs cancer cell growth.</p>Fórmula:C9H8BrF2NForma y color:SolidPeso molecular:248.07FTO-IN-4
CAS:<p>FTO-IN-4 is a potent and selective inhibitor of adiposity and obesity-associated protein (FTO).</p>Fórmula:C22H16Cl2N6O6Forma y color:SolidPeso molecular:531.31CLK1/4-IN-1
<p>CLK1/4-IN-1 inhibits Clk1/4 (IC50: 9.7/6.6 nM), curbing T24 cell growth (GI50: 1.1 μM). Potential cancer research tool.</p>Fórmula:C18H14ClNO4SForma y color:SolidPeso molecular:375.83CHF-6366
CAS:<p>CHF-6366: M3 antagonist & β2 agonist (pKi 10.4/11.4), mild Ca channel blocker, used in COPD study.</p>Fórmula:C42H48N6O8Forma y color:SolidPeso molecular:764.87STING agonist-20
CAS:<p>STING agonist-20: potent, aids in XMT-2056 synthesis, used as a cancer vaccine adjuvant.</p>Fórmula:C36H39N11O8Forma y color:SolidPeso molecular:753.76COX-2-IN-13
<p>COX-2-IN-13 is a potent, selective COX-2 inhibitor with 0.98 μM IC50; shows strong anti-inflammatory properties and low acute toxicity.</p>Fórmula:C19H18N2O5SForma y color:SolidPeso molecular:386.42PD-L1-IN-1
<p>PD-L1-IN-1, potent PD-L1 inhibitor with 115 nM IC50, suppresses tumors, boosts immune response, and spares healthy cells.</p>Fórmula:C21H23N5O2Forma y color:SolidPeso molecular:377.44IDO1-IN-14
<p>IDO1-IN-14 is an IDO1 enzyme inhibitor with an IC50 of 396.9 nM and suppresses HeLa cell activity with an EC50 of 3393 nM.</p>Fórmula:C18H12Cl2FN3O2Forma y color:SolidPeso molecular:392.219(S)-HETE
CAS:<p>9(S)-HETE is an enantiomer of (±)9-HETE, not an enzymatic product, and doesn't promote cell adhesion like 12(S)-HETE. Identified by chiral HPLC.</p>Fórmula:C20H32O3Forma y color:SolidPeso molecular:320.47Teslexivir
CAS:Teslexivir is a topical antiviral agent that is an effective and selective inhibitor of the interaction between two essential viral proteins, E1 and E2.Fórmula:C35H36BrN3O4Pureza:98%Forma y color:SolidPeso molecular:642.58Antitubercular agent-15
<p>Antitubercular agent-15 (5n): low toxicity, fights M. tuberculosis strains; MIC90 values range 0.73-18.8 μg/mL.</p>Fórmula:C21H29FN2Forma y color:SolidPeso molecular:328.47Cacospongionolide B
CAS:<p>Cacospongionolide B from Fasciospongia cavernosa inhibits secretory phospholipase A2, curbing inflammation.</p>Fórmula:C25H36O4Forma y color:SolidPeso molecular:400.55LRRK2-IN-6
<p>LRRK2-IN-6 is an oral, selective LRRK2 inhibitor crossing the blood-brain barrier, targeting GS (IC50: 4.6μM) and WT LRRK2 (IC50: 49μM).</p>Fórmula:C23H24F2N4O2SForma y color:SolidPeso molecular:458.52Antitumor agent-58
<p>Antitumor agent-58 suppresses tumor growth, colony formation, cell migration, and induces mitochondrial dysfunction in MGC-803 cells.</p>Fórmula:C27H28F3N9SForma y color:SolidPeso molecular:567.63MF-592
CAS:<p>MF-592: EP4 receptor antagonist, hEP4 IC50 3 nM, hWB IC50 78 nM, great oral PK, rat arthritis ED50 0.1 mg/kg/day, promising for development.</p>Fórmula:C34H33Cl2N3O6SForma y color:SolidPeso molecular:682.61ALK-IN-23
<p>ALK-IN-23 inhibits ALK (IC50: 1.6-0.71 nM), hinders cancer cell spread, forms colonies in vitro, and reduces tumors in mice with low toxicity.</p>Fórmula:C26H29ClN8O3SForma y color:SolidPeso molecular:569.08GNTI TFA
CAS:<p>GNTI TFA is a selective kappa opioid receptor antagonist.</p>Fórmula:C31H31F6N5O7Forma y color:SolidPeso molecular:699.60CP-608039
CAS:<p>CP-608039 is a selective adenosine A3 receptor agonist for both human A3 and human A1 receptors.</p>Fórmula:C23H25ClN8O5Forma y color:SolidPeso molecular:528.95K252d
CAS:<p>K252d: indolocarbazole alkaloid in Nocardiopsis; inhibits PKC in rat brain and bovine heart phosphodiesterase.</p>Fórmula:C26H23N3O5Forma y color:SolidPeso molecular:457.48C.I. Pigment Red 60
CAS:C.I. Pigment Red 60 is a bright, scarlet, semi-transparent red pigment.Fórmula:C17H9N2Na3O9S2Pureza:98%Forma y color:SolidPeso molecular:518.35Ornoprostil
CAS:Ornoprostil, a prostaglandin E1 analogue, acts as a mucosal protectant.Fórmula:C23H38O6Pureza:98%Forma y color:SolidPeso molecular:410.54iNOS/PGE2-IN-1
<p>iNOS/PGE2-IN-1: iNOS/PGE2 inhibitor, reduces LPS-induced NO, low ulcer risk, anti-inflammatory.</p>Fórmula:C26H22ClN3O4Forma y color:SolidPeso molecular:475.92PptT-IN-2
<p>PptT-IN-2 inhibits PptT enzyme crucial in tuberculosis, with 2.5 μM IC50, showing potential in TB research.</p>Fórmula:C22H29N5O2Forma y color:SolidPeso molecular:395.5EGFR-IN-44
<p>EGFR-IN-44: potent EGFR kinase inhibitor, orally active, IC50 4.11 nM, 33.57% bioavailability, induces apoptosis, for lung cancer study.</p>Fórmula:C27H29ClN6O2SForma y color:SolidPeso molecular:537.08Mimocine
CAS:<p>Mimosine, a plant amino acid, is known to act as a normoxic inducer of hypoxia-inducible factor (HIF).</p>Fórmula:C15H14N2O5Forma y color:SolidPeso molecular:302.28Topoisomerase II inhibitor 5
<p>Topoisomerase II inhibitor 5 (Compound E24) is a DNAtopoisomerase II inhibitor with anticancer effects.</p>Fórmula:C26H27N5O4Forma y color:SolidPeso molecular:473.52BChE-IN-5
<p>BChE-IN-5: potent, selective BChE inhibitor (IC50: 2.8 nM), more effective on hBChE, potential in Alzheimer's research.</p>Fórmula:C30H42N4OForma y color:SolidPeso molecular:474.68Onfasprodil
CAS:<p>Onfasprodil, NR2B inhibitor & GABA regulator, potential for Alzheimer's research. (Patent CN111481543A)</p>Fórmula:C20H23FN2O3Forma y color:SolidPeso molecular:358.41Anti-MRSA agent 3
CAS:<p>Anti-MRSA agent 3 targets MRSA with 0.098 μg/ml MIC, low toxicity, binds DNA, and disrupts cell walls/membranes.</p>Fórmula:C29H18BrN3O2Forma y color:SolidPeso molecular:520.386Ranakinin
CAS:<p>Ranakinin is a novel tachykinin receptor agonist; from the brain of frog, Rana ridibunda.</p>Fórmula:C62H95N17O15SForma y color:SolidPeso molecular:1350.59nAChR antagonist 1
CAS:<p>Compound B15, a potent α7 nAChR antagonist, IC50 = 3.3 μM, promising for research on schizophrenia, Alzheimer's, and inflammation.</p>Fórmula:C19H22N4O2Forma y color:SolidPeso molecular:338.4BAY-179
CAS:<p>BAY-179 is a potent, selective, species cross-reactive complex I inhibitor for the study of cancer.</p>Fórmula:C23H21N5OSPureza:98.29%Forma y color:SolidPeso molecular:415.515-Ph-IAA-AM
<p>5-Ph-IAA-AM, eggshell-permeable analog of 5-Ph-IAA, boosts protein degradation in embryos, useful for studying proteins in C. elegans.</p>Fórmula:C19H17NO4Forma y color:SolidPeso molecular:323.34BM635 mesylate
<p>BM635 mesylate inhibits MmpL3; kills Divergent bacterium with 0.6 µM MIC50; boosts bioavailability.</p>Fórmula:C26H33FN2O4SForma y color:SolidPeso molecular:488.61Acetomycin
CAS:<p>Acetomycin, a γ-lactone from S. ramulosus, halts HCT-8 colon and L1210 leukemia cell growth.</p>Fórmula:C10H14O5Forma y color:SolidPeso molecular:214.22MtTMPK-IN-5
<p>MtTMPK-IN-5 inhibits Mtb TMPK with IC50 of 34 μM and fights tuberculosis with MIC of 12.5 μM, aiding TB research.</p>Fórmula:C21H23N5O2Forma y color:SolidPeso molecular:377.44Thiomuscimol hydrobromide
CAS:<p>Thiomuscimol hydrobromide is an agonist of GABAA receptor.</p>Fórmula:C4H6N2OSPureza:98%Forma y color:SolidPeso molecular:130.17PF-06380101
CAS:<p>PF-06380101, a potent auristatin analog and Dolastatin 10 derivative, shows strong anti-tumor activity and unique ADME attributes.</p>Fórmula:C39H62N6O6SPureza:98%Forma y color:SolidPeso molecular:743.01HDAC/Top-IN-1
CAS:<p>HDAC/Top-IN-1, an oral HDAC/Top inhibitor, targets HDAC1-3,6,8 with low IC50s; blocks S-phase & induces apoptosis in HEL cells.</p>Fórmula:C29H25FN4O4Forma y color:SolidPeso molecular:512.53MALT1-IN-11
CAS:<p>MALT1-IN-11: MALT1 inhibitor, IC50 <10-100 nM, reduces IL10, for cancer/autoimmune research.</p>Fórmula:C20H16F4N8OForma y color:SolidPeso molecular:460.39ML-SI1
CAS:<p>ML-SI1, a racemic mixture of diastereoisomers, is a TRPML inhibitor and acts on TRPML1 (IC50: 15 μM).</p>Fórmula:C23H26Cl2N2O3Forma y color:SolidPeso molecular:449.37LXRβ agonist-3
CAS:<p>LXRβ agonist-3 is a potent and selective LXRβ (liver X receptor β) agonist (EC50: 0.095 μM).</p>Fórmula:C30H33N3O6SForma y color:SolidPeso molecular:563.66Calphostin I
CAS:<p>Calphostins, from Cladosporium fungus, inhibit PKC. Notably, calphostin C is a potent biochemical tool.</p>Fórmula:C44H38O15Forma y color:SolidPeso molecular:806.76MSX-3 free acid
CAS:<p>MSX-3 free acid is an A2A adenosine receptor antagonist and a prodrug of MSX-2.</p>Fórmula:C21H23N4O7PForma y color:SolidPeso molecular:474.40FPI-1465
CAS:<p>FPI-1465: Dual serine-β-lactamase & PBP inhibitor; IC50 PBP2=1.0 μg/mL; Kd CTX-M-15=0.011μM, OXA-48=5.3μM.</p>Fórmula:C11H18N4O7SForma y color:SolidPeso molecular:350.35MDL-100173
CAS:<p>MDL-100173 is a dual angiotensin-converting enzyme (ACE)/neutral endopeptidase (NEP) inhibitor.</p>Fórmula:C24H26N2O4SForma y color:SolidPeso molecular:438.54Monorden diacetate
CAS:<p>Monorden diacetate a Hsp90 Inhibitor. Monorden diacetate is a Promising Lead Compound for the Development of Novel Fungicides.</p>Fórmula:C22H21ClO8Forma y color:SolidPeso molecular:448.85AMS-17
<p>AMS-17, a strong NLRP3 inhibitor, quells microglia activation and cytokines like caspase-1, TNF-α, IL-1β, iNOS in studies.</p>Fórmula:C15H13F3N4O3SForma y color:SolidPeso molecular:386.35Cdc7-IN-19
CAS:<p>Cdc7-IN-19 (compound 1-1) is a potent CDC7 inhibitor with an IC 50 of 1.49 nM [1].</p>Fórmula:C19H21N5O2Forma y color:SolidPeso molecular:351.40TLN-232
CAS:<p>TLN-232, a synthetic heptapeptide, may inhibit cancer by targeting M2PK to disrupt tumor cell energy production.</p>Fórmula:C36H49N9O7S2Forma y color:SolidPeso molecular:783.96HMG499
CAS:<p>HMG499 inhibits HMG-CoA reductase (IC50: 0.41μM), reduces statin-induced HMGCR, lowers cholesterol, and lessens atherosclerosis.</p>Fórmula:C33H54O3Pureza:98%Forma y color:SolidPeso molecular:498.78TRK-IN-12
CAS:<p>TRK-IN-12 (9e), a macrocyclic TRK inhibitor (G595R IC50=13.1 nM), outperforms LOXO-101 in Ba/F3-NTRK1 cells.</p>Fórmula:C18H19ClFN5O3SForma y color:SolidPeso molecular:439.89Canosimibe
CAS:<p>Canosimibe is a cholesterol absorption inhibitor</p>Fórmula:C44H60FN3O10Forma y color:SolidPeso molecular:809.96PF-5177624
CAS:<p>PF-5177624 is a selective and potent PDK1 inhibitor inducing anti-tumor activity in breast cancer cells.</p>Fórmula:C25H25FN8O2Forma y color:SolidPeso molecular:488.52Tubulin polymerization-IN-3
<p>Tubulin polymerization-IN-3 is a potent inhibitor of microtubulin polymerization (IC50: 3.84 μM) and induces apoptosis in colon cancer cells.</p>Fórmula:C20H20ClN5O3Forma y color:SolidPeso molecular:413.86VU6005806
CAS:<p>VU6005806 is a potent M4 PAM with EC50s: 94 nM (human), 28 nM (rat), 87 nM (dog), 68 nM (cyno); studied for neuropsychiatric disorders.</p>Fórmula:C17H16F3N7O2SPureza:98%Forma y color:SolidPeso molecular:439.41NSC 828467
<p>NSC 828467 is one of the top five CA-IX inhibitors with significant in vitro anticancer activity (IC50: 27.2 nM).</p>Fórmula:C21H19N9O2SForma y color:SolidPeso molecular:461.5HDAC-IN-35
<p>HDAC-IN-35 (Compound 14) is an effective and selective inhibitor of VEGFR-2 and HDAC, with IC50 values of 13.2 and 0.166 μM for VEGFR-2 and HDAC6, respectively.</p>Fórmula:C17H13ClF3N3O3Forma y color:SolidPeso molecular:399.75Ambuic acid
CAS:<p>Ambuic acid: cyclohexanone with antifungal, quorum-inhibiting, antibacterial properties, blocks cyclic peptides; reduces MRSA abscesses in mice.</p>Fórmula:C19H26O6Forma y color:SolidPeso molecular:350.41Retezorogant
CAS:<p>Retezorogant is a retinoic acid receptor-related orphan receptor gamma (RORγ) antagonist.</p>Fórmula:C23H33ClN2O3Forma y color:SolidPeso molecular:420.97WEHI-9625
CAS:<p>WEHI-9625 is a tricyclic sulfone small molecule apoptosis inhibitor (EC50: 69 nM).</p>Fórmula:C34H27NO5S2Pureza:98%Forma y color:SolidPeso molecular:593.71KRAS inhibitor-21
CAS:<p>KRAS inhibitor-21 (22b) is a KRAS G12C inhibitor (IC50<0.01 μM) that can be used in cancer research.</p>Fórmula:C33H41N5O3Forma y color:SolidPeso molecular:555.71BI-44370
CAS:<p>BI-44370, a CGRP (calcitonin gene-related peptide) receptor antagonist, can be used to treat migraines and other chronic pain.</p>Fórmula:C35H47N5O6Forma y color:SolidPeso molecular:633.78CHK-IN-1
CAS:CHK-IN-1 is a dual inhibitor of CHK1 and CHK2 with antiproliferative activity.Fórmula:C18H19ClFN5OSPureza:>99.99%Forma y color:SolidPeso molecular:407.89Kalafungin
CAS:<p>Kalafungin inhibits various fungi, yeasts, protozoa, and gram-positive bacteria, less so for gram-negative bacteria.</p>Fórmula:C16H12O6Forma y color:SolidPeso molecular:300.26Anticancer agent 78
<p>Anticancer agent 78: anti-aromatase (IC50=0.9 μM), cytotoxic, potential in breast cancer research.</p>Fórmula:C19H14BrNO4Forma y color:SolidPeso molecular:400.22PDE4B-IN-3
<p>PDE4B-IN-3 is a potent inhibitor of PDE4B (IC50: 0.94 μM) and exhibits anti-inflammatory effects.</p>Fórmula:C30H35N3O4S2Forma y color:SolidPeso molecular:565.75ATR-IN-7
CAS:<p>ATR-IN-7 is a potent inhibitor of ATR.</p>Fórmula:C21H22FN7OForma y color:SolidPeso molecular:407.44Plumbemycin B
CAS:<p>Plumbemycin B is isolated from Streptomyces plumbeus; an L-threonine antagonist.</p>Fórmula:C12H21N4O8PForma y color:SolidPeso molecular:380.29Equisetin
CAS:<p>Equisetin: a QSI from Fusarium equiseti, curbs P. aeruginosa virulence, fights Gram-positive bacteria & HIV-1 integrase; not antibacterial to Gram-negative.</p>Fórmula:C22H31NO4Pureza:98%Forma y color:SolidPeso molecular:373.49Substituted piperidines-1
CAS:<p>Substituted piperidines-1 can promote the release of growth hormone in humans and animals.</p>Fórmula:C29H39N7O2Pureza:98%Forma y color:SolidPeso molecular:517.67CXCR2 antagonist 4
<p>CXCR2 antagonist 4 inhibits CXCR2 (IC50: 0.13 μM) and CXCL8-induced calcium rise (IC50: 27 μM), promising for cancer research.</p>Fórmula:C15H14F2N4OS2Forma y color:SolidPeso molecular:368.42
