Inhibidores
Los inhibidores son moléculas que se unen a enzimas, receptores u otras proteínas para reducir o bloquear su actividad biológica. Estos compuestos se utilizan ampliamente en la investigación para estudiar vías biológicas, comprender los mecanismos de las enfermedades y desarrollar fármacos terapéuticos. Los inhibidores desempeñan un papel crucial en el tratamiento de diversas enfermedades, incluyendo el cáncer, las enfermedades cardiovasculares y las infecciones. En CymitQuimica, ofrecemos una amplia gama de inhibidores de alta calidad para apoyar su investigación en bioquímica, biología celular y desarrollo farmacéutico.
Subcategorías de "Inhibidores"
- Angiogénesis(2.797 productos)
- Apoptosis(6.275 productos)
- Ciclo celular / Checkpoint(4.805 productos)
- Cromatina / Epigenética(2.462 productos)
- Señalización citoesquelética(1.534 productos)
- Daño al ADN / Reparación del ADN(2.959 productos)
- Endocrinología / Hormonas(3.708 productos)
- Enzima(3.670 productos)
- GPCR / proteína G(9.020 productos)
- Inmunología e inflamación(3.884 productos)
- Virus de la gripe(301 productos)
- Señalización JAK / STAT(414 productos)
- Señalización MAPK(1.249 productos)
- Transportador de membrana / canal de iones(3.050 productos)
- Metabolismo(10.206 productos)
- Microbiología / Virología(7.612 productos)
- Neurociencia(10.379 productos)
- Otros inhibidores(36.012 productos)
- Reducción de oxidación(42 productos)
- Señalización PI3K / Akt / mTOR(1.442 productos)
- Proteasas / Proteasoma(1.724 productos)
- Células madre y Derivados(819 productos)
- Tirosina quinasa / adaptadores(2.035 productos)
- Ubiquitinación(1.718 productos)
Mostrar 16 subcategorías más
Se han encontrado 66683 productos de "Inhibidores"
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UCB-35440
CAS:UCB-35440, a 5-lipoxygenase inhibitor and a histamine H1 receptor antagonist, is used potentially for the treatment of dermatitis.Fórmula:C31H34ClN5O4Forma y color:SolidPeso molecular:576.09UU-T01
CAS:UU-T01 inhibits β-catenin/Tcf4 with Ki of 3.14 µM, binds β-catenin directly with KD of 0.531 µM.Fórmula:C10H10N6OForma y color:SolidPeso molecular:230.23GRL-8234
CAS:GRL-8234 is a small-molecule BACE1 inhibitor that reverses memory impairments and age-related cognitive decline.Fórmula:C36H42N4O6SForma y color:SolidPeso molecular:658.81Haloxyfop-P-methyl
CAS:Haloxyfop-P-methyl, an aryloxyphenoxypropionate herbicide, is absorbed through both foliage and roots, where it inhibits lipogenesis and induces oxidativeFórmula:C16H13ClF3NO4Forma y color:SolidPeso molecular:375.73ICMT-IN-15
CAS:ICMT-IN-15 (compound 51) serves as an ICMT inhibitor with an IC50 value of 0.032 μM [1].Fórmula:C21H25ClFNOForma y color:SolidPeso molecular:361.88PF3845yne
CAS:PF3845yne is an alkyne analogue of PF-3845 maintaining high potency for FAAH.Fórmula:C25H24N4O2Forma y color:SolidPeso molecular:412.48Antibacterial agent 94
CAS:Compound 5b, an antibacterial, effectively targets MRSA and disrupts bacterial membranes and PG synthesis.Fórmula:C21H21FO4Forma y color:SolidPeso molecular:356.39Mansonone F
CAS:Mansonone F is a topoisomerase II inhibitor with cytotoxic and topo inhibitory potencies.Fórmula:C15H12O3Forma y color:SolidPeso molecular:240.25KNI-272
CAS:Kynostatin-272 is a HIV protease inhibitor. KNI-272 blocked the maturation of viral particles.Fórmula:C33H41N5O6S2Forma y color:SolidPeso molecular:667.84Diazoketone methotrexate
CAS:Diazoketone methotrexate is an analog of methotrexate with potential antitumor activity.Fórmula:C21H22N10O4Forma y color:SolidPeso molecular:478.46Esterbut-6
CAS:Esterbut-6 is a potent tumor cell proliferation inhibitor in vivo by stabilizes butyric acid.Fórmula:C13H22O7Pureza:98%Forma y color:SolidPeso molecular:290.31VU0029251
CAS:VU0029251 serves as a partial antagonist of mGluR5, exhibiting a binding affinity with a K i of 1.07 μM.Fórmula:C10H11N3S2Forma y color:SolidPeso molecular:237.34Proteasome-IN-5
CAS:<p>Proteasome-IN-5, also known as compound 5, acts as a proteasome inhibitor [1].</p>Fórmula:C20H30BN5O7Pureza:98%Forma y color:SolidPeso molecular:463.29A-424274
CAS:A-424274 is a positive allosteric modulator of α4β2 neuronal nicotinic receptor.Fórmula:C14H15N3Pureza:98%Forma y color:SolidPeso molecular:225.29TLR9-IN-1
CAS:TLR9-IN-1: selective, potent human TLR9 inhibitor (IC50: 7 nM), useful for researching immune-related diseases.Fórmula:C23H31N7OForma y color:SolidPeso molecular:421.54(3S,4S)-Tivantinib
CAS:(3S,4S)-Tivantinib, a potent and highly selective inhibitor of the receptor tyrosine kinase c-MET, targets GSK3α and GSK3β—two novel enzymes implicated in theFórmula:C23H19N3O2Forma y color:SolidPeso molecular:369.42GR-92549
CAS:GR-92549 is an HMG-CoA reductase inhibitor.Fórmula:C25H26F2N2O4Forma y color:SolidPeso molecular:456.48ent-Abacavir
CAS:ent-Abacavir, enantiomer of an anti-HIV carbocyclic nucleoside RT inhibitor, is metabolized in the liver, forms active CBV-TP.Fórmula:C14H18N6OForma y color:SolidPeso molecular:286.33MC-Val-Cit-PAB-NH-C2-NH-Boc
CAS:MC-Val-Cit-PAB-NH-C2-NH-Boc is a cathepsin-cleavable ADC linker utilized in constructing antibody-drug conjugates (ADCs) [1].Fórmula:C36H54N8O10Forma y color:SolidPeso molecular:758.86SHP2-IN-21
CAS:SHP2-IN-21 (compound 208) is an inhibitor of SHP2, exhibiting an IC50 of 3 nM, and is utilized in glioblastoma research [1].Fórmula:C27H26FN7Forma y color:SolidPeso molecular:467.54L-AP4
CAS:L-APB is an effective and specific agonist for the group III mGluRs (EC50s: 0.13, 0.29, 1.0, 249 μM for mGlu4, mGlu8, mGlu6, and mGlu7 receptors, respectively).Fórmula:C4H10NO5PPureza:98%Forma y color:White To Off-White Crystalline PowderPeso molecular:183.1ASGPR ligand-1
CAS:ASGPR ligand-1 is a compound that targets the asialoglycoprotein receptor (ASGPR) and is utilized in various disease research contexts [1].Fórmula:C61H110N10O27Forma y color:SolidPeso molecular:1415.58CH-5137291
CAS:CH-5137291 is a pure AR antagonist with AR nuclear translocation inhibition activity. It suppresses castration and prevents the growth of prostate cancer cells.Fórmula:C18H14F3N5O3S2Forma y color:SolidPeso molecular:469.46GSK321
CAS:GSK321 is an IDH1 inhibitor that prevents cytoplasmic glutamine reductive carboxylation.GSK321 is used in the study of leukemia.Fórmula:C28H28FN5O3Pureza:99.73%Forma y color:SolidPeso molecular:501.55S-Me-DM4
CAS:S-Me-DM4 is an intracellular enzyme S-methylated metabolite of DM4, a maytansinoid with microtubule-depolymerizing properties and potent cytotoxicity, employedFórmula:C39H56ClN3O10SForma y color:SolidPeso molecular:794.39FASN-IN-1
CAS:FASN-in-1 is an effective, specific inhibitor of fatty acid synthase (FASN), a compound specifically designed to target and inhibit the activity of the enzymeFórmula:C18H25N3O3S2Pureza:99.92% - >99.99%Forma y color:SolidPeso molecular:395.54SARS-CoV-2-IN-63
CAS:SARS-CoV-2-IN-63 (Compound R3e) serves as an inhibitor of SARS-CoV-2 replication, demonstrating low cytotoxicity.Fórmula:C20H21N3O3SePureza:98%Forma y color:SolidPeso molecular:430.36MLN-0415
CAS:MLN-0415 is an IKK2 inhibitor which decreases NF-κB activation and down-regulates the expression of a number of inflammatory proteins.Fórmula:C26H32ClN5O4Forma y color:SolidPeso molecular:514.02IIIM-290
CAS:IIIM-290 is an oral CDK inhibitor (IC50s: 90 and 94 nM for CDK2/A and CDK9/T1).Fórmula:C23H21Cl2NO5Pureza:98%Forma y color:SolidPeso molecular:462.32ABP 25
CAS:ABP 25 is a highly potent and selective activity-based probe (ABP) for cathepsin K imaging.Fórmula:C55H66ClN5O3Forma y color:SolidPeso molecular:880.6R1498
CAS:<p>R1498 inhibits CDK2, targets angiogenesis and mitosis, and is an oral treatment for liver and stomach cancer.</p>Fórmula:C18H15ClN4OPureza:98%Forma y color:SolidPeso molecular:338.79Ponicidin
CAS:Ponicidin, a diterpenoid from Rabdosia rubescens, has immunoregulatory, anti-inflammatory, anti-viral, and anti-cancer properties.Fórmula:C20H26O6Pureza:98.98% - 99.92%Forma y color:SolidPeso molecular:362.42Integrin Antagonists 27
CAS:Integrin Antagonists 27 is a small molecule integrin αvβ3 antagonist. It has a binding affinity of 18 nM and as a novel anticancer agent.Fórmula:C24H20N4O5Forma y color:SolidPeso molecular:444.44MDL-19744A
CAS:MDL-19744A is an alpha 1-adrenergic receptor antagonist and renal vasodilator.Fórmula:C21H25NO3SForma y color:SolidPeso molecular:371.49Macimorelin acetate
CAS:Macimorelin acetate (EP-1572) is an oral GHSR agonist for AGHD and CACS research.Fórmula:C28H34N6O5Forma y color:SolidPeso molecular:534.61Brevicompanine B
CAS:Brevicompanine B: fungal metabolite, regulates plant growth/circadian rhythm, inhibits Arabidopsis roots, affects gene transcription, anti-P. falciparum.Fórmula:C22H29N3O2Forma y color:SolidPeso molecular:367.48Unguisin A
CAS:Unguisin A is a cyclic peptide isolated from the marine-derived fungus Emericella unguis [1].Fórmula:C40H54N8O7Forma y color:SolidPeso molecular:758.91LG 83-6-05
CAS:LG 83-6-05 is a novel kind of sodium channel blocking agent.Fórmula:C21H30ClNO3SForma y color:SolidPeso molecular:411.99COH1
CAS:COH1 is a ribonucleotide reductase (RR) inhibitor utilized in research pertaining to cancer, mitochondrial diseases, and neurodegenerative disorders [1].Fórmula:C11H10N2O3SPureza:98%Forma y color:SolidPeso molecular:250.27SREBP/SCAP-IN-2
CAS:SREBP/SCAP-IN-2 (compound 13) acts as a selective inhibitor of SREBP/SCAP [1].Fórmula:C27H37ClF2N4OForma y color:SolidPeso molecular:507.06ASP-8497
CAS:ASP8497 is a potent DPP-IV inhibitor enhancing GLP-1, used for type 2 diabetes and glucose intolerance.Fórmula:C18H27FN4O7SForma y color:SolidPeso molecular:462.49OSMI-1
CAS:OSMI-1: cell-permeable OGT inhibitor, blocks O-GlcNAcylation (IC50: 2.7 μM), no effect on other cell glycans.Fórmula:C28H25N3O6S2Pureza:96.79% - 99.39%Forma y color:SolidPeso molecular:563.64Ref: TM-T16409
1mg40,00€2mg52,00€5mg85,00€10mg124,00€25mg197,00€50mg350,00€100mg522,00€1mL*10mM (DMSO)96,00€Iganidipine
CAS:Iganidipine（NKY 722） is a new water-soluble Ca2+ antagonist with antihypertensive activity for research and neurological related diseases.Fórmula:C28H38N4O6Pureza:96.3%Forma y color:SolidPeso molecular:526.62Sophorose
CAS:Sophorose, a disaccharide within sophorolipids synthesized by yeast, functions as a biosurfactant owing to its hydrophobic properties.Fórmula:C12H22O11Forma y color:SolidPeso molecular:342.3PF-06733804
CAS:PF-06733804 is a potent inhibitor of pan-Trk in cell-based assays (IC50s: 8.4 nM, 6.2 nM, and 2.2 nM for TrkA, TrkB, and TrkC) with anti-hyperalgesic effect.Fórmula:C20H19F5N4O4Pureza:98%Forma y color:SolidPeso molecular:474.38Activated DPG Subunit
CAS:Activated DPG subunit facilitates the synthesis of exon jumping oligomer conjugates targeting specific sites within the human anti-muscular atrophy protein geneFórmula:C51H53ClN7O7PForma y color:SolidPeso molecular:942.44Antitumor agent-93
CAS:Antitumor agent-93 (compound 7D) effectively inhibits the proliferation of multiple tumor cell lines, including MDA-MB-231 and HCT-116 [1].Fórmula:C22H20O8Forma y color:SolidPeso molecular:412.39TMC-649128
CAS:TMC-649128, a RNA polymerase NS5B inhibitor, is used for the treatment of HCV infection.Fórmula:C18H26N6O6Forma y color:SolidPeso molecular:422.44Deoxyharringtonine
CAS:Deoxyharringtonine, an alkaloid extracted from the Cephalotaxus genus, exhibits significant anti-leukemic properties [1].Fórmula:C28H37NO8Forma y color:SolidPeso molecular:515.6
