Inhibidores
Los inhibidores son moléculas que se unen a enzimas, receptores u otras proteínas para reducir o bloquear su actividad biológica. Estos compuestos se utilizan ampliamente en la investigación para estudiar vías biológicas, comprender los mecanismos de las enfermedades y desarrollar fármacos terapéuticos. Los inhibidores desempeñan un papel crucial en el tratamiento de diversas enfermedades, incluyendo el cáncer, las enfermedades cardiovasculares y las infecciones. En CymitQuimica, ofrecemos una amplia gama de inhibidores de alta calidad para apoyar su investigación en bioquímica, biología celular y desarrollo farmacéutico.
Subcategorías de "Inhibidores"
- Angiogénesis(2.797 productos)
- Apoptosis(6.275 productos)
- Ciclo celular / Checkpoint(4.805 productos)
- Cromatina / Epigenética(2.462 productos)
- Señalización citoesquelética(1.534 productos)
- Daño al ADN / Reparación del ADN(2.959 productos)
- Endocrinología / Hormonas(3.708 productos)
- Enzima(3.670 productos)
- GPCR / proteína G(9.020 productos)
- Inmunología e inflamación(3.884 productos)
- Virus de la gripe(301 productos)
- Señalización JAK / STAT(414 productos)
- Señalización MAPK(1.249 productos)
- Transportador de membrana / canal de iones(3.050 productos)
- Metabolismo(10.206 productos)
- Microbiología / Virología(7.612 productos)
- Neurociencia(10.379 productos)
- Otros inhibidores(36.012 productos)
- Reducción de oxidación(42 productos)
- Señalización PI3K / Akt / mTOR(1.442 productos)
- Proteasas / Proteasoma(1.724 productos)
- Células madre y Derivados(819 productos)
- Tirosina quinasa / adaptadores(2.035 productos)
- Ubiquitinación(1.718 productos)
Mostrar 16 subcategorías más
Se han encontrado 66683 productos de "Inhibidores"
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Spectramide
CAS:Spectramide is a dopamine D-2 receptor antagonist.Fórmula:C19H23ClIN3O2Forma y color:SolidPeso molecular:487.76Pristinamycin IA
CAS:Pristinamycin IA (Mikamycin B) is a substrate for the P-glycoprotein and a cyclo-peptidic macrolactone antibiotic.Fórmula:C45H54N8O10Pureza:97.44%Forma y color:SolidPeso molecular:866.96GABA-IN-2
CAS:GABA-IN-2 (Compound 5), a GABA inhibitor, exhibits both larvicidal and insecticidal properties, achieving an 87% mortality rate at a concentration of 50 mg/L [1Fórmula:C12H4Cl2F6N4SeForma y color:SolidPeso molecular:468.04GCC-4401C free base
CAS:GCC-4401C free base is a factor Xa inhibitor similar to rivaroxaban that is currently under development for venous thromboembolic disease (VTE).Fórmula:C18H18ClN5O3SForma y color:SolidPeso molecular:419.89KRIBB3
CAS:KRIBB3: novel anticancer microtubule inhibitor; halts MDA-MB-231 cell migration/invasion by targeting Hsp27 phosphorylation.Fórmula:C19H19NO4Forma y color:SolidPeso molecular:325.36Bcl-2-IN-11
CAS:Bcl-2-IN-11 (compound 6) is a potent and selective inhibitor of Bcl-2 activity, exhibiting an IC50 of 0.9 nM, and demonstrates minimal inhibition against Bcl-xlFórmula:C45H49ClFN7O8SForma y color:SolidPeso molecular:902.43ICI-M247496
CAS:ICI-M247496 is a non-polyglutamated analog of CB3717 and quinazoline-based inhibitor of thymidylate synthase.Fórmula:C19H16N4O3Forma y color:SolidPeso molecular:348.36Maropitant citrate anhydrous
CAS:Maropitant citrate anhydrous is a neurokinin (NK1) receptor antagonist.Fórmula:C38H48N2O8Forma y color:SolidPeso molecular:660.8JA-ACC
CAS:Jasmonyl-ACC (JA-ACC), a derivative of 1-aminocyclopropane-1-carboxylic acid (ACC)—the direct precursor to ethylene—impedes root growth in Arabidopsis, withFórmula:C16H23NO4Forma y color:SolidPeso molecular:293.36TMV-IN-4
CAS:TMV-IN-4, a TMV inhibitor, enhances plant defense and TMV resilience by interacting with helicase, increasing peroxidase and SOD activity.Fórmula:C18H21NO4Forma y color:SolidPeso molecular:315.36Streptovitacin A
CAS:Streptovitacin A boosts growth inhibition against fungi.Fórmula:C15H23NO5Pureza:98%Forma y color:SolidPeso molecular:297.35c-Met/MEK1/Flt-3-IN-1
Antiproliferative Against-3 (comp 33) demonstrates significant activity against Hela (IC 50 = 0.21 µM), A549 (IC 50 = 0.39 µM), and MCF-7 (IC 50 = 0.33 µM) cellFórmula:C39H37FN6O5Forma y color:SolidPeso molecular:688.75ICMT-IN-34
CAS:ICMT-IN-34 (compound 39) serves as an effective inhibitor of ICMT, exhibiting an IC50 value of 0.17 μM [1].Fórmula:C21H25Cl2NOForma y color:SolidPeso molecular:378.34WRNA10
CAS:WRNA10 is a potent binding agent for HIV-1TAR RNA (IC50: 10 μM, CC50: 40 μM).Fórmula:C25H32N4O4Forma y color:SolidPeso molecular:452.55CL2E-SN38
CAS:CL2E-SN-38 is a structurally stable and highly releasable antibody-drug conjugate (ADC) incorporating SN-38, the active metabolite of Irinotecan and a potentFórmula:C87H116N14O24Forma y color:SolidPeso molecular:1741.93Eugenitin
CAS:Eugenitin, a polyketide from Mycoleptodiscus indicus, exhibits inhibitory activity against Leishmania major with an LD50 of 39.9 μM and demonstrates lowFórmula:C12H12O4Pureza:98%Forma y color:SolidPeso molecular:220.22AS100
CAS:AS100 is a bioactive chemical.Fórmula:C23H24Cl3N7O4Forma y color:SolidPeso molecular:568.84PBI-1393
CAS:PBI-1393 can be used as an enhancer for Th1 type cytokine production and primary T cell activation.Fórmula:C19H31N9O4Forma y color:SolidPeso molecular:449.51O-2050
CAS:O-2050: strong CB1 antagonist (Ki 2.5 nM), CB2 inhibitor (Ki 0.2 nM); reduces mouse food intake, increases activity.Fórmula:C23H31NO4SPureza:98%Forma y color:SolidPeso molecular:417.56MK-287
CAS:MK-287 is a PAF antagonist blocking [3H]C18-PAF binding to platelets, PMNs, and lungs; may treat asthma.Fórmula:C25H34O9SForma y color:SolidPeso molecular:510.6HDAC-IN-50
CAS:HDAC-IN-50, a potent FGFR/HDAC inhibitor (IC50: 0.18-13 nM), induces apoptosis, cell cycle arrest, and shows anti-tumor activity.Fórmula:C31H41N7O4Forma y color:SolidPeso molecular:575.7Levuglandin E2
CAS:Levuglandin E2 is a secoprostanoid from prostaglandin endoperoxide.Fórmula:C20H32O5Forma y color:SolidPeso molecular:352.47DNA-PK-IN-10
CAS:DNA-PK-IN-10 is a DNA-PK inhibitor utilized in the research of breast cancer and non-small cell lung cancer [1].Fórmula:C25H28N6O2Pureza:98%Forma y color:SolidPeso molecular:444.53PF-06260414
CAS:PF-06260414 is a selective androgen receptor modulator or SARM used to treat muscle weakness.Fórmula:C14H14N4O2SForma y color:SolidPeso molecular:302.35FLT3-IN-14
CAS:FLT3-IN-14: FLT3 inhibitor; FLT3-WT IC50=5.6nM, FLT3-ITD IC50=1.4nM; blocks Y591 phosphorylation; G1 arrest; pro-apoptotic.Fórmula:C25H24N6O2SForma y color:SolidPeso molecular:472.56RK-0133114
RK-0133114, R-enantiomer of RK-701, is a G9a inhibitor (IC50 = 3.7 μM) for SCD research.Fórmula:C26H30N4O3Forma y color:SolidPeso molecular:446.54AMOR
CAS:AMOR is unique to plant cell walls and enhances plant fertilization efficiency and capacityFórmula:C13H22O12Forma y color:SolidPeso molecular:370.31Glibornuride
CAS:Glibornuride is a blocker of ATP-sensitive K+ channel(pKi: 5.75).Fórmula:C18H26N2O4SPureza:99.5%Forma y color:SolidPeso molecular:366.48Ref: TM-T15385
1mg71,00€5mg152,00€10mg236,00€25mg409,00€50mg580,00€100mg803,00€1mL*10mM (DMSO)167,00€Difethialone
CAS:Difethialone is an anticoagulant rodenticide and a vitamin K antagonist.Fórmula:C31H23BrO2SForma y color:SolidPeso molecular:539.48Glucocorticoid receptor agonist-2 Ala-Ala-Mal
CAS:Glucocorticoid receptor agonist-2 Ala-Ala-Mal (compound 79) serves as a precursor for synthesizing anti-inflammatory antibody-drug conjugate (ADC) molecules andFórmula:C47H50F2N4O12Forma y color:SolidPeso molecular:900.92Isoacitretin
CAS:Isoacitretin is an oral retinoid effective and can be used to treat psoriasis.Fórmula:C21H26O3Forma y color:SolidPeso molecular:326.43DGKα-IN-3
CAS:DGKα-IN-3 (example 25), with an IC50 of 283 nM, is a selective DGKα inhibitor that augments anti-PD-1's anti-tumor activity by promoting T cell proliferationFórmula:C26H27F3N4O3Forma y color:SolidPeso molecular:500.51TH-Z145
CAS:TH-Z145 is a potent FPPS inhibitor for the study of myeloma and lung cancer.Fórmula:C16H28O7P2Pureza:98.29%Forma y color:SolidPeso molecular:394.34Ref: TM-T73450
1mg52,00€5mg103,00€10mg169,00€25mg338,00€50mg543,00€100mg868,00€1mL*10mM (DMSO)114,00€BU-E 75
CAS:BU-E 75 is an agonist of the histamine H2.Fórmula:C21H24F2N6Forma y color:SolidPeso molecular:398.45(S)-Cdc7-IN-18
CAS:'(S)-Cdc7-IN-18 from patent WO2020239107A1 inhibits CDC7, curbing MCM2 and tumor growth.'Fórmula:C19H21N5OSForma y color:SolidPeso molecular:367.47A 56234
CAS:A 56234 is a high-ceiling diuretic.Fórmula:C16H9ClFKNO4Forma y color:SolidPeso molecular:372.8AAK1-IN-4
CAS:AAK1-IN-4 selectively inhibits AAK1 with IC50 of 4.6 nM; penetrates CNS, oral bioactive, potential for studying neuropathic pain.Fórmula:C20H28N4O3Forma y color:SolidPeso molecular:372.46ATI-22-107
CAS:ATI-22-107 is a positive cardiac inotropic agent which may affect myocyte calcium cycling and contractility.Fórmula:C31H32Cl2N4O8Forma y color:SolidPeso molecular:659.51TRPC5 modulator-1
CAS:TRPC5 modulator-1 (Compound 9) is a TRPC5 modulator (IC50<1 nM) that can be used to study neuropsychiatric disorders.Fórmula:C23H27FN2O4Forma y color:SolidPeso molecular:414.47DU172
CAS:DU172 is the tyrosine-targeted covalent adenosine A1 receptor antagonist.Fórmula:C24H30FN5O5SForma y color:SolidPeso molecular:519.59DDR1/2 inhibitor-2
CAS:DDR1/2 Inhibitor-2 (Example 31) serves as an inhibitor of DDR1/DDR2, exhibiting IC50 values below 100 nM.Fórmula:C25H19F3N6O2Forma y color:SolidPeso molecular:492.45VT-1598 tosylate
CAS:VT-1598 tosylate is a selective, orally active antifungal compound that targets CYP51. It demonstrates efficacy against C. auris.Fórmula:C38H28F4N6O5SForma y color:SolidPeso molecular:756.72AMG151 HCl
CAS:ARRY-403 (AMG-151) is an oral glucokinase activator for type 2 diabetes with an EC50 of 79 nM and favorable drug properties.Fórmula:C20H20Cl2N6O3S2Forma y color:SolidPeso molecular:527.439Amauromine
CAS:Amauromine is a peripherally selective and potent cannabinoid receptor type 1 (CB1) receptor antagonist, a novel alkaloid with vasodilatory activity.Fórmula:C32H36N4O2Forma y color:SolidPeso molecular:508.65Dezapelisib
CAS:Dezapelisib, an oral delta PI3K inhibitor, blocks PIP3 production and PI3K/AKT pathway, hindering tumor cell growth and survival.Fórmula:C20H16FN7OSForma y color:SolidPeso molecular:421.45BD-AcAc 2
CAS:BD-AcAc 2 (Ketone Ester) is a ketone monoester and can be used as a source of oral nutritional ketones.Fórmula:C8H16O4Pureza:99.62%Forma y color:SolidPeso molecular:176.21HSP70/SIRT2-IN-2
CAS:<p>HSP70/SIRT2-IN-2 (Compounds 1a), a dual inhibitor of SIRT2 and HSP70, exhibits an IC50 of 45.1±5.0 μM against SIRT2 and demonstrates antitumor activity [1].</p>Fórmula:C17H13N3S3Pureza:98%Forma y color:SolidPeso molecular:355.5CD73-IN-4
CAS:CD73-IN-4 is a potent and selective methylenephosphonic acid CD73 inhibitorFórmula:C16H23ClN5O7PPureza:98.61%Forma y color:SolidPeso molecular:463.81Ref: TM-T9210
1mg97,00€5mg243,00€10mg393,00€25mg702,00€50mg938,00€100mg1.320,00€1mL*10mM (DMSO)245,00€uPSEM 817 tartrate
CAS:Potent α7L-GlyR & PSAM4-5-HT3 agonist (EC50: 0.3/0.5 nM). Reduces cortical neuron activity; induces contralateral rotation in mice (LED 0.1 mg/kg).Fórmula:C20H25N3O7Forma y color:SolidPeso molecular:419.434
