Inhibidores
Los inhibidores son moléculas que se unen a enzimas, receptores u otras proteínas para reducir o bloquear su actividad biológica. Estos compuestos se utilizan ampliamente en la investigación para estudiar vías biológicas, comprender los mecanismos de las enfermedades y desarrollar fármacos terapéuticos. Los inhibidores desempeñan un papel crucial en el tratamiento de diversas enfermedades, incluyendo el cáncer, las enfermedades cardiovasculares y las infecciones. En CymitQuimica, ofrecemos una amplia gama de inhibidores de alta calidad para apoyar su investigación en bioquímica, biología celular y desarrollo farmacéutico.
Subcategorías de "Inhibidores"
- Angiogénesis(2.797 productos)
- Apoptosis(6.275 productos)
- Ciclo celular / Checkpoint(4.805 productos)
- Cromatina / Epigenética(2.462 productos)
- Señalización citoesquelética(1.534 productos)
- Daño al ADN / Reparación del ADN(2.959 productos)
- Endocrinología / Hormonas(3.708 productos)
- Enzima(3.670 productos)
- GPCR / proteína G(9.020 productos)
- Inmunología e inflamación(3.884 productos)
- Virus de la gripe(301 productos)
- Señalización JAK / STAT(414 productos)
- Señalización MAPK(1.249 productos)
- Transportador de membrana / canal de iones(3.050 productos)
- Metabolismo(10.206 productos)
- Microbiología / Virología(7.612 productos)
- Neurociencia(10.379 productos)
- Otros inhibidores(36.012 productos)
- Reducción de oxidación(42 productos)
- Señalización PI3K / Akt / mTOR(1.442 productos)
- Proteasas / Proteasoma(1.724 productos)
- Células madre y Derivados(819 productos)
- Tirosina quinasa / adaptadores(2.035 productos)
- Ubiquitinación(1.718 productos)
Mostrar 16 subcategorías más
Se han encontrado 66683 productos de "Inhibidores"
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cis-9,10-Epoxystearic acid
CAS:cis-9,10-Epoxystearic acid (cis-9,10-Epoxyoctadecanoic acid) is an endogenous component in human urine and blood and can be produced from oleic acid by enzymicFórmula:C18H34O3Pureza:99.93%Forma y color:SolidPeso molecular:298.46ICI-185282
CAS:ICI-185282 is a potent thromboxane receptor antagonist.Fórmula:C18H21F3O5Forma y color:SolidPeso molecular:374.35Glucagon receptor antagonists-3
CAS:Glucagon receptor antagonist -3 is a highly effective glucagon receptor antagonist.Fórmula:C22H30FNO2Pureza:98%Forma y color:SolidPeso molecular:359.48Sardomozide
CAS:Sardomozide is an inhibitor of S-adenosylmethionine decarboxylase (SAMDC)(IC50 of 5 nM).Fórmula:C11H14N6Pureza:98%Forma y color:SolidPeso molecular:230.27Homouridine
CAS:Homouridine, an analogue of uridine, functions as an intermediate in the synthesis of MMP-2 inhibitor (compound I, IC50 = 150 μM).Fórmula:C10H14N2O6Pureza:98%Forma y color:SolidPeso molecular:258.23Rac1-IN-3
CAS:Rac1-IN-3 (Compound 2) is a Rac1 inhibitor exhibiting an inhibitory concentration 50 (IC50) of 46.1 μM [1].Fórmula:C21H23N7O2Pureza:98%Forma y color:SolidPeso molecular:405.45SOS1-IN-16
CAS:SOS1-IN-16 (Comp 54) serves as a selective SOS1 inhibitor exhibiting an IC50 value of 7.2 nM and demonstrates inhibitory activity against CYP3A4 with an IC50 ofFórmula:C30H31F3N4O3Pureza:98%Forma y color:SolidPeso molecular:552.59Durlobactam
CAS:<p>Durlobactam is a drug candidate for beta-lactamase inhibitor.</p>Fórmula:C8H11N3O6SForma y color:SolidPeso molecular:277.25BT424
CAS:BT424, a specific HCK inhibitor, modulates macrophage activation and autophagy in vitro, and mitigates inflammation and renal fibrosis in the UUO model [1].Fórmula:C22H15BCl2N2O2Pureza:98%Forma y color:SolidPeso molecular:421.08Lifirafenib
CAS:Lifirafenib (Beigene-283) is a potent inhibitor of RAF family kinases and EGFR in biochemical assays with IC50 of 23, 29 and 495 nM for the recombinantFórmula:C25H17F3N4O3Pureza:97.99% - 98%Forma y color:SolidPeso molecular:478.42Ref: TM-T22272
1mg35,00€5mg69,00€10mg97,00€25mg190,00€50mgA consultar100mgA consultar1mL*10mM (DMSO)89,00€Nurr1 agonist 7
CAS:Nurr1 agonist 7 is an agonist of Nurr1 (EC50: 0.12 μM), which can be used to study neurological disorders such as Parkinson's disease.Fórmula:C18H20O3Pureza:99.79%Forma y color:SolidPeso molecular:284.35RSV L-protein-IN-2
CAS:RSV L-protein-IN-2 (Compound A), a noncompetitive inhibitor of the RSV polymerase (IC50: 4.5 μM), exhibits antiviral activity against long RSV strains (EC50: 1.Fórmula:C32H36N4O5Pureza:98%Forma y color:SolidPeso molecular:556.65NLRP3-IN-22
CAS:NLRP3-IN-22 (Compound II-4) is an inhibitor of NLRP3, exhibiting a 67% inhibition rate at a concentration of 10 μM [1].Fórmula:C19H12F3NO4SPureza:98%Forma y color:SolidPeso molecular:407.36Glucocorticoid receptor agonist
CAS:Glucocorticoid receptor agonist is an effective glucocorticoid receptor agonist.Fórmula:C20H20F4N2O2Pureza:98%Forma y color:SolidPeso molecular:396.38JNJ-17148066
CAS:JNJ-17148066 is an agonist of estrogen receptor ESR1.Fórmula:C30H31NO5Pureza:98%Forma y color:SolidPeso molecular:485.57MTPG
CAS:Group II/group III metabotropic glutamate receptor antagonistFórmula:C10H11N5O2Pureza:98%Forma y color:SolidPeso molecular:233.23Laxiflorin B
CAS:Laxiflorin B, a novel selective inhibitor of ERK 1/2 derived from herbal sources, exhibits antitumor activity [1].Fórmula:C20H24O5Pureza:98%Forma y color:SolidPeso molecular:344.4CLR-131
CAS:CLR-131, a protein kinase B (PKB) inhibitor, is used potentially for the treatment of non small cell lung cancer, solid tumors.Fórmula:C29H53INO4PPureza:98%Forma y color:SolidPeso molecular:641.62β3-AR agonist 2
CAS:β3-AR agonist 2 is a potent and selective agonist of β3-adrenergic receptor (β3-AR with an EC50 of 8 nM).Fórmula:C27H38N4O7SPureza:98%Forma y color:SolidPeso molecular:562.68Ethylene dimethanesulfonate
CAS:Ethylene dimethanesulfonate has selective pro-apoptotic effects on LCs. Ethylene dimethanesulfonate is a mild alkylating, non-volatile methanesulfonic diesterFórmula:C4H10O6S2Pureza:98.94%Forma y color:SolidPeso molecular:218.25Obestatin(rat) TFA
CAS:<p>Obestatin(rat) TFA, a 23-amino-acid peptide, modulates appetite, gut motility, and body weight; binds GPR39; has anti-inflammatory and antioxidant effects.</p>Fórmula:C116H175F3N34O33Forma y color:SolidPeso molecular:2630.83Trithiozine
CAS:Trithiozine is used in peptic ulcer and hypersecretory disorder research for its antiulcer and antisecretory properties.Fórmula:C14H19NO4SPureza:90% - 99.47%Forma y color:SolidPeso molecular:297.37ROCK2-IN-7
CAS:<p>ROCK2 inhibitor is a chemical compound associated with the therapeutic management of psoriasis.</p>Fórmula:C26H28FN5OPureza:98%Forma y color:SolidPeso molecular:445.53AR234960
CAS:AR234960, also known GTPL7039, is an active biochemical.Fórmula:C27H30FN5O5SForma y color:SolidPeso molecular:555.62GLUT4 activator 1
CAS:GLUT4 activator 1 is a potent glucose transporter type 4 (GLUT4) translocation activator (EC50: 0.14 μM).Fórmula:C23H21FN4O3SPureza:98%Forma y color:SolidPeso molecular:452.5Cathepsin Inhibitor 2
CAS:Cathepsin Inhibitor 2 is a potent Cathepsin S inhibitor (Ki: <20 nM).Fórmula:C19H21F6N3OPureza:98%Forma y color:SolidPeso molecular:421.38GSK2188764
CAS:GSK2188764 is an inhibitor of T. brucei IPMK, partially inhibits rTbIPMK activity.Fórmula:C17H16Cl2N6OPureza:98%Forma y color:SolidPeso molecular:391.25AXL-IN-15
CAS:AXL-IN-15 (cpd391) is a potent inhibitor of Axl, exhibiting both a dissociation constant (K i) and a half-maximal inhibitory concentration (IC50) of less than 1Fórmula:C26H32F3N9O3Pureza:98%Forma y color:SolidPeso molecular:575.59HIV-1 protease-IN-11
CAS:HIV-1 protease-IN-11 (compound 34a), an HIV-1 protease inhibitor, demonstrates potent inhibition with an IC50 of 0.41 nM and maintains substantial efficacyFórmula:C26H37N3O5SPureza:98%Forma y color:SolidPeso molecular:503.65Androgen receptor degrader-1
CAS:Androgen Receptor Degrader-1 (Compound 18) is a potent agent for androgen receptor degradation, applicable in cancer research [1].Fórmula:C15H14ClN3O4Pureza:98%Forma y color:SolidPeso molecular:335.74JNK3 inhibitor-3
CAS:JNK3 Inhibitor-3 selectively blocks JNK3 (>4.1 nM), crosses the blood-brain barrier, is orally active, and improves memory in dementia mice.Fórmula:C26H25N7O2Pureza:98%Forma y color:SolidPeso molecular:467.52A-371191
CAS:A-371191 is an antagonist of Bcl-XL.Fórmula:C36H47N5O5S2Pureza:98%Forma y color:SolidPeso molecular:693.92BAY-204
CAS:BAY-204 is a CSNK1α/δ inhibitor that can be used in the treatment of proliferative diseases.Fórmula:C29H26F3N5O2Forma y color:SolidPeso molecular:533.54MI-219
CAS:MI-219 is a human double minute 2 (HDM2) inhibitor.Fórmula:C27H32Cl2FN3O4Forma y color:SolidPeso molecular:552.47Risvodetinib
CAS:Risvodetinib: potent inhibitor of protein tyrosine kinases c-Abl1, c-Abl2, and c-kit.Fórmula:C33H34N8O2Forma y color:SolidPeso molecular:574.68BMS-317180
CAS:BMS-317180 is a potent, orally active GHS with a great safety profile in preclinical studies, now in clinical development.Fórmula:C21H33N7O5Forma y color:SolidPeso molecular:463.53BMS-830216
CAS:BMS-830216 is a nonbasic melanin hormone receptor 1 antagonist and a prodrug of BMS-819881.Fórmula:C24H22ClN2O7PSForma y color:SolidPeso molecular:548.93O-1057 free base
CAS:O-1057 free base is a water-soluble cannabinoid receptor agonist with antinociceptive properties. RESEARCH USE ONLY.Fórmula:C32H46N2O4Forma y color:SolidPeso molecular:522.72KRAS G12C inhibitor 35
CAS:KRAS G12C inhibitor 35 targets KRAS G12C in cancer research (CN112920183A, compound 3).Fórmula:C31H27ClF2N6O3Forma y color:SolidPeso molecular:605.03HBV-IN-30
CAS:HBV-IN-30, a flavone derivative, inhibits cccDNA in HBV research.Fórmula:C22H18BrClO6Forma y color:SolidPeso molecular:493.73CAY10748
CAS:CAY10748: STING agonist, IC50=0.3794μM, activates STING-pathway, boosts IFN-β/CXCL10/IL-6, inhibits CT26 tumor growth at 0.15mg/kg.Fórmula:C30H37N7O6Forma y color:SolidPeso molecular:591.66Dolastatinol
CAS:Dolastatinol, a synthetic analog of Dolastatin 10, serves as a potent low-nanomolar inhibitor of tubulin polymerization.Fórmula:C43H70N6O7SForma y color:SolidPeso molecular:815.12PD 109488
CAS:PD 109488 is a metabolite of quinapril and is a derivative of Quinapril that acts as an ACE inhibitor.Fórmula:C25H28N2O4Pureza:98%Forma y color:SolidPeso molecular:420.5NaV1.7 Blocker-801
CAS:NaV1.7 Blocker-801 is a potent NaV1.7 blocker.Fórmula:C20H15ClF2N6O3S2Forma y color:SolidPeso molecular:524.95ONO-8539
CAS:ONO-8539 is a prostanoid EP1 receptor antagonist.Fórmula:C25H28N2O5S2Forma y color:SolidPeso molecular:500.63Lotrafiban hydrochloride
CAS:Lotrafiban hydrochloride is an platelet glycoprotein IIb/IIIa blocker with oral activity.Fórmula:C23H33ClN4O4Forma y color:SolidPeso molecular:464.99KW-7158
CAS:KW-7158, a potassium channel activator, is used potentially for the treatment of urinary urgency and frequency.Fórmula:C16H12F3NO5S2Forma y color:SolidPeso molecular:419.42-Furoyl-LIGRLO-amide TFA
CAS:2-Furoyl-LIGRLO-amide TFA is a potent and selective agonist of the proteinase-activated receptor 2 (PAR2), exhibiting a pD2 value of 7.0 [1] [2].Fórmula:C38H64F3N11O10Forma y color:SolidPeso molecular:891.98Lysyl-aspartyl-glutamyl-leucine
CAS:Lysyl-aspartyl-glutamyl-leucine maintains type II surface membrane proteins in the endoplasmic reticulum.Fórmula:C21H37N5O9Forma y color:SolidPeso molecular:503.55
