Inhibidores
Los inhibidores son moléculas que se unen a enzimas, receptores u otras proteínas para reducir o bloquear su actividad biológica. Estos compuestos se utilizan ampliamente en la investigación para estudiar vías biológicas, comprender los mecanismos de las enfermedades y desarrollar fármacos terapéuticos. Los inhibidores desempeñan un papel crucial en el tratamiento de diversas enfermedades, incluyendo el cáncer, las enfermedades cardiovasculares y las infecciones. En CymitQuimica, ofrecemos una amplia gama de inhibidores de alta calidad para apoyar su investigación en bioquímica, biología celular y desarrollo farmacéutico.
Subcategorías de "Inhibidores"
- Angiogénesis(2.542 productos)
- Apoptosis(5.816 productos)
- Ciclo celular / Checkpoint(4.466 productos)
- Cromatina / Epigenética(2.252 productos)
- Señalización citoesquelética(1.381 productos)
- Daño al ADN / Reparación del ADN(2.830 productos)
- Endocrinología / Hormonas(3.518 productos)
- Enzima(3.640 productos)
- GPCR / proteína G(8.362 productos)
- Inmunología e inflamación(3.540 productos)
- Virus de la gripe(296 productos)
- Señalización JAK / STAT(405 productos)
- Señalización MAPK(1.201 productos)
- Transportador de membrana / canal de iones(2.809 productos)
- Metabolismo(9.462 productos)
- Microbiología / Virología(7.003 productos)
- Neurociencia(9.942 productos)
- Otros inhibidores(37.827 productos)
- Reducción de oxidación(40 productos)
- Señalización PI3K / Akt / mTOR(1.399 productos)
- Proteasas / Proteasoma(1.598 productos)
- Células madre y Derivados(830 productos)
- Tirosina quinasa / adaptadores(2.012 productos)
- Ubiquitinación(1.651 productos)
Mostrar 16 subcategorías más
Se han encontrado 66618 productos de "Inhibidores"
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c-Myc inhibitor 8
CAS:<p>c-Myc inhibitor 8 suppresses cell growth in various cancers and is used in research.</p>Fórmula:C19H12BrClF3NO3S2Forma y color:SolidPeso molecular:538.79Adapiprazine
CAS:<p>Adapiprazine is prochlorperazine that works as an anesthetic drug.</p>Fórmula:C29H36ClN3SPureza:98%Forma y color:SolidPeso molecular:494.13L-ANAP hydrochloride (1313516-26-5 free base)
<p>L-ANAP hydrochloride is a polarity-sensitive and genetically encodable fluorescent unnatural amino acid.</p>Fórmula:C15H17ClN2O3Pureza:98%Forma y color:SolidPeso molecular:308.76PPAR agonist 1
CAS:<p>PPAR agonist 1 is an agonist of PPAR α/γ, used for reducing blood glucose, lipid levels, reducing body weight, and lowering cholesterol.</p>Fórmula:C20H25NO6SPureza:98%Forma y color:SolidPeso molecular:407.48Keap1-Nrf2-IN-6
<p>Keap1-Nrf2-IN-6 is a potent, selective inhibitor of the Keap1-Nrf2 protein−protein interaction (PPI), demonstrating an inhibitory concentration (IC50) of 41 nM</p>Fórmula:C30H34N4O8SForma y color:SolidPeso molecular:610.68DYSP-C34
CAS:<p>DYSP-C34, a potent ultrasound (US)-triggered multifunctional molecular machine, exhibits a favorable lipophilic/hydrophilic balance, enhanced US-induced</p>Fórmula:C45H47N5O10Forma y color:SolidPeso molecular:817.88CcpA-IN-1
CAS:<p>CcpA-IN-1 is a Staphylococcus aureus antibiotic exhibiting significant bactericidal activity (MICs=460 nM) [1].</p>Fórmula:C77H82F12N8OP3RuPureza:98%Forma y color:SolidPeso molecular:1557.5MSI-1436
CAS:<p>MSI-1436 is a selective, non-competitive the enzyme protein-tyrosine phosphatase 1B (PTB1B)inhibitor(IC50 of appr 1 μM)</p>Fórmula:C37H72N4O5SPureza:98%Forma y color:SolidPeso molecular:685.06ICMT-IN-18
CAS:<p>ICMT-IN-18 (compound 35) serves as an ICMT inhibitor with an IC50 value of 0.066 μM [1].</p>Fórmula:C22H26N2OForma y color:SolidPeso molecular:334.45L-159884
CAS:<p>L-159884 is a radiolabelled, nonpeptide angiotensin II antagonist that is useful for angiotensin II, AT1 receptor imaging</p>Fórmula:C31H30N4O4SForma y color:SolidPeso molecular:554.66KRAS inhibitor-14
CAS:<p>KRAS inhibitor-14 targets G12C (IC50: 0.249 μM) and inhibits p-ERK in cancer cells; promising for pancreatic, colorectal, lung cancers.</p>Fórmula:C20H15Cl3FN3O2SForma y color:SolidPeso molecular:486.77MK-5757
CAS:<p>MK-5757 is an ORL1 antagonist.</p>Fórmula:C25H35N3O3Forma y color:SolidPeso molecular:425.56AP-24567
CAS:<p>AP-24567 is a CYP3A4-mediated metabolite.</p>Fórmula:C28H25F3N6OForma y color:SolidPeso molecular:518.53S-Fcme
CAS:<p>S-Fcme activates multidrug resistance transporter by boosting ATPase activity and competing for drug binding.</p>Fórmula:C19H33NO2SForma y color:SolidPeso molecular:339.54EMD638683 R-Form
CAS:<p>EMD638683 is a highly selective SGK1 inhibitor with IC50 of 3 μM. EMD638683 R-Form is the R-form of EMD638683.</p>Fórmula:C18H18F2N2O4Forma y color:SolidPeso molecular:364.34DG-041
CAS:<p>DG-041: EP3 receptor antagonist, high affinity (IC50: 4.6 & 8.1 nM), inhibits PGE2 in platelets, blood-brain barrier permeable.</p>Fórmula:C23H15Cl4FN2O3S2Pureza:99.77%Forma y color:SolidPeso molecular:592.32Fenquinotrione
CAS:<p>Fenquinotrione, a 4-hydroxyphenylpyruvate dioxygenase (HPPD) inhibitor, exhibits IC50 values of 27.2 and 44.7 nM against HPPD from rice and Arabidopsis thaliana</p>Fórmula:C22H17ClN2O5Forma y color:SolidPeso molecular:424.83Manoalogue
CAS:<p>Manoalogue is a synthetic analog of manoalide and phospholipase A2 antagonist.</p>Fórmula:C19H26O4Forma y color:SolidPeso molecular:318.41Anticancer agent 40
CAS:<p>Anticancer agent 3e targets SKBR-3, SKOV-3, PC-3, U-87 (IC50 ~0.95 nM) and HDF cells (IC50: 2.13 nM).</p>Fórmula:C25H29NO6Forma y color:SolidPeso molecular:439.5RORγt modulator 4
CAS:<p>RORγt modulator 4 is a RORγt modulator that regulates IL-17A production activity in cells derived from mouse spleen.</p>Fórmula:C26H27N3O4SForma y color:SolidPeso molecular:477.58Dihydrexidine
CAS:<p>Dihydrexidine is a full efficacy D1-like dopamine receptor (D1/D5) agonist (IC50: 10 nM for D1 receptor). It also shows potent antiparkinsonian activity.</p>Fórmula:C17H17NO2Pureza:98%Forma y color:SolidPeso molecular:267.32PRMT5-IN-29
CAS:<p>PRMT5-IN-29 is a potent, orally active inhibitor of PRMT5, exhibiting an IC50 value of 1.5 μM, showing promise for use in advanced cancer research [1].</p>Fórmula:C18H20Cl3N5O5Pureza:98%Forma y color:SolidPeso molecular:492.74ThrRS-IN-3
<p>ThrRS-IN-3: Potent inhibitor of Salmonella enterica ThrRS, IC50 = 19 nM, Kd = 34 nM, with antibacterial effects.</p>Fórmula:C31H30Cl2N6O5Forma y color:SolidPeso molecular:637.51PROTAC IRAK4 degrader-8
CAS:<p>PROTAC IRAK4 Degrader-8 (Compound 2) is a PROTAC designed to target IRAK4 with an IC50 of 15.5 nM [1].</p>Fórmula:C43H50ClF2N11O5Pureza:98%Forma y color:SolidPeso molecular:874.38AMD-3329 free base
CAS:<p>AMD-3329 is a potent anti-HIV agent that blocks virus replication by targeting CXCR4, a key receptor for X4 viruses' entry.</p>Fórmula:C34H50N8Forma y color:SolidPeso molecular:570.81RUNX-IN-1
CAS:<p>RUNX-IN-1, also known as Compound Conjugate 1, covalently attaches to RUNX-binding sequences, thereby preventing RUNX proteins from associating with their</p>Fórmula:C71H88Cl2N24O11Pureza:98%Forma y color:SolidPeso molecular:1524.52L-739758
CAS:<p>L-739758 is a glycoprotein IIb/IIIa inhibitor.</p>Fórmula:C22H26N4O5S3Forma y color:SolidPeso molecular:522.66HDM-201 succinate
CAS:<p>HDM-201 succinate is an orally bioavailable human double minute 2 homolog (HDM2) inhibitor with potential antineoplastic activity.</p>Fórmula:C30H30Cl2N6O8Forma y color:SolidPeso molecular:673.5BDW568
CAS:<p>BDW568, a prodrug of BDW-OH, serves as a stimulator of interferon genes (STING) agonist.</p>Fórmula:C12H12N4O2S2Forma y color:SolidPeso molecular:308.38Ambamustine
CAS:<p>Ambamustine (PTT 119): a tripeptide nitrogen mustard, DNA inhibitor/alkylator with antitumor properties, researched for various disorders.</p>Fórmula:C29H39Cl2FN4O4SPureza:98%Forma y color:SolidPeso molecular:629.61Enpp-1-IN-4
CAS:<p>Enpp-1-IN-4: potent enpp-1 inhibitor with potential in cancer research. See patent WO2019177971A1, compound 1.</p>Fórmula:C19H19N5O5SForma y color:SolidPeso molecular:429.45ICMT-IN-51
CAS:<p>ICMT-IN-51 (compound 43) serves as an ICMT inhibitor with an IC50 value of 0.55 μM [1].</p>Fórmula:C21H26FNOForma y color:SolidPeso molecular:327.44SARS-CoV-2-IN-1
CAS:<p>SARS-CoV-2-IN-1 is a potent inhibitor of Mpro(SARS-CoV-2 Mpro, SARS-CoV Mpro and MERS-CoV Mpro with IC50s of 0.67, 0.90 and 0.58 μM, respectively).</p>Fórmula:C31H39N5O7Pureza:98%Forma y color:SolidPeso molecular:593.67CGC 11093
CAS:<p>CGC 11093: A polyamine analog inhibiting human prostate tumor growth in mice; may help regress choroidal neovascularization.</p>Fórmula:C17H42Cl4N4Forma y color:SolidPeso molecular:444.356-PPD
CAS:<p>6-PPD (Antioxidant 4020) is an antioxidant and the most commonly used additive in rubber. It can induce neurodegeneration in Caenorhabditis elegans.</p>Fórmula:C18H24N2Pureza:98.99% - 99.22%Forma y color:SolidPeso molecular:268.4BChE-IN-20
CAS:<p>BChE-IN-20 (compound 7c) is a potent, selective inhibitor of BChE, demonstrating IC50 values of 105 nM for eqBChE and 2.3 nM for hBChE.</p>Fórmula:C27H39N5O2Forma y color:SolidPeso molecular:465.63L-742001 Hydrochloride
CAS:<p>L-742001 Hydrochloride is an RNA polymerase inhibitor.</p>Fórmula:C23H25Cl2NO4Forma y color:SolidPeso molecular:450.36Sipoglitazar
CAS:<p>Sipoglitazar, a PPARγ agonist, is used potentially for the treatment of diabetes.</p>Fórmula:C25H25N3O4SPureza:98%Forma y color:SolidPeso molecular:463.55Antitrypanosomal agent 14
CAS:Antitrypanosomal agent 14 (Compound 1), a potent T.Fórmula:C14H23N3OSPureza:98%Forma y color:SolidPeso molecular:281.42Alpertine HCl
<p>Alpertine HCl is a small molecule compound with anti-neuropathic properties.</p>Fórmula:C25H32ClN3O4Pureza:98.47%Forma y color:SoildPeso molecular:473.99SARS-CoV-2 3CLpro-IN-5
CAS:<p>SARS-CoV-2 3CLpro-IN-5 is a covalent inhibitor targeting the 3C-like protease (3CLpro), exhibiting potent inhibitory activity with an IC50 of 3.8 nM and</p>Fórmula:C22H26ClF2N5O4Pureza:98%Forma y color:SolidPeso molecular:497.92Melafolone
CAS:<p>Melafolone: natural COX-2/EGFR inhibitor, enhances PD-1 therapy by normalizing tumor vessels, lowers PD-L1.</p>Fórmula:C22H24O7Forma y color:SolidPeso molecular:400.42SARS-CoV-2 Mpro-IN-12
CAS:<p>SARS-CoV-2 Mpro-IN-12 (compound D026) serves as an inhibitor of the main protease (Mpro) of SARS-CoV-2, exhibiting antiviral properties [1].</p>Fórmula:C20H17NO3Pureza:98%Forma y color:SolidPeso molecular:319.35ICI-185282
CAS:<p>ICI-185282 is a potent thromboxane receptor antagonist.</p>Fórmula:C18H21F3O5Forma y color:SolidPeso molecular:374.35SC 67655
CAS:<p>SC 67655 is a peptidomimetic that specifically suppresses human leukocyte antigen DRB10401-restricted T cell proliferation.</p>Fórmula:C37H62N6O9Pureza:98%Forma y color:SolidPeso molecular:734.92Bibw 22
CAS:<p>Bibw 22 is a bifunctional modulator of P-glycoprotein and nucleoside transport.</p>Fórmula:C30H43N7O4Pureza:98%Forma y color:SolidPeso molecular:565.71Pomaglumetad methionil hydrochloride
CAS:<p>LY2140023 hydrochloride: oral methionine prodrug of LY404039, a selective mGlu2/3 agonist, studied for schizophrenia.</p>Fórmula:C12H19ClN2O7S2Pureza:98.57%Forma y color:SolidPeso molecular:402.87TIE-2/VEGFR-2 kinase-IN-4
CAS:<p>TIE-2/VEGFR-2 kinase-IN-4, a benzimidazole derivative, serves as a potent inhibitor of the tyrosine kinase receptors TIE-2 and VEGFR-2, exhibiting inhibitory</p>Fórmula:C26H17F4N5O4Forma y color:SolidPeso molecular:539.44ERK-IN-2 free base
CAS:<p>ERK-IN-2 free base inhibits ERK2 (IC50: 1.8 nM); potential off-target effects at >10 μM.</p>Fórmula:C16H17N5O2Forma y color:SolidPeso molecular:311.34Glucagon receptor antagonists-3
CAS:<p>Glucagon receptor antagonist -3 is a highly effective glucagon receptor antagonist.</p>Fórmula:C22H30FNO2Pureza:98%Forma y color:SolidPeso molecular:359.48
