Inhibidores
Los inhibidores son moléculas que se unen a enzimas, receptores u otras proteínas para reducir o bloquear su actividad biológica. Estos compuestos se utilizan ampliamente en la investigación para estudiar vías biológicas, comprender los mecanismos de las enfermedades y desarrollar fármacos terapéuticos. Los inhibidores desempeñan un papel crucial en el tratamiento de diversas enfermedades, incluyendo el cáncer, las enfermedades cardiovasculares y las infecciones. En CymitQuimica, ofrecemos una amplia gama de inhibidores de alta calidad para apoyar su investigación en bioquímica, biología celular y desarrollo farmacéutico.
Subcategorías de "Inhibidores"
- Angiogénesis(2.542 productos)
- Apoptosis(5.816 productos)
- Ciclo celular / Checkpoint(4.466 productos)
- Cromatina / Epigenética(2.252 productos)
- Señalización citoesquelética(1.381 productos)
- Daño al ADN / Reparación del ADN(2.830 productos)
- Endocrinología / Hormonas(3.518 productos)
- Enzima(3.640 productos)
- GPCR / proteína G(8.362 productos)
- Inmunología e inflamación(3.540 productos)
- Virus de la gripe(296 productos)
- Señalización JAK / STAT(405 productos)
- Señalización MAPK(1.201 productos)
- Transportador de membrana / canal de iones(2.809 productos)
- Metabolismo(9.462 productos)
- Microbiología / Virología(7.003 productos)
- Neurociencia(9.942 productos)
- Otros inhibidores(37.827 productos)
- Reducción de oxidación(40 productos)
- Señalización PI3K / Akt / mTOR(1.399 productos)
- Proteasas / Proteasoma(1.598 productos)
- Células madre y Derivados(830 productos)
- Tirosina quinasa / adaptadores(2.012 productos)
- Ubiquitinación(1.651 productos)
Mostrar 16 subcategorías más
Se han encontrado 66618 productos de "Inhibidores"
Ordenar por
Pureza (%)
0
100
|
0
|
50
|
90
|
95
|
100
PF 04449913 maleate
CAS:<p>Smo antagonist, IC50=5 nM; reduces AML cell leukemia potential and self-renewal in mice.</p>Fórmula:C25H26N6O5Forma y color:SolidPeso molecular:490.52UK-157147
CAS:<p>UK-157147 is a substrate for UGT1A1(Km: 105 μM).</p>Fórmula:C23H24N2O7SPureza:98%Forma y color:SolidPeso molecular:472.51AGN 194310
CAS:AGN 194310 (VTP-194310) is retinioic acid receptors (RARs) pan-antagonist. The Kd values of 3 nM, 2 nM, 5 nM for RARα, RARβ, RARγ, respectively[1][2].Fórmula:C28H24O2SForma y color:SolidPeso molecular:424.553,4'-Dihydroxyflavone
CAS:<p>3,4'-Dihydroxyflavone (3,4'-DHF) is an oral active flavonoid. 3,4'-Dihydroxyflavone (3,4'-DHF) shows antiviral activity against Influenza A virus.</p>Fórmula:C15H10O4Pureza:98.33%Forma y color:SolidPeso molecular:254.24CGS 35066
CAS:<p>endothelin-converting enzyme (ECE) inhibitor</p>Fórmula:C16H16NO6PPureza:98%Forma y color:SolidPeso molecular:349.28Purinostat mesylate
CAS:<p>Purinostat mesylate, a selective HDAC inhibitor (IC50: 0.81-11.5 nM), induces apoptosis and has potent anti-leukemic effects.</p>Fórmula:C24H30N10O6SForma y color:SolidPeso molecular:586.63HPK1-IN-35
CAS:<p>HPK1-IN-35 is a potent, selective inhibitor of HPK1, demonstrating an IC50 value of 3.5 nM.</p>Fórmula:C30H32N8O3SForma y color:SolidPeso molecular:584.69Fmoc-VAP-MMAE
CAS:<p>Fmoc-VAP-MMAE is a conjugate utilized in antibody-drug conjugates (ADCs), comprising a tubulin inhibitor, monomethyl auristatin E (MMAE), connected via an ADC</p>Fórmula:C70H98N8O13Forma y color:SolidPeso molecular:1259.57Ro 31-1118
CAS:<p>Ro 31-1118 is a partial agonist of beta-adrenoceptor.</p>Fórmula:C22H30FNO4Forma y color:SolidPeso molecular:391.48WAY 316606 HCl (915759-45-4 free base)
<p>WAY 316606 HCl is a selective small-molecule inhibitor of secreted frizzled-related protein-1 (EC50: 0.65 μM).</p>Fórmula:C18H19F3N2O4S2·HClPureza:98%Forma y color:SolidPeso molecular:484.94NOX2-IN-2
CAS:<p>NOX2-IN-2 (compound 33) is a potent inhibitor of NOX2, disrupting the p47phox-p22phox protein-protein interaction with a dissociation constant (K i) of 0.24 μM.</p>Fórmula:C25H25N7O3Forma y color:SolidPeso molecular:471.515-Azacytidine 5′-triphosphate
CAS:<p>5-Azacytidine 5′-triphosphate (5-aza-CMP), a cytidine analog, selectively inhibits the incorporation of [^3H]CTP into RNA during the DNA-dependent RNA</p>Fórmula:C8H15N4O14P3Forma y color:SolidPeso molecular:484.14Verzistobart
CAS:<p>Verzistobart, an IgG1κ antibody, specifically targets the hepatitis A virus cellular receptor, HAVCR2.</p>Forma y color:LiquidSARS-CoV-2-IN-66
CAS:<p>SARS-CoV-2-IN-66 (1), a derivative of vitamin K, functions as an inhibitor of SARS-CoV-2, exhibiting an effective concentration (EC50) of 70.8 μM in VeroE6/</p>Fórmula:C28H30O2Pureza:98%Forma y color:SolidPeso molecular:398.54Adenylyl cyclase-IN-1
CAS:<p>Adenylyl cyclase-IN-1 is a potential adenylyl cyclase inhibitor for ocular hypotonia research [1].</p>Fórmula:C9H8N2S3Forma y color:SolidPeso molecular:240.37Casein kinase 1δ-IN-10
CAS:<p>Casein kinase 1δ-IN-10 is an inhibitor of casein kinase 1δ (CK1δ).</p>Fórmula:C21H17N3O3Pureza:98%Forma y color:SolidPeso molecular:359.38Phenoxan
CAS:<p>Phenoxan is isolated from Polyangium; inhibits electron transport at NADH-ubiquinone oxidoreductase.</p>Fórmula:C23H25NO4Forma y color:SolidPeso molecular:379.45WAY-313165
CAS:<p>WAY-313165 is an active molecule.</p>Fórmula:C17H25NO2Forma y color:SolidPeso molecular:275.39FTI-2600
CAS:<p>FTI-2600 is a farnesyltransferase inhibitor.</p>Fórmula:C27H18FN5OForma y color:SolidPeso molecular:447.46MC-VA-PAB-Exatecan
CAS:<p>MC-VA-PAB-Exatecan is an agent-linker conjugate designed for Antibody-Drug Conjugate (ADC) applications, comprising the ADC linker (peptide MC-VA-PAB) and the</p>Fórmula:C50H54FN7O11Forma y color:SolidPeso molecular:948.02FLT3-IN-14
CAS:<p>FLT3-IN-14: FLT3 inhibitor; FLT3-WT IC50=5.6nM, FLT3-ITD IC50=1.4nM; blocks Y591 phosphorylation; G1 arrest; pro-apoptotic.</p>Fórmula:C25H24N6O2SForma y color:SolidPeso molecular:472.56ATR-IN-22
CAS:<p>ATR-IN-22 (Compound 34), an orally active ATR inhibitor, exhibits potent anti-proliferative effects on MIAPaCa-2 cells with an IC50 value of less than 1 μM and</p>Fórmula:C25H31N7OPureza:98%Forma y color:SolidPeso molecular:445.56RK-0133114
<p>RK-0133114, R-enantiomer of RK-701, is a G9a inhibitor (IC50 = 3.7 μM) for SCD research.</p>Fórmula:C26H30N4O3Forma y color:SolidPeso molecular:446.54NF-κB-IN-13
CAS:<p>NF-κB-IN-13 (compound 12) markedly suppresses LPS-induced NF-κB activation and NO synthesis in RAW264.7 macrophages, exhibiting anti-inflammatory properties [1</p>Fórmula:C20H20O5Pureza:98%Forma y color:SolidPeso molecular:340.37Isotianil
CAS:<p>Isotianil is a plant defense inducer that activates typical plant defense responses without direct antimicrobial effects, serving as a plant protection agent</p>Fórmula:C11H5Cl2N3OSForma y color:SolidPeso molecular:298.15Topoisomerase II inhibitor 15
CAS:<p>Topoisomerase II inhibitor 15 (compound 2g) serves as a potent apoptotic inducer, exhibiting heightened selectivity for head and neck tumors [1].</p>Fórmula:C15H11Cl2N5Pureza:98%Forma y color:SolidPeso molecular:332.192,3-dinor-8-iso Prostaglandin F1α
CAS:<p>2,3-Dinor-8-iso Prostaglandin F1α (2,3-dinor-8-iso PGF1α), an isoprostane and active metabolite of arachidonic acid deriving its formation from non-enzymatic</p>Fórmula:C18H32O5Forma y color:SolidPeso molecular:328.402-Quinizarincarboxylic acid
CAS:<p>Compound 15, 2-Quinizarincarboxylic acid, functions as a glucose uptake inhibitor, demonstrating a 24.9% inhibition rate at a concentration of 50 μM [1].</p>Fórmula:C15H8O6Forma y color:SolidPeso molecular:284.22TLR4 agonist-1
CAS:<p>TLR4 agonist-1 (compound 17a) serves as a potent activator of Toll-like Receptor 4 (TLR4) and stimulates the production of MIP-1β in RAW 264.7 and MM6 cells [1</p>Fórmula:C81H158N3O15PForma y color:SolidPeso molecular:1445.11Plecstatin-1
CAS:<p>Plecstatin-1, an organoruthenium compound, serves as a potent anti-cancer agent that selectively targets plectin—a scaffold protein and cytolinker—within tumor</p>Fórmula:C22H23Cl2FN2RuSForma y color:SolidPeso molecular:538.47GLUT4 activator 1
CAS:<p>GLUT4 activator 1 is a potent glucose transporter type 4 (GLUT4) translocation activator (EC50: 0.14 μM).</p>Fórmula:C23H21FN4O3SPureza:98%Forma y color:SolidPeso molecular:452.5Phosphazide
CAS:<p>Phosphazide is a zidovudine prodrug.</p>Fórmula:C10H14N5O6PForma y color:SolidPeso molecular:331.22BI-11634
CAS:<p>BI-11634 is a factor Xa inhibitor.</p>Fórmula:C22H23ClN4NaO4Pureza:98%Forma y color:SolidPeso molecular:465.89URAT1 inhibitor 1
CAS:URAT1 inhibitor 1 (1g) is an inhibitor of uric acid transporter 1 (URAT1) (IC50: 32 nM), has the potential to treat hyperuricemia associated with gout.Fórmula:C19H15Br2N5O2S2Pureza:98%Forma y color:SolidPeso molecular:569.29Lexitropsin 1
CAS:<p>Lexitropsin 1 is a new anticancer drug.</p>Fórmula:C15H19N7O3SPureza:98%Forma y color:SolidPeso molecular:377.42P2X3 antagonist 38
CAS:<p>Compound 38, also known as Compound 4, is a potent, orally active P2X3 antagonist that demonstrates inhibitory activity with IC50 values of 0.132 µM, 0.165 µM,</p>Fórmula:C22H25F3N6O3Pureza:98%Forma y color:SolidPeso molecular:478.47WAY-658674
CAS:<p>WAY-658674 is a bioactive molecule utilized in the research of amyloid diseases and synucleinopathies.</p>Fórmula:C12H13ClN2O2SForma y color:SolidPeso molecular:284.76ICMT-IN-47
CAS:<p>ICMT-IN-47 (compound 26) acts as an ICMT inhibitor with an IC50 value of 0.76 μM [1].</p>Fórmula:C25H35NOForma y color:SolidPeso molecular:365.551-Myristoyl-3-chloropropanediol
CAS:<p>1-Myristoyl-3-chloropropanediol, a 3-monochloropropanediol (3-MCPD) fatty acid ester, induces nephropathy, tubular hyperplasia, and adenomas through chronic</p>Fórmula:C17H33ClO3Forma y color:SolidPeso molecular:320.9AM-156
CAS:<p>AM-156 is a bio-active chemical.</p>Fórmula:C23H24F3NNaO4Forma y color:SolidPeso molecular:458.433RORγt Inverse agonist 6
CAS:<p>RORγt Inverse agonist 6 is an agonist of RORγt inverse. RORγt Inverse agonist 6 can be used in research on Th17-driven autoimmune diseases.</p>Fórmula:C28H29ClN6O5Pureza:99.52%Forma y color:SolidPeso molecular:565.02SRI 6409-94
CAS:<p>SRI 6409-94, a teratogenic analogue of Ro 13-6298, is orally active and utilized as a molecular tool to investigate the impact of retinol's three-dimensional</p>Fórmula:C24H29NO3Pureza:98%Forma y color:SolidPeso molecular:379.49Keap1-Nrf2-IN-6
<p>Keap1-Nrf2-IN-6 is a potent, selective inhibitor of the Keap1-Nrf2 protein−protein interaction (PPI), demonstrating an inhibitory concentration (IC50) of 41 nM</p>Fórmula:C30H34N4O8SForma y color:SolidPeso molecular:610.68RIP2 kinase inhibitor 2
CAS:<p>RIP2 kinase inhibitor 2 is a receptor-interacting protein-2 kinase inhibitor.</p>Fórmula:C21H28N4O4SPureza:98%Forma y color:SolidPeso molecular:432.54TC-5115
CAS:<p>TC-5115 inhibits MLL1 enzyme at 16 nM, promising for treating MLL leukemia.</p>Fórmula:C23H32N8O5SForma y color:SolidPeso molecular:532.62LY 134046
CAS:<p>LY 134046 is an inhibitor of phenylethanolamine-N-methyltransferase (PNMT).</p>Fórmula:C10H11Cl2NPureza:98%Forma y color:SolidPeso molecular:216.11Dendrogenin A
CAS:<p>Dendrogenin A (DDA) is a compound acting as a selective liver X receptor (LXR) modulator, cholesterol epoxide hydrolase inhibitor (Ki = 120 nM), and a metabolic</p>Fórmula:C32H55N3O2Forma y color:SolidPeso molecular:513.80FK706
CAS:<p>FK706, a human neutrophil elastase inhibitor (IC50: 83 nM, Ki: 4.2 nM), also blocks mouse and porcine elastases. Anti-inflammatory.</p>Fórmula:C26H33F3N4NaO7Forma y color:SolidPeso molecular:593.556Ardisin
CAS:<p>Ardisin is a Topoisomerase I and II enzyme inhibitor. Ardisin may have antioxidant effects.</p>Fórmula:C20H32O2Forma y color:SolidPeso molecular:304.47NUC-7738
CAS:<p>NUC-7738 is a 5'-aryloxyphosphoamidoester prodrug of 3'-dA, which regulates 尾-catenin signaling and can be used in cancer research.</p>Fórmula:C26H29N6O7PPureza:97.32% - 97.32%Forma y color:SolidPeso molecular:568.52
