Inhibidores
Los inhibidores son moléculas que se unen a enzimas, receptores u otras proteínas para reducir o bloquear su actividad biológica. Estos compuestos se utilizan ampliamente en la investigación para estudiar vías biológicas, comprender los mecanismos de las enfermedades y desarrollar fármacos terapéuticos. Los inhibidores desempeñan un papel crucial en el tratamiento de diversas enfermedades, incluyendo el cáncer, las enfermedades cardiovasculares y las infecciones. En CymitQuimica, ofrecemos una amplia gama de inhibidores de alta calidad para apoyar su investigación en bioquímica, biología celular y desarrollo farmacéutico.
Subcategorías de "Inhibidores"
- Angiogénesis(2.542 productos)
- Apoptosis(5.816 productos)
- Ciclo celular / Checkpoint(4.466 productos)
- Cromatina / Epigenética(2.252 productos)
- Señalización citoesquelética(1.381 productos)
- Daño al ADN / Reparación del ADN(2.830 productos)
- Endocrinología / Hormonas(3.518 productos)
- Enzima(3.640 productos)
- GPCR / proteína G(8.362 productos)
- Inmunología e inflamación(3.540 productos)
- Virus de la gripe(296 productos)
- Señalización JAK / STAT(405 productos)
- Señalización MAPK(1.201 productos)
- Transportador de membrana / canal de iones(2.809 productos)
- Metabolismo(9.462 productos)
- Microbiología / Virología(7.003 productos)
- Neurociencia(9.942 productos)
- Otros inhibidores(37.827 productos)
- Reducción de oxidación(40 productos)
- Señalización PI3K / Akt / mTOR(1.399 productos)
- Proteasas / Proteasoma(1.598 productos)
- Células madre y Derivados(830 productos)
- Tirosina quinasa / adaptadores(2.012 productos)
- Ubiquitinación(1.651 productos)
Mostrar 16 subcategorías más
Se han encontrado 66618 productos de "Inhibidores"
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U-46619
CAS:U-46619 is an effective thromboxane A2 (TXA2) agonist and a thromboxane A2 analog (endoperoxide), capable of inducing contraction in the aortic smooth muscle (Fórmula:C21H34O4Pureza:98%Forma y color:SolidPeso molecular:350.49LY52
CAS:LY52 is a matrix metalloproteinase-2 inhibitor. It acts by suppressing tumor invasion and metastasis.Fórmula:C22H24N4O6Pureza:98%Forma y color:SolidPeso molecular:440.45Todralazine hydrochloride
CAS:Todralazine hydrochloride, a β2AR blocker with antioxidant properties, is used in hypertension studies.Fórmula:C11H13ClN4O2Pureza:99.91%Forma y color:SolidPeso molecular:268.7Anticancer agent 128
CAS:<p>Anticancer agent 128 (compound 1) is an IAP inhibitor that covalently binds to the BIR3 domains of XIAP, cIAP1, and cIAP2, exhibiting IC50 values of 24.9 nM, 19</p>Fórmula:C26H38N4O4Pureza:98%Forma y color:SolidPeso molecular:470.6CYT296
CAS:<p>CYT296 is a chromatin de-condensation agent that enhances the efficiency of induced pluripotent stem cell (iPSC) generation mediated by defined factors (OSKM)</p>Fórmula:C18H16O2SPureza:98%Forma y color:SolidPeso molecular:296.38Zandelisib
CAS:<p>Zandelisib is an inhibitor of phosphatidylinositol 3-kinase (PI3K)(p110δ, IC50 of 3.5 nM), and with antineoplastic activity.</p>Fórmula:C31H38F2N8OPureza:99.88%Forma y color:SolidPeso molecular:576.68Homonojirimycin
CAS:<p>Homonojirimycin is an alpha-glucosidase inhibitor.</p>Fórmula:C7H15NO5Pureza:98%Forma y color:SolidPeso molecular:193.2Antituberculosis agent-1
CAS:<p>Antituberculosis Agent-1 (Compound 8a) is an effective antituberculosis agent, demonstrating a minimum inhibitory concentration (MIC) of 3.84 μg/mL against</p>Fórmula:C21H21NO4Forma y color:SolidPeso molecular:351.4SB-682330A
CAS:<p>SB-682330A is a Raf kinase inhibitor.</p>Fórmula:C28H27N3O3Forma y color:SolidPeso molecular:453.53RO5068760
CAS:<p>RO5068760, a selective MEK1/2 inhibitor, effectively targets a range of tumors, particularly B-RafV600E mutants, with an IC50 of 0.025 μM.</p>Fórmula:C28H27FIN3O6Forma y color:SolidPeso molecular:647.43ATR-IN-5
CAS:<p>ATR-IN-5 is a potent inhibitor of ATR, a member of the PIKK family of proteins involved in genome stability and DNA damage repair.</p>Fórmula:C27H32F3N9OForma y color:SolidPeso molecular:555.6Famitinib malate
CAS:<p>Famitinib malate (SHR1020) is a potent oral kinase inhibitor targeting c-kit, VEGFR-2, and PDGFRβ, with IC50s 2.3, 4.7, 6.6 nM, useful for cancer research.</p>Fórmula:C27H33FN4O7Forma y color:SolidPeso molecular:544.57M867
CAS:<p>M867 is a selective, reversible caspase-3 inhibitor, possessing an IC50 of 1.4 nM and a Ki value of 0.7 nM, demonstrating anti-apoptotic activity [1].</p>Fórmula:C27H43N7O6Pureza:98%Forma y color:SolidPeso molecular:561.67pan-KRAS-IN-3
CAS:<p>Pan-KRAS-IN-3 (Example 84) is a pan-KRAS inhibitor suitable for cancer research [1].</p>Fórmula:C33H32F3N5O2Pureza:98%Forma y color:SolidPeso molecular:587.63TPC-144
CAS:<p>TPC-144: Potent, selective reversible LSD1 inhibitor with antitumor effects in AML/SCLC cells and xenografts.</p>Fórmula:C31H31F2N3O2Pureza:98%Forma y color:SolidPeso molecular:515.59Antitumor agent-73
CAS:<p>Antitumor Agent-73, derived from Diosgenin, blocks STAT3 and activates Pdia3, showing strong cancer cell line efficacy.</p>Fórmula:C50H82BrO4PPureza:98%Forma y color:SolidPeso molecular:858.06Catechin 3-rhamnoside
CAS:Catechin 3-rhamnoside has antioxidant activity.Fórmula:C21H24O10Pureza:98%Forma y color:SolidPeso molecular:436.41VU0531245
CAS:<p>VU0531245 is a potent inhibitor of the SLACK (Sequence Like A Calcium-activated K+) channel, exhibiting an IC50 of 2.1 μM [1].</p>Fórmula:C17H17N3O4S2Forma y color:SolidPeso molecular:391.47PDK4-IN-1 hydrochloride
CAS:<p>PDK4-IN-1 hydrochloride is an anthraquinone derivative and a potent and orally active inhibitor of pyruvate dehydrogenase kinase 4 (PDK4, IC50 value = 84 nM).</p>Fórmula:C22H20ClN3O2Pureza:99.67%Forma y color:SolidPeso molecular:393.87IIIM-8
CAS:<p>IIIM-8 is a melanogenesis inhibitor that suppresses pigment production in both in vitro and in vivo settings, exhibiting no cytotoxic effects on Human Adult</p>Fórmula:C14H17NO4Pureza:98%Forma y color:SolidPeso molecular:263.29PDE12-IN-3
CAS:<p>PDE12-IN-3 is an inhibitor of phosphodiesterase 12 (PDE12) (pXC50 of 7.68),with antiviral activity.</p>Fórmula:C29H25N5O3Pureza:98%Forma y color:SolidPeso molecular:491.54Cochliodone A
CAS:<p>Cochliodone A, a bioactive compound isolated from the deep-sea fungus Chaetomium sp., exhibits both antibacterial and anticancer properties.</p>Fórmula:C34H38O12Forma y color:SolidPeso molecular:638.66Nurr1 agonist 4
CAS:<p>Nurr1 agonist 4 (compound 8) serves as a potent Nurr1 agonist, exhibiting an EC50 value of 2.1 μM [1].</p>Fórmula:C12H10O4Pureza:98%Forma y color:SolidPeso molecular:218.21BMS-189664
CAS:<p>BMS-189664 is an inhibitor of thrombin.</p>Fórmula:C22H34N6O4SPureza:98%Forma y color:SolidPeso molecular:478.61CGS 35066
CAS:<p>endothelin-converting enzyme (ECE) inhibitor</p>Fórmula:C16H16NO6PPureza:98%Forma y color:SolidPeso molecular:349.28ICMT-IN-4
CAS:<p>ICMT-IN-4 (compound 28) serves as an inhibitor of ICMT, exhibiting an IC50 value of 0.27 μM [1].</p>Fórmula:C22H29NO2Forma y color:SolidPeso molecular:339.47S1P1 agonist 6 hemicalcium
CAS:<p>Compound I (S1P1 agonist 6 hemicalcium) is an S1P1 agonist that diminishes autoimmune activity by inhibiting lymphocyte trafficking, and serves as an</p>Fórmula:C25H26F3NO3CaPureza:98%Forma y color:SolidPeso molecular:465.51T-448 free base
CAS:<p>T-448 free base is a specific, orally active and irreversible lysine-specific demethylase 1 (LSD1, an H3K4 demethylase) inhibitor(IC50 of 22 nM).</p>Fórmula:C17H20N4OSPureza:98%Forma y color:SolidPeso molecular:328.43HIV-IN-8
CAS:<p>HIV-IN-8 (Compound 9) acts as an HIV inhibitor, suppressing HIV replication with an effective concentration (EC50) of 13 μg/mL [1].</p>Fórmula:C36H30O16Forma y color:SolidPeso molecular:718.61KRAS G12C inhibitor 5
CAS:<p>KRAS G12C inhibitor 5 is a KRas G12C inhibitor.</p>Fórmula:C32H37N7O2Pureza:98%Forma y color:SolidPeso molecular:551.68Z1078601926
CAS:<p>Z1078601926 is an allosteric inhibitor of the human dopamine transporter (hDAT) and exhibits a synergistic effect when combined with Nomifensine [1].</p>Fórmula:C14H19FN2OForma y color:SolidPeso molecular:250.31WEHI-345 analog
CAS:<p>WEHI-345 analog is an Src inhibitor.</p>Fórmula:C23H25N7OPureza:98%Forma y color:SolidPeso molecular:415.49FAAH/cPLA2α-IN-1
CAS:<p>FAAH/cPLA2α-IN-1 is a compound that simultaneously inhibits both FAAH and cPLA2α, demonstrating potent activity with half-maximal inhibitory concentrations (</p>Fórmula:C19H26N4O5Pureza:98%Forma y color:SolidPeso molecular:390.43PAC1R antagonist 1
CAS:<p>PAC1R antagonist 1 is a PAC1 receptor antagonist that inhibits the activation of peptides by pituitary adenylate cyclase and can be used to study tumours.</p>Fórmula:C17H17ClN6O2Pureza:98.43%Forma y color:SolidPeso molecular:372.81CXCR4 antagonist 7
CAS:<p>Compound PARA-B, a CXCR4 antagonist with IC50 = 9.3 nM, targets HIV, cancer, inflammatory diseases, and WHIM syndrome.</p>Fórmula:C15H17N5O3Forma y color:SolidPeso molecular:315.33A81988
CAS:A81988 is an antagonist of angiotensin AT1 receptors.Fórmula:C23H22N6O2Pureza:98%Forma y color:SolidPeso molecular:414.46D-Ala-Lys-AMCA
CAS:<p>D-Ala-Lys-AMCA, a PEPT1 substrate, transports into Caco-2/liver cancer cells with blue fluorescence.</p>Fórmula:C21H28N4O6Pureza:98%Forma y color:SolidPeso molecular:432.47FR-234938
CAS:<p>FR-234938 is a non-nucleoside adenosine deaminase inhibitor with anti-inflammatory activity.</p>Fórmula:C19H21N3O2Pureza:98%Forma y color:SolidPeso molecular:323.39Piperidione
CAS:<p>Piperidione is a cough-suppressing agent [1].</p>Fórmula:C9H15NO2Forma y color:SolidPeso molecular:169.22L-826141
CAS:<p>L-826141 is an inhibitor of phosphodiesterase 4.</p>Fórmula:C25H19F10NO4Pureza:98%Forma y color:SolidPeso molecular:587.41BMS 433796
CAS:<p>BMS 433796 is a γ-secretase inhibitor that demonstrates Aβ-lowering activity within a transgenic mouse model of Alzheimer's disease.</p>Fórmula:C21H20F2N4O4Pureza:99.17%Forma y color:SolidPeso molecular:430.4BN 52256
CAS:<p>BN 52256 helps reduce arrhythmias.</p>Fórmula:C19H19NOSeForma y color:SolidPeso molecular:356.32LY2033298
CAS:<p>LY2033298 enhances oximoline's effect on hamster circadian rhythms, aiding neurosystem disorders.</p>Fórmula:C13H14ClN3O2SPureza:99.06%Forma y color:SolidPeso molecular:311.79Anti-inflammatory agent 46
CAS:<p>Anti-inflammatory agent 46 (compound 7h), exhibiting nitric oxide (NO) inhibitory properties, demonstrates a high affinity for iNOS through low binding energies</p>Fórmula:C24H19FN2O3SPureza:98%Forma y color:SolidPeso molecular:434.48FR-181157
CAS:<p>FR-181157, a novel prostaglandin (PG) mimetic, shows high potency and agonist efficacy at the IP receptor and has good bioavailability.</p>Fórmula:C30H27NNaO4Pureza:98%Forma y color:SolidPeso molecular:488.539Lp-PLA2-IN-2
CAS:Lp-PLA2-IN-2 is a selective and potent lipoprotein-associated phospholipase A2 (Lp-PLA2) inhibitor, with an IC50 0f 120 nM for recombinant human Lp-PLA2.Fórmula:C19H23FN2O4SPureza:98%Forma y color:SolidPeso molecular:394.46p-Tolylmaleimide
CAS:<p>p-Tolylmaleimide (p Tolylmaleimide) is an inhibitor of the water channel and binds to Aquaporin Z.</p>Fórmula:C11H9NO2Pureza:99.94%Forma y color:SolidPeso molecular:187.19Delmitide acetate
CAS:<p>Delmitide acetate (RDP58) is an orally active d-isomer decapeptide that exhibits potent anti-inflammatory properties.</p>Fórmula:C61H109N17O13Pureza:98%Forma y color:SolidPeso molecular:1288.62Ilaprazole sodium hydrate
CAS:<p>Ilaprazole sodium hydrate (IY-81149 sodium hydrate) is a proton pump inhibitor that blocks the transport of HSV particles.</p>Fórmula:C19H21N4NaO4SPureza:99.2%Forma y color:SolidPeso molecular:424.45LM-1484
CAS:<p>LM-1484 displays a higher affinity for 3H-LTC4 sites and is an antagonist of CysLT1 receptor.</p>Fórmula:C28H24N4O3Pureza:98%Forma y color:SolidPeso molecular:464.52
